G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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S1P1 agonist 6 hemicalcium
CAS:2941310-03-6
Compound I (S1P1 agonist 6 hemicalcium) is an S1P1 agonist that diminishes autoimmune activity by …
Formula:
C25H26F3NO3Ca
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
465.51
Ref: TM-T79817
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 6 May 2025
RBC10
CAS:362503-73-9
RBC10 inhibits the binding of Ral to its effector RALBP1, as well as inhibiting Ral-mediated …
Formula:
C24H25ClN2O2
Purity:
98.38%
Color and Shape:
Solid
Molecular weight:
408.92
Ref: TM-T24706
| 1mg | 34.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 80.00 € | ||
| 10mg | 116.00 € | ||
| 25mg | 259.00 € | ||
| 50mg | 374.00 € | ||
| 100mg | 545.00 € | ||
| 200mg | 740.00 € | ||
| 1mL*10mM (DMSO) | 86.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
Talibegron hydrochloride
CAS:178600-17-4
Talibegron hydrochloride: β3 adrenoceptor agonist, pD2 3.72, relaxes rat arteries, reduces leptin in mice.
Formula:
C18H22ClNO4
Purity:
99.82%
Color and Shape:
Solid
Molecular weight:
351.83
Ref: TM-T23557
| 1mg | 35.00 € | ||
| 5mg | 71.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 248.00 € | ||
| 100mg | 338.00 € | ||
| 200mg | 460.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
Ubrogepant
CAS:1374248-77-7
Ubrogepant (MK-1602) is an antagonist of calcitonin gene-related peptide receptor that can be used in …
Formula:
C29H26F3N5O3
Purity:
99.79%
Color and Shape:
Solid
Molecular weight:
549.54
Ref: TM-T17194
| 1mg | 153.00 € | ||
| 5mg | 378.00 € | ||
| 10mg | 597.00 € | ||
| 25mg | 929.00 € | ||
| 50mg | 1,225.00 € | ||
| 100mg | 1,681.00 € | ||
| 1mL*10mM (DMSO) | 487.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
5-HT2A receptor agonist-3
CAS:1391499-52-7
5-HT2A receptor agonist-3 represents the highest selectivity for the human 5-HT2A receptor currently identified, exhibiting …
Formula:
C21H26BrNO3
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
420.34
Ref: TM-T79155
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 6 May 2025
Selvigaltin
CAS:1978336-95-6
Selvigaltin (GB1211) is a Gal-3 inhibitor with potential anticancer activity. Selvigaltin is used in the …
Formula:
C19H16BrF3N4O4S
Purity:
99.97%
Color and Shape:
Liquid
Molecular weight:
533.32
Ref: TM-T63751
| 1mg | 274.00 € | ||
| 5mg | 655.00 € | ||
| 10mg | 1,121.00 € | ||
| 25mg | 2,365.00 € | ||
| 50mg | 3,753.00 € | ||
| 100mg | 5,663.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
Tedalinab
CAS:916591-01-0
Tedalinab is an effective and selective cannabinoid receptor 2 agonist.
Formula:
C19H21F2N3O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
345.39
Ref: TM-T17027
| 25mg | 1,084.00 € | ||
| 50mg | 1,415.00 € | ||
| 100mg | 2,242.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
Brilaroxazine
CAS:1239729-06-6
Brilaroxazine (RP5063): multimodal dopamine/5-HT modulator, partial agonist at D2/D3/D4, 5-HT1A/2A, and antagonist at 5-HT2B/7.
Formula:
C22H25Cl2N3O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
450.36
Ref: TM-T14782
| 1mg | 105.00 € | ||
| 5mg | 250.00 € | ||
| 10mg | 406.00 € | ||
| 25mg | 700.00 € | ||
| 50mg | 1,008.00 € | ||
| 100mg | 1,378.00 € | ||
| 500mg | 2,737.00 € | ||
| 1mL*10mM (DMSO) | 368.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
MOR agonist-1
CAS:2305781-14-8
MOR Agonist-1 is a μ-opioid receptor (MOR) agonist noted for its potent analgesic properties and …
Formula:
C22H26ClFN2O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
404.91
Ref: TM-T79060
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 6 May 2025
(±)-N-Methylcoclaurine
CAS:1472-62-4
N-Methylcoclaurine (±) acts as a selective antagonist at the α2-adrenoceptor [1].
Formula:
C18H21NO3
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
299.36
Ref: TM-T79641
| 25mg | 1,872.00 € | ||
| 50mg | 2,452.00 € | ||
| 100mg | 3,230.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
NKP608
CAS:177707-12-9
NKP608 is a NK-1 receptor antagonist with anticancer and anxiolytic activities.
Formula:
C31H24ClF6N3O2
Purity:
99.88% - 99.88%
Color and Shape:
Solid
Molecular weight:
619.99
Ref: TM-TQ0087
| 2mg | 149.00 € | ||
| 5mg | 246.00 € | ||
| 25mg | 727.00 € | ||
| 50mg | 945.00 € | ||
| 100mg | 1,501.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
BLT2 antagonist-1
CAS:2069220-61-5
BLT2 antagonist-1 (compound 15b) is a selective inhibitor of the BLT2 receptor, impeding the chemotaxis …
Formula:
C26H26FNO4
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
435.49
Ref: TM-T79418
| 25mg | 1,586.00 € | ||
| 50mg | 2,072.00 € | ||
| 100mg | 2,660.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
PSB-603
CAS:1092351-10-4
PSB-603 is a selective antagonist of Adenosine A2B receptor(Ki = 0.553 nM) with anti-inflammatory effects.
Formula:
C24H25ClN6O4S
Purity:
97.13%
Color and Shape:
Solid
Molecular weight:
529.01
Ref: TM-T23203
| 1mg | 37.00 € | ||
| 5mg | 97.00 € | ||
| 10mg | 160.00 € | ||
| 25mg | 344.00 € | ||
| 50mg | 562.00 € | ||
| 100mg | 938.00 € | ||
| 200mg | 1,264.00 € | ||
| 1mL*10mM (DMSO) | 111.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
LPA1 receptor antagonist 1
CAS:1396006-71-5
LPA1 receptor antagonist 1(LPA1 R antagonist 1) is a lysophosphatidic acid receptor antagonist for the …
Formula:
C28H26N4O4
Purity:
99.46% - 99.58%
Color and Shape:
Solid
Molecular weight:
482.53
Ref: TM-T15785
| 1mg | 144.00 € | ||
| 5mg | 349.00 € | ||
| 10mg | 557.00 € | ||
| 25mg | 873.00 € | ||
| 50mg | 1,169.00 € | ||
| 100mg | 1,586.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
(±)-Prenalterol
CAS:57526-81-5
(±)-Prenalterol (H 80/62) is an agonist of beta-2- and beta-1-adrenergic receptors and is used to …
Formula:
C12H19NO3
Purity:
99.71%
Color and Shape:
Liquid
Molecular weight:
225.28
Ref: TM-T25984
| 1mg | 88.00 € | ||
| 5mg | 187.00 € | ||
| 10mg | 303.00 € | ||
| 25mg | 507.00 € | ||
| 50mg | 722.00 € | ||
| 100mg | 938.00 € | ||
| 200mg | 1,311.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
Cenerimod
CAS:1262414-04-9
Cenerimod (ACT-334441) is an S1P1 agonist used in the study of murine experimental autoimmune encephalomyelitis …
Formula:
C25H31N3O5
Purity:
97.43%
Color and Shape:
Solid
Molecular weight:
453.53
Ref: TM-T14924
| 2mg | 42.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 94.00 € | ||
| 1mL*10mM (DMSO) | 67.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
Ogremorphin
CAS:352563-21-4
Ogremorphin (GPR68-IN-1) is a potent inhibitor of GPR68, exhibiting an EC50 of 170 nM.it is …
Formula:
C21H17N3OS
Purity:
99.65% - 99.65%
Color and Shape:
Liquid
Molecular weight:
359.44
Ref: TM-T79209
| 1mg | 379.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
BMS-960
CAS:1265321-86-5
BMS-960 is an S1P agonist with potential anti-tumour activity for cancer research.
Formula:
C26H23F3N4O5
Purity:
97.74% - 99.28%
Color and Shape:
Solid
Molecular weight:
528.48
Ref: TM-T26866
| 1mg | 712.00 € | ||
| 5mg | 1,483.00 € | ||
| 25mg | 2,688.00 € | ||
| 50mg | 4,019.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
PAC1R antagonist 1
CAS:2305204-24-2
PAC1R antagonist 1 is a PAC1 receptor antagonist that inhibits the activation of peptides by …
Formula:
C17H17ClN6O2
Purity:
98.43%
Color and Shape:
Liquid
Molecular weight:
372.81
Ref: TM-T78105
| 1mg | 146.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
PZ-1190
CAS:1852517-78-2
PZ-1190, a multitarget ligand for serotonin and dopamine receptors, exhibits potential antipsychotic activity in rodents …
Formula:
C27H30N4O2S2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
506.68
Ref: TM-T81336
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 6 May 2025
