G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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GLPG0974
CAS:1391076-61-1
GLPG0974 is an antagonist of FFA2/GPR43 with IC50 of 9 nM.
Formula:
C25H25ClN2O4S
Purity:
99.58%
Color and Shape:
Solid
Molecular weight:
484.99
Ref: TM-T15388
| 1mg | 55.00 € | ||
| 1ml | 125.00 € | ||
| 5mg | 118.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 368.00 € | ||
| 50mg | 547.00 € |
Estimated delivery in United States, on Friday 3 Jan 2025
Norbinaltorphimine dihydrochloride
CAS:113158-34-2
Norbinaltorphimine dihydrochloride is a selective and potent κ opioid receptor antagonist that induces itch-associated responses …
Formula:
C40H45Cl2N3O6
Purity:
≥98%
Color and Shape:
Solid
Molecular weight:
734.71
Ref: TM-T12241
| 1mg | 40.00 € | ||
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 3 Jan 2025
Rodatristat ethyl
CAS:1673571-51-1
Rodatristat ethyl is an oral TPH1 inhibitor reducing 5-HT levels & lowering PAH at low …
Formula:
C29H31ClF3N5O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
590.04
Ref: TM-T16779
| 25mg | 2,233.00 € | ||
| 50mg | 3,615.00 € | ||
| 100mg | 5,781.00 € |
Estimated delivery in United States, on Friday 3 Jan 2025
SB 243213 dihydrochloride
CAS:1780372-25-9
SB 243213 dihydrochloride is an orally active, selective and high-affinity antagonist of 5-hydroxytryptamine (5-HT)2C receptor(pKi …
Formula:
C22H21Cl2F3N4O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
501.33
Ref: TM-T12859L
| 1mg | 108.00 € | ||
| 5mg | 313.00 € |
Estimated delivery in United States, on Friday 3 Jan 2025
Befiradol hydrochloride
CAS:2436760-81-3
Befiradol HCl (NLX-112) is a selective 5-HT1A receptor agonist with anxiolytic effects and prevents ATXN3 …
Formula:
C20H23Cl2F2N3O
Purity:
99.1%
Color and Shape:
Solid
Molecular weight:
430.32
Ref: TM-T62385
| 1mg | 149.00 € | ||
| 2mg | 213.00 € | ||
| 5mg | 357.00 € | ||
| 10mg | 522.00 € | ||
| 25mg | 841.00 € | ||
| 50mg | 1,160.00 € | ||
| 100mg | 1,556.00 € |
Estimated delivery in United States, on Friday 3 Jan 2025
PF-4693627
CAS:1312815-93-2
PF-4693627 is an effective and selective microsomal prostaglandin E synthase-1 inhibitor (IC50=3 nM).
Formula:
C26H29Cl2N3O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
502.43
Ref: TM-T16504
| 1mg | 167.00 € | ||
| 5mg | 757.00 € | ||
| 10mg | 1,413.00 € | ||
| 500µg | 92.00 € |
Estimated delivery in United States, on Friday 3 Jan 2025
Taranabant
CAS:701977-09-5
Taranabant: potent CB1 receptor inverse agonist; inhibits agonists with 0.13 nM Ki in vitro.
Formula:
C27H25ClF3N3O2
Purity:
99.06% - 99.06%
Color and Shape:
Solid
Molecular weight:
515.96
Ref: TM-T13080L
| 1mg | 98.00 € |
Estimated delivery in United States, on Friday 3 Jan 2025
AZD5462
CAS:2787501-83-9
AZD5462 is a potent orally available relaxin receptor RXFP1 agonist for the study of heart …
Formula:
C30H41FN2O6
Purity:
99.63%
Color and Shape:
Solid
Molecular weight:
544.65
Ref: TM-T63838
| 1mg | 355.00 € | ||
| 5mg | 836.00 € | ||
| 10mg | 1,207.00 € | ||
| 25mg | 1,882.00 € | ||
| 50mg | 2,642.00 € | ||
| 100mg | 3,268.00 € |
Estimated delivery in United States, on Friday 3 Jan 2025
BMS-986141
CAS:1478711-48-6
BMS-986141(UDM-003183) is a selective and potent protease-activated receptor-4 (PAR-4) antagonist with oral activity and an …
Formula:
C27H23N5O5S2
Purity:
98.36% - 99.11%
Color and Shape:
Solid
Molecular weight:
561.63
Ref: TM-T63966
| 1mg | 894.00 € | ||
| 2mg | 1,189.00 € | ||
| 5mg | 1,792.00 € | ||
| 10mg | 2,210.00 € | ||
| 25mg | 2,962.00 € | ||
| 50mg | 3,678.00 € |
Estimated delivery in United States, on Friday 3 Jan 2025
LY2794193
CAS:2173037-97-1
LY2794193 is a highly effective and selective agonist of the mGlu3 receptor (hmGlu3 Ki=0.927 nM,EC50=0.47 …
Formula:
C16H18N2O6
Color and Shape:
Solid
Molecular weight:
334.32
Ref: TM-T15807
| 5mg | 490.00 € | ||
| 25mg | 1,679.00 € | ||
| 50mg | 2,209.00 € | ||
| 100mg | 3,061.00 € |
Estimated delivery in United States, on Friday 3 Jan 2025
H3R-IN-1 Hydrochloride
CAS:2319790-07-1
H3R-IN-1 Hydrochloride is an inverse agonist of histamine receptor 3( H3R ) .
Formula:
C19H24ClN3O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
377.87
Ref: TM-T11531
| 25mg | 1,030.00 € | ||
| 50mg | 1,356.00 € | ||
| 100mg | 2,131.00 € |
Estimated delivery in United States, on Friday 3 Jan 2025
SGL5213
CAS:1240305-17-2
SGL5213 is a potent oral SGLT1 inhibitor (IC50: 29 nM) with potential for treating type …
Formula:
C37H55N3O8
Purity:
98%
Color and Shape:
Solid
Molecular weight:
669.85
Ref: TM-T12892
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Friday 3 Jan 2025
Rolapitant hydrochloride
CAS:858102-79-1
Rolapitant HCl is a potent NK1 antagonist, non-CYP3A4 interactive, with anti-emetic effects and a Ki …
Formula:
C25H27ClF6N2O2
Purity:
98.35% - 99.79%
Color and Shape:
Solid
Molecular weight:
536.94
Ref: TM-T3724
| 1mg | 240.00 € | ||
| 1ml | 727.00 € | ||
| 5mg | 596.00 € | ||
| 10mg | 848.00 € | ||
| 25mg | 1,280.00 € | ||
| 50mg | 1,719.00 € | ||
| 100mg | 2,336.00 € |
Estimated delivery in United States, on Friday 17 Jan 2025
Chlorcyclizine hydrochloride
CAS:14362-31-3
Chlorcyclizine hydrochloride is an antagonist of histamine H1.
Formula:
C18H22Cl2N2
Molecular weight:
337.29
Ref: TM-T10794
| 25mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
Cyclizine dihydrochloride
CAS:5897-18-7
Cyclizine dihydrochloride (Marzine hydrochloride) is a histamine H1 antagonist. It is given by mouth or …
Formula:
C18H24Cl2N2
Color and Shape:
Solid
Molecular weight:
339.3
Ref: TM-T3037
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 200mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
Cyclobenzaprine hydrochloride
CAS:6202-23-9
Cyclobenzaprine hydrochloride (MK130 hydrochloride) , a centrally acting muscle relaxant with antidepressant activity, leads to …
Formula:
C20H22ClN
Purity:
99.98%
Color and Shape:
Crystalline Solid
Molecular weight:
311.86
Ref: TM-T1509
| 500mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
Desmopressin
CAS:16679-58-6
Desmopressin (DDAVP)(DDAVP) is the synthetic analogue of the antidiuretic hormone arginine vasopressin.Vasopressin Receptor The antidiuretic …
Formula:
C46H64N14O12S2
Purity:
97.45%
Color and Shape:
Solid
Molecular weight:
1069.22
Ref: TM-T5019
| 1mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information |
Xylazine hydrochloride
CAS:23076-35-9
Xylazine hydrochloride (BAY 1470 hydrochloride) is an adrenergic alpha-2 agonist used as a sedative, analgesic …
Formula:
C12H16N2S·HCl
Purity:
99.9%
Color and Shape:
Solid
Molecular weight:
256.79
Ref: TM-T1500
| 10mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 200mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
Naloxone hydrochloride
CAS:357-08-4
Naloxone hydrochloride (Naloxone HCl) is a specific opiate antagonist that has no agonist activity. It …
Formula:
C19H21NO4·HCl
Purity:
97.91%
Color and Shape:
White To Off-White/Powder
Molecular weight:
363.84
Ref: TM-T0102
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 200mg | Discontinued | Request information |
Nalfurafine
CAS:152657-84-6
Nalfurafine (TRK-820) is an effective and selective agonist of G protein-biased κ-opioid receptor with high …
Formula:
C28H32N2O5
Purity:
99.18%
Color and Shape:
Solid
Molecular weight:
476.56
Ref: TM-T41284
| 1mg | Discontinued | Request information | |
| 2mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
