G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
Found 5957 products for "G-protein Coupled Receptors and 7-TM Receptors".
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NESS 0327
CAS:NESS 0327 is a high selectivity antagonist of the cannabinoid CB1 receptor. NESS 0327 is more than 60,000-fold selective for the CB1 receptor.Formula:C24H23Cl3N4OPurity:99.78%Color and Shape:SolidMolecular weight:489.82Ghrelin receptor full agonist-2
CAS:Ghrelin receptor full agonist-2 is a highly potent Ghrelin receptor full agonist.Formula:C26H28ClN5O5SColor and Shape:SolidMolecular weight:558.05ABT 724 trihydrochloride
CAS:ABT-724 trihydrochloride: selective D4 agonist; EC50=12.4nM(human),14.3nM(rat),23.2nM(ferret); for erectile dysfunction research.Formula:C17H22Cl3N5Purity:99.91%Color and Shape:White SolidMolecular weight:402.75Ref: TM-T22019
5mg38.00€1mL*10mM (DMSO)42.00€10mg62.00€25mg119.00€50mg178.00€100mg268.00€200mg398.00€Hemopressin(rat)
CAS:Peptide inhibitor for ep24.15, neurolysin & ACE with Ki 27.76, 3.43, 1.87 μM. Lowers blood pressure, modulates CB1 receptor, reduces pain & food intake.Formula:C53H77N13O12Purity:98%Color and Shape:SolidMolecular weight:1088.27BQ-123 TFA
BQ-123 TFA: Potent ETA antagonist, IC50 = 7.3 nM, Ki = 25 nM, inhibits ET-1 cell proliferation, lowers rat BP.Formula:C33H43F3N6O9Color and Shape:SolidMolecular weight:724.72M40
CAS:Potent, non-selective galanin receptor antagonist (Ki values are 1.82 and 5.1 nM at GAL1 and GAL2 respectively) that inhibits galanin (1-29) binding in ratFormula:C94H145N23O24Purity:98%Color and Shape:SolidMolecular weight:1981.33MAO-B-IN-3
MAO-B-IN-3 is a reversible, selective inhibitor of monoamine oxidase B (MAO-B) with an IC50 of 96 nM and demonstrates affinity for the 5-HT6 receptor with a KiFormula:C24H25N3O2Purity:98%Color and Shape:SolidMolecular weight:387.47BAY-6672 hydrochloride
CAS:BAY-6672 hydrochloride is a potent, selective antagonist of the human Prostaglandin F (FP) receptor, exhibiting an IC50 value of 11 nM.Formula:C26H28BrCl2N3O3Color and Shape:SolidMolecular weight:581.33(R)-(+)-Atenolol
CAS:(R)-(+)-Atenolol ((R)-Atenolol) is a cardioselective beta-1 adrenergic blocker, which properties are similar to propranolol, but without a negative inotropic effect.Formula:C14H22N2O3Purity:98.72%Color and Shape:SolidMolecular weight:266.34Leukotriene B4 Ethanolamide
CAS:LTB4 binds to BLT1 (high affinity) and BLT2. LTB4-EA, a metabolite, is a stronger BLT1 antagonist, suggesting anti-inflammatory properties.Formula:C22H37NO4Color and Shape:SolidMolecular weight:379.541HHS-0701
CAS:HHS-0701: SuTEx ligand, strong PTGR2 inhibitor, blocks 15-Keto-PGE2 metabolism.Formula:C20H20N4O3SPurity:97.24%Color and Shape:SolidMolecular weight:396.46Cetirizine Impurity C dihydrochloride
CAS:Cetirizine Impurity C dihydrochloride is a Cetirizine metabolite and long-acting H1-antihistamine.Formula:C21H27Cl3N2O3Color and Shape:SolidMolecular weight:461.81Spantide II
CAS:Spantide II is an antagonist of tachykinin.Formula:C86H104Cl2N18O13Purity:98%Color and Shape:SolidMolecular weight:1668.77AG 045572
CAS:AG 045572 is a potent GnRH receptor antagonist that inhibits the GnRH receptor in humans and rats with Ki values of 6.0 nM and 3.8 nM, respectively.AG 045572 isFormula:C30H37NO5Purity:99.96%Color and Shape:White SolidMolecular weight:491.62Conessine hydrobromide
CAS:Conessine hydrobromide is a naturally occurring steroid alkaloid and has been used in traditional herbal medicine as a treatment for amoebic dysentery.Formula:C24H41BrN2Color and Shape:SolidMolecular weight:437.51Pancreatic Polypeptide, human
CAS:Endogenous high affinity agonist for human NPY Y4 receptor (Ki = 0.056 nM). Believed to play an important role in the function of the gastrointestinal tract.Formula:C185H287N53O54S2Purity:98%Color and Shape:SolidMolecular weight:4181.71LH-RH (4-10)
CAS:LH-RH (4-10), a heptapeptide from LHRH degradation, is made in macrophages and type II pneumocytes.Formula:C33H53N11O9Color and Shape:SolidMolecular weight:747.84Prolactin-Releasing Peptide (1-31), bovine
Prolactin-Releasing Peptide (1-31), bovine, is a fragment of prolactin-releasing peptide (PrRP).Formula:C44H80N14O15Color and Shape:SolidMolecular weight:1044.59276LAS190792
CAS:LAS190792 (AZD8999) is a dual muscarinic antagonist/β2-agonist, pIC50s (M1-M5, β1-β3): 8.9-5.6; used as a bronchodilator.Formula:C39H43ClN4O9S2Color and Shape:SolidMolecular weight:811.36(Asp28)-Glucagon (1-29) (human, rat, porcine)
CAS:"(Asp28)-Glucagon (1-29) (human, rat, porcine)" is an analog of glucagon with an aspartic acid (Asp) substitution at position 28, notably enhancing its aqueousFormula:C153H224N42O50SColor and Shape:SolidMolecular weight:3483.73
