G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Oxmetidine
CAS:72830-39-8
Oxmetidine (SKF 92994) is an H2R antagonist that inhibits transmembrane calcium flux in the cardiovascular …
Formula:
C19H21N5O3S
Purity:
99.67%
Color and Shape:
Liquid
Molecular weight:
399.47
Ref: TM-T68122
| 1mg | 371.00 € | ||
| 5mg | 881.00 € | ||
| 10mg | 1,188.00 € | ||
| 25mg | 1,745.00 € | ||
| 50mg | 2,385.00 € | ||
| 100mg | 3,211.00 € | ||
| 500mg | 6,449.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Benzquinamide
CAS:63-12-7
Benzquinamide (P2647), an antiemetic agent with anticancer activity, inhibits p-glycoprotein-mediated drug efflux and potentiates the …
Formula:
C22H32N2O5
Purity:
94.86%
Color and Shape:
Solid
Molecular weight:
404.5
Ref: TM-T12343
| 1mg | 651.00 € | ||
| 5mg | 1,674.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
![[Orn5]-URP acetate](https://static.cymitquimica.com/products/TM/thumb/TP1928L1.jpg)
[Orn5]-URP acetate
[Orn5]-URP acetate is an effective and selective Urotensin-II receptor (UT) antagonist (pEC50 = 7.24). [Orn5]-URP …
Formula:
C50H66N10O12S2
Purity:
98.43%
Color and Shape:
Solid
Molecular weight:
1063.25
Ref: TM-TP1928L1
| 1mg | 169.00 € | ||
| 5mg | 367.00 € | ||
| 10mg | 547.00 € | ||
| 25mg | 813.00 € | ||
| 50mg | 1,089.00 € | ||
| 100mg | 1,473.00 € | ||
| 200mg | 1,985.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Gancaonin I
CAS:126716-36-7
Gancaonin I exhibits anti-BsFtsZ GTPase activities; it also shows significant inhibitory activity against B. subtilis, …
Formula:
C21H22O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
354.4
Ref: TM-TN4098
| 5mg | 1,879.00 € | ||
| 1mL*10mM (DMSO) | 2,349.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Galanin-Like Peptide (human)
CAS:245114-99-2
Galanin-Like Peptide (human) is a neuropeptide consisting of 60 amino acids, instrumental in regulating feeding, …
Formula:
C292H451N83O84S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
6500.28
Ref: TM-T80144
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
CYM 50769
CAS:1421365-63-0
CYM 50769 is a neuropeptide W/B receptor 1 (NPBWR1, GPR7) antagonist(IC50 = 0.12 μM).
Formula:
C24H17ClN2O3
Purity:
98% - 98.76%
Color and Shape:
Solid
Molecular weight:
416.86
Ref: TM-T22702
| 1mg | 52.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 171.00 € | ||
| 25mg | 369.00 € | ||
| 50mg | 551.00 € | ||
| 100mg | 783.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
YT 146
CAS:90596-75-1
YT 146 is a biochemical.
Formula:
C18H25N5O4
Purity:
98.81% - 99.72%
Color and Shape:
Solid
Molecular weight:
375.42
Ref: TM-T35282
| 1mg | 274.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 920.00 € | ||
| 25mg | 1,417.00 € | ||
| 50mg | 1,846.00 € | ||
| 100mg | 2,572.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
CAY10678
CAS:1268709-57-4
CAY10678 is an mPGES-1 inhibitor that inhibits PD-1.CAY10678 reduces collagen deposition and T-cell depletion, and …
Formula:
C23H34N4O
Purity:
99.66%
Color and Shape:
Liquid
Molecular weight:
382.54
Ref: TM-T38369
| 1mg | 52.00 € | ||
| 5mg | 119.00 € | ||
| 10mg | 176.00 € | ||
| 25mg | 346.00 € | ||
| 50mg | 523.00 € | ||
| 100mg | 737.00 € | ||
| 500mg | 1,515.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
LE 300
CAS:274694-98-3
LE 300 represents a structurally novel type of antagonists acting preferentially at the dopamine D(1)/D(5)receptors …
Formula:
C20H22N2
Purity:
98.08% - 98.35%
Color and Shape:
Solid
Molecular weight:
290.4
Ref: TM-T22921
| 1mg | 87.00 € | ||
| 5mg | 206.00 € | ||
| 10mg | 306.00 € | ||
| 25mg | 512.00 € | ||
| 50mg | 730.00 € | ||
| 100mg | 994.00 € | ||
| 500mg | 1,988.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
D3R ligand 1
D3R Ligand 1 (compound 23b) is a potent, selective antagonist of the dopamine D3 receptor …
Formula:
C27H37NO5
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
455.59
Ref: TM-T78736
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
2-PCCA hydrochloride
CAS:1609563-70-3
2-PCCA hydrochloride, a racemate, is a potent and selective GPR88 receptor agonist showing inhibition of …
Formula:
C30H39Cl2N3O
Purity:
99.65% - 99.96%
Color and Shape:
Soild
Molecular weight:
528.56
Ref: TM-T80666
| 1mg | 183.00 € | ||
| 5mg | 452.00 € | ||
| 10mg | 647.00 € | ||
| 25mg | 1,003.00 € | ||
| 50mg | 1,392.00 € | ||
| 100mg | 1,828.00 € | ||
| 500mg | 3,671.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
PF-4348235 HCl
PF-4348235 HCl (β2AR/M-receptor agonist-2 HCl) is a muscarinic M3 receptor antagonist (Ki: 0.73 nM) and …
Formula:
C36H50Cl2N4O7S
Purity:
99.66%
Color and Shape:
Liquid
Molecular weight:
753.78
Ref: TM-T72226L
| 1mg | 197.00 € | ||
| 5mg | 488.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
AT-121 hydrochloride
CAS:2099681-71-5
AT-121 hydrochloride: dual nociception/mu-opioid agonist, Ki 3.67/16.49 nM, safe, non-addictive pain reliever with analgesic effects.
Formula:
C24H39ClN4O3S
Purity:
100% - 97.28%
Color and Shape:
Liquid
Molecular weight:
499.11
Ref: TM-T39529
| 1mg | 326.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,050.00 € | ||
| 25mg | 1,487.00 € | ||
| 50mg | 1,852.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
PY-60
CAS:2765218-56-0
PY-60 can effectively activate YAP transcriptional activity against annexin A2 (ANXA2).Cost-effective and quality-assured.
Formula:
C16H15N3O2S
Purity:
98.86% - 99.32%
Color and Shape:
Liquid
Molecular weight:
313.37
Ref: TM-T9566
| 1mg | 112.00 € | ||
| 5mg | 269.00 € | ||
| 10mg | 447.00 € | ||
| 25mg | 733.00 € | ||
| 50mg | 1,003.00 € | ||
| 100mg | 1,380.00 € | ||
| 500mg | 2,756.00 € | ||
| 1mL*10mM (DMSO) | 301.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
PSB 0777 ammonium hydrate
PSB 0777 ammonium hydrate is a potent and selective adenosine A2A receptor full agonist, exhibiting …
Formula:
C18H20N5O7S2·NH4·75H2O
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
532.09
Ref: TM-T78084
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
PSB-1114 triethylamine
PSB-1114 triethylamine is a potent, enzymatically stable, P2Y2 receptor agonist with a 134 nM EC50, …
Formula:
C10H15F2N3O13P3S·xC6H15N
Purity:
98%
Color and Shape:
Liquid
Ref: TM-T78080
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
α-helical CRF 9-41 acetate
α-helical CRF 9-41 acetate is a competitive antagonist of CRF2 (KB = 100 nM) and …
Purity:
96.60%
Color and Shape:
Liquid
Molecular weight:
#N/A
Ref: TM-TP2048L
| 1mg | 200.00 € | ||
| 5mg | 479.00 € | ||
| 10mg | 645.00 € | ||
| 25mg | 974.00 € | ||
| 50mg | 1,301.00 € | ||
| 100mg | 1,775.00 € | ||
| 200mg | 2,393.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Emoghrelin
CAS:928262-58-2
Emoghrelin, extracted from Heshouwu (Polygonum multiflorum), promotes the secretion of growth hormone by activating the …
Formula:
C24H22O13
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
518.42
Ref: TM-T80006
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Pobilukast
CAS:107023-41-6
Pobilukast (SKF 104353) is a cysteinyl leukotriene receptor antagonist that can be used to study …
Formula:
C26H34O5S
Purity:
99.65% - 99.84%
Color and Shape:
Liquid
Molecular weight:
458.61
Ref: TM-T68130
| 1mg | 317.00 € | ||
| 5mg | 751.00 € | ||
| 10mg | 1,065.00 € | ||
| 25mg | 1,584.00 € | ||
| 50mg | 2,068.00 € | ||
| 100mg | 2,647.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
KB-5492 FA
KB-5492 FA is a selective sigma receptor inhibitor with antiulcerogenic effects.CAS 번호128-52-56-8
Formula:
C24H32N2O8
Purity:
98.54%
Color and Shape:
Liquid
Molecular weight:
476.52
Ref: TM-T62396L
| 5mg | 62.00 € | ||
| 10mg | 97.00 € | ||
| 25mg | 189.00 € | ||
| 1mL*10mM (DMSO) | 68.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
