G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Apadenoson TFA
Apadenoson TFA is a potent adenosine A2A receptor (A2AR) agonist that can be used to …
Formula:
C25H31F3N6O8
Purity:
98.40%
Color and Shape:
Soild
Molecular weight:
600.55
Ref: TM-T26641L
| 1mg | 735.00 € | ||
| 5mg | 1,834.00 € | ||
| 25mg | 3,167.00 € | ||
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
AT-121 hydrochloride
CAS:2099681-71-5
AT-121 hydrochloride: dual nociception/mu-opioid agonist, Ki 3.67/16.49 nM, safe, non-addictive pain reliever with analgesic effects.
Formula:
C24H39ClN4O3S
Purity:
100% - 97.28%
Color and Shape:
Solid
Molecular weight:
499.11
Ref: TM-T39529
| 1mg | 326.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,050.00 € | ||
| 25mg | 1,487.00 € | ||
| 50mg | 1,852.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
JHU 75528
CAS:947696-17-5
JHU 75528 (JHU-75528) is a novel PET tracer with inhibitory effects on CB that can …
Formula:
C23H21Cl2N5O2
Purity:
99.97%
Color and Shape:
Solid
Molecular weight:
470.35
Ref: TM-T77634
| 1mg | 183.00 € | ||
| 5mg | 400.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 916.00 € | ||
| 50mg | 1,263.00 € | ||
| 100mg | 1,699.00 € | ||
| 500mg | 3,418.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
AL 34662
CAS:210580-75-9
AL 34662 is a selective and potent 5-HT2A receptor agonist with IC50s of 0.77 nM …
Formula:
C10H13N3O
Purity:
99.77%
Color and Shape:
Solid
Molecular weight:
191.23
Ref: TM-T22029
| 1mg | 41.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | 212.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Latozinemab
Latozinemab (AL001) is a humanized monoclonal antibody targeting Sortilin to study dementia and Alzheimer's.
Purity:
95%
Ref: TM-T77053
| 1mg | 301.00 € | ||
| 5mg | 787.00 € | ||
| 10mg | 1,264.00 € | ||
| 25mg | 1,850.00 € | ||
| 50mg | 2,527.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Quercetin-3'-o-phosphate TEA
Quercetin-3'-o-phosphate TEA (Quercetin 3'-phosphate TEA) is an adenosine A receptor antagonist that can be used …
Formula:
C21H26NO10P
Purity:
95.50%
Color and Shape:
Soild
Molecular weight:
483.41
Ref: TM-T68132L
| 1mg | 182.00 € | ||
| 5mg | 399.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 922.00 € | ||
| 50mg | 1,263.00 € | ||
| 100mg | 1,700.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Stressin I TFA
Stressin I (Cyclo(31-34)[DPhe12, Nle21, 38, Glu31, Lys34]Ac-hCRF(4-41)) TFA, with a K i of 1.7 nM, …
Purity:
98%
Ref: TM-T81081
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
(Iso)-Landipirdine
CAS:1000308-09-7
(Iso)-Landipirdine((Iso)-RO5025181) is a selective and potent 5-HT6R antagonist.
Formula:
C18H19FN2O3S
Purity:
97.27%
Color and Shape:
Soild
Molecular weight:
362.42
Ref: TM-T27795L
| 1mg | 182.00 € | ||
| 5mg | 449.00 € | ||
| 10mg | 643.00 € | ||
| 25mg | 1,003.00 € | ||
| 50mg | 1,384.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
TUG-499
CAS:1206629-08-4
TUG-499 is a selective free fatty acid receptor 1 (FFAR1 or GPR40) agonist (EC50: 7.39).TUG-499 …
Formula:
C16H11Cl2NO2
Purity:
99.59%
Color and Shape:
Soild
Molecular weight:
320.17
Ref: TM-T60184
| 1mg | 52.00 € | ||
| 1ml | 114.00 € | ||
| 5mg | 109.00 € | ||
| 10mg | 157.00 € | ||
| 25mg | 258.00 € | ||
| 50mg | 346.00 € | ||
| 100mg | 453.00 € | ||
| 500mg | 984.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
SLB1122168 formic
SLB1122168 is a potent inhibitor of Spns2-mediated sphingosine-1-phosphate (S1P) release, exhibiting an IC50 value of …
Formula:
C23H37N3O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
403.56
Ref: TM-T78160
| 2mg | 125.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Sonepcizumab
CAS:1031360-18-5
Sonepcizumab, a human monoclonal antibody, targets S1P to combat cancer and prevent post-glaucoma eye scarring.
Purity:
SDS-PAGE:95% SEC-HPLC:98.90%
Color and Shape:
Solid
Ref: TM-T76828
| 1mg | 269.00 € | ||
| 5mg | 616.00 € | ||
| 10mg | 829.00 € | ||
| 25mg | 1,255.00 € | ||
| 50mg | 1,691.00 € | ||
| 100mg | 2,277.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Galanin-Like Peptide (human)
CAS:245114-99-2
Galanin-Like Peptide (human) is a neuropeptide consisting of 60 amino acids, instrumental in regulating feeding, …
Formula:
C292H451N83O84S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
6500.28
Ref: TM-T80144
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
![[DPro10] Dynorphin A (1-11)acetate,porcine](https://static.cymitquimica.com/products/TM/thumb/T76341L.jpg)
[DPro10] Dynorphin A (1-11)acetate,porcine
[DPro10] Dynorphin A (1-11)acetate,porcine is a highly potent κ-opioid receptor agonist with a Ki value …
Formula:
C65H107N21O15
Purity:
99.05%
Color and Shape:
Soild
Molecular weight:
1422.7
Ref: TM-T76341L
| 1mg | 60.00 € | ||
| 5mg | 124.00 € | ||
| 10mg | 176.00 € | ||
| 25mg | 296.00 € | ||
| 50mg | 444.00 € | ||
| 100mg | 646.00 € | ||
| 500mg | 1,364.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
S1R agonist 2 hydrochloride
Compound 8b hydrochloride, a selective S1R agonist, exhibits affinity with K i s of 1.1 …
Formula:
C21H28ClNO
Purity:
98%
Color and Shape:
Solid
Molecular weight:
345.91
Ref: TM-T78087
| 2mg | 94.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Mogamulizumab
CAS:1159266-37-1
Mogamulizumab is a monoclonal antibody targeting CC chemokine receptor 4 with anticancer effects, used in …
Purity:
SDS-PAGE:97.3%;SEC-HPLC:99.4%
Color and Shape:
Solid
Ref: TM-T76782
| 1mg | 445.00 € | ||
| 5mg | 916.00 € | ||
| 10mg | 1,281.00 € | ||
| 25mg | 1,839.00 € | ||
| 50mg | 2,591.00 € | ||
| 100mg | 3,533.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
D3R ligand 1
D3R Ligand 1 (compound 23b) is a potent, selective antagonist of the dopamine D3 receptor …
Formula:
C27H37NO5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
455.59
Ref: TM-T78736
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Samidorphan HCl
CAS:2328045-02-7
Samidorphan HCl is an orally active and highly potent modulator of the opioid system that …
Formula:
C21H27ClN2O4
Purity:
98.25% - 99.60%
Color and Shape:
Soild
Molecular weight:
406.9
Ref: TM-T67888L
| 1mg | 162.00 € | ||
| 5mg | 386.00 € | ||
| 10mg | 573.00 € | ||
| 25mg | 909.00 € | ||
| 50mg | 1,225.00 € | ||
| 100mg | 1,652.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
PSB 0777 ammonium hydrate
PSB 0777 ammonium hydrate is a potent and selective adenosine A2A receptor full agonist, exhibiting …
Formula:
C18H20N5O7S2·NH4·75H2O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
532.09
Ref: TM-T78084
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Galcanezumab
CAS:1578199-75-3
Galcanezumab: humanized IgG4 antibody that targets CGRP for migraine and cluster headache prevention/treatment.
Purity:
SDS-PAGE:95% SEC-HPLC:95%
Color and Shape:
Solid
Ref: TM-T76682
| 1mg | 184.00 € | ||
| 5mg | 551.00 € | ||
| 10mg | 880.00 € | ||
| 25mg | 1,282.00 € | ||
| 50mg | 1,754.00 € | ||
| 100mg | 2,366.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Dazmegrel HCl
Dazmegrel HCl is a platelet thromboxane inhibitor used in the study of myocardial infarction and …
Formula:
C16H18ClN3O2
Purity:
98.63%
Color and Shape:
Solid
Molecular weight:
319.79
Ref: TM-T31213L
| 1mg | 182.00 € | ||
| 5mg | 451.00 € | ||
| 10mg | 645.00 € | ||
| 25mg | 1,007.00 € | ||
| 50mg | 1,389.00 € | ||
| 100mg | 1,836.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
