G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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PSB-1114 triethylamine
PSB-1114 triethylamine is a potent, enzymatically stable, P2Y2 receptor agonist with a 134 nM EC50, …
Formula:
C10H15F2N3O13P3S·xC6H15N
Purity:
98%
Color and Shape:
Solid
Ref: TM-T78080
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Emoghrelin
CAS:928262-58-2
Emoghrelin, extracted from Heshouwu (Polygonum multiflorum), promotes the secretion of growth hormone by activating the …
Formula:
C24H22O13
Purity:
98%
Color and Shape:
Solid
Molecular weight:
518.42
Ref: TM-T80006
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
CB2 receptor agonist 2
CAS:1314230-75-5
CB2 receptor agonist 2 (ZINC72105556): potent, Ki=8.5 nM, high selectivity for CB2.
Formula:
C30H36N2O4
Purity:
98.07%
Color and Shape:
Solid
Molecular weight:
488.62
Ref: TM-T22009
| 1mg | 114.00 € | ||
| 2mg | 172.00 € | ||
| 5mg | 262.00 € | ||
| 10mg | 384.00 € | ||
| 25mg | 603.00 € | ||
| 50mg | 810.00 € | ||
| 100mg | 1,089.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Fenclozine Maleate
CAS:76823-82-0
Fenclozine Maleate (S 1429) is a potential histamine H1 receptor antagonist , which can be …
Formula:
C45H47ClN2O12
Purity:
98.47%
Color and Shape:
Soild
Molecular weight:
843.314
Ref: TM-T83975
| 1mg | 184.00 € | ||
| 5mg | 455.00 € | ||
| 10mg | 651.00 € | ||
| 25mg | 1,016.00 € | ||
| 50mg | 1,401.00 € | ||
| 100mg | 1,853.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
PF-9184
CAS:1221971-47-6
PF-9184 inhibits human mPGES-1 selectively, with an IC50 of 16.5 nM, and reduces IL-1β-stimulated PGE2 …
Formula:
C21H14Cl2N2O4S
Purity:
97.64%
Color and Shape:
Solid
Molecular weight:
461.32
Ref: TM-T21738
| 1mg | 35.00 € | ||
| 5mg | 75.00 € | ||
| 10mg | 102.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Galantide acetate
Galantide acetate, a non-specific galanin receptor antagonist, is a peptide consisting of fragments of galanin …
Formula:
C106H155N25O28S
Purity:
97.8%
Color and Shape:
Solid
Molecular weight:
2259.58
Ref: TM-T15368L
| 1mg | 150.00 € | ||
| 5mg | 382.00 € | ||
| 10mg | 543.00 € | ||
| 25mg | 807.00 € | ||
| 50mg | 1,080.00 € | ||
| 100mg | 1,464.00 € | ||
| 200mg | 1,976.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
difelikefalin acetate(1024828-77-0 Free base)
is a ketone and a building block.
Formula:
C38H57N7O8
Purity:
96.94%
Color and Shape:
Solid
Molecular weight:
739.9
Ref: TM-TP2485
| 1mg | 162.00 € | ||
| 5mg | 325.00 € | ||
| 10mg | 506.00 € | ||
| 25mg | 821.00 € | ||
| 50mg | 1,105.00 € | ||
| 100mg | 1,514.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
SNC 80
CAS:156727-74-1
SNC 80, a non-peptide δ-opioid agonist (Ki=1.78 nM, IC50=2.73 nM), also targets μ-δ heteromers (EC50=52.8 …
Formula:
C28H39N3O2
Purity:
98.67%
Color and Shape:
Solid
Molecular weight:
449.63
Ref: TM-T8414
| 1mg | 41.00 € | ||
| 5mg | 80.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 389.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
(d(CH2)51,Tyr(Me)2,Orn8)-Oxytocin
CAS:77327-45-8
(d(CH2)51,Tyr(Me)2, Orn8)-Oxytocin (OVT) is an antagonist of the oxytocin receptor that finds application in the …
Formula:
C48H74N12O12S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1075.3
Ref: TM-T80126
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Semaglutide Acetate
CAS:1997361-85-9
Semaglutide Acetate is an agonist of a glucagon-like peptide 1 (GLP-1) receptor and can be …
Formula:
C189H295N45O61
Purity:
98.42%
Color and Shape:
Solid
Molecular weight:
4174.68
Ref: TM-T19850L
| 1mg | 222.00 € | ||
| 5mg | 463.00 € | ||
| 10mg | 676.00 € | ||
| 25mg | 1,056.00 € | ||
| 50mg | 1,412.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Azepexole hydrochloride
CAS:147663-20-5
Azepexole hydrochloride (4H-Oxazolo[4,5-d]azepin-2-amine, 6-ethyl-5,6,7,8-tetrahydro-, hydrochloride (1:1)) is a potent α2-Adrenoceptor agonist with anaesthetic
Formula:
C9H16ClN3O
Purity:
98.03% - 99.72%
Color and Shape:
Soild
Molecular weight:
217.7
Ref: TM-T21787L
| 1ml | 42.00 € | ||
| 5mg | 35.00 € | ||
| 10mg | 49.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
FFN246
CAS:2210244-83-8
FFN246, a fluorescent probe, concurrently targets the serotonin transporter (SERT) and vesicular monoamine transporter 2 …
Formula:
C15H13FN2O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
256.27
Ref: TM-T78684
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
WAY-620645
CAS:742116-45-6
WAY-620645 is a CCK antagonist with antitumor and analgesic activities.
Formula:
C22H22N4O2
Purity:
99.91%
Color and Shape:
Solid
Molecular weight:
374.44
Ref: TM-T9991
| 1mg | 39.00 € | ||
| 1ml | 107.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 228.00 € | ||
| 50mg | 324.00 € | ||
| 100mg | 470.00 € | ||
| 200mg | 639.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
DOTA-CXCR4-L
DOTA-CXCR4-L, a peptide targeting the CXCR4 receptor, is utilized in cancer research, notably in the …
Formula:
C58H78N16O14
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1223.34
Ref: TM-T80216
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Patecibart
CAS:2642374-04-5
Patecibart is a humanized immunoglobulin G4-kappa monoclonal antibody that functions as an antagonist to the …
Purity:
98%
Color and Shape:
Solid
Ref: TM-T81538
| 1mg | To inquire | ||
| 5mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Anatibant 2HCl
CAS:209788-45-4
Anatibant 2HCl is a small molecule bradykinin B2 receptor antagonist for the treatment of neurological …
Formula:
C34H36Cl2N6O5S·2ClH
Purity:
99.18% - 99.71%
Color and Shape:
Soild
Molecular weight:
784.58
Ref: TM-T26627L
| 1mg | 327.00 € | ||
| 5mg | 901.00 € | ||
| 10mg | 1,119.00 € | ||
| 25mg | 1,477.00 € | ||
| 50mg | 1,839.00 € | ||
| 100mg | 2,322.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
(3aR,9aR)-Fluparoxan
CAS:105182-47-6
(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration …
Formula:
C10H10FNO2
Purity:
98.68%
Color and Shape:
Soild
Molecular weight:
195.19
Ref: TM-T77566
| 1mg | 182.00 € | ||
| 5mg | 401.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 920.00 € | ||
| 50mg | 1,267.00 € | ||
| 100mg | 1,699.00 € | ||
| 500mg | 3,416.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
6'-GNTI dihydrochloride
CAS:2410327-94-3
6'-GNTI dihydrochloride is a κ-opioid receptor (KOR) agonist that favors activation of G-protein-mediated signaling over …
Formula:
C27H29N5O3·2ClH
Purity:
99.08%
Color and Shape:
Solid
Molecular weight:
544.47
Ref: TM-T39988
| 1mg | 325.00 € | ||
| 5mg | 788.00 € | ||
| 10mg | 1,082.00 € | ||
| 25mg | 1,606.00 € | ||
| 50mg | 2,164.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Spns2-IN-1
Spns2-IN-1 is a potent Spns2 inhibitor, effectively impeding Spns2-dependent S1P transport with an IC50 value …
Purity:
98%
Ref: TM-T81114
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Setmelanotide
CAS:920014-72-8
Setmelanotide (BIM-22493) is a selective agonist of melanocortin 4 receptor (MC4R)(human and rat MC4R with …
Formula:
C49H68N18O9S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1117.31
Ref: TM-T12882
| 1mg | 95.00 € | ||
| 1ml | 448.00 € | ||
| 5mg | 241.00 € | ||
| 10mg | 376.00 € | ||
| 25mg | 679.00 € | ||
| 50mg | 1,099.00 € | ||
| 100mg | 1,497.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
