G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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JHU 75528
CAS:947696-17-5
JHU 75528 (JHU-75528) is a novel PET tracer with inhibitory effects on CB that can …
Formula:
C23H21Cl2N5O2
Purity:
99.97%
Color and Shape:
Liquid
Molecular weight:
470.35
Ref: TM-T77634
| 1mg | 183.00 € | ||
| 5mg | 400.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 916.00 € | ||
| 50mg | 1,263.00 € | ||
| 100mg | 1,699.00 € | ||
| 500mg | 3,418.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Fluparoxan hydrochloride
CAS:105227-44-9
Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or …
Formula:
C10H11ClFNO2
Purity:
99.44%
Color and Shape:
Soild
Molecular weight:
231.65
Ref: TM-T77565
| 1mg | 182.00 € | ||
| 5mg | 401.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 916.00 € | ||
| 50mg | 1,262.00 € | ||
| 100mg | 1,698.00 € | ||
| 500mg | 3,431.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Linzagolix choline
CAS:1321816-57-2
Linzagolix choline is a GnRH antagonist. It can be used to study pain associated with …
Formula:
C27H28F3N3O8S
Purity:
99.64%
Color and Shape:
Solid
Molecular weight:
611.59
Ref: TM-T25742
| 1mg | 185.00 € | ||
| 5mg | 459.00 € | ||
| 10mg | 657.00 € | ||
| 25mg | 1,025.00 € | ||
| 50mg | 1,413.00 € | ||
| 100mg | 1,869.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
(d(CH2)51,Tyr(Me)2,Orn8)-Oxytocin
CAS:77327-45-8
(d(CH2)51,Tyr(Me)2, Orn8)-Oxytocin (OVT) is an antagonist of the oxytocin receptor that finds application in the …
Formula:
C48H74N12O12S2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
1075.3
Ref: TM-T80126
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 12 Dec 2024
Quercetin-3'-o-phosphate TEA
Quercetin-3'-o-phosphate TEA (Quercetin 3'-phosphate TEA) is an adenosine A receptor antagonist that can be used …
Formula:
C21H26NO10P
Purity:
95.50%
Color and Shape:
Soild
Molecular weight:
483.41
Ref: TM-T68132L
| 1mg | 182.00 € | ||
| 5mg | 399.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 922.00 € | ||
| 50mg | 1,263.00 € | ||
| 100mg | 1,700.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
TUG-499
CAS:1206629-08-4
TUG-499 is a selective free fatty acid receptor 1 (FFAR1 or GPR40) agonist (EC50: 7.39).TUG-499 …
Formula:
C16H11Cl2NO2
Purity:
99.59%
Color and Shape:
Soild
Molecular weight:
320.17
Ref: TM-T60184
| 1mg | 52.00 € | ||
| 5mg | 109.00 € | ||
| 10mg | 157.00 € | ||
| 25mg | 258.00 € | ||
| 50mg | 346.00 € | ||
| 100mg | 453.00 € | ||
| 500mg | 984.00 € | ||
| 1mL*10mM (DMSO) | 114.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
SLB1122168 formic
SLB1122168 is a potent inhibitor of Spns2-mediated sphingosine-1-phosphate (S1P) release, exhibiting an IC50 value of …
Formula:
C23H37N3O3
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
403.56
Ref: TM-T78160
| 2mg | 125.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
S1R agonist 2 hydrochloride
Compound 8b hydrochloride, a selective S1R agonist, exhibits affinity with K i s of 1.1 …
Formula:
C21H28ClNO
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
345.91
Ref: TM-T78087
| 2mg | 94.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Astressin acetate
Astressin acetate is an antagonist of corticotropin releasing factor (CRF) with low affinity for the …
Formula:
C163H273N49O44
Purity:
96.87%
Color and Shape:
Liquid
Molecular weight:
3623.21
Ref: TM-TP1448L
| 1mg | 220.00 € | ||
| 5mg | 875.00 € | ||
| 10mg | 1,309.00 € | ||
| 25mg | 2,358.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
CB2 receptor agonist 2
CAS:1314230-75-5
CB2 receptor agonist 2 (ZINC72105556): potent, Ki=8.5 nM, high selectivity for CB2.
Formula:
C30H36N2O4
Purity:
98.07%
Color and Shape:
Solid
Molecular weight:
488.62
Ref: TM-T22009
| 1mg | 114.00 € | ||
| 2mg | 172.00 € | ||
| 5mg | 262.00 € | ||
| 10mg | 384.00 € | ||
| 25mg | 603.00 € | ||
| 50mg | 810.00 € | ||
| 100mg | 1,089.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Fenclozine Maleate
CAS:76823-82-0
Fenclozine Maleate (S 1429) is a potential histamine H1 receptor antagonist , which can be …
Formula:
C45H47ClN2O12
Purity:
98.47%
Color and Shape:
Soild
Molecular weight:
843.314
Ref: TM-T83975
| 1mg | 184.00 € | ||
| 5mg | 455.00 € | ||
| 10mg | 651.00 € | ||
| 25mg | 1,016.00 € | ||
| 50mg | 1,401.00 € | ||
| 100mg | 1,853.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Galantide acetate
Galantide acetate, a non-specific galanin receptor antagonist, is a peptide consisting of fragments of galanin …
Formula:
C106H155N25O28S
Purity:
97.8%
Color and Shape:
Liquid
Molecular weight:
2259.58
Ref: TM-T15368L
| 1mg | 150.00 € | ||
| 5mg | 382.00 € | ||
| 10mg | 543.00 € | ||
| 25mg | 807.00 € | ||
| 50mg | 1,080.00 € | ||
| 100mg | 1,464.00 € | ||
| 200mg | 1,976.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Azepexole hydrochloride
CAS:147663-20-5
Azepexole hydrochloride (4H-Oxazolo[4,5-d]azepin-2-amine, 6-ethyl-5,6,7,8-tetrahydro-, hydrochloride (1:1)) is a potent α2-Adrenoceptor agonist with anaesthetic
Formula:
C9H16ClN3O
Purity:
98.03% - 99.72%
Color and Shape:
Soild
Molecular weight:
217.7
Ref: TM-T21787L
| 5mg | 35.00 € | ||
| 10mg | 49.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 42.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
WAY-620645
CAS:742116-45-6
WAY-620645 is a CCK antagonist with antitumor and analgesic activities.
Formula:
C22H22N4O2
Purity:
99.91%
Color and Shape:
Liquid
Molecular weight:
374.44
Ref: TM-T9991
| 1mg | 62.00 € | ||
| 5mg | 132.00 € | ||
| 10mg | 186.00 € | ||
| 25mg | 388.00 € | ||
| 50mg | 553.00 € | ||
| 100mg | 802.00 € | ||
| 500mg | 1,558.00 € | ||
| 1mL*10mM (DMSO) | 176.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Setmelanotide
CAS:920014-72-8
Setmelanotide (BIM-22493) is a selective agonist of melanocortin 4 receptor (MC4R)(human and rat MC4R with …
Formula:
C49H68N18O9S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1117.31
Ref: TM-T12882
| 1mg | 95.00 € | ||
| 5mg | 241.00 € | ||
| 10mg | 376.00 € | ||
| 25mg | 679.00 € | ||
| 50mg | 1,099.00 € | ||
| 100mg | 1,497.00 € | ||
| 1mL*10mM (DMSO) | 448.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Nemifitide diTFA
CAS:204992-09-6
Nemifitide diTFA is a synthetic pentapeptide with antidepressant properties, resembling MIF, that crosses the blood-brain …
Formula:
C37H45F7N10O10
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
922.8
Ref: TM-TP1127
| 1mg | 91.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Tipelukast
CAS:125961-82-2
Tipelukast (KCA 757), an oral drug for asthma research, blocks leukotrienes and fights inflammation and …
Formula:
C29H38O7S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
530.67
Ref: TM-T15647
| 1mg | 301.00 € | ||
| 5mg | 735.00 € | ||
| 10mg | 1,007.00 € | ||
| 25mg | 1,519.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
β-Endorphin (1-27) (human) acetate
β-Endorphin (1-27) (human) acetate, existing in the hypophysis cerebri and hypothalamus, exhibits antinociception activity.
Formula:
C141H221N33O42S
Purity:
96.52%
Color and Shape:
Liquid
Molecular weight:
3082.52
Ref: TM-T38193L
| 1mg | 111.00 € | ||
| 2mg | 157.00 € | ||
| 5mg | 240.00 € | ||
| 10mg | 355.00 € | ||
| 25mg | 542.00 € | ||
| 50mg | 758.00 € | ||
| 100mg | 1,016.00 € | ||
| 200mg | 1,354.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Sarizotan 2HCl
CAS:177976-12-4
Sarizotan 2HCl is an hERG channel inhibitor and 5-hydroxytryptamine 5-HT1A receptor agonist with potential antidepressant …
Formula:
C22H23Cl2FN2O
Purity:
98.83%
Color and Shape:
Soild
Molecular weight:
421.34
Ref: TM-T70044L
| 1mg | 182.00 € | ||
| 5mg | 451.00 € | ||
| 10mg | 645.00 € | ||
| 25mg | 1,007.00 € | ||
| 50mg | 1,389.00 € | ||
| 100mg | 1,836.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Sincalide ammonium
CAS:70706-98-8
Sincalide ammonium, a CCK analog, stimulates bile release, gallbladder contraction, and sphincter relaxation, aiding in …
Formula:
C49H65N11O16S3
Purity:
98.46%
Color and Shape:
Solid
Molecular weight:
1160.3
Ref: TM-TP1198
| 1mg | 96.00 € | ||
| 5mg | 231.00 € | ||
| 10mg | 369.00 € | ||
| 25mg | 608.00 € | ||
| 50mg | 853.00 € | ||
| 100mg | 1,142.00 € | ||
| 500mg | 2,285.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
