G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Picumeterol FA
picumeterol FA is a potent and selective β2-adrenergic receptor agonist.
Formula:
C22H31Cl2N3O4
Purity:
99.80%
Color and Shape:
Soild
Molecular weight:
472.4
Ref: TM-T68129L1
| 1mg | 182.00 € | ||
| 5mg | 452.00 € | ||
| 10mg | 647.00 € | ||
| 25mg | 1,009.00 € | ||
| 50mg | 1,384.00 € | ||
| 100mg | 1,828.00 € | ||
| 500mg | 3,648.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Tropanserin
CAS:85181-40-4
Tropanserin (MDL 72422) is a 5-hydroxytryptamine receptor antagonist with anxiolytic activity that is used to …
Formula:
C17H23NO2
Purity:
99.74%
Color and Shape:
Solid
Molecular weight:
273.37
Ref: TM-T8451
| 1mg | 45.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 138.00 € | ||
| 25mg | 222.00 € | ||
| 50mg | 333.00 € | ||
| 100mg | 491.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
A 77636 hydrochloride
CAS:145307-34-2
A 77636 hydrochloride is a potent, orally active, selective and long acting dopamine D1 receptor …
Formula:
C20H28ClNO3
Purity:
99.62%
Color and Shape:
Solid
Molecular weight:
365.89
Ref: TM-T21782
| 1mg | 94.00 € | ||
| 5mg | 213.00 € | ||
| 10mg | 310.00 € | ||
| 25mg | 523.00 € | ||
| 50mg | 736.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
CXCL-CXCR1/2-IN-1
CAS:2415653-55-1
CXCL-CXCR1/2-IN-1 is an ELR+CXCL-CXCR1/2 pathway inhibitor with anticancer activity and can be used in the …
Formula:
C14H8Cl2N4O3S
Purity:
99.40%
Color and Shape:
Soild
Molecular weight:
383.21
Ref: TM-T84325
| 5mg | 47.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 124.00 € | ||
| 50mg | 198.00 € | ||
| 100mg | 295.00 € | ||
| 500mg | 705.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Neocarzinostatin
CAS:9014-02-2
Neocarzinostatin is an effective DNA-damaging, anti-tumor antibiotic.
Purity:
98%
Color and Shape:
Solid
Molecular weight:
N/A
Ref: TM-T16283
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Monday 16 Dec 2024
NPS ALX Compound 4a hydrochloride(1:1)
NPS ALX Compound 4a hydrochloride(1:1) is a potent and selective 5-hydroxytryptamine6 (5-HT6) receptor antagonist, with …
Formula:
C25H26ClN3O2S
Purity:
99.8%
Color and Shape:
Soild
Molecular weight:
468.01
Ref: TM-T12262L1
| 1mg | 51.00 € | ||
| 5mg | 110.00 € | ||
| 10mg | 165.00 € | ||
| 25mg | 272.00 € | ||
| 50mg | 394.00 € | ||
| 100mg | 539.00 € | ||
| 200mg | 713.00 € | ||
| 1mL*10mM (DMSO) | 132.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
GLP-1R Antagonist 1
CAS:488097-06-9
GLP-1R Antagonist 1 is an orally active, CNS penetrant and non-competitive glucagon-like peptide 1 receptor …
Formula:
C16H11ClF6N4O2
Purity:
90%
Color and Shape:
Solid
Molecular weight:
440.73
Ref: TM-T15387
| 1mg | 45.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 142.00 € | ||
| 25mg | 267.00 € | ||
| 50mg | 423.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Apelin-12 acetate
Apelin-12 acetate possesses a high affinity to orphan receptor APJ receptor.
Formula:
C66H107N21O16S
Purity:
98.82%
Color and Shape:
Liquid
Molecular weight:
1482.75
Ref: TM-T39823L
| 1mg | 217.00 € | ||
| 5mg | 305.00 € | ||
| 10mg | 473.00 € | ||
| 25mg | 755.00 € | ||
| 50mg | 1,076.00 € | ||
| 100mg | 1,447.00 € | ||
| 1mL*10mM (DMSO) | 759.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
CTOP acetate
CTOP acetate is a somatostatin analogue and a μ-opioid receptor antagonist.
Formula:
C52H71N11O13S2
Purity:
99.87%
Color and Shape:
Soild
Molecular weight:
1122.32
Ref: TM-TP2052L
| 1mg | 211.00 € | ||
| 5mg | 627.00 € | ||
| 10mg | 924.00 € | ||
| 25mg | 1,705.00 € | ||
| 50mg | 2,558.00 € | ||
| 100mg | 3,457.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Physalaemin
CAS:2507-24-6
Physalaemin is a non-mammalian tachykinin.
Formula:
C58H84N14O16S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1265.45
Ref: TM-T19518
| 25mg | 1,435.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Tabernanthalog
CAS:2483829-58-7
TBG is a 5-HT2A agonist reducing alcohol/heroin cravings and promoting neuroplasticity with antidepressant effects in …
Formula:
C14H18N2O
Purity:
98.57%
Color and Shape:
Soild
Molecular weight:
230.31
Ref: TM-T60221
| 1mg | 182.00 € | ||
| 2mg | 273.00 € | ||
| 5mg | 418.00 € | ||
| 10mg | 613.00 € | ||
| 25mg | 922.00 € | ||
| 50mg | 1,282.00 € | ||
| 100mg | 1,766.00 € | ||
| 500mg | 3,511.00 € | ||
| 1mL*10mM (DMSO) | 361.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
BPR1M97
CAS:2059904-66-2
BPR1M97 is a mu opioid receptor (MOP) and neuropeptide-orphin FQ (NOP) receptor agonist with blood-brain …
Formula:
C18H18Cl2N2O
Purity:
98.13% - 99.15%
Color and Shape:
Solid
Molecular weight:
349.25
Ref: TM-T10593
| 1mg | 94.00 € | ||
| 5mg | 223.00 € | ||
| 10mg | 352.00 € | ||
| 25mg | 647.00 € | ||
| 50mg | 1,014.00 € | ||
| 100mg | 1,423.00 € | ||
| 500mg | 2,762.00 € | ||
| 1mL*10mM (DMSO) | 215.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Lintitript
CAS:136381-85-6
Lintitript (SR 27897) is a selective antagonist of CCK1 with EC50s of 6 nM and …
Formula:
C20H14ClN3O3S
Purity:
98.48%
Color and Shape:
Solid
Molecular weight:
411.86
Ref: TM-T15759
| 1mg | 113.00 € | ||
| 2mg | 154.00 € | ||
| 5mg | 230.00 € | ||
| 10mg | 344.00 € | ||
| 25mg | 549.00 € | ||
| 50mg | 741.00 € | ||
| 100mg | 994.00 € | ||
| 1mL*10mM (DMSO) | 258.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
PG 931 acetate
PG 931 acetate is a potent agonist of melanocortin 4 (MC4) receptors.
Formula:
C61H89N15O13
Purity:
98.74%
Color and Shape:
Liquid
Molecular weight:
1240.45
Ref: TM-TP1953L
| 1mg | 399.00 € | ||
| 5mg | 898.00 € | ||
| 10mg | 1,218.00 € | ||
| 25mg | 1,813.00 € | ||
| 50mg | 2,446.00 € | ||
| 100mg | 3,290.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Prostaglandin F2α 1,11-lactone
CAS:62410-84-8
Prostaglandin F2α 1,11-lactone (PGF2α 1,11-lactone) is a lipid-soluble prodrug of Prostaglandin F2α and can be …
Formula:
C20H32O4
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
336.47
Ref: TM-T37326
| 10mg | 1,613.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
SB 216641
CAS:170230-39-4
SB 216641 is a 5-HT (1B/1D) antagonist with anxiolytic activity for the study of anxiety …
Formula:
C28H30N4O4
Purity:
98.01%
Color and Shape:
Liquid
Molecular weight:
486.56
Ref: TM-T85323
| 1mg | 196.00 € | ||
| 5mg | 486.00 € | ||
| 10mg | 682.00 € | ||
| 25mg | 1,064.00 € | ||
| 50mg | 1,467.00 € | ||
| 100mg | 1,878.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
DPDPE
CAS:88373-73-3
DPDPE is selective δ-opioid receptor agonist peptide.
Formula:
C30H39N5O7S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
645.79
Ref: TM-TP2036
| 1mg | 376.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
TDI-10229
CAS:2810887-45-5
TDI-10229: potent oral sAC inhibitor, IC50=195 nM. Good mouse pharmacokinetics for in vivo use.
Formula:
C16H16ClN5
Purity:
97.77%
Color and Shape:
Soild
Molecular weight:
313.78
Ref: TM-T64355
| 1mg | 41.00 € | ||
| 5mg | 159.00 € | ||
| 10mg | 233.00 € | ||
| 25mg | 416.00 € | ||
| 50mg | 625.00 € | ||
| 100mg | 903.00 € | ||
| 200mg | 1,246.00 € | ||
| 1mL*10mM (DMSO) | 171.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Tecastemizole
CAS:75970-99-9
Tecastemizole (R 43512) is a selective antagonist of H1 receptor and a major metabolite of …
Formula:
C19H21FN4
Purity:
99.66%
Color and Shape:
Solid
Molecular weight:
324.4
Ref: TM-T26253
| 1mg | 56.00 € | ||
| 5mg | 123.00 € | ||
| 10mg | 174.00 € | ||
| 25mg | 297.00 € | ||
| 50mg | 428.00 € | ||
| 100mg | 603.00 € | ||
| 500mg | 1,201.00 € | ||
| 1mL*10mM (DMSO) | 138.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
NUCC-390 dihydrochloride (1060524-97-1 free base)
NUCC-390 dihydrochloride is selective agonist of small-molecule CXCR4 receptor.
Formula:
C23H35Cl2N5O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
468.46
Ref: TM-T12269L
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Monday 16 Dec 2024
