G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Ceruletide Ammonium Salt
Ceruletide Ammonium Salt is a decapeptide, originating from the skin of tropical frogs, which is …
Formula:
C58H77N14O21S2
Purity:
98.47%
Color and Shape:
Soild
Molecular weight:
1370.44
Ref: TM-T14932L1
| 1mg | 96.00 € | ||
| 5mg | 323.00 € | ||
| 10mg | 480.00 € | ||
| 25mg | 769.00 € | ||
| 50mg | 1,013.00 € | ||
| 100mg | 1,374.00 € | ||
| 500mg | 2,719.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
(2R,3S)-Azelaprag
CAS:2049979-31-7
(2R,3S)-N-(4-(2,6-dimethoxyphenyl)-5-(5-methylpyridin-3-yl)-4H-1,2,4-triazol-3-yl)-3-(5-methylpyrimidin-2-yl)butane-2-sulfonamide is an Apelin receptor agonist
Formula:
C25H29N7O4S
Purity:
98.69%
Color and Shape:
Soild
Molecular weight:
523.61
Ref: TM-T14390L
| 5mg | 2,325.00 € | ||
| 10mg | 2,975.00 € | ||
| 25mg | 3,719.00 € | ||
| 50mg | 5,020.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Edg-2 receptor inhibitor 1
CAS:1195941-38-8
Edg-2 receptor inhibitor 1 (SAR-100842) is an Edg-2 receptor inhibitor extracted (IC50: <0.1 μM).
Formula:
C27H27NO5
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
445.51
Ref: TM-T4521
| 1mg | 95.00 € | ||
| 2mg | 171.00 € | ||
| 5mg | 268.00 € | ||
| 10mg | 419.00 € | ||
| 25mg | 648.00 € | ||
| 50mg | 925.00 € | ||
| 100mg | 1,240.00 € | ||
| 1mL*10mM (DMSO) | 286.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
B-Raf IN 14
CAS:326918-98-3
B-Raf IN 14 is a BRAF inhibitor.
Formula:
C15H14BrN5O3S
Purity:
98.32%
Color and Shape:
Solid
Molecular weight:
424.27
Ref: TM-T72070
| 1mg | 182.00 € | ||
| 5mg | 411.00 € | ||
| 10mg | 602.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,299.00 € | ||
| 100mg | 1,737.00 € | ||
| 500mg | 3,463.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Picumeterol FA
picumeterol FA is a potent and selective β2-adrenergic receptor agonist.
Formula:
C22H31Cl2N3O4
Purity:
99.80%
Color and Shape:
Soild
Molecular weight:
472.4
Ref: TM-T68129L1
| 1mg | 182.00 € | ||
| 5mg | 452.00 € | ||
| 10mg | 647.00 € | ||
| 25mg | 1,009.00 € | ||
| 50mg | 1,384.00 € | ||
| 100mg | 1,828.00 € | ||
| 500mg | 3,648.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Mogamulizumab
CAS:1159266-37-1
Mogamulizumab is a monoclonal antibody targeting CC chemokine receptor 4 with anticancer effects, used in …
Purity:
SDS-PAGE:97.3%;SEC-HPLC:99.4%
Color and Shape:
Solid
Ref: TM-T76782
| 1mg | 445.00 € | ||
| 5mg | 916.00 € | ||
| 10mg | 1,281.00 € | ||
| 25mg | 1,839.00 € | ||
| 50mg | 2,591.00 € | ||
| 100mg | 3,533.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Deltorphin acetate
Deltorphin acetate is a substance obtained from the skin secretions of a frog, Phyllomedusa bicolor …
Formula:
C46H66N10O12S2
Purity:
98.93%
Color and Shape:
Solid
Molecular weight:
1015.21
Ref: TM-T20166L
| 1mg | 184.00 € | ||
| 5mg | 412.00 € | ||
| 10mg | 617.00 € | ||
| 25mg | 1,110.00 € | ||
| 50mg | 1,665.00 € | ||
| 100mg | 2,497.00 € | ||
| 200mg | 3,746.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
![5-Bromoimidazo[1,2-A]Pyrazine](https://static.cymitquimica.com/products/TM/thumb/T77641.jpg)
5-Bromoimidazo[1,2-A]Pyrazine
CAS:87597-26-0
5-Bromoimidazo[1,2-a]pyrazine inhibits phosphodiesterase and beta-adrenergic receptors.5-Bromoimidazo[1,2-a]pyrazine shows antibronchospastic activity in vitro.
Formula:
C6H4BrN3
Purity:
97.04%
Color and Shape:
Liquid
Molecular weight:
198.02
Ref: TM-T77641
| 1mg | 182.00 € | ||
| 5mg | 400.00 € | ||
| 10mg | 595.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,263.00 € | ||
| 100mg | 1,706.00 € | ||
| 500mg | 3,431.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Vazegepant
CAS:1337918-83-8
Vazegepant is an intranasal CGRP receptor antagonist utilized for conducting acute migraine research.
Formula:
C36H46N8O3
Purity:
98.61%
Color and Shape:
Solid
Molecular weight:
638.80
Ref: TM-T38734
| 1mg | 102.00 € | ||
| 5mg | 222.00 € | ||
| 10mg | 330.00 € | ||
| 25mg | 599.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Samidorphan HCl
CAS:2328045-02-7
Samidorphan HCl is an orally active and highly potent modulator of the opioid system that …
Formula:
C21H27ClN2O4
Purity:
98.25% - 99.60%
Color and Shape:
Soild
Molecular weight:
406.9
Ref: TM-T67888L
| 1mg | 162.00 € | ||
| 5mg | 386.00 € | ||
| 10mg | 573.00 € | ||
| 25mg | 909.00 € | ||
| 50mg | 1,225.00 € | ||
| 100mg | 1,652.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Tiflucarbine
CAS:89875-86-5
Tiflucarbine is a potential non-selective 5-HT agonist with antidepressant activity.Tiflucarbine dose-dependently increased the specific activity …
Formula:
C16H17FN2S
Purity:
100%
Color and Shape:
Liquid
Molecular weight:
288.38
Ref: TM-T68162
| 1mg | 260.00 € | ||
| 5mg | 640.00 € | ||
| 10mg | 919.00 € | ||
| 25mg | 1,361.00 € | ||
| 50mg | 1,828.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Galcanezumab
CAS:1578199-75-3
Galcanezumab: humanized IgG4 antibody that targets CGRP for migraine and cluster headache prevention/treatment.
Purity:
> 95%
Color and Shape:
Solid
Ref: TM-T76682
| 1mg | 125.00 € | ||
| 5mg | 370.00 € | ||
| 10mg | 594.00 € | ||
| 25mg | 919.00 € | ||
| 50mg | 1,233.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
D3R ligand 1
D3R Ligand 1 (compound 23b) is a potent, selective antagonist of the dopamine D3 receptor …
Formula:
C27H37NO5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
455.59
Ref: TM-T78736
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
Talastine
CAS:16188-61-7
Talastine is an antihistamine compound that can induce an allergic rash.
Formula:
C19H21N3O
Purity:
99.30% - 99.37%
Color and Shape:
Liquid
Molecular weight:
307.39
Ref: TM-T68150
| 1mg | 91.00 € | ||
| 5mg | 195.00 € | ||
| 10mg | 289.00 € | ||
| 25mg | 545.00 € | ||
| 50mg | 728.00 € | ||
| 100mg | 1,012.00 € | ||
| 500mg | 2,023.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
PACAP-related Peptide (rat) (trifluoroacetate salt)
PRP, a 29-amino acid peptide in the secretin/glucagon family, is found in rat brain regions …
Color and Shape:
Solid
Ref: TM-T37435
| 1mg | 473.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Spns2-IN-1
Spns2-IN-1 is a potent Spns2 inhibitor, effectively impeding Spns2-dependent S1P transport with an IC50 value …
Purity:
98%
Ref: TM-T81114
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
Cortistatin-8 acetate
Cortistatin-8 acetate: synthetic corticosteroid analog, GHS-R antagonist; doesn't affect acyl GH release or hesperidin response.
Formula:
C49H72N12O11S2
Purity:
99.01%
Color and Shape:
Soild
Molecular weight:
1069.3
Ref: TM-TP2236L
| 1mg | 223.00 € | ||
| 5mg | 548.00 € | ||
| 10mg | 783.00 € | ||
| 25mg | 1,189.00 € | ||
| 50mg | 1,613.00 € | ||
| 100mg | 2,172.00 € | ||
| 500mg | 4,353.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Mesoridazine Besylate
CAS:32672-69-8
Mesoridazine Besylate (Serentil), a piperidine antipsychotic and phenothiazine, treats schizophrenia; it's a thioridazine metabolite.
Formula:
C27H32N2O4S3
Purity:
99.58%
Color and Shape:
Solid
Molecular weight:
544.75
Ref: TM-T3086
| 5mg | 75.00 € | ||
| 10mg | 127.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
PF-9184
CAS:1221971-47-6
PF-9184 inhibits human mPGES-1 selectively, with an IC50 of 16.5 nM, and reduces IL-1β-stimulated PGE2 …
Formula:
C21H14Cl2N2O4S
Purity:
97.64%
Color and Shape:
Solid
Molecular weight:
461.32
Ref: TM-T21738
| 1mg | 35.00 € | ||
| 5mg | 75.00 € | ||
| 10mg | 102.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
PSB 0777 ammonium hydrate
PSB 0777 ammonium hydrate is a potent and selective adenosine A2A receptor full agonist, exhibiting …
Formula:
C18H20N5O7S2·NH4·75H2O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
532.09
Ref: TM-T78084
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
