Membrane Transport Protein
Found 68 products for "Membrane Transport Protein".
DL-Dapoxetine HCl - Bio-X ™
CAS:Controlled ProductDapoxetine is a serotonin reuptake inhibitor drug that is used to treat premature ejaculation. This drug works by increasing the levels of serotonin in the brain, which in turn can help to delay the reflex that triggers ejaculation. As a result, it delays ejaculation and improves control over this.Formula:C21H23NO•HClPurity:Min. 95%Color and Shape:PowderMolecular weight:341.87 g/molElacridar hydrochloride
CAS:Inhibitor of ABC transporters; oral bioenhancer for anti-cancer therapyFormula:C34H34ClN3O5Purity:Min. 98 Area-%Color and Shape:Yellow PowderMolecular weight:600.11 g/molReboxetine mesylate - Bio-X ™
CAS:Controlled ProductReboxetine mesylate is a drug that belongs to the class of tricyclic antidepressants. It is a selective and potent inhibitor of neuronal reuptake of norepinephrine (noradrenaline). Reboxetine also interacts with neurokinin-1 receptors, which may affect locomotor activity and hippocampal formation, resulting in effects to memory and learning. It has been shown to be effective in the treatment of symptoms related to depression and Parkinson's disease.Formula:C20H27NO6SPurity:Min. 98 Area-%Molecular weight:409.5 g/molMaprotiline HCl - Bio-X ™
CAS:Controlled ProductMaprotiline is a tetracyclic antidepressant that is used for the treatment of major depressive disorder and anxiety that is associated with depression. This drug inhibits noradrenaline reuptake and has anticholinergic properties. Additionally, Maprotiline inhibits the amine transporter which allows for a delay in the reuptake of noradrenaline.
Formula:C20H23N•HClPurity:Min. 95%Color and Shape:PowderMolecular weight:313.86 g/molPF 03463275
CAS:Orally available and central nervous system-penetrant inhibitor of GlyT1 glycine transporter SLC6A9. PF 03463275 was shown to enhance neuroplasticity and cognitive remediation in schizophrenia patients. In animal studies, PF 03463275 also influenced retina as changes in electroretinogram were detected in albino rats.Formula:C19H22ClFN4OPurity:Min. 95%Molecular weight:376.86 g/molEvacetrapib monohydrate
CAS:Inhibitor of CETP exchange protein
Formula:C31H36F6N6O2•H2OPurity:Min. 95 Area-%Color and Shape:Off-White PowderMolecular weight:656.66 g/molUK 5099
CAS:Specific inhibitor of the mitochondrial pyruvate carrier complexes MPC1 and MPC2. The compound blocks the pyruvate transport across the inner mitochondrial membrane and therefore reduces pyruvate influx into the gluconeogenesis. It supresses glucose production in hepatocytes and was proposed for the control of hyperglycaemia in diabetic patients. Also used for the sensitisation of cancer cell lines to chemotherapy.Formula:C18H12N2O2Purity:Min. 95%Color and Shape:Off-White Yellow PowderMolecular weight:288.3 g/molValspodar
CAS:P-glycoprotein (MDR1) inhibitor; non-immunosuppressive cyclosporin A analog
Formula:C63H111N11O12Purity:Min. 98 Area-%Color and Shape:PowderMolecular weight:1,214.62 g/molDihydrokainic acid
CAS:Non-transportable inhibitor of GLT-1 glutamate transporterFormula:C10H17NO4Purity:Min. 95%Molecular weight:215.25 g/molTariquidar
CAS:Potent P-glycoprotein (P-gp) inhibitor
Formula:C38H38N4O6Purity:Min. 97 Area-%Color and Shape:PowderMolecular weight:646.73 g/molMethyl-d3-magnesium iodide solution, 1.0 M in diethyl ether
CAS:Controlled ProductMethyl-d3-magnesium iodide solution, 1.0 M in diethyl ether, is a specialized organometallic reagent used extensively in synthetic chemistry. This compound is a labeled Grignard reagent, where the methyl group is fully deuterated. It is sourced through the synthesis involving the reaction of deuterated methyl iodide with magnesium in an anhydrous diethyl ether solvent.
Formula:CD3IMgPurity:Min. 95%Molecular weight:169.26 g/molDalcetrapib
CAS:Inhibitor of CETP exchange protein
Formula:C23H35NO2SPurity:Min. 98 Area-%Molecular weight:389.6 g/molBrefeldin A
CAS:Inhibits protein translocation from ER to Golgi; fungal metabolite
Formula:C16H24O4Purity:Min. 95%Color and Shape:PowderMolecular weight:280.36 g/molRef: 3D-AB15917
Discontinued productBAY 876
CAS:Selective and potent inhibitor of glucose transporter GLUT1 with IC50 of 2 nM. The compound limits glucose uptake and is able to block basal as well as stress-regulated glycolysis in ovarian cancer cells. It supresses proliferation, viability and tumorigenicity of ovarian cancer cells.Formula:C24H16F4N6O2Purity:Min. 95%Color and Shape:SolidMolecular weight:496.42 g/molClomipramine hydrochloride - Bio-X ™
CAS:Controlled ProductClomipramine is a tricyclic antidepressant drug that inhibits the reuptake of serotonin, norepinephrine, and dopamine. It is used to treat obsessive compulsive disorder, panic disorders and cataplexy. Additionally, Clomipramine is shown to modulate immune activation and shows constant anti-inflammatory properties at therapeutic concentrations by consistently decreasing pro-inflammatory cytokines.
Formula:C19H24Cl2N2Purity:Min. 95%Color and Shape:White PowderMolecular weight:351.31 g/molCitalopram HBr - Bio-X ™
CAS:Controlled ProductCitalopram is a selective serotonin reuptake inhibitor that is used for the treatment of depression. It has also been found to relieve and manage symptoms of anxiety, eating disorders and OCD. Citalopram targets serotonin by inhibiting its reuptake in the synaptic cleft. In vitro studies demonstrate that citalopram is a strong and selective inhibitor of neuronal serotonin reuptake and has weak effects on norepinephrine and dopamine central reuptake. .Formula:C20H21FN2O•HBrPurity:Min. 95%Color and Shape:PowderMolecular weight:405.3 g/molGBR 12909 dihydrochloride
CAS:Dopamine reuptake inhibitor; ligand of sigma receptorsFormula:C28H34Cl2F2N2OPurity:Min. 97 Area-%Color and Shape:White PowderMolecular weight:523.49 g/molRef: 3D-FG65030
Discontinued productGBR 12935 dihydrochloride
CAS:Dopamine reuptake inhibitorFormula:C28H34N2O•(HCl)2Purity:Min. 95%Color and Shape:PowderMolecular weight:487.5 g/molBI 01383298
CAS:Potent inhibitor of the sodium-coupled citrate cotransporter SLC13A5 (NaCT, INDY). The compound is not structurally related to citrate and is selective for SLC13A over other related transporters.
Formula:C19H19Cl2FN2O3SPurity:Min. 95%Color and Shape:SolidMolecular weight:445.34 g/molParoxetine hydrochloride
CAS:Controlled ProductA serotonin reuptake inhibitor with anticholinergic activity and mild inhibitory activity on noradrenaline reuptake. Paroxetine has been used for the treatment of depression, anxiety disorders, post-traumatic stress disorder, premenstrual dysphoric disorder and obsessive-compulsive disorder. Also inhibits nitric oxide synthase and cytochrome isoenzyme P450 2D6.
Formula:C19H20FNO3·HClPurity:Min. 97%Color and Shape:White PowderMolecular weight:365.83 g/molRef: 3D-FP38223
Discontinued product
