
Transportador de membrana / canal de iones
Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.
Subcategorías de "Transportador de membrana / canal de iones"
- ABC(3 productos)
- ATPasa(93 productos)
- Receptor de adiponectina(5 productos)
- CFTR(64 productos)
- Receptor CGRP(52 productos)
- Canal de calcio(496 productos)
- Canal de cloruro(49 productos)
- Receptor GABA(336 productos)
- Transportador de monoamina(23 productos)
- Transportador de monocarboxilato(17 productos)
- NKCC(2 productos)
- NPC1L1(3 productos)
- Cotransportador de Na-K-Cl(8 productos)
- OAT(27 productos)
- OCT(7 productos)
- P-gp(53 productos)
- Canal de potasio(277 productos)
- Bomba de protones(39 productos)
- SGLT(30 productos)
- Canal de sodio(202 productos)
- Canal TRP / TRPV(93 productos)
Mostrar 13 subcategorías más
Se han encontrado 2290 productos de "Transportador de membrana / canal de iones"
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CS-526
CAS:<p>CS-526 is a reversible proton pump inhibitor targeting the K+ site on H+,K+-ATPase, reducing gastric acid secretion and preventing mucosal lesions.</p>Fórmula:C20H22FN3OForma y color:SolidPeso molecular:339.41Pumaprazole
CAS:<p>Pumaprazole (BY-841) is an antagonist of a reversible proton pump.</p>Fórmula:C19H22N4O2Pureza:99.91%Forma y color:SolidPeso molecular:338.4L 691121
CAS:<p>L 691121 is a class III antiarrhythmic compound. It also blocks potassium currents.</p>Fórmula:C22H25ClN4O5SPureza:98%Forma y color:SolidPeso molecular:492.98Caroverine
CAS:Caroverine is a potential chemotherapeutical agent in HNSCC cell lines.Fórmula:C22H27N3O2Forma y color:SolidPeso molecular:365.47TCS 46b
CAS:<p>TCS 46b is a NR1A/NR2B NMDA receptor antagonist with oral activity.</p>Fórmula:C22H23N3OPureza:99.78% - 99.78%Forma y color:SolidPeso molecular:345.44BPO-27 racemate
CAS:<p>BPO-27 racemate (BPO-27 (racemate)) is an effective CFTR inhibitor with IC50 of 8 nM.</p>Fórmula:C26H18BrN3O6Pureza:97.67% - 98.86%Forma y color:SolidPeso molecular:548.34Diproqualone
CAS:<p>Diproqualone, analogous to methaqualone, exhibits sedative, anxiolytic, anti-inflammatory, and analgesic properties [1].</p>Fórmula:C12H14N2O3Forma y color:SolidPeso molecular:234.255XR9051 Hydrochloride
CAS:<p>XR9051 Hydrochloride, a potent modulator of P-glycoprotein-mediated multidrug resistance (MDR), inhibits the binding of cytotoxics to P-glycoprotein.</p>Fórmula:C39H39ClN4O5Forma y color:SolidPeso molecular:679.216-Iodoamiloride
CAS:<p>6-Iodoamiloride is a potent inhibitor of acid-sensing ion channel 1 (ASIC1), exhibiting an IC50 value of 88 nM.</p>Fórmula:C6H8IN7OPureza:98%Forma y color:SolidPeso molecular:321.08NPBA
CAS:<p>NPBA, a potassium K2P channel TASK-3 (KCNK9) agonist, concurrently functions as a blocker of the tandem pore domain weak inward rectifying K+ channel (TWIK2). This compound effectively inhibits NLRP3 inflammasome activation in macrophages [1].</p>Fórmula:C16H14F3N3O3Forma y color:SolidPeso molecular:353.3Crobenetine hydrochloride
CAS:<p>Crobenetine hydrochloride, a sodium channel antagonist, is used potentially for the treatment of stroke.</p>Fórmula:C25H34ClNO2Forma y color:SolidPeso molecular:416Nalanthalide
CAS:<p>Nalanthalide, serving as a voltage-gated potassium channel Kv1.3 blocker (IC50 = 3.9 µM) with potential immunosuppressive properties, is applicable in the research of inflammatory immune diseases including neuroinflammation [1] [2].</p>Fórmula:C30H44O5Forma y color:SolidPeso molecular:484.67COR659
CAS:<p>COR659: suppresses alcohol/chocolate intake in rats; enhances GABAB receptor, blocks CB1 receptor.</p>Fórmula:C16H16ClNO3SPureza:99.75%Forma y color:SolidPeso molecular:337.82Ebio1
CAS:<p>Ebio1, a selective activator of the voltage-gated potassium channel KCNQ2, enhances channel conductance by promoting the formation of an expanded gate at a saturation voltage of +50 mV, leading to increased channel activity [1].</p>Fórmula:C19H14FNOForma y color:SolidPeso molecular:291.32GSK 2833503A
CAS:<p>GSK 2833503A: potent TRPC6/3 antagonist; IC50: 3-16/21-100 nM; >63x selective; inhibits cardiac hypertrophy signaling.</p>Fórmula:C18H21ClFN3OSForma y color:SolidPeso molecular:381.9Iganidipine HCl
CAS:NKY-722 (HCl), also known as Iganidipine, is a calcium channel blocker potentially for the treatment of glaucoma.Fórmula:C28H40Cl2N4O6Forma y color:SolidPeso molecular:599.55PU-48
CAS:<p>PU-48 is a potent inhibitor of urea transporters A (UT-A) with an IC50 value of 0.32 μM, exhibiting a significant diuretic effect in mouse models without</p>Fórmula:C14H12N2O3SForma y color:SolidPeso molecular:288.32URAT1 inhibitor 8
CAS:<p>URAT1 Inhibitor 8 (example 247) serves as a highly potent inhibitor of URAT1, demonstrating an IC50 value of 0.001 μM.</p>Fórmula:C19H13ClFN3O4SForma y color:SolidPeso molecular:433.84NaV1.7 Blocker-801
CAS:<p>NaV1.7 Blocker-801 is a potent NaV1.7 blocker.</p>Fórmula:C20H15ClF2N6O3S2Forma y color:SolidPeso molecular:524.95MCT1-IN-2
CAS:<p>SR13800 is a monocarboxylate transporter 1 (MCT1) inhibitor with cell-permeable.</p>Fórmula:C25H29N3O2SForma y color:SolidPeso molecular:435.58
