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Transportador de membrana / canal de iones

Transportador de membrana / canal de iones

Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.

Subcategorías de "Transportador de membrana / canal de iones"

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Se han encontrado 2272 productos de "Transportador de membrana / canal de iones"

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  • N-Depropylpropafenone
    Targetmol
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    N-Depropylpropafenone

    CAS:
    <p>N-Depropylpropafenone, an active metabolite of Propafenone, is produced through the metabolism by the CYP450 enzyme system (primarily CYP2D6). It functions by blocking sodium ion channels, thereby delaying the depolarization process in myocardial cells and exhibiting antiarrhythmic properties.</p>
    Fórmula:C18H21NO3
    Forma y color:Solid
    Peso molecular:299.36

    Ref: TM-T201563

  • Desmethylflunitrazepam
    Targetmol
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    Desmethylflunitrazepam

    CAS:
    <p>Desmethylflunitrazepam (Norflunitrazepam) is a benzodiazepine derivative and an active metabolite of Flunitrazepam.</p>
    Fórmula:C15H10FN3O3
    Forma y color:Solid
    Peso molecular:299.26

    Ref: TM-T201723

  • Tizolemide
    Targetmol
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    Tizolemide

    CAS:
    <p>Tizolemide, a sulfonamide diuretic compound with alkaline properties, is cleared through the tubular transport system. It induces changes in the passive transport components across the basolateral membrane of isolated frog skin.</p>
    Fórmula:C11H14ClN3O3S2
    Forma y color:Solid
    Peso molecular:335.83

    Ref: TM-T201590

  • cis-KV1.3-IN-1
    Targetmol
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    cis-KV1.3-IN-1

    CAS:
    <p>cis-KV1.3-IN-1, also known as Compound cis-18, is the cis-isomer of KV1.3-IN-1 and functions as an inhibitor of the KV1.3 channel. In Xenopus laevis oocytes expressing human hKV1.3, cis-KV1.3-IN-1 (10 μM) achieves an inhibition rate of 25.53% against KV1.3.</p>
    Fórmula:C23H30N2O4S
    Forma y color:Solid
    Peso molecular:430.56

    Ref: TM-T201783

  • Cyazofamid
    Targetmol
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    Cyazofamid

    CAS:
    <p>Cyazofamid functions as a fungicide by impairing the production of ATP. It inhibits Organic Cation Transporter 3 (OCT3) and OAT1 with IC50 values of 1.54 and 17.3 μM, respectively.</p>
    Fórmula:C13H13ClN4O2S
    Forma y color:Solid
    Peso molecular:324.79

    Ref: TM-T201605

  • Lu AF90103
    Targetmol
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    Lu AF90103

    CAS:
    <p>Lu AF90103 (Compound 42e) is the methyl ester prodrug of compound 42d, capable of crossing the blood-brain barrier. Compound 42d acts as a partial agonist of the GluN1/GluN2B complex, with an efficacy of 24% and an EC50 value of 78 nM. Lu AF90103 plays a significant role in neuropsychiatric disorder research.</p>
    Fórmula:C13H15N3O3S
    Forma y color:Solid
    Peso molecular:293.342

    Ref: TM-T204820

  • Logo de CymitQuimica
    Targetmol
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    Cav 2.2/3.2 blocker 1

    <p>Compound 9e is a Cav 2.2/3.2 blocker; IC50: 1.22 μM &amp; 80 μM, respectively; penetrates CNS.</p>
    Fórmula:C28H30N2O3
    Forma y color:Solid
    Peso molecular:442.55

    Ref: TM-T62586

  • Ro-51
    Targetmol
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    Ro-51

    CAS:
    <p>dual P2X3 and P2X2/3 antagonist</p>
    Fórmula:C17H23IN4O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:474.29

    Ref: TM-T23245

  • Quinacainol dihydrochloride
    Targetmol
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    Quinacainol dihydrochloride

    CAS:
    <p>Quinacainol dihydrochloride (PK 10139 dihydrochloride) is the bis(2 hydrochloride) salt form of Quinacainol. It acts as an inhibitor of the sodium current, with an EC50 of 95 µM. This compound displays antiarrhythmic activity by modulating the electrophysiological properties of the heart.</p>
    Fórmula:C21H32Cl2N2O
    Forma y color:Solid
    Peso molecular:399.398

    Ref: TM-T204878

  • Logo de CymitQuimica
    Targetmol
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    IAB15

    CAS:
    <p>IAB15 is a potent inhibitor of T-type calcium channel that can be used in the research of epilepsy [1].</p>
    Fórmula:C15H14F3NO2
    Forma y color:Solid
    Peso molecular:297.27

    Ref: TM-T60648

  • SGE-516
    Targetmol
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    SGE-516

    CAS:
    <p>SGE516: neuroactive steroid, enhances GABAA, lowers neuronal activity, protects from seizures.</p>
    Fórmula:C23H35N3O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:385.54

    Ref: TM-T28766

  • TTA-P1
    Targetmol
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    TTA-P1

    CAS:
    <p>TTA-P1: potent T-type calcium channel inhibitor; impacts neuron firing, hormone secretion, cell growth; potential in absence epilepsy research.</p>
    Fórmula:C19H27Cl2FN2O
    Forma y color:Solid
    Peso molecular:389.33

    Ref: TM-T61747

  • YY-23
    Targetmol
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    YY-23

    CAS:
    <p>YY-23 is a selective NMDAR (containing GluN2C or GluN2D) inhibitor. By inhibiting NMDARs with GluN2D on GABAergic interneurons in the prefrontal cortex, YY-23 suppresses GABAergic neurotransmission and enhances excitatory transmission. YY-23 exhibits antidepressant activity and is useful for neurological disease research.</p>
    Fórmula:C33H54O8
    Forma y color:Solid
    Peso molecular:578.777

    Ref: TM-T206120

  • LY3130481
    Targetmol
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    LY3130481

    CAS:
    <p>LY3130481: TARP γ-8 dependent AMPA receptor blocker; selectively targets AMPA/TARP γ-8 with 65 nM IC50.</p>
    Fórmula:C19H18N4O3S
    Forma y color:Solid
    Peso molecular:382.44

    Ref: TM-T15814

  • Logo de CymitQuimica
    Targetmol
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    Cav 3.2 inhibitor 2

    <p>Cav 3.2 inhibitor 2 blocks T-type Ca2+ channels (IC50=0.09339 μM) and reduces mouse somatic/visceral pain. Used for intractable pain studies.</p>
    Fórmula:C32H37F2N3O
    Forma y color:Solid
    Peso molecular:517.65

    Ref: TM-T63606

  • MSK-195
    Targetmol
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    MSK-195

    CAS:
    <p>MSK-195 is an effective TRPV1 agonist.</p>
    Fórmula:C28H40N2O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:484.63

    Ref: TM-T24504

  • Kv7.2/Kv7.3 modulator-1
    Targetmol
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    Kv7.2/Kv7.3 modulator-1

    CAS:
    <p>Kv7.2/Kv7.3 modulator-1 (compound 6a) acts as a modulator for Kv7.2/Kv7.3 channels, with a pEC50 value of 7.96 for opening these channels. Kv7.2/Kv7.3 modulator-1 is applicable in research related to epilepsy, depression, brain injury, and pain.</p>
    Fórmula:C20H21F4N3O3
    Forma y color:Solid
    Peso molecular:427.393

    Ref: TM-T206950

  • SR 33805 oxalate
    Targetmol
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    SR 33805 oxalate

    CAS:
    <p>Ca2+ channel antagonist</p>
    Fórmula:C34H42N2O9S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:654.77

    Ref: TM-T23391

  • Logo de CymitQuimica
    Targetmol
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    T-Type calcium channel inhibitor 2

    <p>Compound 6g inhibits T-type Ca channels (IC50: Cav3.1-31μM, Cav3.2-83μM), cytotoxic to A549 (IC50: 5μM) &amp; HCT-116 cells (IC50: 6.4μM).</p>
    Fórmula:C36H39FN4OS
    Forma y color:Solid
    Peso molecular:594.78

    Ref: TM-T64203

  • ATP synthase inhibitor 2
    Targetmol
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    ATP synthase inhibitor 2

    CAS:
    <p>ATP synthase inhibitor 2 blocks P. aeruginosa ATP synthase; IC50=10 μg/mL, fully inhibits at 128 μg/mL.</p>
    Fórmula:C21H22N2O3S
    Forma y color:Solid
    Peso molecular:382.48

    Ref: TM-T61649