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Transportador de membrana / canal de iones

Transportador de membrana / canal de iones

Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.

Subcategorías de "Transportador de membrana / canal de iones"

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Se han encontrado 2430 productos de "Transportador de membrana / canal de iones"

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  • Logo de CymitQuimica
    Targetmol
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    Analgesic/antidepressant agent-1

    <p>Analgesic/antidepressant agent-1 (Compound k1) is an orally active N-acetylamino chloro ketone derivative capable of crossing the blood-brain barrier. It exhibits high affinity for NMDA receptors and demonstrates analgesic, anti-inflammatory, and antidepressant properties, with low psychotomimetic activity.</p>
    Fórmula:C22H25ClN2O2
    Forma y color:Solid
    Peso molecular:384.9

    Ref: TM-T205604

  • TRPA1-IN-1
    Targetmol
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    TRPA1-IN-1

    CAS:
    <p>TRPA1-IN-1 is a potent, selective antagonist of the TRPA1 channel, demonstrating significant oral bioavailability as a small molecule.</p>
    Fórmula:C19H17ClN6O3
    Forma y color:Solid
    Peso molecular:412.83

    Ref: TM-T39935

  • BKCa activator-1
    Targetmol
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    BKCa activator-1

    <p>BKCa activator-1 (Compound 51b) is an orally active activator of BKCa calcium-activated potassium channels with an EC50 of 2.82 μM. It promotes K+ efflux, leading to cell membrane hyperpolarization and inhibition of smooth muscle contraction. In a spontaneous hypertensive rat (SHR) model, it alleviates urinary incontinence and exhibits antitussive effects in a guinea pig cough model.</p>
    Fórmula:C22H23F7N2O3
    Forma y color:Solid
    Peso molecular:496.418

    Ref: TM-T205564

  • Conantokin G
    Targetmol
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    Conantokin G

    CAS:
    GluN2B-specific NMDA receptor blocker; IC50=480 nM in neurons, ~300 nM in oocytes; neuroprotective.
    Fórmula:C88H138N26O44
    Pureza:98%
    Forma y color:White Lyophilised Solid
    Peso molecular:2264.21

    Ref: TM-TP2060

  • CALP3
    Targetmol
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    CALP3

    CAS:
    Cell-permeable CaM agonist, binds EF-hand, activates phosphodiesterase without Ca2+, inhibits Ca2+ toxicity, IC50=33μM.
    Fórmula:C44H68N10O9
    Pureza:98%
    Forma y color:Solid
    Peso molecular:881.08

    Ref: TM-TP1911

  • (+)-Lycoctonine
    Targetmol
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    (+)-Lycoctonine

    CAS:
    Compound TJS1874 is a useful organic compound for research related to life sciences. The catalog number is TJS1874 and the CAS number is 26000-17-9.
    Fórmula:C25H41NO7
    Forma y color:Solid
    Peso molecular:467.6

    Ref: TM-TJS1874

  • Albanin A
    Targetmol
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    Albanin A

    <p>Albanin A is a useful organic compound for research related to life sciences and the catalog number is T124310.</p>
    Fórmula:C20H18O6
    Forma y color:Solid
    Peso molecular:354.358

    Ref: TM-T124310

  • Lei-Dab7
    Targetmol
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    Lei-Dab7

    CAS:
    Selective KCa2.2 channel blocker with Kd 3.8 nM, >200-fold specificity, enhances LTP, convulsive in vivo.
    Fórmula:C141H236N46O39S6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:3392.06

    Ref: TM-TP2007

  • GeX-2
    Targetmol
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    GeX-2

    CAS:
    <p>GeX-2 is a truncated analogue of αO-conotoxin. It has the ability to activate GABAB receptors and inhibit α9α10nAChR as well as CaV2.2 channels. Additionally, GeX-2 is effective in alleviating pain in a rat model of chronic constriction injury.</p>
    Fórmula:C103H169N43O27
    Forma y color:Solid
    Peso molecular:2441.72

    Ref: TM-TP3132

  • 1-(1-Methyl-1h-pyrazol-4-yl)-ethanone
    Targetmol
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    1-(1-Methyl-1h-pyrazol-4-yl)-ethanone

    CAS:
    1-(1-Methyl-1h-pyrazol-4-yl)-ethanone is a high purity biochemical reagent that can be used in research related to life sciences.
    Fórmula:C6H8N2O
    Pureza:99.92%
    Forma y color:Solid
    Peso molecular:124.14

    Ref: TM-TN9428

  • GX 201
    Targetmol
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    GX 201

    CAS:
    <p>GX 201 is a selective NaV1.7 inhibitor, IC50 of &lt; 3.2 nM for hNaV1.7.</p>
    Fórmula:C25H27ClF4N2O4S
    Pureza:99.81%
    Forma y color:Solid
    Peso molecular:563

    Ref: TM-T9647

  • SLC26A3-IN-2
    Targetmol
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    SLC26A3-IN-2

    CAS:
    <p>Vilobelimab (CaCP-29) is a human-mouse chimeric IgG antibody targeting human complement component 5a, a C5a inhibitor that inhibits neutrophil activation.</p>
    Fórmula:C19H13ClN2O2S
    Pureza:99.86%
    Forma y color:Solid
    Peso molecular:368.84

    Ref: TM-T74815

  • Logo de CymitQuimica
    Targetmol
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    Ebio3

    <p>Ebio3 is a selective potassium ion channel (KCNQ2) inhibitor with an IC50 of 1.2 nM. It binds to the KCNQ2 channel via its hydrophobic tail, causing the inward movement of the S6 helix, which results in the closure of the internal gate. The inhibitory effect of Ebio3 is equally effective on pathogenic KCNQ2 mutants, such as R75C and I238L, reducing their outward current by approximately 80%. Ebio3 holds potential for research in neurological disorders like epilepsy.</p>
    Fórmula:C19H23F2N3O2
    Forma y color:Solid
    Peso molecular:363.4

    Ref: TM-T205242

  • Homocarnosine
    Targetmol
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    Homocarnosine

    CAS:
    Homocarnosine is an endogenous dipeptide in cerebral regions and cerebrospinal fluid.
    Fórmula:C10H16N4O3
    Forma y color:Solid
    Peso molecular:240.26

    Ref: TM-T32098

  • α5-GABAA receptor modulator 1
    Targetmol
    + Info

    α5-GABAA receptor modulator 1

    <p>α5-GABAA receptor modulator 1 (Compound A-4) is a selective silent allosteric modulator (SAM) targeting the α5 subunit of GABAA receptors, useful for research into central nervous system (CNS) disorders.</p>
    Fórmula:C21H20FN3O4
    Forma y color:Solid
    Peso molecular:397.4

    Ref: TM-T205217

  • LY-466195
    Targetmol
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    LY-466195

    CAS:
    LY-466195 is a competitive antagonist of GLUK5 receptor.
    Fórmula:C16H24F2N2O4
    Forma y color:Solid
    Peso molecular:346.37

    Ref: TM-T27958

  • Oleoyl-D-lysine
    Targetmol
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    Oleoyl-D-lysine

    CAS:
    Oleoyl-D-lysine: lipid-based GlyT2 inhibitor, eases neuropathic pain in mice, safe, non-sedative, no respiratory depression.
    Fórmula:C24H46N2O3
    Forma y color:Solid
    Peso molecular:410.63

    Ref: TM-T74739

  • Levamlodipine besylate Hemipentahydrate
    Targetmol
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    Levamlodipine besylate Hemipentahydrate

    CAS:
    <p>Levamlodipine besylate hemipentahydrate is the besylate hemipentahydrate salt form of Levamlodipine. It is an orally effective calcium channel blocker with antioxidative and vasodilatory properties. This compound can reduce serum malondialdehyde (MDA) levels, enhance the activity of superoxide dismutase (SOD), and alleviate oxidative stress. Levamlodipine besylate hemipentahydrate is relevant for research in vascular dementia, hypertension, and cerebrovascular diseases.</p>
    Fórmula:C20H25ClN2O5·C6H6O3SH2O
    Forma y color:Solid
    Peso molecular:1224.18

    Ref: TM-T204904

  • GaTx2
    Targetmol
    + Info

    GaTx2

    CAS:
    High-affinity ClC-2 blocker (KD ~50 pM), selective over other ClCs/CFTR/GABAC/CaCC/KV1.2; slows activation, no effect on open channels.
    Fórmula:C125H199N39O47S6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:3192.54

    Ref: TM-TP2027

  • PNU-140975
    Targetmol
    + Info

    PNU-140975

    CAS:
    PNU-140975 is a bio-active chemical.
    Fórmula:C3H9N5O2
    Forma y color:Solid
    Peso molecular:147.138

    Ref: TM-T34096