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Transportador de membrana / canal de iones

Transportador de membrana / canal de iones

Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.

Subcategorías de "Transportador de membrana / canal de iones"

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Se han encontrado 2293 productos de "Transportador de membrana / canal de iones"

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  • KCC2 potentiators-1
    Targetmol
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    KCC2 potentiators-1

    CAS:
    <p>Compound 2, known as KCC2 potentiators-1, acts as an enhancer of the potassium chloride cotransporter-2 (KCC2). It holds potential for applications in studies related to neurological disorders.</p>
    Fórmula:C15H17N3OS
    Forma y color:Solid
    Peso molecular:287.38

    Ref: TM-T203414

  • A 80915A
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    A 80915A

    CAS:
    <p>A80915A: Semi-naphthoquinone antibiotic, blocks gastric (H(+)-K+)-ATPase; potency varies with enzyme conformation; K+ reduces binding rate.</p>
    Fórmula:C26H31Cl3O5
    Forma y color:Solid
    Peso molecular:529.88

    Ref: TM-T26450

  • Logo de CymitQuimica
    Targetmol
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    ω-Conotoxin MVIIC TFA

    <p>ω-Conotoxin MVIIC TFA is a peptide and neurotoxin blocks P-type and q-type voltage-sensitive neuronal Ca ++ channels (VGCCs) radiolabel immunoprecipitation.</p>
    Fórmula:C106H178N40O32S7·C2HF3O2
    Forma y color:Solid
    Peso molecular:2863.27

    Ref: TM-T75726

  • FD 12-9
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    FD 12-9

    CAS:
    FD 12-9, Anti-glioblastoma activity. is a flavonoid dimer, acts as a dual inhibitor of P-gp and BCRP, with EC50s of 285 nM and 0.9 nM, respectively.
    Fórmula:C51H47N3O11
    Pureza:98%
    Forma y color:Solid
    Peso molecular:877.93

    Ref: TM-T11268

  • JC-229
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    JC-229

    CAS:
    <p>JC-229 is a potent and selective TbRPA1 inhibitor that can inhibit RPA1 in Trypanosoma brucei. JC-229 can be used to study human African Trypanosomiasis (HAT).</p>
    Fórmula:C20H14Cl4N2O3S
    Pureza:97.14%
    Forma y color:Solid
    Peso molecular:504.21

    Ref: TM-T77645

  • Logo de CymitQuimica
    Targetmol
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    Urease-IN-19

    <p>Urease-IN-19 (Compound 3c) is a potent inhibitor of urease, demonstrating an IC50 value of 2.7 µM. It shows potential for use in research related to kidney stones and gastric ulcers.</p>
    Fórmula:C17H16FN3S
    Forma y color:Solid
    Peso molecular:313.39

    Ref: TM-T205469

  • CPI1
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    CPI1

    <p>CPI1 is an effective and highly specific inhibitor of multidrug resistance protein 1 (MRP1). It exhibits inhibitory activity against MRP1 at the nanomolar level (Ki: 100 nM) and has minimal effect on P-glycoprotein (Pgp). CPI1 competes with LTC4 for binding to the same site on MRP1, inhibiting ATP hydrolysis and substrate transport. It is useful in research related to drug delivery and addressing cancer chemotherapy resistance.</p>
    Fórmula:C111H131N23O30S
    Forma y color:Solid
    Peso molecular:2299.43

    Ref: TM-TP3085

  • Chlorotoxin
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    Chlorotoxin

    CAS:
    <p>Chlorotoxin: 36-amino acid peptide from deathstalker scorpion venom; blocks small chloride channels.</p>
    Fórmula:C158H249N53O47S11
    Pureza:98%
    Forma y color:Solid
    Peso molecular:3995.71

    Ref: TM-TP1431

  • Logo de CymitQuimica
    Targetmol
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    Huwentoxin I

    CAS:
    <p>Huwentoxin I (HWTX-I) is a peptide toxin that targets and inhibits both voltage-gated sodium channels and N-type calcium channels.</p>
    Fórmula:C161H246N48O44S6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:3750.36

    Ref: TM-T80185

  • Mambalgin 1
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    Mambalgin 1

    CAS:
    <p>ASIC1a inhibitor; IC50: 192 nM (human), 72 nM (dimer); inactive channel binding; selective; pain response delay.</p>
    Fórmula:C272H429N85O84S10
    Pureza:98%
    Forma y color:Solid
    Peso molecular:6554.51

    Ref: TM-TP2003

  • TRPA1 Antagonist 3
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    TRPA1 Antagonist 3

    CAS:
    <p>TRPA1 Antagonist 3 is a compound with photoswitchable properties that acts as an agonist on the TRPA1 channel, providing the ability for optical control.</p>
    Fórmula:C11H8ClN3
    Forma y color:Solid
    Peso molecular:217.66

    Ref: TM-T40822

  • Atagabalin
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    Atagabalin

    CAS:
    <p>Atagabalin (PD 0200390), a gabamimetic for insomnia treatment and related to gabapentin, was halted due to poor trial outcomes.</p>
    Fórmula:C10H19NO2
    Forma y color:Solid
    Peso molecular:185.26

    Ref: TM-T30188

  • S-Sulfo-L-cysteine sodium salt
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    S-Sulfo-L-cysteine sodium salt

    CAS:
    <p>S-Sulfo-L-cysteine sodium salt shows a weak affinity for mGluR1α and mGluR5a at high concentrations and has potential antioxidant activity.</p>
    Fórmula:C3H6NNaO5S2
    Pureza:99.88%
    Forma y color:Solid
    Peso molecular:223.2

    Ref: TM-T23303

  • ω-Conotoxin GVIA
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    ω-Conotoxin GVIA

    CAS:
    <p>Peptide neurotoxin; selectively and reversibly blocks N-type calcium channels (IC50 = 0.15 nM). Reduces (RS)-3,5-DHPG -induced long term depression in vivo.</p>
    Fórmula:C120H182N38O43S6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:3037

    Ref: TM-TP2062

  • N-Arachidonoyl Taurine
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    N-Arachidonoyl Taurine

    CAS:
    <p>N-Arachidonoyl taurine, an amino acid, activates TRPV1/TRPV4, is metabolized by lipoxygenase, and affects insulin secretion and calcium flux.</p>
    Fórmula:C22H37NO4S
    Forma y color:Solid
    Peso molecular:411.6

    Ref: TM-T35918

  • Carbonic anhydrase inhibitor 32
    Targetmol
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    Carbonic anhydrase inhibitor 32

    <p>Carbonic anhydrase inhibitor32 (compound 5B) is an orally active, selective inhibitor of hCA (carbonic anhydrase) II/VII, with Ki values of 6.3 nM for hCA II, 10.1 nM for hCA VII, and 681 nM for hCA I. It shows potential for neuroprotection and anticonvulsant effects by reducing mTOR activation and increasing hippocampal KCC2 levels.</p>
    Fórmula:C17H16N6O3S
    Forma y color:Solid
    Peso molecular:384.41

    Ref: TM-T207684

  • AQP4 (201-220)
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    AQP4 (201-220)

    CAS:
    <p>AQP4 (201-220) is the encephalitogenic epitope of AQP-4. AQP4 (201-220) can induce experimental autoimmune encephalomyelitis (EAE), characterized by midline brain lesions, retinal lesions, and lesions at the gray matter/white matter boundary of the spinal cord. AQP-4 is the target antigen in neuromyelitis optica.</p>
    Fórmula:C97H143N27O27S
    Forma y color:Solid
    Peso molecular:2151.4

    Ref: TM-TP3213

  • Cavα2δ-IN-1
    Targetmol
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    Cavα2δ-IN-1

    CAS:
    <p>Cavα2δ-IN-1 demonstrates exceptional specificity for voltage-gated calcium channels Cavα2δ-1 (with a Ki value of 6 nM), in comparison to Cavα2δ-2 (with a Ki</p>
    Fórmula:C18H27N5O
    Forma y color:Solid
    Peso molecular:329.448

    Ref: TM-T40071

  • NF864
    Targetmol
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    NF864

    CAS:
    NF864, a suramin analog, is a P2X1 receptor inhibitor.
    Fórmula:C57H28N6Na12O41S12
    Pureza:98%
    Forma y color:Solid
    Peso molecular:2113.5

    Ref: TM-T25863

  • (S)-ABT 102
    Targetmol
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    (S)-ABT 102

    CAS:
    <p>N-[(1S)-1H-inden-1-yl]-N'-indazol-4-ylurea is a strong TRPV1 blocker with a 123 nM IC50 against capsaicin.</p>
    Fórmula:C21H24N4O
    Pureza:99.65% - 99.77%
    Forma y color:Soild
    Peso molecular:348.44

    Ref: TM-T29522L