
Transportador de membrana / canal de iones
Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.
Subcategorías de "Transportador de membrana / canal de iones"
- ABC(3 productos)
- ATPasa(93 productos)
- Receptor de adiponectina(5 productos)
- CFTR(64 productos)
- Receptor CGRP(51 productos)
- Canal de calcio(493 productos)
- Canal de cloruro(49 productos)
- Receptor GABA(336 productos)
- Transportador de monoamina(23 productos)
- Transportador de monocarboxilato(17 productos)
- NKCC(2 productos)
- NPC1L1(3 productos)
- Cotransportador de Na-K-Cl(8 productos)
- OAT(27 productos)
- OCT(7 productos)
- P-gp(53 productos)
- Canal de potasio(276 productos)
- Bomba de protones(39 productos)
- SGLT(30 productos)
- Canal de sodio(202 productos)
- Canal TRP / TRPV(93 productos)
Mostrar 13 subcategorías más
Se han encontrado 2277 productos de "Transportador de membrana / canal de iones"
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SDZ 220-581 Ammonium salt
CAS:<p>SDZ 220-581 Ammonium salt is a potent, orally active and competitive antagonist of NMDA receptor(pKi : 7.7).</p>Fórmula:C16H20ClN2O5PPureza:98%Forma y color:SolidPeso molecular:386.77Lansoprazole-d4
CAS:<p>Lansoprazole D4 (AG-1749 D4) is a deuterium labeled Lansoprazole. Lansoprazole is an inhibitor of proton pump which prevents the stomach from producing acid.</p>Fórmula:C16H14F3N3O2SPureza:98%Forma y color:SolidPeso molecular:373.39SDZ 220-581 hydrochloride
CAS:<p>SDZ 220-581 hydrochloride is a potent, orally active and competitive antagonist of NMDA receptor(pKi : 7.7).</p>Fórmula:C16H18Cl2NO5PPureza:98%Forma y color:SolidPeso molecular:406.2N-Methyl-DL-aspartic acid
CAS:<p>N-Methyl-DL-aspartic acid, a glutamate analogue and NMDA receptor agonist, is utilized in neurological disease research.</p>Fórmula:C5H9NO4Pureza:99.85%Forma y color:SolidPeso molecular:147.13Lansoprazole Sulfide D4
CAS:<p>Lansoprazole Sulfide D4 is a deuterium labeled Lansoprazole Sulfide. Lansoprazole Sulfide is an orally active anti-TB (Mycobacterium tuberculosis) agent with IC50 values of 0.59 μM intracellularly and 0.46 μM in broth.Lansoprazole Sulfide is an active metabolite of the proton pump inhibitor Lansoprazole.</p>Fórmula:C16H14F3N3OSPureza:98%Forma y color:SolidPeso molecular:357.39Cabotegravir sodium
CAS:<p>Cabotegravir sodium inhibits HIV integrase (IC50: 2.5 nM), metabolized by UGT1A1, with minimal ARV interaction.</p>Fórmula:C19H16F2N3NaO5Forma y color:SolidPeso molecular:427.34UBP608
CAS:<p>UBP608 selectively inhibits NMDA GluN1/GluN2A receptors, 23x more than GluN1/GluN2D.</p>Fórmula:C10H5BrO4Forma y color:SolidPeso molecular:269.05γ-DGG
CAS:<p>gamma-DGG is a competitive blocker of AMPA receptor.</p>Fórmula:C7H12N2O5Pureza:98%Forma y color:SolidPeso molecular:204.18Rapastinel
CAS:<p>Rapastinel (TPPT-amide) (GLYX-13) is an N-methyl-D-aspartate receptor (NMDAR) modulator.</p>Fórmula:C18H31N5O6Pureza:97.18%Forma y color:SolidPeso molecular:413.47Piretanide
CAS:<p>Piretanide, an oral loop diuretic, effective and potassium-sparing, heart failure and hypertension with reduced electrolyte imbalance risk.</p>Fórmula:C17H18N2O5SForma y color:Pale Yellow PowderPeso molecular:362.4SKA-121
CAS:<p>SKA-121 is a selective KCa3.1 activator (EC50s: 109 nM and 4.4 μM for KCa3.1 and KCa2.3, respectively).</p>Fórmula:C12H10N2OPureza:98%Forma y color:SolidPeso molecular:198.22Mexiletine-d6 hydrochloride
CAS:<p>Mexiletine D6 hydrochloride is a non-selective voltage-gated sodium channel blocker,is a Class IB antianhythmic.</p>Fórmula:C11H18ClNOPureza:98%Forma y color:SolidPeso molecular:221.76Jedi2
CAS:<p>Jedi2 is a Piezo1 activator rather than a specific Piezo2 activator. Jedi2 binds to the mouse Piezo1 proteins with a K d of 2770 μM [1].</p>Fórmula:C10H8O3SPureza:97.85%Forma y color:SolidPeso molecular:208.23β-D-Glucopyranosyl abscisate
CAS:<p>β-D-Glucopyranosyl abscisate (ABA-GE) is a hydrolyzable conjugate of abscisic acid (ABA), which predominantly accumulates in the vacuole and likely in the</p>Fórmula:C21H30O9Forma y color:SolidPeso molecular:426.46Etifoxine
CAS:<p>Etifoxine targets β2/β3 GABAA receptors, is anxiolytic in humans/rodents, boosts GABAA, binds TSPO, aids axon regeneration, no sedative effects.</p>Fórmula:C17H17ClN2OPureza:98%Forma y color:SolidPeso molecular:300.78SDZ 220-581
CAS:<p>SDZ 220-581 is a potent, orally active and competitive antagonist of NMDA receptor(pKi : 7.7).</p>Fórmula:C16H17ClNO5PPureza:98%Forma y color:SolidPeso molecular:369.74Perfluoroenanthic acid
CAS:<p>Perfluoroenanthic acid (Perfluoroheptanoic acid) is a perfluoroalkyl substance (PFAS) that negatively impacts spermatogenic development and testicular m6A RNA methylation in offspring exposed during gestation, thus impeding spermatogenesis and inducing reproductive toxicity. Additionally, in primary cortical neuron cultures, Perfluoroenanthic acid alters dendritic spine morphology and synaptogenesis, enhances neural activity and synaptic transmission, and increases the expression of excitatory synapse-associated proteins Synaptophysin and PSD95.</p>Fórmula:C7HF13O2Forma y color:SolidPeso molecular:364.063,3-Diethylthiacarbocyanine iodide
CAS:<p>3, 3-diethylthiacarbocyanine iodide is a cyanine dye. Can be used for photochemical methods.</p>Fórmula:C21H21IN2S2Pureza:99.79%Forma y color:SolidPeso molecular:492.44MSC-4381
CAS:<p>MSC-4381 (MCT4-IN-1) is an orally available and selectively modeled highly potent inhibitor of monocarboxylic acid transporter protein 4 (MCT4/SLC16A3) with potential anticancer and antitumor activity for the study of osteosarcoma.</p>Fórmula:C26H20ClN3O6SPureza:99.04%Forma y color:SolidPeso molecular:537.97
