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Transportador de membrana / canal de iones

Transportador de membrana / canal de iones

Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.

Subcategorías de "Transportador de membrana / canal de iones"

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Se han encontrado 2277 productos de "Transportador de membrana / canal de iones"

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  • Enflurane

    CAS:
    <p>Enflurane (Efrane), a volatile anaesthetic, inhibits Ca2+-activated K+ channels and is used to gauge anesthesia levels in gas chromatography.</p>
    Fórmula:C3H2ClF5O
    Pureza:99.64%
    Forma y color:Clear Colorless Liquid Ordinary Temperature And Pressure Bp 56 8°C Density 1 50 G Cm-3 At Room Temperature Used As An
    Peso molecular:184.49
  • Aptiganel hydrochloride

    CAS:
    <p>Aptiganel hydrochloride(Cerestat) is the salt form of Aptiganel.Aptiganel is a non-competitive NMDA antagonist with neuroprotective effects used in the treatment of stroke and focal cerebral ischemia.</p>
    Fórmula:C20H22ClN3
    Pureza:99.89%
    Forma y color:Solid
    Peso molecular:339.86
  • UBP710

    CAS:
    <p>UBP710 is an effective and selective NMDA receptor modulator.</p>
    Fórmula:C18H14O2
    Pureza:98.05%
    Forma y color:Solid
    Peso molecular:262.3
  • AZ194

    CAS:
    <p>CRMP2-Ubc9-NaV1.7 inhibitor 194, is a CRMP2-Ubc9-NaV1.7 inhibitor.</p>
    Fórmula:C34H31F2N3O3
    Pureza:99.61%
    Forma y color:Solid
    Peso molecular:567.62
  • SKF89976A hydrochloride

    CAS:
    <p>SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = 0.28 μM), GAT-2 (IC50s = 137.34 μM) and</p>
    Fórmula:C22H26ClNO2
    Pureza:98.02%
    Forma y color:Solid
    Peso molecular:371.9
  • Basmisanil

    CAS:
    <p>Basmisanil (RG1662) is a negative allosteric modulator/inverse agonist of GABAAα5 receptors.Formulations containing basmisanil are in clinical trials for the</p>
    Fórmula:C21H20FN3O5S
    Pureza:99.21% - 99.42%
    Forma y color:Solid
    Peso molecular:445.46
  • Pipequaline hydrochloride

    CAS:
    <p>Pipequaline hydrochloride (PK-8165 hydrochloride) is an anticonflict &amp; anticonvulsant quinoline derivative.</p>
    Fórmula:C22H25ClN2
    Pureza:99.46%
    Forma y color:Solid
    Peso molecular:352.9
  • Tezacaftor

    CAS:
    <p>Tezacaftor (VX661) is a small molecule that can be used as a corrector of the cystic fibrosis transmembrane conductance regulator (CFTR) gene function.</p>
    Fórmula:C26H27F3N2O6
    Pureza:98.84% - >99.99%
    Forma y color:Solid
    Peso molecular:520.5
  • SG-209

    CAS:
    <p>SG 209 is an analog of nicorandil and acts as a K+ channel opener and nitrate-free coronary vasodilator.</p>
    Fórmula:C10H12N2O3
    Pureza:99.84%
    Forma y color:Solid
    Peso molecular:208.21
  • Memantine

    CAS:
    <p>Memantine treats moderate to severe Alzheimer's; it's an amantadine derivative blocking NMDA receptors.</p>
    Fórmula:C12H21N
    Pureza:≥98%
    Forma y color:White Powder
    Peso molecular:179.3
  • Trans-ACBD

    CAS:
    <p>Trans-ACBD (Trans-1-aminocyclobutane-1,3-dicarboxylic acid) is an effective and specific N-methyl-D-aspartate receptor agonist.</p>
    Fórmula:C6H9NO4
    Pureza:99.47%
    Forma y color:Solid
    Peso molecular:159.14
  • Esomeprazole potassium salt

    CAS:
    <p>Esomeprazole potassium, a potent oral proton pump inhibitor, curbs acid secretion in stomach cells, aiding GERD research.</p>
    Fórmula:C17H18KN3O3S
    Forma y color:Solid
    Peso molecular:383.51
  • AC1903

    CAS:
    <p>AC1903 is a specific inhibitor of TRPC5 channel, and has been shown to suppress severe proteinuria and prevent podocyte loss.</p>
    Fórmula:C19H17N3O
    Pureza:98.45%
    Forma y color:Solid
    Peso molecular:303.36
  • Dihydroergotoxine mesylate

    CAS:
    Dihydroergotoxine mesylate (Ergoloid mesylates) is mainly used to improve symptoms and physical symptoms of mental degeneration related to aging.
    Fórmula:C20H29N3O5S
    Pureza:99.39% - ≥95%
    Forma y color:Solid
    Peso molecular:423.53
  • (S)-(-)-5-Fluorowillardiine hydrochloride

    CAS:
    <p>(S)-(-)-5-Fluorowillardiine hydrochloride is a potent and specific agonist of AMPAR.</p>
    Fórmula:C7H9ClFN3O4
    Forma y color:Solid
    Peso molecular:253.62
  • GNE-131

    CAS:
    <p>GNE-131 is a potent and specific inhibitor of human sodium channel NaV1.7 (IC50: 3 nM).</p>
    Fórmula:C23H30N4O3S
    Pureza:98.54% - 99.59%
    Forma y color:Solid
    Peso molecular:442.57
  • XEN907

    CAS:
    <p>XEN907 is a novel spiro oxindole NaV1.7 blocker. XEN907 also inhibits hNaV1.7 (IC50: 3 nM).</p>
    Fórmula:C21H21NO4
    Pureza:99.92%
    Forma y color:Solid
    Peso molecular:351.4
  • Trofinetide

    CAS:
    <p>Trofinetide (NNZ-2566) is a synthetic analog of the endogenous N-terminus tripeptide. It has been shown to be neuroprotective in animal models of brain injury.</p>
    Fórmula:C13H21N3O6
    Pureza:98.70% - 99.50%
    Forma y color:Solid
    Peso molecular:315.32
  • Mitiglinide

    CAS:
    <p>Mitiglinide (KAD-1229), an insulinotropic ATP-sensitive K+ channel antagonist, targets Kir6.2/SUR1; used in type 2 diabetes research.</p>
    Fórmula:C19H25NO3
    Forma y color:Solid
    Peso molecular:315.41
  • Esomeprazole magnesium salt

    CAS:
    <p>Esomeprazole magnesium, an oral proton pump inhibitor, curbs gastric acid by blocking H+, K+-ATPase; used in treating GERD.</p>
    Fórmula:C17H21MgN3O3S
    Forma y color:Solid
    Peso molecular:371.74