
Transportador de membrana / canal de iones
Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.
Subcategorías de "Transportador de membrana / canal de iones"
- ABC(3 productos)
- ATPasa(93 productos)
- Receptor de adiponectina(5 productos)
- CFTR(64 productos)
- Receptor CGRP(51 productos)
- Canal de calcio(493 productos)
- Canal de cloruro(49 productos)
- Receptor GABA(336 productos)
- Transportador de monoamina(23 productos)
- Transportador de monocarboxilato(17 productos)
- NKCC(2 productos)
- NPC1L1(3 productos)
- Cotransportador de Na-K-Cl(8 productos)
- OAT(27 productos)
- OCT(7 productos)
- P-gp(53 productos)
- Canal de potasio(276 productos)
- Bomba de protones(39 productos)
- SGLT(30 productos)
- Canal de sodio(202 productos)
- Canal TRP / TRPV(92 productos)
Mostrar 13 subcategorías más
Se han encontrado 2272 productos de "Transportador de membrana / canal de iones"
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Fluxametamide
CAS:<p>Fluxametamide, an isoxazoline insecticide, targets insect chloride channels with IC50s of 1.95 nM (GABA) and 225 nM (glutamate).</p>Fórmula:C20H16Cl2F3N3O3Pureza:99.49%Forma y color:SolidPeso molecular:474.26γ-Aminobutyric acid
CAS:<p>γ-Aminobutyric acid (4-Aminobutyric acid) is the most common inhibitory neurotransmitter in the central nervous system.</p>Fórmula:C4H9NO2Pureza:99.95%Forma y color:White Or Almost White(According To Quality Test Specification It Can Be White Or Almost White ) Solid PowderPeso molecular:103.12Cycloleucine
CAS:<p>Cycloleucine is an antagonist of NMDA receptor associated glycine receptor with a Ki of 600 μM.</p>Fórmula:C6H11NO2Pureza:99.90%Forma y color:SolidPeso molecular:129.164-Aminopyridine
CAS:<p>4-Aminopyridine (Dalfampridine) is a nonselective potassium (K+) channel blocker that binds to the cytoplasmic side of the cell membrane.</p>Fórmula:C5H6N2Pureza:91.61%Forma y color:SolidPeso molecular:94.11Disopyramide
CAS:<p>Disopyramide, or Triombrin, a class I anti-arrhythmic with membrane-stabilizing effects, has heart depressant, anticholinergic, and anesthetic properties.</p>Fórmula:C21H29N3OPureza:99.62%Forma y color:SolidPeso molecular:339.47DCEBIO
CAS:<p>DCEBIO, a 1-EBIO derivative, enhances Cl- secretion via hIK1 K+ channel and apical conductance in T84 cells.</p>Fórmula:C9H8Cl2N2OPureza:99.89%Forma y color:SolidPeso molecular:231.08Ciclopirox olamine
CAS:<p>Ciclopirox olamine is a broad-spectrum antifungal agent with additional antibacterial and anti-inflammatory activities.</p>Fórmula:C14H24N2O3Pureza:99.16% - >99.99%Forma y color:White To Yellow Solid Solid Particulate/PowderPeso molecular:268.35Dooku1
CAS:<p>Dooku1, Yoda1 analog, blocks Piezo1 channels, halting Ca2+ entry. IC50: 1.3μM in HEK 293, 1.5μM in HUVEC, stops Yoda1's aortic relaxation.</p>Fórmula:C13H9Cl2N3OSPureza:98.87% - 99.74%Forma y color:SolidPeso molecular:326.2Eleclazine hydrochloride
CAS:<p>Eleclazine hydrochloride (GS 6615 hydrochloride) is a novel inhibitor of late Na+ current (IC50: 0.7 uM).</p>Fórmula:C21H17ClF3N3O3Pureza:99.86%Forma y color:SolidPeso molecular:451.83IK1 inhibitor PA-6
CAS:<p>IK1 inhibitor PA-6 (PA-6) is a selective and potent inhibitor of IK1 (KIR2.x ion-channel-carried inward rectifier current)(IC50 of 12-15 nM for human and mouse</p>Fórmula:C31H32N4O2Pureza:98.9%Forma y color:SolidPeso molecular:492.61Penicillin G sodium salt
CAS:<p>Penicillin G sodium(Benzylpenicillin sodium) salt is a penicillin derivative commonly used in the form of its sodium or potassium salts in the treatment of a</p>Fórmula:C16H17N2NaO4SPureza:98.11%Forma y color:White To Off-White Crystalline PowderPeso molecular:356.37Trichlormethiazide
CAS:<p>Trichlormethiazide (Naqua) is a short-acting, 3-dichloromethyl derivative of hydrochlorothiazide, belonging to the class of thiazide diuretics.</p>Fórmula:C8H8Cl3N3O4S2Pureza:98.8% - 99.54%Forma y color:SolidPeso molecular:380.66AZD 7009
CAS:<p>AZD 7009 is a novel antiarrhythmic compound that inhibits the sodium current of hNav1.5 in CHO K1 cells with an IC50 of 11 uM.</p>Fórmula:C23H34N4O5Pureza:98.42% - 98.51%Forma y color:SoildPeso molecular:446.54Ethaverine hydrochloride
CAS:<p>Ethaverine hydrochloride is a homologue of papaverine and is used as a vasodilator and antispasmodic.Cost-effective and quality-assured.</p>Fórmula:C24H30ClNO4Pureza:99.66% - 99.90%Forma y color:SolidPeso molecular:431.96Prilocaine hydrochloride
CAS:<p>Prilocaine HCl: local amino amide anesthetic, blocks voltage-gated sodium channels in neurons, inhibits Na+ permeability.</p>Fórmula:C13H21ClN2OPureza:99.97%Forma y color:Needles White Or Off White Crystalline PowderPeso molecular:256.77CIQ
CAS:<p>CIQ is a subunit-selective potentiator of NMDA receptors containing the NR2C or NR2D subunit. EC50 value: 2.7 μM for NR2C and 2.8 μM for NR2D.</p>Fórmula:C26H26ClNO5Pureza:99.5%Forma y color:SolidPeso molecular:467.94Bupivacaine hydrochloride
CAS:<p>Bupivacaine hydrochloride (Vivacaine) is a long-lasting, amide local anesthetic that blocks sodium channels, inhibiting nerve impulses and sensation.</p>Fórmula:C18H28N2O·HClPureza:99.9% - >99.99%Forma y color:SolidPeso molecular:324.89BMS-195270
CAS:<p>BMS-195270 is a bio-active chemical.</p>Fórmula:C15H9ClF3N3O2Pureza:98.7%Forma y color:SolidPeso molecular:355.7Bemegride
CAS:<p>Bemegride (3-Ethyl-3-methylglutarimide), a central nervous system stimulant, serves as an antidote for barbiturate poisoning.</p>Fórmula:C8H13NO2Pureza:99.89%Forma y color:Physical Description White Crystalline Solid Sublimes At 212°F And 200 Mm Pressure (Ntp 1992)Peso molecular:155.19FG 7142
CAS:<p>FG 7142 (LSU-65), a benzodiazepine inverse agonist, targets α1 subunit GABAA receptors (EC50=137 nM, Ki=91 nM) and upregulates β-adrenoceptors.</p>Fórmula:C13H11N3OPureza:98.75%Forma y color:SolidPeso molecular:225.25
