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Transportador de membrana / canal de iones

Transportador de membrana / canal de iones

Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.

Subcategorías de "Transportador de membrana / canal de iones"

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Se han encontrado 2272 productos de "Transportador de membrana / canal de iones"

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  • Fluxametamide

    CAS:
    <p>Fluxametamide, an isoxazoline insecticide, targets insect chloride channels with IC50s of 1.95 nM (GABA) and 225 nM (glutamate).</p>
    Fórmula:C20H16Cl2F3N3O3
    Pureza:99.49%
    Forma y color:Solid
    Peso molecular:474.26
  • γ-Aminobutyric acid

    CAS:
    <p>γ-Aminobutyric acid (4-Aminobutyric acid) is the most common inhibitory neurotransmitter in the central nervous system.</p>
    Fórmula:C4H9NO2
    Pureza:99.95%
    Forma y color:White Or Almost White(According To Quality Test Specification It Can Be White Or Almost White ) Solid Powder
    Peso molecular:103.12
  • Cycloleucine

    CAS:
    <p>Cycloleucine is an antagonist of NMDA receptor associated glycine receptor with a Ki of 600 μM.</p>
    Fórmula:C6H11NO2
    Pureza:99.90%
    Forma y color:Solid
    Peso molecular:129.16
  • 4-Aminopyridine

    CAS:
    <p>4-Aminopyridine (Dalfampridine) is a nonselective potassium (K+) channel blocker that binds to the cytoplasmic side of the cell membrane.</p>
    Fórmula:C5H6N2
    Pureza:91.61%
    Forma y color:Solid
    Peso molecular:94.11
  • Disopyramide

    CAS:
    <p>Disopyramide, or Triombrin, a class I anti-arrhythmic with membrane-stabilizing effects, has heart depressant, anticholinergic, and anesthetic properties.</p>
    Fórmula:C21H29N3O
    Pureza:99.62%
    Forma y color:Solid
    Peso molecular:339.47
  • DCEBIO

    CAS:
    <p>DCEBIO, a 1-EBIO derivative, enhances Cl- secretion via hIK1 K+ channel and apical conductance in T84 cells.</p>
    Fórmula:C9H8Cl2N2O
    Pureza:99.89%
    Forma y color:Solid
    Peso molecular:231.08
  • Ciclopirox olamine

    CAS:
    <p>Ciclopirox olamine is a broad-spectrum antifungal agent with additional antibacterial and anti-inflammatory activities.</p>
    Fórmula:C14H24N2O3
    Pureza:99.16% - >99.99%
    Forma y color:White To Yellow Solid Solid Particulate/Powder
    Peso molecular:268.35
  • Dooku1

    CAS:
    <p>Dooku1, Yoda1 analog, blocks Piezo1 channels, halting Ca2+ entry. IC50: 1.3μM in HEK 293, 1.5μM in HUVEC, stops Yoda1's aortic relaxation.</p>
    Fórmula:C13H9Cl2N3OS
    Pureza:98.87% - 99.74%
    Forma y color:Solid
    Peso molecular:326.2
  • Eleclazine hydrochloride

    CAS:
    <p>Eleclazine hydrochloride (GS 6615 hydrochloride) is a novel inhibitor of late Na+ current (IC50: 0.7 uM).</p>
    Fórmula:C21H17ClF3N3O3
    Pureza:99.86%
    Forma y color:Solid
    Peso molecular:451.83
  • IK1 inhibitor PA-6

    CAS:
    <p>IK1 inhibitor PA-6 (PA-6) is a selective and potent inhibitor of IK1 (KIR2.x ion-channel-carried inward rectifier current)(IC50 of 12-15 nM for human and mouse</p>
    Fórmula:C31H32N4O2
    Pureza:98.9%
    Forma y color:Solid
    Peso molecular:492.61
  • Penicillin G sodium salt

    CAS:
    <p>Penicillin G sodium(Benzylpenicillin sodium) salt is a penicillin derivative commonly used in the form of its sodium or potassium salts in the treatment of a</p>
    Fórmula:C16H17N2NaO4S
    Pureza:98.11%
    Forma y color:White To Off-White Crystalline Powder
    Peso molecular:356.37
  • Trichlormethiazide

    CAS:
    <p>Trichlormethiazide (Naqua) is a short-acting, 3-dichloromethyl derivative of hydrochlorothiazide, belonging to the class of thiazide diuretics.</p>
    Fórmula:C8H8Cl3N3O4S2
    Pureza:98.8% - 99.54%
    Forma y color:Solid
    Peso molecular:380.66
  • AZD 7009

    CAS:
    <p>AZD 7009 is a novel antiarrhythmic compound that inhibits the sodium current of hNav1.5 in CHO K1 cells with an IC50 of 11 uM.</p>
    Fórmula:C23H34N4O5
    Pureza:98.42% - 98.51%
    Forma y color:Soild
    Peso molecular:446.54
  • Ethaverine hydrochloride

    CAS:
    <p>Ethaverine hydrochloride is a homologue of papaverine and is used as a vasodilator and antispasmodic.Cost-effective and quality-assured.</p>
    Fórmula:C24H30ClNO4
    Pureza:99.66% - 99.90%
    Forma y color:Solid
    Peso molecular:431.96
  • Prilocaine hydrochloride

    CAS:
    <p>Prilocaine HCl: local amino amide anesthetic, blocks voltage-gated sodium channels in neurons, inhibits Na+ permeability.</p>
    Fórmula:C13H21ClN2O
    Pureza:99.97%
    Forma y color:Needles White Or Off White Crystalline Powder
    Peso molecular:256.77
  • CIQ

    CAS:
    <p>CIQ is a subunit-selective potentiator of NMDA receptors containing the NR2C or NR2D subunit. EC50 value: 2.7 μM for NR2C and 2.8 μM for NR2D.</p>
    Fórmula:C26H26ClNO5
    Pureza:99.5%
    Forma y color:Solid
    Peso molecular:467.94
  • Bupivacaine hydrochloride

    CAS:
    <p>Bupivacaine hydrochloride (Vivacaine) is a long-lasting, amide local anesthetic that blocks sodium channels, inhibiting nerve impulses and sensation.</p>
    Fórmula:C18H28N2O·HCl
    Pureza:99.9% - >99.99%
    Forma y color:Solid
    Peso molecular:324.89
  • BMS-195270

    CAS:
    <p>BMS-195270 is a bio-active chemical.</p>
    Fórmula:C15H9ClF3N3O2
    Pureza:98.7%
    Forma y color:Solid
    Peso molecular:355.7
  • Bemegride

    CAS:
    <p>Bemegride (3-Ethyl-3-methylglutarimide), a central nervous system stimulant, serves as an antidote for barbiturate poisoning.</p>
    Fórmula:C8H13NO2
    Pureza:99.89%
    Forma y color:Physical Description White Crystalline Solid Sublimes At 212°F And 200 Mm Pressure (Ntp 1992)
    Peso molecular:155.19
  • FG 7142

    CAS:
    <p>FG 7142 (LSU-65), a benzodiazepine inverse agonist, targets α1 subunit GABAA receptors (EC50=137 nM, Ki=91 nM) and upregulates β-adrenoceptors.</p>
    Fórmula:C13H11N3O
    Pureza:98.75%
    Forma y color:Solid
    Peso molecular:225.25