Transportador de membrana / canal de iones
Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.
Subcategorías de "Transportador de membrana / canal de iones"
- ABC(3 productos)
- ATPasa(93 productos)
- Receptor de adiponectina(5 productos)
- CFTR(64 productos)
- Receptor CGRP(51 productos)
- Canal de calcio(493 productos)
- Canal de cloruro(49 productos)
- Receptor GABA(336 productos)
- Transportador de monoamina(23 productos)
- Transportador de monocarboxilato(17 productos)
- NKCC(2 productos)
- NPC1L1(3 productos)
- Cotransportador de Na-K-Cl(8 productos)
- OAT(27 productos)
- OCT(7 productos)
- P-gp(53 productos)
- Canal de potasio(276 productos)
- Bomba de protones(39 productos)
- SGLT(30 productos)
- Canal de sodio(202 productos)
- Canal TRP / TRPV(92 productos)
Mostrar 13 subcategorías más
Se han encontrado 2270 productos de "Transportador de membrana / canal de iones"
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VRT-532
CAS:<p>VRT-532 (CFpot-532) is an effective modulator of CFTR and is commonly used in studies of cystic fibrosis (CF) caused by CFTR defects.</p>Fórmula:C16H14N2OPureza:99.88% - 99.93%Forma y color:SolidPeso molecular:250.3CFTR corrector 8
CAS:<p>CFTR corrector 8: potent for cystic fibrosis research, modulates CFTR protein.</p>Fórmula:C29H27F2NO7Pureza:99.57%Forma y color:SolidPeso molecular:539.52L-838417
CAS:<p>L-838417 is a GABAA receptor subtype-selective benzodiazepine site-selective ligand and GABAA receptor-positive modulator used in the study of anxiety disorders</p>Fórmula:C19H19F2N7OPureza:98.12% - 99.70%Forma y color:SolidPeso molecular:399.4FEMA-4809
CAS:<p>FEMA-4809 activates TRPM8, the ion channel for cold sensation, and is used as a cooling agent.</p>Fórmula:C17H17N3O2SPureza:99.9%Forma y color:SolidPeso molecular:327.4ABT 102
CAS:<p>ABT 102 (CHEMBL398338) is a selective antagonist of transient receptor potential vanilloid 1 (TRPV1) receptor.</p>Fórmula:C21H24N4OPureza:98.38% - 99.86%Forma y color:SolidPeso molecular:348.44Elpetrigine
CAS:<p>Elpetrigine (GW273293) is a potential sodium channel blocker with antiepileptic activity that can be used to study epilepsy.</p>Fórmula:C10H7Cl3N4Pureza:99.04% - 99.43%Forma y color:SolidPeso molecular:289.55Stepronin
CAS:<p>Stepronin (TTPG) shows expectorant activities and inhibits airway secretion.</p>Fórmula:C10H11NO4S2Pureza:99.59%Forma y color:White Or Off White CrystallinePeso molecular:273.33VU 0240551
CAS:<p>VU 0240551 is a selective antagonist of neuronal K-Cl cotransporter KCC2 inhibitor with an IC50 of 560 nM. VU 0240551 inhibits L-type calcium channels and hERG.</p>Fórmula:C16H14N4OS2Pureza:99.9%Forma y color:SolidPeso molecular:342.44Mavatrep
CAS:<p>Mavatrep (JNJ-39439335) is a selective antagonist of TRPV1 with Ki of 6.5 nM and can be used for studies about inflammatory pain.</p>Fórmula:C25H21F3N2OPureza:98.51% - 99.31%Forma y color:SolidPeso molecular:422.44TAK-653
CAS:<p>TAK-653 is a selective AMPA receptor PAM with minimal agonist activity, showing antidepressant-like effects and safety in rats.</p>Fórmula:C19H23N3O3SPureza:99.89%Forma y color:SolidPeso molecular:373.47N106
CAS:<p>N106 is an activator of the SUMO-activating enzyme, E1 ligase, and triggers intrinsic sumoylation of SERCA2a. N106 can be used in studies about heart failure.</p>Fórmula:C17H14N4O3SPureza:99.69%Forma y color:SolidPeso molecular:354.38Butibufen
CAS:<p>Butibufen (FF-106) is a non-steroidal anti-inflammatory compound and LOX inhibitor with analgesic and antipyretic activity for the study of rheumatic diseases.</p>Fórmula:C14H20O2Pureza:98.11% - 98.91%Forma y color:SolidPeso molecular:220.31L-Cysteine S-sulfate
CAS:<p>L-Cysteine S-sulfate (S-Sulfo-L-cysteine) is an effective N-methyl-d-aspartate (NMDA) glutamatergic receptors agonist.</p>Fórmula:C3H7NO5S2Pureza:99.90% - 99.92%Forma y color:SolidPeso molecular:201.22Divaplon
CAS:<p>Divaplon is a GABA receptor agonist (IC50: 0.056 µM) that displays non-sedating anxiolytic behavioral characteristics in a rat model of anxiety.</p>Fórmula:C17H17N3O2Pureza:97.44% - 98.25%Forma y color:SolidPeso molecular:295.34Saripidem
CAS:<p>Saripidem (SL-85.0274) is a compound with anxiolytic activity.</p>Fórmula:C19H20ClN3OPureza:99.45%Forma y color:SolidPeso molecular:341.83Riluzole hydrochloride
CAS:<p>Riluzole hydrochloride, an anticonvulsant Na+ channel blocker, inhibits GABA uptake (IC50: 43 µM).</p>Fórmula:C8H6ClF3N2OSPureza:99.76%Forma y color:SolidPeso molecular:270.66Enecadin
CAS:<p>Enecadin is a neuroprotective agent.</p>Fórmula:C21H28FN3OPureza:98.53%Forma y color:SolidPeso molecular:357.46Sipatrigine
CAS:<p>Sipatrigine (619C89) is an inhibitor of glutamate release, TREK ion channels, TRESK channels, sodium channels, and calcium channels.</p>Fórmula:C15H16Cl3N5Pureza:98.64% - 99.77%Forma y color:SolidPeso molecular:372.68SKF96067
CAS:<p>SKF96067 is a reversible gastric H+/K+-ATPase inhibitor that can induce relaxation of human airway smooth muscle in vitro.</p>Fórmula:C21H22N2O2Pureza:99.89%Forma y color:SolidPeso molecular:334.41ANO1-IN-1
CAS:<p>ANO1-IN-1 blocks ANO1/2 channels (IC50: 2.56/15.43 μM) and hinders glioma cell growth.</p>Fórmula:C18H28N2O2SPureza:99.66%Forma y color:SolidPeso molecular:336.49KT-362 fumarate
CAS:<p>KT-362 fumarate, a novel antagonist of Ca, K, and Na channels, induces vasodilation and relaxes rabbit arterial strips.</p>Fórmula:C26H32N2O7SPureza:99.75% - 99.98%Forma y color:SolidPeso molecular:516.61AV-101
CAS:<p>AV-101 (4-Cl-KYN) is a prodrug antagonist at the glycine site of the NMDA receptor with antidepressant activity that reduces dyskinesia.</p>Fórmula:C10H11ClN2O3Pureza:97.78% - 98.27%Forma y color:SolidPeso molecular:242.66MSP3
CAS:<p>MSP3 is an agonist of TRPV1 (EC50 = 0.87 μM) and shows antinociceptive and neuroprotective effects.</p>Fórmula:C16H19NO3SPureza:99.89%Forma y color:SolidPeso molecular:305.39KR-32568
CAS:<p>KR-32568 is a sodium/hydrogen exchanger 1 (NHE-1) inhibitor (IC50: 230 nM).</p>Fórmula:C13H12FN3O2Pureza:99.91%Forma y color:SolidPeso molecular:261.25Quinacainol
CAS:<p>Quinacainol (RP 54272) is a new antiarrhythmic compound with class I antiarrhythmic effects in rats.</p>Fórmula:C21H30N2OPureza:99.64%Forma y color:SolidPeso molecular:326.48Alpidem
CAS:<p>Alpidem (Ananxyl), a non-sedative imidazopyridine anxiolytic, treats anxiety with high benzodiazepine receptor affinity.</p>Fórmula:C21H23Cl2N3OPureza:99.56% - 99.97%Forma y color:White To Off-White SolidPeso molecular:404.33GNE-8324
CAS:<p>GNE-8324 is a GluN2A selective positive allosteric modulator that enhances NMDAR-mediated synaptic responses in inhibitory, but not excitatory, neurons.</p>Fórmula:C18H18FN3OSPureza:98.68% - 99.34%Forma y color:SolidPeso molecular:343.42Tiludronate disodium
CAS:<p>Tiludronate disodium: osteoclast inhibitor for metabolic bone disorder research.</p>Fórmula:C7H7ClNa2O6P2SPureza:>99.99% - >99.99%Forma y color:Fine White To Off-White Crystalline PowderPeso molecular:362.57Neboglamine hydrochloride
CAS:<p>Neboglamine (CR-2249, XY-2401) hydrochloride boosts NMDA receptor, aids schizophrenia research, and is orally active.</p>Fórmula:C13H25ClN2O3Pureza:99.19%Forma y color:SolidPeso molecular:292.8Nelonemdaz
CAS:<p>Nelonemdaz (Neu2000) is an NMDA receptor antagonist with antioxidant activity that can be used to study cerebral infarction reperfusion injury.</p>Fórmula:C15H8F7NO3Pureza:99.52%Forma y color:SolidPeso molecular:383.22DMT1 blocker 1
CAS:<p>DMT1 blocker 1 inhibits DMT1; IC50=0.64μM; may prevent intestinal iron absorption.</p>Fórmula:C16H14N4O2Pureza:99.73%Forma y color:SolidPeso molecular:294.31Temiverine hydrochloride
CAS:<p>Temiverine hydrochloride is a potential calcium channel antagonist with anticholinergic effects that inhibits some of the functions of atropine.</p>Fórmula:C24H36ClNO3Pureza:99.26% - 99.43%Forma y color:SolidPeso molecular:422ZTZ240
CAS:<p>ZTZ240 is a KCNQ2 channel activator used in the study of epilepsy.</p>Fórmula:C12H8ClFN2OPureza:99.89%Forma y color:SolidPeso molecular:250.66S 18986
CAS:<p>S 18986 is a selective, orally active, brain penetrant positive allosteric modulator of AMPA-type receptors, showcasing cognitive-enhancing properties in</p>Fórmula:C10H12N2O2SPureza:99.64%Forma y color:SolidPeso molecular:224.28NC-1300-B
CAS:<p>NC-1300-B inhibits H(+)-K(+)-ATPase and is used in the study of gastric ulcers.</p>Fórmula:C17H19N3OSPureza:99.50%Forma y color:SolidPeso molecular:313.42ELB-139
CAS:<p>ELB-139 is a GABA A receptor agonist. ELB139 increases 5-HT in the striatum and prefrontal cortex of rats.</p>Fórmula:C14H16ClN3OPureza:>99.99%Forma y color:SolidPeso molecular:277.75CNS-5161 hydrochloride
CAS:<p>CNS-5161 hydrochloride (CNS 5161A) is a new antagonist of NMDA ion-channel.</p>Fórmula:C16H19Cl2N3S2Pureza:99.53%Forma y color:SolidPeso molecular:388.38Indecainide
CAS:<p>Indecainide (Ricainid) is an antiarrhythmic compound that is carcinogenic and may be used in studies secondary to coronary artery disease.</p>Fórmula:C20H24N2OPureza:98.01% - 98.96%Forma y color:SolidPeso molecular:308.42Suriclone
CAS:<p>Suriclone (RP 31264), a cyclic pyrrolidone for anxiety, modulates GABA-A receptors without major sedation.</p>Fórmula:C20H20ClN5O3S2Pureza:99.21% - 99.73%Forma y color:SolidPeso molecular:477.99Panadiplon
CAS:<p>Panadiplon (FG 10571) is a selective gamma-aminobutyric acid receptor agonist and partial agonist of 5GABAA, a benzodiazepine receptor, used in the treatment of</p>Fórmula:C18H17N5O2Pureza:98.30% - 98.94%Forma y color:SolidPeso molecular:335.36Bamocaftor
CAS:<p>Bamocaftor corrects CFTR in CF, restoring F508del-CFTR function, used with tezacaftor and VX-561 for F508del/MF patients.</p>Fórmula:C28H32F3N5O4SPureza:99.71%Forma y color:SolidPeso molecular:591.65Progabide
CAS:<p>Progabide (SL 76002) is an agonist of the gamma-aminobutyric acid receptor.</p>Fórmula:C17H16ClFN2O2Pureza:99.68%Forma y color:SolidPeso molecular:334.77Protonstatin-1
CAS:<p>Protonstatin-1: treats hypoglycemia & Alzheimer's, inhibits IGFIR kinase, used in cancer studies.</p>Fórmula:C8H5NO2S2Pureza:99.77%Forma y color:SolidPeso molecular:211.26Rilmakalim
CAS:<p>Rilmakalim is a potassium channel opener. Rilmakalim shows antivasoconstrictor effect.</p>Fórmula:C21H23NO5SPureza:99.8% - 99.9%Forma y color:SolidPeso molecular:401.48Elismetrep
CAS:<p>Elismetrep (MT-8554) is an orally available TRPM8 inhibitor with potential analgesic activity for the study of vasomotor symptoms in postmenopausal women.</p>Fórmula:C27H21F3N2O5SPureza:99.37% - 99.93%Forma y color:SolidPeso molecular:542.53AZD-1305
CAS:<p>AZD-1305: novel anti-arrhythmic blocking IKr, Ca, Na currents; useful in arrhythmia research.</p>Fórmula:C22H31FN4O4Pureza:99.31% - 99.86%Forma y color:SolidPeso molecular:434.5PD-118057
CAS:<p>PD-118057, a potent hERG activator, may treat long QT syndrome and heart failure without hERG activity inhibition.</p>Fórmula:C21H17Cl2NO2Pureza:99.16% - 99.97%Forma y color:SolidPeso molecular:386.27TASK-1-IN-1
CAS:<p>TASK-1-IN-1: Potent, selective TASK-1 blocker (IC50: 148 nM), weaker on TASK-3 (IC50: 1750 nM), anticancer properties.</p>Fórmula:C22H20N2O2Pureza:99.57%Forma y color:SoildPeso molecular:344.41GW 542573X
CAS:<p>GW 542573X is a potent and selective small molecule Ca2+-activated K+ 2 (SK2) channel activator.GW 542573X induces a leftward shift in the Ca2+ response curve</p>Fórmula:C19H28N2O5Pureza:99.91%Forma y color:SolidPeso molecular:364.44(+)-KCC2 blocker 1
CAS:<p>(+)-KCC2 blocker 1 is a selective blocker of KCC2 (IC50 = 0.4 μM).</p>Fórmula:C22H25NO5SPureza:99.88%Forma y color:SolidPeso molecular:415.5Cerebrocrast
CAS:<p>Cerebrocrast (IOS-11212) has anti-inflammatory and hypoglycemic activity, blocks human platelet activation, and is used in the study of diabetes.</p>Fórmula:C26H35F2NO7Pureza:99.71%Forma y color:SolidPeso molecular:511.56Nerisopam
CAS:<p>Nerisopam is an agonist of gamma-aminobutyric acid (GABA) receptor.</p>Fórmula:C18H19N3O2Pureza:97.07%Forma y color:SolidPeso molecular:309.36SCH28080
CAS:<p>SCH28080 is a reversible and K+-competitive inhibitor of gastric H+/K+-ATPase with an IC50 value of 20 nM (rabbit microsomal membrane).SCH28080 is a potent</p>Fórmula:C17H15N3OPureza:99.24%Forma y color:SolidPeso molecular:277.32SKA-111
CAS:<p>SKA-111 activates KCa3.1 potassium channels, modulates membrane potential in endothelial cells, and dilates rat coronary arteries.</p>Fórmula:C12H10N2SPureza:99.9%Forma y color:SolidPeso molecular:214.29PG01
CAS:<p>PG01 is a potent CFTR Cl-channel potentiator, effective against ΔF508 (Ka 0.3 μM), and also against E193K, G970R and G551D (CFTR mutants), with Kd values of 0.</p>Fórmula:C28H29N3O2Pureza:99.87%Forma y color:SolidPeso molecular:439.55Saviprazole
CAS:<p>Saviprazole (Hoe-731), a proton pump inhibitor, is used potentially for treatment of gastric ulcer.</p>Fórmula:C15H10F7N3O2S2Pureza:97.07% - 97.17%Forma y color:SolidPeso molecular:461.38SET 2
CAS:<p>SET 2 is an antagonist of transient receptor potential vanilloid type 2(TRPV2) with an IC50 of 0.46 μM. SET 2 shows selectivity over TRPV1, TRPV3 and TRPV4.</p>Fórmula:C17H21F3N4O2SPureza:99.77%Forma y color:SolidPeso molecular:402.43Muscimol HBr
CAS:<p>Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.</p>Fórmula:C4H7BrN2O2Pureza:98.13%Forma y color:Off-White PowderPeso molecular:195.01MK-0448
CAS:<p>MK-0448 is a novel and selective blocker of the Kv1.5 (KCNA5) channel, a key channel involved in cardiac repolarization current I Kur.</p>Fórmula:C24H21FN4O2SPureza:99.25% - 99.79%Forma y color:SolidPeso molecular:448.51RWJ-51204
CAS:<p>RWJ-51204: potent adenosine A2A blocker, GABA(A) partial agonist (IC50: 0.2-2 nM), neuroprotective, may treat Parkinson's.</p>Fórmula:C21H19F2N3O3Pureza:99.57% - 99.95%Forma y color:SolidPeso molecular:399.39Fengabine
CAS:<p>Fengabine (SL-79229) is a GABA receptor agonist with antidepressant activity and is used to treat depression.</p>Fórmula:C17H17Cl2NOPureza:99%Forma y color:SolidPeso molecular:322.23HC-070
CAS:<p>HC-070 is a TRPC5 and TRPC4 antagonist (IC50 = 9.3 nM and 46 nM).</p>Fórmula:C22H20Cl2N4O4Pureza:98.48%Forma y color:SolidPeso molecular:475.32Abeprazan hydrochloride
CAS:<p>Abeprazan hydrochloride (Fexuprazan hydrochloride) is an effective reversible potassium-competitive acid blocker with oral activity, inhibiting H+, K+ -atPase</p>Fórmula:C19H18ClF3N2O3SPureza:98.57%Forma y color:SolidPeso molecular:446.87RL648_81
CAS:<p>RL648_81 is a selective activator of KCNQ2/3 channels (EC50 = 190 nM). RL648_81 can be used in studies about neuronal hyperexcitability neurologic disorders.</p>Fórmula:C17H17F4N3O2Pureza:99.82%Forma y color:SolidPeso molecular:371.33Sarmazenil
CAS:<p>Sarmazenil (Ro 15-3505) is a partial inverse agonist at the benzodiazepine receptor and is used in the study of chronic hepatic encephalopathy.</p>Fórmula:C15H14ClN3O3Pureza:99.46%Forma y color:SolidPeso molecular:319.74Pyr3
CAS:<p>Pyr3 selectively blocks TRPC3 channels, reducing Ca2+ influx; it's effective at 700 nM.</p>Fórmula:C16H11Cl3F3N3O3Pureza:98.04%Forma y color:SolidPeso molecular:456.63Losigamone
CAS:<p>Losigamone (AO-33) is an agonist of GABA receptor and can be used in studies about the treatment of partial seizures.</p>Fórmula:C12H11ClO4Pureza:99.98%Forma y color:SolidPeso molecular:254.67Sulcardine sulfate
CAS:<p>Sulcardine sulfate (B-87823) is a multi-ion channel blocker with antiarrhythmic activity that inhibits Na+, K+, and Ca2+ channels.</p>Fórmula:C24H35N3O8S2Pureza:98.74%Forma y color:SolidPeso molecular:557.68FR-167356
CAS:<p>FR-167356 inhibits a3 isoform H⁺-ATPase (IC50: 170-370 nM), targeting osteoclasts, kidneys, macrophages; reduces B16-F10 bone metastasis.</p>Fórmula:C19H17Cl2NO3Pureza:98.44% - 99.74%Forma y color:SolidPeso molecular:378.25Ani9
CAS:<p>Ani9 selectively blocks ANO1/TMEM16A with a 77 nM IC50, useful for ANO1 research and treating cancer, hypertension, pain, diarrhea, asthma.</p>Fórmula:C17H17ClN2O3Pureza:99.73%Forma y color:SolidPeso molecular:332.78Trombodipine
CAS:<p>Trombodipine (PCA-4230) is a platelet aggregation inhibitor with antithrombotic activity and protection against Listeria monocytogenes.</p>Fórmula:C21H24N2O7SPureza:98.73% - 99.14%Forma y color:SolidPeso molecular:448.49DFP00173
CAS:<p>DFP00173: Potent, selective AQP3 inhibitor; IC50 ~0.1-0.4 μM; less effective on AQP7, AQP9.</p>Fórmula:C11H7Cl2N3O3SPureza:99.53% - 99.53%Forma y color:SolidPeso molecular:332.16DMP-543
CAS:<p>DMP-543 (XR-543) is a potassium channel (KV7 channel) blocker that enhances the release of neurotransmitters.</p>Fórmula:C26H18F2N2OPureza:99.89%Forma y color:SolidPeso molecular:412.43Leminoprazole
CAS:<p>Leminoprazole is an orally available H+,K(+)-ATPase inhibitor that protects gastric mucosal cells from various cellular damages.</p>Fórmula:C19H23N3OSPureza:99.08% - 99.56%Forma y color:SolidPeso molecular:341.47UK 66914
CAS:<p>UK 66914 is a K(+) channel blocker for the study of cardiac arrhythmias.</p>Fórmula:C18H24N4O3SPureza:99.75%Forma y color:SolidPeso molecular:376.47ZM 226600
CAS:<p>ZM 226600 is an ATP-sensitive potassium channel opener with an EC50 value of 500 nM. ZM226600 has an inhibitory effect on spontaneous bladder activity.</p>Fórmula:C16H14F3NO4SPureza:99.87%Forma y color:SolidPeso molecular:373.35NNC 05-711
CAS:<p>NNC 05-711 (NO-711 hydrochloride) is a potent and selective inhibitor of GAT-1 (GABA transporter 1), exerting anticonvulsant and analgesic effects.</p>Fórmula:C21H23ClN2O3Pureza:99.92%Forma y color:SolidPeso molecular:386.87Quinabactin
CAS:<p>Quinabactin (LC-66C6): ABA agonist, induces guard cell closure, reduces water loss, hinders germination, boosts drought resistance in Arabidopsis/soybean.</p>Fórmula:C20H24N2O3SPureza:99.63%Forma y color:SolidPeso molecular:372.48NaV1.2/1.6 channel blocker-1
CAS:<p>NaV1.2/1.6 channel blocker-1 is a NaV1.2/1.6 channel blocker that inhibits rNaV1.6 and can be used to study generalised epilepsy and movement disorders.</p>Fórmula:C14H14N2OSPureza:99.54%Forma y color:SolidPeso molecular:258.34XE991
CAS:<p>XE991 is a Kv7 (KCNQ) channel blocker.XE 991 dihydrochloride inhibits Kv7.1 (KCNQ1) and M-current and can be used in the study of neurological disorders.</p>Fórmula:C26H20N2OPureza:98.87%Forma y color:SolidPeso molecular:376.45Silperisone HCl
CAS:<p>Silperisone HCl is a muscle relaxant and vasodilator, treating myoclonus, hypertonia, dystonia, and myospasm by blocking Na+ and Ca2+ channels.</p>Fórmula:C15H25ClFNSiPureza:99.62%Forma y color:SolidPeso molecular:301.9Ru-32514
CAS:<p>Ru-32514 is a benzodiazepine receptor agonist.</p>Fórmula:C18H17N3O2Pureza:99.21%Forma y color:SolidPeso molecular:307.35TWIK-1/TREK-1-IN-3
CAS:<p>TWIK-1/TREK-1-IN-3 is a potassium channel TREK-1 inhibitor TWIK-1/TREK-1-IN-3 has antidepressant activity and can be used to study depression.</p>Fórmula:C19H27F3N2O2Pureza:99.04%Forma y color:SolidPeso molecular:372.43IKs124
CAS:<p>IKs124 is a KCNE2/KCNQ1 potassium channel blocker, for hKCNE1 and hKCNE3, and can be used to study peptic ulcers.</p>Fórmula:C18H26N2O3SPureza:99.53%Forma y color:SolidPeso molecular:350.48UCL 2077
CAS:<p>UCL 2077 blocks KCNQ channels, related to epilepsy, and selective slow-afterhyperpolarization channels, with 500 nM IC50, sparing Ca2+ channels.</p>Fórmula:C25H22N2Pureza:99.58%Forma y color:SolidPeso molecular:350.46Aptiganel
CAS:<p>Aptiganel (CNS-1102) is a non-competitive NMDA antagonist, a peptide that may be used to study acute ischemic stroke.</p>Fórmula:C20H21N3Pureza:98.13% - 98.90%Forma y color:SolidPeso molecular:303.4Cirsimaritin
CAS:<p>Cirsimaritin has anti-bacterial, anti-inflammatory, anti-tumor, antioxidant effects, and protects kidneys; it weakly targets GABAA receptors.</p>Fórmula:C17H14O6Pureza:99.9%Forma y color:SolidPeso molecular:314.29YM758
CAS:<p>YM758 is an inhibitor of If current channel.</p>Fórmula:C26H32FN3O4Pureza:99.65%Forma y color:SolidPeso molecular:469.55Golexanolone
CAS:<p>Golexanolone can be used to study neurological diseases.</p>Fórmula:C21H31NO2Pureza:99.90% - 99.99%Forma y color:SolidPeso molecular:329.48BPDBA
CAS:<p>BPDBA is an effective, selective, and non-competitive inhibitor of the betaine/GABA transporter (BGT-1), displaying inhibitory activity against human BGT-1 and</p>Fórmula:C19H20Cl2N2OPureza:99.37% - 99.95%Forma y color:SolidPeso molecular:363.28TC-I 2014
CAS:<p>TC-I 2014 shows antiallodynic properties in pain models.</p>Fórmula:C23H19F6N3OPureza:99.07%Forma y color:SolidPeso molecular:467.41R 56865
CAS:<p>R 56865 is a weak potential-operated channel inhibitor that inhibits the late sodium current in human isolated cardiomyocytes.</p>Fórmula:C23H28FN3OSPureza:99.52%Forma y color:SolidPeso molecular:413.55Orphenadrine
CAS:<p>Orphenadrine is a noncompetitive N-methyl-D-aspartate (NMDA) receptor antagonist that inhibits clonal HERG channels in a concentration-dependent manner,</p>Fórmula:C18H23NOPureza:98.91% - 99.11%Forma y color:SolidPeso molecular:269.38Linaprazan
CAS:<p>Linaprazan (AZD0865) inhibits gastric H+,K+-ATPase by K+-competitive binding with an IC50 of 1.0 μM.</p>Fórmula:C21H26N4O2Pureza:99.54%Forma y color:SolidPeso molecular:366.46OADS
CAS:<p>OADS is an inhibitor of ClC-ec1 with low micromolar affinity. OADS has no specific effect on a CLC channel (ClC-1).</p>Fórmula:C30H42N2O8S2Forma y color:SolidPeso molecular:622.79PU-48
CAS:<p>PU-48 is a potent inhibitor of urea transporters A (UT-A) with an IC50 value of 0.32 μM, exhibiting a significant diuretic effect in mouse models without</p>Fórmula:C14H12N2O3SForma y color:SolidPeso molecular:288.32URAT1 inhibitor 8
CAS:<p>URAT1 Inhibitor 8 (example 247) serves as a highly potent inhibitor of URAT1, demonstrating an IC50 value of 0.001 μM.</p>Fórmula:C19H13ClFN3O4SForma y color:SolidPeso molecular:433.84NaV1.7 Blocker-801
CAS:<p>NaV1.7 Blocker-801 is a potent NaV1.7 blocker.</p>Fórmula:C20H15ClF2N6O3S2Forma y color:SolidPeso molecular:524.95MCT1-IN-2
CAS:<p>SR13800 is a monocarboxylate transporter 1 (MCT1) inhibitor with cell-permeable.</p>Fórmula:C25H29N3O2SForma y color:SolidPeso molecular:435.58mGAT3/4-IN-2
CAS:<p>mGAT3/4-IN-2 are potent inhibitors of mGAT3/mGAT4 with their pIC50 values of 5.44 and 5.25, respectively.</p>Fórmula:C26H32ClN3OS2Forma y color:SolidPeso molecular:502.13GDC-6599
CAS:<p>GDC-6599 (Example 8) is an orally active inhibitor of the TRPA1 channel, potentially useful for researching TRPA1-mediated conditions, including pain [1].</p>Fórmula:C20H19ClN6O3Forma y color:SolidPeso molecular:426.86MONIRO-1
CAS:<p>MONIRO-1 blocks T/N-type Ca²⁺ channels: hCav2.2 (IC50: 34μM), hCav3.1 (3.3μM), hCav3.2 (1.7μM), hCav3.3 (7.2μM).</p>Fórmula:C23H24ClFN4O3Forma y color:SolidPeso molecular:458.92γ-Kainylglutamic acid
CAS:<p>gamma-Kainylglutamic acid is a selective amino acid-induced neuroexcitation antagonist.</p>Fórmula:C15H22N2O7Pureza:98%Forma y color:SolidPeso molecular:342.34(-)-Bicuculline methochloride
CAS:<p>(-)-Bicuculline methochloride is a potent antagonist of GABAA receptor.</p>Fórmula:C21H20ClNO6Pureza:98%Forma y color:SolidPeso molecular:417.84Y-27152
CAS:<p>Y-27152 is a prodrug of the KATP (Kir6) channel opener Y-26763 and is a long-acting K+ channel opener.</p>Fórmula:C21H22N2O4Pureza:98%Forma y color:SolidPeso molecular:366.41P-1075
CAS:<p>P-1075 activates SUR2-KIR6 channels at 45 nM; may open mitoKATP channels and protect the heart.</p>Fórmula:C12H17N5Pureza:99.85%Forma y color:SolidPeso molecular:231.3FGIN-1-27
CAS:<p>FGIN-1-27 is a high-affinity agonist of the translocator protein and a specific peripheral benzodiazepine receptor (PBR) ligand(Ki = 5.0 nM).</p>Fórmula:C28H37FN2OPureza:99.86%Forma y color:SolidPeso molecular:436.6CS-526
CAS:<p>CS-526 is a reversible proton pump inhibitor targeting the K+ site on H+,K+-ATPase, reducing gastric acid secretion and preventing mucosal lesions.</p>Fórmula:C20H22FN3OForma y color:SolidPeso molecular:339.41NMDA receptor modulator 6
CAS:<p>NMDA receptor regulator 6 (Compound 183) is an effective NMDA receptor regulator and has research value in neurological disorders.</p>Fórmula:C20H17FN2O4SForma y color:SolidPeso molecular:400.42Pumaprazole
CAS:<p>Pumaprazole (BY-841) is an antagonist of a reversible proton pump.</p>Fórmula:C19H22N4O2Pureza:99.91%Forma y color:SolidPeso molecular:338.4ROMK-IN-32
CAS:<p>ROMK-IN-32 is an inhibitor of the extra-renal medullary potassium channel (ROMK) (IC50: 35 nM) and also inhibits hERG (IC50: 22 μM).</p>Fórmula:C24H28N4O5Forma y color:SolidPeso molecular:452.5N-Linolenoylethanolamine
CAS:<p>N-Linolenoylethanolamine (18:3 NAE), an endocannabinoid, functions as a vanillin receptor (TRPV1) agonist [1].</p>Fórmula:C20H35NO2Forma y color:SolidPeso molecular:321.505BMS-986169
CAS:<p>BMS-986169 is a high-affinity and selective negative allosteric modulator of the NMDA receptor GluN2B subunit, depression.</p>Fórmula:C23H27FN2O2Pureza:97.61%Forma y color:SolidPeso molecular:382.47DNDS
CAS:<p>DNDS is a channel blocker of voltage-dependent cystic fibrosis transmembrane conductance regulator (CFTR).</p>Fórmula:C14H8N2Na2O10S2Pureza:99.92%Forma y color:Physical Description White Powder (Ntp 1992)Peso molecular:474.33Pristinamycin IA
CAS:<p>Pristinamycin IA (Mikamycin B) is a substrate for the P-glycoprotein and a cyclo-peptidic macrolactone antibiotic.</p>Fórmula:C45H54N8O10Pureza:97.44%Forma y color:SolidPeso molecular:866.96CFTR corrector 6
CAS:<p>CFTR corrector 6, a potent CFTR potentiator, aids cystic fibrosis research and related disorders.</p>Fórmula:C22H13F4N9Forma y color:SolidPeso molecular:479.39SLC13A5-IN-1
CAS:<p>SLC13A5-IN-1 is a selective inhibitor of sodium-citrate co-transporter (SLC13A5),completely blocks the uptake of 14C-citrate(IC50 : 0.022 μM in HepG2 cells).</p>Fórmula:C19H19Cl3N2O3SPureza:99.67%Forma y color:SolidPeso molecular:461.79TRPC5 modulator-1
CAS:<p>TRPC5 modulator-1 (Compound 9) is a TRPC5 modulator (IC50<1 nM) that can be used to study neuropsychiatric disorders.</p>Fórmula:C23H27FN2O4Forma y color:SolidPeso molecular:414.47AC-4
CAS:<p>AC-4 is a blocker of photoswitchable TRPV1 channel.</p>Fórmula:C26H25F3N4O2SForma y color:SolidPeso molecular:514.56PF 04531083
CAS:<p>PF 04531083 is a selective blocker of the NaV1.8 channel. PF 04531083 can be used for neuropathic and inflammatory pain studies.</p>Fórmula:C17H16ClN5O2Pureza:99.85%Forma y color:SolidPeso molecular:357.79CP 154526
CAS:<p>CRF1 receptor antagonist</p>Fórmula:C23H33ClN4Pureza:98%Forma y color:SolidPeso molecular:400.99AMPA receptor modulator-2
CAS:<p>AMPA receptor modulator-2 is a modulator of AMPA receptor. The pIC50 value for TARPγ2 dependent AMPA receptor is 10.1.</p>Fórmula:C15H6F6N4OSPureza:99.8%Forma y color:SolidPeso molecular:404.29TRPC3/6-IN-2
CAS:<p>TRPC3/6-IN-2 is a potent inhibitor of TRPC3 and TRPC6, exhibiting IC50 values of 16 nM for TRPC3 and 29.8 nM for TRPC6, respectively [1].</p>Fórmula:C18H23F2N5Forma y color:SolidPeso molecular:347.41Antiarrhythmic agent-1
CAS:<p>Antiarrhythmic agent-1 (example I), functioning as an antiarrhythmic agent and an IKr potassium channel blocker (IC 50 <1 μM), effectively inhibits cardiac</p>Fórmula:C25H27N3O4SForma y color:SolidPeso molecular:465.56A-1165442
CAS:<p>A-1165442 is a competitive TRPV1 antagonist. For human TRPV, the IC50 values is 9 nM.</p>Fórmula:C22H20ClF2N3O2Forma y color:SolidPeso molecular:431.86Dibutyryl-cGMP sodium
CAS:<p>Bt2cGMP sodium is a cGMP analog, activates PKG, inhibits platelet [3H]-arachidonate, and induces analgesia via K+ channels.</p>Fórmula:C18H24N5NaO9PPureza:98%Forma y color:SolidPeso molecular:508.38NMDA receptor modulator 4
CAS:<p>NMDA receptor modulator 4 (Compound 169) can be used for the research of neurological disorder that is a potent modulator of NMDA receptor [1].</p>Fórmula:C13H9F3N2O3SForma y color:SolidPeso molecular:330.28P2X3 antagonist 34
CAS:<p>Potent P2X3 antagonist 34, oral, selective for human, rat, guinea pig receptors; IC50s: 25/92/126 nM; strong anti-tussive, no taste change.</p>Fórmula:C24H26F2N4O3Pureza:98%Forma y color:SolidPeso molecular:456.48ML-252 hydrochloride
CAS:<p>ML-252 is a potent, selective inhibitor of the Kv7.2 voltage-gated potassium channel, demonstrating an IC50 value of 69 nM in patch clamp assays. It exists as the (S)-enantiomer, which is significantly more effective than both its (R)-enantiomer counterpart and the racemic mixture, with respective IC50 values of 944 nM and 160 nM. ML-252 exhibits high selectivity for Kv7.2 over other potassium channel subtypes and shows minimal activity against more than 68 G protein-coupled receptors, various transporters, L- and N-type calcium channels, K_ATP, and hERG potassium channels. However, it does inhibit the melatonin MT1 receptor by 61% at a 10 µM concentration.</p>Fórmula:C20H24N2OHClForma y color:SolidPeso molecular:344.9Licostinel
CAS:<p>Licostinel (CGP 63446) is a glutamate receptor antagonist. Licostinel protects against permanent focal cerebral ischemia.</p>Fórmula:C8H3Cl2N3O4Pureza:98.02%Forma y color:SolidPeso molecular:276.033′-Acetate-ATP
CAS:<p>3’-Acetate-ATP, an analogue of ATP and its acetylation product, exhibits maximum ultraviolet absorption at 259 nm in neutral aqueous solutions.</p>Fórmula:C12H18N5O14P3Forma y color:SolidPeso molecular:549.22GMA-839
CAS:<p>GMA-839 is a selective modulator of gamma-aminobutyric acid(A) receptors.</p>Fórmula:C21H31F3O3Pureza:98%Forma y color:SolidPeso molecular:388.46Biricodar
CAS:<p>Biricodar is a P-glycoprotein and MRP-1 modulator.</p>Fórmula:C34H41N3O7Pureza:98%Forma y color:SolidPeso molecular:603.71ADX71441
CAS:<p>ADX71441, a GABAB PAM, lengthens urinary latencies, lessens events & volume, and may aid in alcoholism and bladder pain.</p>Fórmula:C19H15ClF2N4O4Forma y color:SolidPeso molecular:436.8Cavα2δ1&NET-IN-3
CAS:<p>Cavα2δ1&NET-IN-3 (example 216) is an inhibitor targeting both the α2δ subunit of voltage-gated calcium channels (VGCC) and the noradrenaline transporter (NET).</p>Fórmula:C24H30N6O2SForma y color:SolidPeso molecular:466.6p-fin4
CAS:<p>p-fin4, a peptide, inhibits STEP-GluA2 interaction, Ki 0.4 μM; may enhance cognition, has anxiolytic and antidepressant effects.</p>Fórmula:C39H53N8O18PForma y color:SolidPeso molecular:952.85Adipiplon
CAS:<p>Adipiplon(NG2-73, NG273) is a novel selective gamma-aminobutyric acid (GABA) partial agonist.</p>Fórmula:C18H18FN7Forma y color:SolidPeso molecular:351.38CGP 64213
CAS:<p>CGP 64213 is a GABAb receptor agonist.</p>Fórmula:C26H36IN2O7PPureza:98%Forma y color:SolidPeso molecular:646.45PF-06456384
CAS:<p>PF-06456384 is a highly potent and selective NaV1.7 inhibitor with IC50 value of 0.01 nM.</p>Fórmula:C35H32F3N7O3S2Pureza:98%Forma y color:SolidPeso molecular:719.8AGN-201904Z
CAS:<p>AGN-201904Z is a slow-release, acid-resistant pro-PPI that turns into omeprazole, offering extended acid suppression.</p>Fórmula:C25H25N3NaO8S2Pureza:98%Forma y color:SolidPeso molecular:582.6VU6007477
CAS:<p>VU6007477: M1 PAM, EC50=230 nM, min. agonist activity, penetrates CNS, no seizure AEs.</p>Fórmula:C24H26N6O2Forma y color:SolidPeso molecular:430.5AR-C141990
CAS:<p>AR-C141990 is a lactate transporters inhibitor.</p>Fórmula:C26H28N4O4SForma y color:SolidPeso molecular:492.59Piprofurol
CAS:<p>Piprofurol is used as a Calcium channel blocker.</p>Fórmula:C26H33NO6Pureza:98%Forma y color:SolidPeso molecular:455.54(Rac)-AMG8379
CAS:<p>(Rac)-AMG8379 ((Rac)-AMG8380) is a racemate of AMG8379 which is an orally active and selective sulfonamide NaV1.7 antagonist.</p>Fórmula:C25H16ClF2N3O5SPureza:99.6%Forma y color:SolidPeso molecular:543.93Nepaprazole
CAS:<p>Nepaprazole (TY-11345) is a potent proton pump inhibitor; IC50: 5.8µM at pH 6.0, 9.9µM at pH 7.4. Better inhibition in weak acid.</p>Fórmula:C18H19N3O2SPureza:98%Forma y color:SolidPeso molecular:341.43RS 5773
CAS:<p>RS 5773 is a benzothiazepine derivative with antianginal effects.</p>Fórmula:C29H33ClN2O4SPureza:98%Forma y color:SolidPeso molecular:541.1JT010
CAS:<p>JT010 is an effective agonist of TRPA1 (EC50 = 0.65 nM).</p>Fórmula:C16H19ClN2O3SPureza:99.75%Forma y color:SolidPeso molecular:354.85BTG 502
CAS:<p>BTG 502 is an alkylamide insecticide that binds to voltage-gated sodium channels, antagonising the activation of sodium channels by Batrachotoxin (BTX).</p>Fórmula:C21H24BrNOPureza:99.30%Forma y color:SolidPeso molecular:386.33TROX-1
CAS:<p>TROX-1 is the activation state-dependent Cav2 channel antagonist.</p>Fórmula:C22H16ClFN6OPureza:98%Forma y color:SolidPeso molecular:434.85Dasolampanel etibutil
CAS:<p>Dasolampanel etibutil is a novel selective antagonist of ionotropic glutamate receptor 5 (iGluR5).</p>Fórmula:C23H32ClN5O3Forma y color:SolidPeso molecular:461.98U 89843A
CAS:<p>U 89843A is a positive allosteric modulator of gamma-aminobutyric acid (GABA)A receptors.</p>Fórmula:C16H23N5Pureza:99.62%Forma y color:SolidPeso molecular:285.39(R)-3,4-DCPG
CAS:<p>AMPA receptor antagonist with weak activity at NMDA receptors and little activity at kainate receptors</p>Fórmula:C10H9NO6Pureza:98%Forma y color:SolidPeso molecular:239.18JM-1232
CAS:<p>JM-1232 is a sedative and hypnotic drug being researched as a potential anesthetic.</p>Fórmula:C24H27N3O2Forma y color:SolidPeso molecular:389.49Afizagabar
CAS:<p>Afizagabar, a first-in-class α5-GABAAR antagonist, IC50: 585 nM, Ki: 66 nM, may boost memory.</p>Fórmula:C19H12FN3O2SForma y color:SolidPeso molecular:365.38CGP-54626 free base
CAS:<p>CGP-54626 is a selective antagonist of the GABAB receptor (IC50 = 4 nM ).</p>Fórmula:C18H28Cl2NO3PPureza:98%Forma y color:SolidPeso molecular:408.3CFTR corrector 12
CAS:<p>CFTR corrector 12 is a CFTR corrector that rescues all mutant proteins except M760R ABCA3 and can be used to study cystic fibrosis.</p>Fórmula:C19H21ClN4O2S2Pureza:99.47%Forma y color:SolidPeso molecular:436.98M084 hydrochloride
CAS:<p>M084 hydrochloride, a TRPC4/5 channel blocker, exhibits IC50 values of 10.3 μM and 8.2 μM, respectively. This compound is noted for its antidepressant and anxiolytic effects [1] [2].</p>Fórmula:C11H16ClN3Forma y color:SolidPeso molecular:225.72PPADS tetrasodium
CAS:<p>PPADS tetrasodiuma is a P2X receptor antagonist and an inhibitor of the inverse mode of Na/Ca²⁺ exchange in guinea pig airway smooth muscle.</p>Fórmula:C14H10N3Na4O12PS2Pureza:95% - ≥95%Forma y color:SolidPeso molecular:599.3NaPi2b-IN-2
CAS:<p>NaPi2b-IN-2 (compound 5) serves as a potent inhibitor of the sodium-dependent transport protein 2b (SLC34A2, NaPi2b), exhibiting an IC50 of 38 nM against human</p>Fórmula:C41H47ClF3N5O5SPureza:98%Forma y color:SolidPeso molecular:814.36Crobenetine hydrochloride
CAS:<p>Crobenetine hydrochloride, a sodium channel antagonist, is used potentially for the treatment of stroke.</p>Fórmula:C25H34ClNO2Forma y color:SolidPeso molecular:416CGP 55845 hydrochloride
CAS:<p>CGP55845 hydrochloride is a potent and selective GABAB receptor antagonist with an IC 50 of 6 nM which can be used in neurological research [1] [2].</p>Fórmula:C18H23Cl3NO3PForma y color:SolidPeso molecular:438.71XR9051 Hydrochloride
CAS:<p>XR9051 Hydrochloride, a potent modulator of P-glycoprotein-mediated multidrug resistance (MDR), inhibits the binding of cytotoxics to P-glycoprotein.</p>Fórmula:C39H39ClN4O5Forma y color:SolidPeso molecular:679.21α,β-Methylene ATP trisodium
CAS:<p>α,β-Methylene ATP trisodium is a ligand of P2X3 and P2X7 receptor.</p>Fórmula:C11H15N5Na3O12P3Pureza:99.66%Forma y color:SolidPeso molecular:571.15Dimethylamiloride
CAS:<p>Dimethylamiloride is a specific inhibitor of antiporters [1].</p>Fórmula:C8H12ClN7OPureza:98%Forma y color:SolidPeso molecular:257.68PF-05105679
CAS:<p>PF-05105679 is a selective TRPM8 antagonist (IC50 = 103 nM). PF-05105679 can be used in research on cold-related pain.</p>Fórmula:C26H21FN2O3Pureza:99.84%Forma y color:SolidPeso molecular:428.45L 691121
CAS:<p>L 691121 is a class III antiarrhythmic compound. It also blocks potassium currents.</p>Fórmula:C22H25ClN4O5SPureza:98%Forma y color:SolidPeso molecular:492.98mGAT-IN-1
CAS:<p>mGAT-IN-1 is a potent, non-selective GAT inhibitor that inhibits mGAT3 activity well (IC50: 2.5 μM, pIC50: 5.61).</p>Fórmula:C28H34ClN3O2S2Forma y color:SolidPeso molecular:544.17Risevistinel
CAS:<p>Risevistinel (NYX-783), a positive allosteric modulator of the N-methyl-D-aspartate (NMDA) receptor, may mitigate cognitive deficits in neurodegenerative</p>Fórmula:C14H23N3O4Pureza:98%Forma y color:SolidPeso molecular:297.35LOE 908 hydrochloride
CAS:<p>Broad spectrum cation channel blocker</p>Fórmula:C41H49ClN2O9Pureza:98%Forma y color:SolidPeso molecular:749.29Piperidine-4-sulfonic acid
CAS:<p>Piperidine-4-sulfonic acid is a potent GABA agonist, demonstrating an IC50 value of 0.034 μM for the inhibition of H-GABA binding [1].</p>Fórmula:C5H11NO3SPureza:98%Forma y color:SolidPeso molecular:165.21NPEC-caged-(S)-AMPA
CAS:<p>AMPA receptor agonist</p>Fórmula:C16H17N3O8Pureza:98%Forma y color:SolidPeso molecular:379.32Sodium Channel inhibitor 4
CAS:<p>Sodium Channel Inhibitor 4 is a compound that functions as a sodium channel inhibitor [1].</p>Fórmula:C19H18ClN3O4S2Pureza:98%Forma y color:SolidPeso molecular:451.95ZM 260384
CAS:<p>ZM 260384 is a potassium channel opener.</p>Fórmula:C15H11F4N3O4Forma y color:SolidPeso molecular:373.26NCS-382 sodium
CAS:<p>NCS-382 (sodium) is a potent antagonist of the GABA receptor, exhibiting anti-sedative and anti-hypnotic properties, with applications in neurological disease</p>Fórmula:C13H13NaO3Pureza:98%Forma y color:SolidPeso molecular:240.23CGP 54626 hydrochloride
CAS:<p>CGP 54626 hydrochloride is a GABAB receptor antagonist.</p>Fórmula:C18H29Cl3NO3PPureza:98%Forma y color:SolidPeso molecular:444.76S-Pantoprazole sodium trihydrate
CAS:<p>S-Pantoprazole (sodium trihydrate), a variant of Pantoprazole, is pivotal in managing diseases associated with gastric acid secretion disorders, serving as a</p>Fórmula:C16H20F2N3NaO7SPureza:98%Forma y color:SolidPeso molecular:459.4TRPV2-selective blocker 1
CAS:<p>TRPV2-selective blocker 1 (compound IV2-1) is a selective inhibitor of the TRPV2 channel, exhibiting an IC50 value of 6.3 μM.</p>Fórmula:C15H18OS2Forma y color:SolidPeso molecular:278.43CP-409092
CAS:<p>CP-409092 is a partial GABAA receptor agonist. It has anti-anxiety activity.</p>Fórmula:C17H19N3O2Pureza:98%Forma y color:SolidPeso molecular:297.35Aneratrigine
CAS:<p>Aneratrigine is a blocker of the sodium channel protein type 9 subunit alpha, utilized in research on neuropathic pain diseases [1].</p>Fórmula:C19H20ClF2N5O2S2Pureza:98%Forma y color:SolidPeso molecular:487.97(R)-Elexacaftor
CAS:<p>(R)-Elexacaftor (compound 37) is the enantiomer of Elexacaftor (compound 1). (R)-Elexacaftor is a CFTR modulator with an EC50 of 0.29 μM for CFTR dF508.</p>Fórmula:C26H34F3N7O4SPureza:98.991%Forma y color:SolidPeso molecular:597.65SCS
CAS:<p>SCS is a GABAA receptor antagonist.</p>Fórmula:C14H12N2O3Pureza:99.73%Forma y color:SolidPeso molecular:256.26KVI-020
CAS:<p>KVI-020: oral Kv1.5 blocker (IC50: 480nM), hERG inhibitor (IC50: 15100nM), potent antiarrhythmic for AF studies.</p>Fórmula:C20H25N3O5SForma y color:SolidPeso molecular:419.49Chromanol 293B
CAS:<p>slow delayed rectifier K+ current (IKs) blocker</p>Fórmula:C15H20N2O4SPureza:98%Forma y color:SolidPeso molecular:324.4GDC-0310
CAS:<p>GDC-0310 is a selective, orally available Nav1.7 inhibitor with an IC50 of 0.6 nM for human Nav1.7, suitable for pain research.</p>Fórmula:C25H29Cl2FN2O4SPureza:99.877%Forma y color:SolidPeso molecular:543.48GNE-0723
CAS:<p>GNE-0723 is a selective positive allosteric modulator of the NMDA receptor, GluN2A.blood-brain barrier (BBB) and Dravet syndrome and Alzheimer's disease (AD).</p>Fórmula:C16H8ClF6N5OSPureza:97.29% - 99.91%Forma y color:SolidPeso molecular:467.78PF-4778574
CAS:<p>PF-4778574 is a positive AMPA receptor allosteric modulation (EC50: 45 to 919 nM in different cells).</p>Fórmula:C19H22N2O3S2Pureza:98%Forma y color:SolidPeso molecular:390.52Mioflazine
CAS:<p>Mioflazine suppresses nucleoside uptake. Mioflazine is an orally active nucleoside transport inhibitor. It has the potential for sleep disorders treatment.</p>Fórmula:C29H30Cl2F2N4O2Pureza:98%Forma y color:SolidPeso molecular:575.48DPO-1
CAS:<p>DPO-1 可以高效抑制电压门控钾离子通道Kv1.5，也可以阻断超快速延迟整流钾电流。它能够预防房性心律失常。</p>Fórmula:C22H29OPPureza:99.78%Forma y color:SolidPeso molecular:340.44CLP257
CAS:<p>CLP257 is a selective K+-Cl− cotransporter KCC2 activator (EC50: 616 nM) and it is inactive against NKCC1, GABAA receptors, KCC1, KCC3 or KCC4.</p>Fórmula:C14H14FN3O2SPureza:99.5%Forma y color:SolidPeso molecular:307.348-Pcpt-cGMP
CAS:<p>8-Pcpt-cGMP acts as an agonist for cyclic nucleotide-gated (CNG) channels with an EC50 of 0.5 μM and exhibits good membrane permeability. This compound is utilized in research to explore the role of CNG channels in visual and olfactory signal transduction.</p>Fórmula:C16H15ClN5O7PSForma y color:SolidPeso molecular:487.81BMS-199264 hydrochloride
CAS:<p>BMS-199264 hydrochloride is selective inhibitor of mitochondrial F1F0 ATP hydrolase,inhibit decline of ATP and myocardial necrosis during myocardial ischemia.</p>Fórmula:C26H32Cl2N4O4SPureza:99.86%Forma y color:SolidPeso molecular:567.53Co 102862
CAS:<p>Co 102862 is a voltage-gated sodium channel blocker. Co 102862 can be used for anticonvulsant studies.</p>Fórmula:C14H12FN3O2Pureza:99.82%Forma y color:SolidPeso molecular:273.26Mesendogen
CAS:<p>Mesendogen is an inhibitor of transient receptor potential cation channel, subfamily M, member 6 (TRPM6) and 7 (TRPM7) and acts by inhibiting TRPM6/TRPM7</p>Fórmula:C18H16ClF3N2OSPureza:99.66%Forma y color:SolidPeso molecular:400.85GSK3395879
CAS:<p>GSK3395879 is a selective and orally bioavailable antagonist of transient receptor potential vanilloid-4 (TRPV4) (IC50: 1 nM for hTRPV4).</p>Fórmula:C20H15F4N3O5SPureza:98%Forma y color:SolidPeso molecular:485.41BPO-27 racemate
CAS:<p>BPO-27 racemate (BPO-27 (racemate)) is an effective CFTR inhibitor with IC50 of 8 nM.</p>Fórmula:C26H18BrN3O6Pureza:97.67% - 98.86%Forma y color:SolidPeso molecular:548.34LG 83-6-05
CAS:<p>LG 83-6-05 is a novel kind of sodium channel blocking agent.</p>Fórmula:C21H30ClNO3SForma y color:SolidPeso molecular:411.99Sudoterb free base
CAS:<p>Sudoterb free base (Sudoterb) , also known as LL3858, is an anti-tubercular drug candidate.</p>Fórmula:C29H28F3N5OPureza:97.26% - 98.85%Forma y color:SolidPeso molecular:519.56URAT1 inhibitor 1
CAS:<p>URAT1 inhibitor 1 (1g) is an inhibitor of uric acid transporter 1 (URAT1) (IC50: 32 nM), has the potential to treat hyperuricemia associated with gout.</p>Fórmula:C19H15Br2N5O2S2Pureza:98%Forma y color:SolidPeso molecular:569.29Clobutinol hydrochloride
CAS:<p>Clobutinol hydrochloride, an antitussive agent, influences heart rate and blood pressure, and is utilized in cough-related research [1] [2] [3].</p>Fórmula:C14H23Cl2NOPureza:98%Forma y color:SolidPeso molecular:292.25Xeniafaraunol A
CAS:<p>Xeniafaraunol A (compound 31) is a potent inhibitor of the transient receptor potential melastatin 7 (TRPM7) channel [1].</p>Fórmula:C20H28O2Forma y color:SolidPeso molecular:300.44
