Transportador de membrana / canal de iones
Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.
Subcategorías de "Transportador de membrana / canal de iones"
- ABC(3 productos)
- ATPasa(98 productos)
- Receptor de adiponectina(5 productos)
- CFTR(66 productos)
- Receptor CGRP(53 productos)
- Canal de calcio(525 productos)
- Canal de cloruro(51 productos)
- Receptor GABA(355 productos)
- Transportador de monoamina(26 productos)
- Transportador de monocarboxilato(18 productos)
- NKCC(2 productos)
- NPC1L1(3 productos)
- Cotransportador de Na-K-Cl(9 productos)
- OAT(28 productos)
- OCT(7 productos)
- P-gp(52 productos)
- Canal de potasio(280 productos)
- Bomba de protones(40 productos)
- SGLT(31 productos)
- Canal de sodio(202 productos)
- Canal TRP / TRPV(94 productos)
Mostrar 13 subcategorías más
Se han encontrado 2430 productos de "Transportador de membrana / canal de iones"
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Apcin A HCL
CAS:<p>Apcin A HCL is an Apcin derivative. Apcin A HCL is an anaphase-promoting complex (APC) inhibitor. Apcin-A HCL interacts strongly with Cdc20, and inhibits the ubiquitination of Cdc20 substrates. Apcin-A HCL can be used to synthesize the PROTAC CP5V [1].</p>Fórmula:C10H15Cl4N5O2Pureza:99.30%Forma y color:SolidPeso molecular:379.07Indoxacarb
CAS:Indoxacarb is an Oxadiazine insecticide.Fórmula:C22H17ClF3N3O7Pureza:98%Forma y color:SolidPeso molecular:527.83Alfadolone acetate
CAS:Alfadolone acetate is a gamma-aminobutyric acid (GABA) receptor agonist.Fórmula:C23H34O5Forma y color:SolidPeso molecular:390.51Filapixant
CAS:Filapixant, a purinoreceptor antagonist. This compound serves as the active reference substance for Eliapixant.Fórmula:C24H26F3N5O3SForma y color:SolidPeso molecular:521.56Dexivacaine
CAS:Dexivacaine is an type of anesthetic.Fórmula:C15H22N2OForma y color:SolidPeso molecular:246.35(±)-Vasicine
CAS:<p>(±)-Vasicine, the racemate of Vasicine, is isolated from Peganum harmala seeds and exhibits anti-ulcer activity.</p>Fórmula:C11H12N2OPureza:98%Forma y color:SolidPeso molecular:188.23PF-06761281
CAS:PF-06761281 is a partially selective sodium-coupled citrate transporter protein (NaCT/SLC13A5) inhibitor, oral, reducing plasma glucose concentration.Fórmula:C13H17NO6Forma y color:SolidPeso molecular:283.28Verapamil EP Impurity C hydrochloride
CAS:<p>NSC-609249 hydrochloride, an impurity of Verapamil, is a calcium channel blocker with potent orally active properties. It also functions as a first-generation P-glycoprotein (P-gp) inhibitor.</p>Fórmula:C12H20ClNO2Forma y color:SolidPeso molecular:245.752-AEMP TFA
CAS:2-AEMP TFA is a potent and rapidly acting antagonist of GABA(A)-ρ1 receptors. 2-AEMP is an analog of GABA.Fórmula:C3H10NO3PPureza:98%Forma y color:SolidPeso molecular:139.0913-Methylglutaconic acid
CAS:<p>3-Methylglutaconic acid, a primary metabolite accumulating in 3-Methylglutaconic aciduria (MGTA), induces lipid and protein oxidation, while diminishing non-enzymatic antioxidant defenses in cerebral cortex supernatants, thereby promoting oxidative stress in the cerebral cortex. This compound is utilized in research concerning brain damage diseases [1].</p>Fórmula:C6H8O4Pureza:98%Forma y color:SolidPeso molecular:144.13Zastaprazan
CAS:<p>Zastaprazan (JP-1366, compound 6) is a potassium-competitive acid blocker and proton pump inhibitor that suppresses gastric acid secretion, indicated for GERD.</p>Fórmula:C22H26N4OPureza:99.97%Forma y color:SolidPeso molecular:362.48GNE-9278
CAS:<p>GNE-9278 is a highly selective NMDAR orthosteric modulator that targets the GluN1 transmembrane structural domain (TMD), enhancing peak current and agonist affinity in activated NMDAR.</p>Fórmula:C21H27N5O3SForma y color:SolidPeso molecular:429.54Vonoprazan fumarate
CAS:<p>Vonoprazan fumarate (TAK-438) is a novel P-CAB (potassium-competitive acid blocker) that reversibly inhibits H+/K+, ATPase.</p>Fórmula:C17H16FN3O2S·C4H4O4Pureza:99.16% - 99.98%Forma y color:SolidPeso molecular:461.46Fostedil
CAS:Fostedil enhances heart function, maintains blood flow during partial/total coronary occlusions, and lowers aortic pressure.Fórmula:C18H20NO3PSPureza:98%Forma y color:SolidPeso molecular:361.4Motugivatrep
CAS:<p>Motugivatrep is a potent and selective TRPV1 antagonist that can be used to study TRPV1-related respiratory diseases.</p>Fórmula:C22H20F3NO3Pureza:99.22%Forma y color:SolidPeso molecular:403.39CMPDA
CAS:CMPDA is a positive allosteric modulator of AMPA receptors [EC50s: 45.4 nM/63.4 nM for GluA2i/GluA2o receptor].Fórmula:C16H28N2O4S2Pureza:98%Forma y color:SolidPeso molecular:376.53Phenamil methanesulfonate
CAS:TRPP3 channel inhibitorFórmula:C13H16ClN7O4SPureza:98%Forma y color:SolidPeso molecular:401.83Pipequaline
CAS:Pipequaline (PK-8165) is an anticonflict & anticonvulsant quinoline derivative. It is an anxiolytic drug that was never marketed. It possesses a novel chemical structure that is not closely related to other drugs of this type. The drug has a similar pharmacological profile to the benzodiazepine family of drugs, but with mainly anxiolytic properties and very little sedative, amnestic or anticonvulsant effects, and so is classified as a nonbenzodiazepine anxiolytic.Fórmula:C22H24N2Pureza:98%Forma y color:SolidPeso molecular:316.44Ref: TM-T4655
Producto descatalogadoT16A(inh)-C01
CAS:<p>T16A(inh)-C01 is the Ca(2+)-activated Cl(-) Channel, Ano1 class C inhibitor.</p>Fórmula:C18H16O5Pureza:98%Forma y color:SolidPeso molecular:312.32CGP 44532
CAS:CGP 44532 a GABAB receptor agonist.Fórmula:C4H12NO3PPureza:98%Forma y color:SolidPeso molecular:153.12Gacyclidine
CAS:Gacyclidine (OTO311), an NMDA receptor blocker, treats tinnitus and injuries in the brain and spinal cord.Fórmula:C16H25NSPureza:99.85% - 99.92%Forma y color:SolidPeso molecular:263.44Tifenazoxide
CAS:Tifenazoxide is an effective and SUR1/Kir6.2 selective KATP channels opener. Tifenazoxide has an anti-diabetic effect, can inhibit glucose-stimulated insulin release in vitro and in vivo.Fórmula:C9H10ClN3O2S2Pureza:98%Forma y color:SolidPeso molecular:291.78Pazinaclone
CAS:<p>Pazinaclone is a non-benzodiazepine (GABAA) partial agonist with sedative and anxiolytic activity.</p>Fórmula:C25H23ClN4O4Pureza:97.79% - 99.07%Forma y color:SolidPeso molecular:478.93Belfosdil
CAS:Belfosdil is a blocker of antihypertensive calcium channel.Fórmula:C27H50O7P2Pureza:98%Forma y color:SolidPeso molecular:548.63LFS-1107
CAS:<p>LFS-1107, a reversible CRM1 inhibitor (Kd: 12.5 pM), selectively targets and eliminates ENKTL cells, offering potential for cancer research applications [1].</p>Fórmula:C12H11N5OS2Pureza:98%Forma y color:SolidPeso molecular:305.38Bumetanide sodium
CAS:Bumetanide sodium, a potent diuretic, blocks NKCC1 (IC50: 0.68 μM) and NKCC2 (IC50: 4.0 μM).Fórmula:C17H19N2NaO5SForma y color:SolidPeso molecular:386.4CGP 56999A
CAS:CGP 56999A is a GABA(B) receptor antagonist; it boosts BDNF and reduces dopamine loss in rat striatum.Fórmula:C19H30NO5PPureza:98%Forma y color:SolidPeso molecular:383.42Xilmenolone
CAS:<p>Xilmenolone acts as a positive allosteric modulator of the GABA_A receptor [1].</p>Fórmula:C26H37N3O2Pureza:98%Forma y color:SolidPeso molecular:423.59Ref: TM-T78670
Producto descatalogadoHMR 1556
CAS:HMR 1556 is a chromanol derivative and is an IKs blocker (IC50s of 10.5 nM and 34 nM in canine and guinea pig left ventricular myocytes, respectively).Fórmula:C17H24F3NO5SForma y color:SolidPeso molecular:411.44VMAT2-IN-2 tosylate
CAS:<p>VMAT2-IN-2 tosylate is a potent inhibitor of VMAT2 and is applicable in the research of tardive dyskinesia [1].</p>Fórmula:C27H36F3NO6SPureza:98%Forma y color:SolidPeso molecular:559.64Ref: TM-T79061
Producto descatalogado
