Transportador de membrana / canal de iones
Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.
Subcategorías de "Transportador de membrana / canal de iones"
- ABC(3 productos)
- ATPasa(98 productos)
- Receptor de adiponectina(5 productos)
- CFTR(66 productos)
- Receptor CGRP(53 productos)
- Canal de calcio(525 productos)
- Canal de cloruro(51 productos)
- Receptor GABA(355 productos)
- Transportador de monoamina(26 productos)
- Transportador de monocarboxilato(18 productos)
- NKCC(2 productos)
- NPC1L1(3 productos)
- Cotransportador de Na-K-Cl(9 productos)
- OAT(28 productos)
- OCT(7 productos)
- P-gp(52 productos)
- Canal de potasio(280 productos)
- Bomba de protones(40 productos)
- SGLT(31 productos)
- Canal de sodio(202 productos)
- Canal TRP / TRPV(94 productos)
Mostrar 13 subcategorías más
Se han encontrado 2430 productos de "Transportador de membrana / canal de iones"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
D-AP4
CAS:broad spectrum excitatory amino acid receptor antagonistFórmula:C4H10NO5PPureza:98%Forma y color:White PowderPeso molecular:183.1GSK-5503A
CAS:GSK-5503A is a novel channel blocker of CRAC.Fórmula:C23H17F2N3O2Pureza:98%Forma y color:SolidPeso molecular:405.4UT-B-IN-1
CAS:<p>UT-B-IN-1: reversible UT-B inhibitor, IC50: 10 nM (human), 25 nM (mouse), low toxicity, diuretic research tool.</p>Fórmula:C20H17N5O2S3Forma y color:SolidPeso molecular:455.58Quinine hemisulfate
CAS:Quinidine: antiarrhythmic, orally active, inhibits cytochrome P450db, blocks K+ channels (IC50: 19.9μM), may aid in malaria research.Fórmula:C40H50N4O8SPureza:98%Forma y color:SolidPeso molecular:746.92(RS)-CPP
CAS:(RS)-CPP is a NMDA antagonist.Fórmula:C8H17N2O5PPureza:98%Forma y color:SolidPeso molecular:252.2PF-05214030
CAS:PF-05214030 is a novel potent TRPV4 antagonist (hTRPV4 IC50 4nM; rTRPV4 IC50 27nM).Fórmula:C17H13Cl2FN2O4SForma y color:SolidPeso molecular:431.27FG8119
CAS:FG8119 is a novel benzodiazepine agonist with potential anticonvulsant and antiepileptic activity for the study of neurological disorders.Fórmula:C17H15N5O2Pureza:>99.99%Forma y color:SolidPeso molecular:321.33GABAA receptor agent 6
CAS:GABAA receptor agent 6 (compound 2027) is a potent γ-GABAAR antagonist with low cellular membrane permeability (Ki = 0.56 μM) [1].Fórmula:C18H25N3O2Forma y color:SolidPeso molecular:315.41GSK-5498A
CAS:GSK-5498A: Selective CARC blocker, inhibits release of mediators from mast cells and cytokines from T-cells (IC50, 1 μM).Fórmula:C18H11F6N3OForma y color:SolidPeso molecular:399.29TB 21007
CAS:GABAA receptor inverse agonistFórmula:C15H17NO2S3Pureza:98%Forma y color:SolidPeso molecular:339.5D-3263
CAS:D-3263 is an agonist of transient receptor potential melatonin member 8 (TRPM8) with potential antitumor activity.Fórmula:C21H31N3O3Pureza:98%Forma y color:SolidPeso molecular:373.49Gea 857
CAS:<p>Gea 857 is a potassium conductance putative blocker.</p>Fórmula:C15H22ClNO2Pureza:98%Forma y color:SolidPeso molecular:283.79N20C hydrochloride
CAS:<p>N20C hydrochloride (2-((3,3-diphenylpropyl)amino)acetamide hydrochloride) is a non-competitive NMDA receptor open-channel blocker.</p>Fórmula:C17H21ClN2OPureza:99.9%Forma y color:SolidPeso molecular:304.81PNU 37883 hydrochloride
CAS:Kir6 (KATP) channel antagonistFórmula:C21H36ClN3OPureza:98%Forma y color:SolidPeso molecular:381.98TRPC5-IN-1
CAS:TRPC5-IN-1 is a TRPC5 inhibitor active in various animal models of chronic kidney disease.Fórmula:C20H16N4OForma y color:SolidPeso molecular:328.374-(Phenyldiazenyl)benzoic acid
CAS:<p>4-(Phenyldiazenyl)benzoic acid is a photosensitive and photoswitchable TRPA1 agonist that can be used as pharmacological tool to study pain signaling.</p>Fórmula:C13H10N2O2Forma y color:SolidPeso molecular:226.23MPO-IN-5
CAS:<p>MPO-IN-5: strong, irreversible MPO blocker; IC50s: 0.22 μM for peroxidation, 2.8 μM for hERG.</p>Fórmula:C24H24N6O2Forma y color:SolidPeso molecular:428.49KC 12291 hydrochloride
CAS:voltage-gated sodium channel blockerFórmula:C22H28ClN3O3SPureza:98%Forma y color:SolidPeso molecular:449.99NMDA receptor potentiator-1
CAS:Compound 1368 is a selective NMDA receptor enhancer; IC50s: 4 μM for NR2C, 5 μM for NR2D.Fórmula:C26H26ClNO5Forma y color:SolidPeso molecular:467.94(RS)-3,4-DCPG
CAS:antagonist of AMPA receptors and agonist of mGluR8Fórmula:C10H9NO6Pureza:98%Forma y color:SolidPeso molecular:239.18SOCE inhibitor 1
CAS:SOCE inhibitor 1 is a inhibitor of store-operated calcium entry (SOCE)(IC50 of 4.4 μM).Fórmula:C25H22F3N5O4Pureza:98%Forma y color:SolidPeso molecular:513.47ZAPA sulfate
CAS:GABAA receptors agonistFórmula:C4H8N2O6S2Pureza:98%Forma y color:SolidPeso molecular:244.25NMDA receptor modulator 5
CAS:NMDA receptor modulator 5 (Compound 195), a potent NMDA receptor modulator, exhibits potential for neurological disorder research [1].Fórmula:C14H11F3N2O3SForma y color:SolidPeso molecular:344.31Glisoxepide
CAS:Glisoxepide: sulphonamide, oral K(ATP) blocker, antihyperglycemic, affects heart.Fórmula:C20H27N5O5SPureza:98%Forma y color:SolidPeso molecular:449.52JNJ-55511118
CAS:<p>JNJ-55511118 is a TARP γ8 allosteric modulator with anticonvulsant activity, which can be used in research on chronic operant alcohol self-administration.</p>Fórmula:C14H8ClF3N2O2Forma y color:SolidPeso molecular:328.67S3337
CAS:<p>S3337 is an inhibitor of H+, K+-ATPase</p>Fórmula:C18H21N3O3SPureza:98%Forma y color:SolidPeso molecular:359.44(2R,3S)-Chlorpheg
CAS:(2R,3S)-Chlorpheg is a NMDA receptor antagonist.Fórmula:C11H12ClNO4Pureza:98%Forma y color:SolidPeso molecular:257.67PF-0713
CAS:PF 0713, a GABAA receptor agonist, is used as an intravenous sedative-hypnotic for general anaesthesia, ICU sedation, procedural sedation, chemotherapy.Fórmula:C14H22OPureza:98%Forma y color:SolidPeso molecular:206.32Lidoflazine
CAS:Lidoflazine: antianginal, blocks HERG K+ & Ca channels, risks QT prolongation & arrhythmia.Fórmula:C30H35F2N3OPureza:98%Forma y color:SolidPeso molecular:491.62NMDA receptor modulator 3
CAS:NMDA receptor modulator 3 (Compound 99) is a potent modulator of NMDA receptor that can be used in the research of neurological disorder [1].Fórmula:C12H9F3N2O2SForma y color:SolidPeso molecular:302.27Corrector C4
CAS:Corrector C4, a corrector commonly used to study cystic fibrosis mutants, works by alleviating the interaction between CFTR transmembrane domain mutants andFórmula:C21H17ClN4O2S2Pureza:98.36%Forma y color:SolidPeso molecular:456.97CAY10719
CAS:CAY10719 selectively inhibits ABCG2 (IC50 = 0.23 μM), reverses SN 38 resistance, and inhibits ATPase, with low ABCG1 activity.Fórmula:C25H20Cl2N2O2Forma y color:SolidPeso molecular:451.34TG41
CAS:TG41 is a GABAA receptors positive modulator.Fórmula:C18H13BrCl2N2O2Pureza:98%Forma y color:SolidPeso molecular:440.12MK-7145
CAS:MK-7145 is an inhibitor of ROMK(IC50 of 0.045 μM).Fórmula:C26H30N2O6Pureza:98%Forma y color:SolidPeso molecular:466.53RN-9893 (hydrochloride)
CAS:<p>RN-9893 is a TRPV4 antagonist with human/rat IC50s of 0.42/0.66 μM; selective over TRPV1, TRPV3, TRPM8. Reduces rat TRPV4 activity (IC50: 0.57-2.1 μM).</p>Fórmula:C21H24ClF3N4O5SForma y color:SolidPeso molecular:536.95(S)-Lercanidipine hydrochloride
CAS:<p>(S)-Lercanidipine hydrochloride is the S-enantiomer of Lercanidipine hydrochloride. (S)-lercanidipine hydrochloride is a potent blocker of calcium channel.</p>Fórmula:C36H42ClN3O6Pureza:98%Forma y color:SolidPeso molecular:648.19Kadethrin
CAS:Kadethrin is a synthetic pyrethroid. It was used as a pesticide.Fórmula:C23H24O4SPureza:98%Forma y color:Yellow-Brown Viscous Oil SolidPeso molecular:396.5HZ166
CAS:HZ-166 is a positive GABAA receptor modulator and a GABAA receptor subtype-selective benzodiazepine site ligand.Fórmula:C21H16N4O2Pureza:98%Forma y color:SolidPeso molecular:356.38NCS-382
CAS:γ-Hydroxybutyric acid antagonistFórmula:C13H14O3Pureza:98%Forma y color:SolidPeso molecular:218.25L-trans-2,4-PDC
CAS:L-trans-2,4-PDC is an EAAT1-4 inhibitor/non-transportable EAAT5 inhibitor.Fórmula:C6H9NO4Pureza:98%Forma y color:SolidPeso molecular:159.14Anipamil
CAS:Anipamil is a long-acting blocker of calcium channel,and for the treatment of cardiovascular disease.Fórmula:C34H52N2O2Pureza:98%Forma y color:SolidPeso molecular:520.79SL-651498
CAS:SL-651498, a GABAA receptor agonist, is used potentially for the treatment of anxiety.Fórmula:C23H20FN3O2Pureza:98%Forma y color:SolidPeso molecular:389.42Norbormide
CAS:Norbormide is a toxic compound used as a rodenticide. It has several mechanisms of action, acting as a vasoconstrictor and calcium channel blocker.Fórmula:C33H25N3O3Pureza:98%Forma y color:Crystals From Methylene Chloride + Ether Norbormide Is A Colorless To Off-White Crystalline Powder Used As A Selective Rat Poison (Epa 1998)Peso molecular:511.57Neramexane Mesylate
CAS:<p>Neramexane: NMDA & nicotinic receptor blocker with neuroprotective, antidepressant, and cognitive-enhancing effects.</p>Fórmula:C12H27NO3SPureza:98%Forma y color:SolidPeso molecular:265.41Dofequidar
CAS:<p>Dofequidar (MS-209 free base) is a quinoline derivative that inhibits the efflux of chemotherapeutic agents.</p>Fórmula:C30H31N3O3Pureza:98%Forma y color:SolidPeso molecular:481.59MRS4719
CAS:<p>MRS4719: potent P2X4 antagonist, IC50 0.503 μM. Reduces infarct, brain atrophy, Ca2+ influx. Used in ischemic stroke research.</p>Fórmula:C26H13N5O3S·C6H15NForma y color:SolidPeso molecular:504.6Clathrodin
CAS:Clathrodin is a voltage-gated sodium (NaV) channels modulator.Fórmula:C11H13N5OForma y color:SolidPeso molecular:231.25GABAA receptor agent 4
CAS:<p>Compound 1e is a potent γ-GABAAR antagonist with a Ki of 0.18 µM, offering immunomodulatory effects on T cell proliferation.</p>Fórmula:C17H24N2OForma y color:SolidPeso molecular:272.39UBP 302
CAS:<p>UBP 302 is a selective GLUK5 kainate receptor antagonist with Kd 402 nM; low GluK2 affinity.</p>Fórmula:C15H15N3O6Pureza:98%Forma y color:SolidPeso molecular:333.3
