Transportador de membrana / canal de iones
Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.
Subcategorías de "Transportador de membrana / canal de iones"
- ABC(3 productos)
- ATPasa(97 productos)
- Receptor de adiponectina(5 productos)
- CFTR(64 productos)
- Receptor CGRP(53 productos)
- Canal de calcio(520 productos)
- Canal de cloruro(51 productos)
- Receptor GABA(351 productos)
- Transportador de monoamina(26 productos)
- Transportador de monocarboxilato(18 productos)
- NKCC(2 productos)
- NPC1L1(3 productos)
- Cotransportador de Na-K-Cl(9 productos)
- OAT(28 productos)
- OCT(7 productos)
- P-gp(53 productos)
- Canal de potasio(280 productos)
- Bomba de protones(40 productos)
- SGLT(31 productos)
- Canal de sodio(203 productos)
- Canal TRP / TRPV(94 productos)
Mostrar 13 subcategorías más
Se han encontrado 2402 productos de "Transportador de membrana / canal de iones"
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Alilusem
CAS:Alilusem is a new diuretic that is beneficial to the clinical treatment of hypertension.Fórmula:C17H15ClKN2O5SForma y color:SolidPeso molecular:433.92TRPV antagonist 1
CAS:TRPV antagonist 1 is an antagonist of transient receptor potential vanilloid (TRPV; IC50 < 250 nM).Fórmula:C26H21F3N2O4SPureza:98%Forma y color:SolidPeso molecular:514.52URAT1 inhibitor 4
CAS:<p>URAT1 inhibitor 4 is a potent, orally active Lesinurad derivative with a 7.56 μM IC50, showing greater in vivo efficacy.</p>Fórmula:C27H20BrN3O4S3Forma y color:SolidPeso molecular:626.56UK-52831
CAS:UK-52831, a calcium channel antagonist, is used potentially for the treatment of hypertension and myocardia ischemia.Fórmula:C22H26Cl2N6O5Pureza:98%Forma y color:SolidPeso molecular:525.39DS2
CAS:Positive allosteric modulator of δ-subunit containing GABAA receptorsFórmula:C18H12ClN3OSPureza:98%Forma y color:SolidPeso molecular:353.83ATPA
CAS:<p>ATPA activates GluR5 glutamate receptors; EC50s range 0.66-32 μM across GluR5 variants.</p>Fórmula:C10H16N2O4Pureza:98%Forma y color:SolidPeso molecular:228.24Ro 19-4603
CAS:Benzodiazepine inverse agonistFórmula:C15H17N3O3SPureza:98%Forma y color:SolidPeso molecular:319.38CGS8216
CAS:<p>CGS8216 shows analgesic activity at high doses, has anxiolytic activity, and can be used to study immune system disorders.</p>Fórmula:C16H11N3OPureza:98.53%Forma y color:SolidPeso molecular:261.28LY382884
CAS:<p>LY382884 is a selective and potent GluR5 kainate receptor antagonist with anxiolytic activity.LY382884 blocks blockade of mossy fibre LTP induction.</p>Fórmula:C18H23NO4Pureza:98.32% - 98.71%Forma y color:SolidPeso molecular:317.38Remacemide hydrochloride
CAS:Remacemide hydrochloride is a NMDA receptor antagonist.Fórmula:C17H21ClN2OPureza:98%Forma y color:SolidPeso molecular:304.81NS 3763
CAS:NS 3763 is a kainate receptor antagonist.Fórmula:C22H16N2O6Pureza:98%Forma y color:SolidPeso molecular:404.37Traxoprodil Mesylate
CAS:Traxoprodil Mesylate is a potent noncompetitive N-methyl-D-aspartate (NMDA) receptors antagonist and has selective for the NR2B subunit.Fórmula:C21H29NO6SPureza:98%Forma y color:SolidPeso molecular:423.525,7-Dichlorokynurenic acid sodium salt
CAS:5,7-Dichlorokynurenic acid sodium salt is a NMDA receptor antagonist.Fórmula:C10H5Cl2NNaO3Pureza:98%Forma y color:SolidPeso molecular:281.05F15845
CAS:<p>F 15845: potent sodium current blocker, anti-ischemic, offers short/long-term post-infarction cardioprotection.</p>Fórmula:C20H25NO2S2Forma y color:SolidPeso molecular:375.55TRPC6-IN-1
CAS:TRPC6-IN-1 is an inhibitor of the Transient Receptor Potential Canonical 6 Channel (TRPC6) (EC50: 4.66 μM).Fórmula:C21H23FN4O3Pureza:98%Forma y color:SolidPeso molecular:398.43GV-196771A
CAS:<p>GV-196771A A novel NMDA receptor glycine site antagonist with potent antinociceptive activity.</p>Fórmula:C20H13Cl2N2NaO3Pureza:96.43%Forma y color:SolidPeso molecular:423.23AMG-628
CAS:AMG-628 inhibits RAF kinase, halts growth, and triggers apoptosis in B-RAFV600E mutant colon/melanoma cells.Fórmula:C25H25FN6O2SForma y color:SolidPeso molecular:492.57Ethacrynate Sodium
CAS:Ethacrynate Sodium, a sodium salt, blocks chloride, potassium, and sodium transport mainly in Henle's loop.Fórmula:C13H12Cl2NaO4Pureza:98%Forma y color:SolidPeso molecular:326.12Y-26763
CAS:Y-26763 is a K+ channel opener and active metabolite of Y-27152. This is an ATP-sensitive K+ (KATP) channel activator.Fórmula:C14H16N2O4Pureza:98%Forma y color:SolidPeso molecular:276.29FCPT
CAS:FCPT is an ATP competitive kinesin-5 inhibitor.Fórmula:C17H13FN2SPureza:98%Forma y color:SolidPeso molecular:296.36BHF-177
CAS:<p>BHF-177 is a positive allosteric modulator of the GABAB receptor. BHF-177 reduces self-administration of nicotine in animal studies.</p>Fórmula:C19H20F3N3Forma y color:SolidPeso molecular:347.38SKF 97541
CAS:<p>GABAB agonist</p>Fórmula:C4H12NO2PPureza:98%Forma y color:SolidPeso molecular:137.12Galicaftor
CAS:<p>ABBV-2222 is a CFTR corrector which is studied for the treatment of cystic fibrosis (CF).</p>Fórmula:C28H21F4NO7Pureza:98%Forma y color:SolidPeso molecular:559.46UBP-282
CAS:AMPA and kainate receptor antagonistFórmula:C15H15N3O6Pureza:98%Forma y color:SolidPeso molecular:333.3Norverapamil
CAS:Norverapamil is a blocker of L-type calcium channel and an inhibitor of P-glycoprotein (P-gp) function .Fórmula:C26H36N2O4Pureza:98%Forma y color:SolidPeso molecular:440.58JNJ-39729209
CAS:<p>JNJ-39729209 is a TRPV1 antagonist.</p>Fórmula:C19H11Cl2F3N4SForma y color:SolidPeso molecular:455.28Zonampanel
CAS:<p>Zonampanel is a selective glutamate receptor subtype, α-amino-3-hydroxy-5-methylisoxazole-4-propionic acid receptor antagonist.</p>Fórmula:C13H9N5O6Pureza:98%Forma y color:SolidPeso molecular:331.24mGAT3/4-IN-1
CAS:<p>mGAT3/4-IN-1 inhibits mGAT3/4 with pIC50: 5.31/5.24, reduces neuropathic pain in diabetic mice.</p>Fórmula:C26H31ClN2O2S2Forma y color:SolidPeso molecular:503.1217-PA
CAS:17-PA is a GABAA receptor antagonist.Fórmula:C25H34OPureza:98%Forma y color:SolidPeso molecular:350.54MK-0343
CAS:MK0343 is an orally bioavailable GABAA receptor subtype-selective partial agonist and is a non-sedating anxiolytic.Fórmula:C19H17F2N7OPureza:98%Forma y color:SolidPeso molecular:397.38Sematilide
CAS:Sematilide is a blocker of selective IKr channel.Fórmula:C14H23N3O3SPureza:98%Forma y color:SolidPeso molecular:313.42Posenacaftor
CAS:<p>Posenacaftor (PTI-801) regulates CFTR protein for cystic fibrosis research.</p>Fórmula:C27H27NO5Forma y color:SolidPeso molecular:445.51Cavα2δ1&NET-IN-1
CAS:<p>Cavα2δ1&NET-IN-1 .</p>Fórmula:C23H26N4O2SForma y color:SolidPeso molecular:422.54CGS 20625
CAS:partial agonist for the benzodiazepine binding site of the GABAA receptorFórmula:C18H19N3O2Pureza:99.61%Forma y color:SolidPeso molecular:309.36CXL-1020
CAS:CXL-1020, a HNO prodrug, enhances heart muscle function & relaxation, aiding in heart failure research.Fórmula:C7H9NO5S2Forma y color:SolidPeso molecular:251.282-Hydroxysaclofen
CAS:2-Hydroxysaclofen is a GABAB receptor antagonist.Fórmula:C9H12ClNO4SPureza:98%Forma y color:White SolidPeso molecular:265.71AMG9090
CAS:<p>AMG9090 is a transient receptor potential ankyrin 1 (TRPA1) antagonist.</p>Fórmula:C15H11Cl4NOSPureza:98%Forma y color:SolidPeso molecular:395.13CGP 7930
CAS:Positive allosteric modulator of GABAB receptorsFórmula:C19H32O2Pureza:98%Forma y color:SolidPeso molecular:292.46Perzinfotel
CAS:<p>Perzinfotel, a neuroprotective NMDA antagonist with high affinity (IC50=30 nM), is selective and competitive.</p>Fórmula:C9H13N2O5PForma y color:SolidPeso molecular:260.18Ro15-4513
CAS:Ro15-4513 is imidazobenzodiazepinone derivative and is a partial inverse agonist of benzodiazepine receptors. Ro15-4513 is an effective ethanol antagonist.Fórmula:C15H14N6O3Pureza:98%Forma y color:SolidPeso molecular:326.31Alaproclate, (S)-
CAS:Alaproclate, (S)- is a selective inhibitor of serotonin reuptake.Fórmula:C13H18ClNO2Pureza:98%Forma y color:SolidPeso molecular:255.74S-8921
CAS:S-8921 is an inhibitor of ileal Na+/bile acid cotransporter.Fórmula:C30H36O9Pureza:98%Forma y color:SolidPeso molecular:540.65'-Iodoresiniferatoxin
CAS:TRPV1 (VR1) receptor antagonistFórmula:C37H39IO9Pureza:98%Forma y color:SolidPeso molecular:754.6TPA-023B
CAS:TPA-023B: oral GABAA α2/α3 agonist (Kis: 0.73/2 nM), α1 antagonist (Ki: 1.8 nM), non-sedating anxiolytic.Fórmula:C21H15F2N5OPureza:98%Forma y color:SolidPeso molecular:391.37P-gp inhibitor 5
CAS:<p>P-gp inhibitor 5 strongly blocks P-glycoprotein, enhances drug sensitivity, and reverses cancer cell drug resistance.</p>Fórmula:C28H20ClNO5SForma y color:SolidPeso molecular:517.98U-101017
CAS:<p>U-101017 is a partial benzodiazepine receptor and GABAA receptor agonist.</p>Fórmula:C23H27ClN4O3Pureza:98%Forma y color:SolidPeso molecular:442.94Posenacaftor sodium
CAS:Posenacaftor (PTI-801) sodium, a CFTR modulator for CF research, corrects CFTR protein folding and trafficking.Fórmula:C27H27NNaO5Forma y color:SolidPeso molecular:468.505Org 20599
CAS:<p>GABAA receptor agonist</p>Fórmula:C25H40ClNO3Pureza:98%Forma y color:SolidPeso molecular:438.04NC 1100
CAS:NC 1100 is a calcium channel antagonist.Fórmula:C27H34Cl2N2O3Pureza:98%Forma y color:SolidPeso molecular:505.48CNS-5161
CAS:CNS-5161 is an NMDA antagonist.Fórmula:C16H18ClN3S2Pureza:98%Forma y color:SolidPeso molecular:351.92
