Transportador de membrana / canal de iones
Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.
Subcategorías de "Transportador de membrana / canal de iones"
- ABC(3 productos)
- ATPasa(93 productos)
- Receptor de adiponectina(5 productos)
- CFTR(64 productos)
- Receptor CGRP(52 productos)
- Canal de calcio(496 productos)
- Canal de cloruro(49 productos)
- Receptor GABA(337 productos)
- Transportador de monoamina(23 productos)
- Transportador de monocarboxilato(17 productos)
- NKCC(2 productos)
- NPC1L1(3 productos)
- Cotransportador de Na-K-Cl(8 productos)
- OAT(27 productos)
- OCT(7 productos)
- P-gp(53 productos)
- Canal de potasio(277 productos)
- Bomba de protones(39 productos)
- SGLT(30 productos)
- Canal de sodio(202 productos)
- Canal TRP / TRPV(93 productos)
Mostrar 13 subcategorías más
Se han encontrado 2293 productos de "Transportador de membrana / canal de iones"
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PF-06649298
CAS:<p>PF-06649298 inhibits NaCT, blocking citrate transport in hepatocytes, IC50: 16.2 μM, affects glucose and lipid metabolism.</p>Fórmula:C16H22O5Forma y color:SolidPeso molecular:294.34P2X3 antagonist 36
CAS:<p>P2X3 antagonist 36 is a P2X3 antagonist.</p>Fórmula:C20H18ClF3N6O3Forma y color:SolidPeso molecular:482.84UBP618
CAS:<p>UBP618 is a GluN1/GluN2 receptors pan-inhibitor.</p>Fórmula:C17H11BrO3Pureza:98%Forma y color:SolidPeso molecular:343.17LY 233053
CAS:<p>LY 233053 is a Competitive NMDA receptor antagonist.</p>Fórmula:C8H13N5O2Pureza:98%Forma y color:SolidPeso molecular:211.22GS-462808
CAS:<p>GS-462808: Cardiac Nav1.5 inhibitor, less brain penetration/activity.</p>Fórmula:C17H12F3N5O3Forma y color:SolidPeso molecular:391.3Pipazethate
CAS:<p>Pipipyrazine is a nonnarcotic oral cough suppressant, cough suppressant.</p>Fórmula:C21H25N3O3SForma y color:SolidPeso molecular:399.51Cavα2δ1&NET-IN-2
CAS:<p>Cavα2δ1&NET-IN-2 .</p>Fórmula:C22H26N6O2SForma y color:SolidPeso molecular:438.55Bliretrigine
CAS:<p>Bliretrigine, a sodium channel blocker, effectively relieves pain [1] [2] [3].</p>Fórmula:C20H24N4O2Forma y color:SolidPeso molecular:352.43AJG-049 HCl
CAS:<p>AJG-049 HCl is a calcium channel antagonist that inhibits L-type Ca2+ channels via diltiazem-binding site(s).</p>Fórmula:C27H31ClN2O2Forma y color:SolidPeso molecular:451.01NNC052090
CAS:<p>NNC052090 inhibits GABA uptake, favoring hBGT-1 (Ki=1.4μM), affects α1/D2 receptors (IC50=266/1632nM).</p>Fórmula:C27H30N2O2Forma y color:SolidPeso molecular:414.54A 784168
CAS:<p>A-784168: potent, oral TRPV1 inhibitor with good CNS penetration.</p>Fórmula:C19H15F6N3O3SForma y color:SolidPeso molecular:479.4Arachidonyl serotonin
CAS:<p>Dual FAAH inhibitor/TRPV1 antagonist</p>Fórmula:C30H42N2O2Pureza:98%Forma y color:SolidPeso molecular:462.67P-CAB agent 1
CAS:<p>Compound B19, a P-CAB, inhibits H+/K+-ATPase with IC50 of 60.50 nM, useful in ARD research.</p>Fórmula:C26H23FN4OForma y color:SolidPeso molecular:426.49UR-MB108
CAS:<p>UR-MB108 is a potent and selective inhibitor of ABCG2 (BCRP), displaying an IC50 value of 79 nM, and exhibits stability in blood plasma.</p>Fórmula:C40H38N6O4Forma y color:SolidPeso molecular:666.77Cariporide Mesylate
CAS:<p>Cariporide Mesylate is a selective inhibitor of the Na+/H+ exchanger isoform 1.</p>Fórmula:C13H21N3O6S2Forma y color:SolidPeso molecular:379.45U89232
CAS:<p>U-89232 is an opener of the cardioselective KATP channel.</p>Fórmula:C19H25N5O2Pureza:98%Forma y color:SolidPeso molecular:355.43TC-P 262
CAS:<p>P2X3 and P2X2/3 receptor antagonist</p>Fórmula:C14H18N4OPureza:98%Forma y color:SolidPeso molecular:258.32Azimilide
CAS:<p>class III anti-arrhythmic drug</p>Fórmula:C23H28ClN5O3Pureza:98%Forma y color:SolidPeso molecular:457.95DDO-02001
CAS:<p>DDO-02001 can be used in anti-arrhythmia research. DDO-02001 is a moderately potent inhibitor of Kv1.5 potassium channel with an IC50 value of 17.7 μM [1].</p>Fórmula:C20H24N2O2Forma y color:SolidPeso molecular:324.42ASIC-IN-1
CAS:<p>ASIC-IN-1 is a potent inhibitor of acid-sensing ion channels, demonstrating an IC 50 value of less than 10 μM.</p>Fórmula:C23H25N3O2Forma y color:SolidPeso molecular:375.46Becampanel
CAS:<p>Becampanel (AMP397) is the first competitive AMPA antagonist. Becampanel (AMP397) also is an antiepileptic agent.</p>Fórmula:C10H11N4O7PPureza:98%Forma y color:SolidPeso molecular:330.19MRK-623
CAS:<p>MRK-623 (14k) is an oral GABA A agonist with high affinity for α1/α2/α3/α5 subunits and anxiolytic properties.</p>Fórmula:C20H17FN4OForma y color:SolidPeso molecular:348.37CAY10608
CAS:<p>CAY10608 selectively blocks NR2B NMDA receptors (IC50 = 50 nM), is neuroprotective, and reduces brain infarct size in ischemia.</p>Fórmula:C18H22Cl2N2O4SForma y color:SolidPeso molecular:433.356'-Iodoresiniferatoxin
CAS:<p>TRPV1 (VR1) vanilloid receptor partial agonist</p>Fórmula:C37H39IO9Pureza:98%Forma y color:SolidPeso molecular:754.6LUF7244
CAS:<p>LUF7244 is a K v 11.1 channel modulator with anti-arrhythmia research potential, curbing early afterdepolarizations.</p>Fórmula:C20H15ClN2O3Forma y color:SolidPeso molecular:366.8PMPA (NMDA antagonist)
CAS:<p>PMPA (NMDA antagonist) is a Competitive NMDA receptor antagonist.</p>Fórmula:C6H13N2O5PPureza:98%Forma y color:SolidPeso molecular:224.15piCRAC-1
CAS:<p>piCRAC-1 is a powerful inhibitor of the photoinducible Ca2+ release-activated Ca2+ (CRAC) channel.</p>Fórmula:C17H10F6N4Forma y color:SolidPeso molecular:384.28RyRs activator 3
CAS:<p>RyRs activator 3 (compound A4) serves as an insecticide highly effective against both the diamondback moths, M.</p>Fórmula:C23H19BrCl2N6O3Pureza:98%Forma y color:SolidPeso molecular:578.25Ned-K
CAS:<p>Ned-K blocks NAADP, reduces heart ischemia-reperfusion calcium waves.</p>Fórmula:C31H31N5O3Forma y color:SolidPeso molecular:521.61Relutrigine
CAS:<p>Relutrigine (PRAX-562) is an oral persistent sodium channel inhibitor with anticonvulsant properties, IC50 of 141 nM/75 nM for ATX-II/SCN8A-N1768D.</p>Fórmula:C15H11F6N5O2Forma y color:SolidPeso molecular:407.27(R)-(+)-HA-966
CAS:<p>(R)-(+)-HA-966 ((+)-HA-966) is a partial agonist/antagonist of glycine site of the N-methyl-D-aspartate (NMDA) receptor complex. (R)-(+)-HA-966 selectively blocks the activation of the mesolimbic dopamine system by amphetamine, has the potential for neuro</p>Fórmula:C4H8N2O2Forma y color:White SolidPeso molecular:116.12Otaplimastat
CAS:<p>SP-8203 is a reactive oxygen species inhibitor and superoxide dismutase stimulant.</p>Fórmula:C28H34N6O5Pureza:98%Forma y color:SolidPeso molecular:534.61DL-AP5 Sodium salt
CAS:DL-AP5 Sodium salt is a NMDA receptor antagonist.Fórmula:C5H12NNaO5PPureza:98%Forma y color:SolidPeso molecular:220.12Linopirdine dihydrochloride
CAS:<p>KV7 (KCNQ) voltage-gated potassium channels blocker</p>Fórmula:C26H22ClN3OPureza:98%Forma y color:SolidPeso molecular:427.93TDN345
CAS:<p>TDN345 is a antagonist of Ca2+, for the treatment of vascular and senile dementia including Alzheimer's disease.</p>Fórmula:C28H34F2N2O2Pureza:98%Forma y color:SolidPeso molecular:468.58PK-THPP
CAS:<p>PK-THPP is a channel blocker of TASK-3.</p>Fórmula:C29H32N4O2Forma y color:SolidPeso molecular:468.59MPX-007
CAS:<p>MPX-007, a potent NMDA inhibitor, inhibits GluN2A-containing NMDA receptors expressed in HEK cells with IC50s of 27 nM.</p>Fórmula:C18H17F2N5O3S2Forma y color:SolidPeso molecular:453.49NS5818
CAS:<p>NS5818 inhibits ClC.</p>Fórmula:C23H19Cl2N7O2Pureza:98%Forma y color:SolidPeso molecular:496.35P-CAB agent 2
CAS:<p>Potent P-CAB agent 2 blocks gastric acid secretion; H+/K+-ATPase IC50 <100 nM, hERG IC50 18.69 μM; non-toxic.</p>Fórmula:C22H25FN2O4SForma y color:SolidPeso molecular:432.51RS 029
CAS:<p>RS 029 is a nitroimidazole that has been exhibited to significantly inhibit (Na+K+) ATP-ase activity.</p>Fórmula:C13H16N6O6Pureza:98%Forma y color:SolidPeso molecular:352.3CP 339818 hydrochloride
CAS:<p>KV1.3 channel antagonist</p>Fórmula:C21H25ClN2Pureza:98%Forma y color:SolidPeso molecular:340.89Vincanol
CAS:<p>Vincanol is a potent voltage-gated Na+ channels blocker.</p>Fórmula:C19H24N2OPureza:98%Forma y color:SolidPeso molecular:296.41NS004
CAS:<p>NS004 is a large-conductance K+ channel opener, it inhibits mitochondrial function in glioma cells.</p>Fórmula:C14H8ClF3N2O2Pureza:98%Forma y color:SolidPeso molecular:328.67KCa2 channel modulator 1
CAS:<p>Compound 2o, a selective K/Ca2 channel enhancer, boosts rat K Ca 2.2 (EC50: 0.99 μM) and human K Ca 2.3 (EC50: 0.19 μM).</p>Fórmula:C16H15ClFN5Forma y color:SolidPeso molecular:331.78Leconotide
CAS:<p>Leconotide is a calcium channel blocker and antihyperalgesia agent; isolated from the venom of the cone snail, Conus catus.</p>Fórmula:C107H179N35O36S7Forma y color:SolidPeso molecular:2756.23TTA-P2
CAS:<p>TTA-P2: potent CNS-penetrating T-type Ca2+ channel blocker; eliminates Cav3.1 window currents.</p>Fórmula:C21H29Cl2FN2O2Forma y color:SolidPeso molecular:431.37NAV26
CAS:<p>NAV26 is a selective blocker of the Nav1.7 channel.</p>Fórmula:C22H21F3N2O4Pureza:98%Forma y color:SolidPeso molecular:434.41GABAA receptor modulator-2
CAS:<p>Compound 20: Selective, oral α5-GABAAR inhibitor, Ki: 4.1 nM. High stability, CNS safe.</p>Fórmula:C22H22FN3O5SForma y color:SolidPeso molecular:459.49ANO1-IN-2
CAS:<p>ANO1-IN-2: potent ANO1 blocker (IC50: 1.75 μM), less effective on ANO2 (IC50: 7.43 μM), inhibits glioblastoma cell growth.</p>Fórmula:C16H14ClN3O2S2Forma y color:SolidPeso molecular:379.88BMS-284640
CAS:<p>BMS-284640 is a NHE inhibitor that protects against MI in animal studies.</p>Fórmula:C15H19N3O2Forma y color:SolidPeso molecular:273.33
