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Transportador de membrana / canal de iones

Transportador de membrana / canal de iones

Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.

Subcategorías de "Transportador de membrana / canal de iones"

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Se han encontrado 2272 productos de "Transportador de membrana / canal de iones"

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  • 264W94
    Targetmol
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    264W94

    CAS:
    <p>264W94 robustly inhibits IBAT, induces CYP7A1, and significantly reduces cholesterol.</p>
    Fórmula:C23H31NO4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:417.56

    Ref: TM-T10090

  • CFTR corrector 18
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    CFTR corrector 18

    CAS:
    <p>CFTRcorrector 18 (Compound I-99) acts as a modulator of the cystic fibrosis transmembrane conductance regulator (CFTR). It enhances the processing and trafficking of CFTR, thereby increasing the amount of CFTR present on the cell surface. CFTRcorrector 18 holds potential for research in cystic fibrosis (CF).</p>
    Fórmula:C38H40N6O5S
    Forma y color:Solid
    Peso molecular:692.826

    Ref: TM-T206874

  • P2X4-IN-1
    Targetmol
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    P2X4-IN-1

    CAS:
    <p>P2X4-IN-1 is an orally active P2X4 inhibitor. P2X4-IN-1 is applicable in research focused on disease prevention.</p>
    Fórmula:C18H14ClN5O3S
    Forma y color:Solid
    Peso molecular:415.85

    Ref: TM-T207340

  • ML-SI1
    Targetmol
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    ML-SI1

    CAS:
    <p>ML-SI1, a racemic mixture of diastereoisomers, is a TRPML inhibitor and acts on TRPML1 (IC50: 15 μM).</p>
    Fórmula:C23H26Cl2N2O3
    Forma y color:Solid
    Peso molecular:449.37

    Ref: TM-T62692

  • 3-Bromoamphetamine hydrochloride
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    3-Bromoamphetamine hydrochloride

    CAS:
    <p>3-Bromoamphetamine hydrochloride is a para-substituted amphetamine that functions as a monoamine releaser.</p>
    Fórmula:C9H13BrClN
    Forma y color:Solid
    Peso molecular:250.563

    Ref: TM-T206868

  • Logo de CymitQuimica
    Targetmol
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    PF-06305591 dihydrate

    <p>PF-06305591 dihydrate is a potent and highly selective voltage gated sodium channel NaV1.8 blocker (IC 50 = 15 nM) with an excellent preclinical in vitro ADME</p>
    Fórmula:C15H26N4O3
    Forma y color:Solid
    Peso molecular:310.39

    Ref: TM-T60761

  • Mibefradil dihydrochloride hydrate
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    Mibefradil dihydrochloride hydrate

    CAS:
    <p>Mibefradil dihydrochloride hydrate is a long-acting antihypertensive blocking high-voltage L calcium channels.</p>
    Fórmula:C29H42Cl2FN3O4
    Forma y color:Solid
    Peso molecular:586.57

    Ref: TM-T64151

  • LY 235959
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    LY 235959

    CAS:
    <p>LY 235959 is a NMDA receptor antagonist.</p>
    Fórmula:C11H20NO5P
    Pureza:98%
    Forma y color:Solid
    Peso molecular:277.25

    Ref: TM-T22944

  • Logo de CymitQuimica
    Targetmol
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    CRM1 degrader 1

    <p>CRM1 degrader 1 (1l) is a low-toxic CRM1 degrader that induces apoptosis in gastric carcinoma and selectively inhibits the proliferation of gastric cancer[1].</p>
    Fórmula:C16H20O3
    Forma y color:Solid
    Peso molecular:260.33

    Ref: TM-T60416

  • PDE2 inhibitor 6
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    PDE2 inhibitor 6

    CAS:
    <p>PDE2 inhibitor6 (Compound 1) is an orally active phosphodiesterase (PDE) inhibitor, effectively inhibiting PDE2A, PDE3B, and PDE10A2 with IC50 values of 0.95 nM, 6.17 μM (pIC50=5.21), and 87.1 nM (pIC50=7.06), respectively. It modulates AMPA receptor activity, enhances synaptic plasticity, and improves learning and memory in rat models. Furthermore, PDE2 inhibitor6 possesses blood-brain barrier permeability.</p>
    Fórmula:C20H22F2N6O
    Forma y color:Solid
    Peso molecular:400.425

    Ref: TM-T206498

  • Metaphit methylsulfate
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    Metaphit methylsulfate

    CAS:
    <p>Metaphit methylsulfate is a specific PCP antagonist and an acylating agent for the [3H] phencyclidine binding site in rat brain homogenate. It inhibits PCP-induced motor activity through a presynaptic mechanism.</p>
    Fórmula:C19H28N2O3S2
    Forma y color:Solid
    Peso molecular:396.567

    Ref: TM-T204740

  • Logo de CymitQuimica
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    URAT1 inhibitor 3

    <p>URAT1 inhibitor 3: potent oral URAT1 blocker, IC50=0.8 nM, for gout/hyperuricemia study.</p>
    Fórmula:C14H8Cl2N2O2
    Forma y color:Solid
    Peso molecular:307.13

    Ref: TM-T60724

  • Unoprostone
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    Unoprostone

    CAS:
    <p>Unoprostone is a prostaglandin F2α analogs (PGAs), and reduces intraocular pressure and is used topically for glaucoma or ocular hypertension.</p>
    Fórmula:C22H38O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:382.53

    Ref: TM-T13955

  • S-8510 phosphate
    Targetmol
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    S-8510 phosphate

    CAS:
    <p>S-8510 phosphate is an agonist of inverse Benzodiazepine (BDZ) receptor(Kis of 34.6 nM, 36.2 nM for –GABA and +GABA respectively).</p>
    Fórmula:C12H13N4O6P
    Pureza:98%
    Forma y color:Solid
    Peso molecular:340.23

    Ref: TM-T12792

  • Gabaculine HCl
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    Gabaculine HCl

    CAS:
    <p>Gabaculine, an irreversible GABA-T inhibitor (Ki: 2.9 μM), impacts plastid development and affects DPOR/GluTR levels.</p>
    Fórmula:C7H10ClNO2
    Forma y color:Solid
    Peso molecular:175.61

    Ref: TM-T24080

  • EMD-95885
    Targetmol
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    EMD-95885

    CAS:
    <p>EMD-95885 is a selective antagonist of NMDA receptors containing NR2B subunits, with an IC50 of 3.9 nM. It does not interact with other sites on the NMDA receptor.</p>
    Fórmula:C22H23FN2O3
    Forma y color:Solid
    Peso molecular:382.428

    Ref: TM-T205291

  • RO-275
    Targetmol
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    RO-275

    CAS:
    <p>RO-275 is an HCN1 inhibitor that also inhibits HCN2, HCN3, and HCN4, improving working memory deficits and being used in research on cognitive disorders.</p>
    Fórmula:C18H14ClN5O
    Pureza:98.12% - 98.3%
    Forma y color:Solid
    Peso molecular:351.79

    Ref: TM-T87339

  • Olorigliflozin
    Targetmol
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    Olorigliflozin

    CAS:
    <p>Olorigliflozin is a sodium glucose co-transporter (SGLT) inhibitor with antihyperglycemic properties.</p>
    Fórmula:C23H27ClO7
    Forma y color:Solid
    Peso molecular:450.909

    Ref: TM-T205428

  • ARN23765
    Targetmol
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    ARN23765

    CAS:
    <p>ARN23765 is an F508del-CFTR corrector with an EC50 of 38 pM in human bronchial epithelial cells. It enhances the maturation and function of F508del-CFTR at the cell membrane, influencing ion transport and secretion, thereby addressing the pathological mechanisms of cystic fibrosis (CF).</p>
    Fórmula:C30H22F5N3O6
    Forma y color:Solid
    Peso molecular:615.504

    Ref: TM-T205032

  • Pyrimidinone 8
    Targetmol
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    Pyrimidinone 8

    CAS:
    <p>Pyrimidinone 8 is a reversible, linear non-competitive inhibitor of divalent metal transporter 1 (DMT1) with a Ki of 20 μM (hDMT1). It does not affect the surface expression of hDMT1 and is not influenced by extracellular pH. Pyrimidinone 8 inhibits hDMT1-mediated iron uptake, with an IC50 of 13.8 μM.</p>
    Fórmula:C10H12N4O
    Forma y color:Solid
    Peso molecular:204.229

    Ref: TM-T205042