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Metabolismo

Metabolismo

Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.

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Se han encontrado 8625 productos de "Metabolismo"

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  • Hydroxypyruvic acid

    CAS:
    <p>Hydroxypyruvic acid: a metabolic intermediate for glycine, serine, threonine; used by serine-pyruvate aminotransferase, glyoxylate reductase.</p>
    Fórmula:C3H4O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:104.06
  • Methiocarb

    CAS:
    <p>Methiocarb is a carbamate insecticide acting as a reversible AChE or ChE inhibitor, inducing oxidative stress in rats.</p>
    Fórmula:C11H15NO2S
    Pureza:98.49%
    Forma y color:Colorless Crystals Immobilizing Agent For Birds Acaricide And Molluscicide (Epa 1998)
    Peso molecular:225.31
  • Decanoyl coenzyme A

    CAS:
    <p>Decanoyl coenzyme A (Decanoyl CoA) serves as a primer for the fatty acid elongation system in Mycobacterium smegmatis [1].</p>
    Fórmula:C31H54N7O17P3S
    Forma y color:Solid
    Peso molecular:921.78
  • Abiraterone sulfate

    CAS:
    <p>Abiraterone sulfate is a metabolite of Abiraterone . Abiraterone is a potent and irreversible CYP17A1 inhibitor with antiandrogen activity [1] .</p>
    Fórmula:C24H31NO4S
    Forma y color:Solid
    Peso molecular:429.57
  • Naroparcil

    CAS:
    <p>Naroparcil, an oral thioglycoside, has antithrombotic properties and alters thrombin complex formation.</p>
    Fórmula:C19H17NO4S2
    Pureza:98.71% - 99.88%
    Forma y color:Solid
    Peso molecular:387.47
  • β-Glucosidase

    CAS:
    <p>β-Glucosidase is a glucoside bond hydrolase involved in glucose metabolism and can be used to study diseases caused by abnormal glucose metabolism.</p>
    Fórmula:C24H44O12
    Forma y color:Solid
    Peso molecular:524.6
  • AMG-529


    <p>AMG-529 is a humanized monoclonal antibody targeting ASGR1, capable of binding to ASGR1 and inhibiting ligand attachment, which subsequently results in an increase in ALP (ASGR1-inhibited biomarker) levels.</p>
    Forma y color:Odour Liquid
  • Sofosbuvir impurity E


    <p>Sofosbuvir impurity E, a less active byproduct, inhibits HCV RNA replication with potent anti-HCV effects.</p>
    Fórmula:C22H29FN3O9P
    Pureza:98%
    Forma y color:Solid
    Peso molecular:529.45
  • Octocog alfa

    CAS:
    <p>Octocog alfa, a second-generation, full-length recombinant antihemophilic factor VIII (AHF), is utilized for the treatment of Hemophilia A [1].</p>
    Forma y color:Solid
  • Setosusin

    CAS:
    <p>Setosusin, a meroterpenoid from C. setosus, reduces Aβ-induced neurotoxicity in PC12 cells (EC50 = 112.6 μM).</p>
    Fórmula:C29H38O8
    Forma y color:Solid
    Peso molecular:514.615
  • Calcium 2-oxoglutarate

    CAS:
    <p>Calcium 2-oxoglutarate is an intermediate in the production of GTP or ATP in the Krebs cycle. It is a reversible inhibitor of tyrosinase (IC50: 15 mM).</p>
    Fórmula:C5H8CaO5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:188.192
  • MK-8262

    CAS:
    <p>MK-8262: oral CETP inhibitor, potent (IC50 = 53 nM, log D = 5.3), may impact HDL/LDL and CHD research.</p>
    Fórmula:C35H25F9N2O5
    Forma y color:Solid
    Peso molecular:724.58
  • Dansylphenylalanine

    CAS:
    <p>Dansylphenylalanine is a typical fluorescent analyte.</p>
    Fórmula:C21H22N2O4S
    Forma y color:Solid
    Peso molecular:398.48
  • Dihydrocarminomycin

    CAS:
    <p>Dihydrocarminomycin is an anthracycline antibiotics.</p>
    Fórmula:C26H29NO10
    Pureza:98%
    Forma y color:Solid
    Peso molecular:515.515
  • Pepticinnamin E

    CAS:
    <p>Pepticinnamin E is a naturally occurring bisubstrate farnesyltransferase inhibitor.</p>
    Fórmula:C49H54ClN5O10
    Pureza:98%
    Forma y color:Solid
    Peso molecular:908.43
  • 9AzNue5Ac

    CAS:
    <p>9AzNue5Ac is a Neu5Ac analog that is metabolized in vivo in living cells and in mice.9AzNue5Ac binds to sialoglycans.</p>
    Fórmula:C11H18N4O8
    Pureza:≥98%
    Forma y color:Solid
    Peso molecular:334.28
  • Aschantin

    CAS:
    <p>Aschantin is a useful organic compound for research related to life sciences. The catalog number is T126072 and the CAS number is 13060-15-6.</p>
    Fórmula:C22H24O7
    Forma y color:Solid
    Peso molecular:400.427
  • DPP-4-IN-11


    <p>DPP-4-IN-11 (compound 10) is an orally active DPP-4 inhibitor (IC50=2.75 μM) with anti-type 2 diabetes activity. This compound exerts its hypoglycemic effects by inhibiting the activity of α-glucosidase (IC50=3.02 μM) and α-amylase (IC50=3.3 μM).</p>
    Forma y color:Odour Solid
  • Relzomostat

    CAS:
    <p>Relzomostat inhibits MetAP2, with research potential for obesity and type 2 diabetes.</p>
    Fórmula:C24H36F2N2O5
    Forma y color:Solid
    Peso molecular:470.558
  • Defensin HNP-2 human

    CAS:
    <p>Defensin HNP-2 is a naturally occurring antibiotic and monocyte chemotactic peptide synthesized by human neutrophils.</p>
    Fórmula:C147H223N43O37S6
    Forma y color:Solid
    Peso molecular:3377.03
  • (±)14-HDHA

    CAS:
    <p>(±)14-HDHA is an oxidized metabolite of DHA and can be further oxidized to the 14-oxoDHA, 14-HDoHE inhibits LPS-induced IL-6 mRNA expression.</p>
    Fórmula:C22H32O3
    Forma y color:Solid
    Peso molecular:344.49
  • α-2,3-Sialyltransferase (PmST3)

    CAS:
    <p>PmST3 is a beta-galactoside enzyme adding sialic acid to glycoproteins and glycolipids.</p>
    Forma y color:Solid
  • BDM_92499


    <p>BDM_92499 is a nanomolar, selective IRAP inhibitor with an IC50 of 3.4 nM. It also inhibits ERAP1 and ERAP2, with IC50 values of 0.46 μM and 4.2 μM, respectively.</p>
    Forma y color:Odour Solid
  • 6-Azathymine acid

    CAS:
    <p>6-Azathymine is a metabolite of Pymetrozine, an insecticide targeting aphids and whiteflies by disrupting feeding.</p>
    Fórmula:C4H3N3O4
    Forma y color:Solid
    Peso molecular:157.08
  • CAIX/CAXII-IN-3


    <p>CAIX/CAXII-IN-3 (compound 11) serves as an inhibitor for CAIX/CAXII, exhibiting an IC50 value of less than 65 nM. Additionally, this compound effectively inhibits the proliferation of human melanoma cells.</p>
    Forma y color:Odour Solid
  • N-Desethyl Bimatoprost

    CAS:
    <p>N-Desethyl Bimatoprost (17-phenyl trinor PGF2α amide) is an F-series PG analog in which the C-1 carboxyl group has been modified to an unsubstituted amide.</p>
    Fórmula:C23H33NO4
    Forma y color:Solid
    Peso molecular:387.51
  • α-1,4-Galactosyltransferase (LgtC)

    CAS:
    <p>A4GALT (LgtC) adds galactose to lactosylceramide, forming globotriaosylceramide; used in P1 antigen synthesis.</p>
    Forma y color:Solid
  • 10 FTHF disodium

    CAS:
    <p>10 FTHF disodium (10-Formyltetrahydrofolic acid disodium) is a form of tetrahydrofolate that is involved in the synthesis of purine compounds.</p>
    Fórmula:C20H21N7Na2O7
    Forma y color:Solid
    Peso molecular:517.4
  • 4,8-Dioxa-3H-perfluorononanoic acid

    CAS:
    <p>4,8-Dioxa-3H-perfluorononanoic acid, a type of per- and polyfluoroalkyl substance (PFAS), exhibits affinity for the human pregnane X receptor (hPXR) and demonstrates potential agonistic activity.</p>
    Fórmula:C7H2F12O4
    Forma y color:Solid
    Peso molecular:378.07
  • 1-Palmitoyl Lysophosphatidic Acid

    CAS:
    <p>1-Palmitoyl Lysophosphatidic Acid boosts antibiotics against P. aeruginosa by binding Ca2+ and Mg2+.</p>
    Fórmula:C19H39O7P
    Pureza:98%
    Forma y color:Solid
    Peso molecular:410.48
  • PPARγ-IN-3


    <p>PPARγ-IN-3 (compound 9ga), a potent and orally active PPARγ inhibitor, effectively reduces triglyceride (TG) accumulation and exhibits low cytotoxicity. Additionally, it prevents excessive body weight gain, lessens fat and liver mass, and decreases lipid accumulation in both the liver and blood. PPARγ-IN-3 holds promise for research into diet-induced obesity.</p>
    Fórmula:C23H28FN7O3
    Forma y color:Solid
    Peso molecular:469.51
  • Monoglyceride lipase

    CAS:
    <p>Monoglyceridelipase is a crucial enzyme involved in lipid metabolism, catalyzing the hydrolysis of monoglycerides (especially 2-AG, or 2-arachidonoylglycerol) into glycerol and free fatty acids. By regulating the levels of 2-AG, this enzyme impacts neural signaling, pain perception, inflammatory responses, and metabolic processes.</p>
    Forma y color:Solid
  • α-Glucosidase-IN-72


    <p>α-Glucosidase-IN-72 (compound 5i), a 2,4-dichloro-N-phenylacetamide derivative, functions as an α-glucosidase inhibitor with an inhibitory concentration (IC 50) of 6 μM. Notably, it does not adhere to Lipinski's "rule of five" and is not a cancer inducer.</p>
    Fórmula:C37H26Cl2N4O9
    Forma y color:Solid
    Peso molecular:741.53
  • PP5-IN-2


    <p>PP5-IN-2, a selective and orally active inhibitor of protein phosphatase 5 (PP5), exhibits an IC 50 of 0.9 μM. This compound activates p53 and leads to the downregulation of cyclin D1 and MGMT, thereby inducing cell cycle arrest and reversing Temozolomide (TMZ) resistance in the U87 MG cell line. Additionally, PP5-IN-2 has demonstrated effective inhibition of tumor growth in the xenograft mouse model.</p>
    Fórmula:C16H15NO4
    Forma y color:Solid
    Peso molecular:285.29
  • Penicillinase

    CAS:
    <p>Penicillinase is a β-lactamase and secretory enzyme capable of degrading and inactivating penicillin and similar compounds.</p>
    Forma y color:Solid
  • C-Type Natriuretic Peptide (1-53), Porcine, Rat,mouse

    CAS:
    <p>C-Type Natriuretic Peptide (1-53), from porcine, rat, and mouse sources, serves as an activator of particulate guanylate cyclase B (pGC-B), prominently found in endothelial cells, kidneys, and the heart. This peptide efficiently mediates a potent anti-fibrotic effect in human cardiac and renal fibroblasts through the production of the second messenger cGMP.</p>
    Forma y color:Solid
  • N-acetyl Leukotriene E4

    CAS:
    <p>N-acetyl Leukotriene E4 is an endogenous metabolite of Leukotriene E4, less active than Leukotriene E4, causing constriction of the airways.</p>
    Fórmula:C25H39NO6S
    Forma y color:Solid
    Peso molecular:481.65
  • Bacterial α-Amylase

    CAS:
    <p>Bacterial α-Amylase is an enzyme that catalyzes the hydrolysis reaction of starch into smaller sugar molecules such as maltose and glucose.</p>
    Forma y color:Solid
  • (S)-ICMT-IN-3


    <p>'(S)-ICMT-IN-3 (compound ent 1-27) is an ICMT inhibitor with an IC50 value of 0.23 μM [1].'</p>
    Forma y color:Odour Solid
  • Estriol 3-glucuronide

    CAS:
    <p>Estriol-3-glucuronide, a natural compound found in urine, is also present in amniotic fluid during normal pregnancy [1][2].</p>
    Fórmula:C24H32O9
    Forma y color:Solid
    Peso molecular:464.511
  • N1-Acetylspermine

    CAS:
    <p>N1-Acetylspermine, an endogenous metabolite found in urine, has applications in leukemia research [1] [2].</p>
    Fórmula:C12H28N4O
    Forma y color:Solid
    Peso molecular:244.38
  • 3-O-Dihydro-p-coumaroyltohogenol


    <p>3-O-Dihydro-p-coumaroyltohogenol functions as a PTP1B inhibitor (IC50 = 6.27 μM), exhibiting anti-diabetic and anti-obesity activities.</p>
    Fórmula:C39H60O5
    Forma y color:Solid
    Peso molecular:608.89
  • ADP-specific glucokinase

    CAS:
    <p>ADP-specific glucokinase, expressed in thermophilic archaea, is an ADP-specific enzyme that catalyzes the conversion of glucose to glucose-6-phosphate, thereby facilitating glycolysis. This enzyme can activate T cells and enhance the phagocytic activity of macrophages. It is used in research related to metabolic disorders, neurological diseases, and tumors.</p>
    Forma y color:Solid
  • Phosphofructokinase

    CAS:
    <p>Phosphofructokinase, a crucial glycolytic enzyme, catalyzes the conversion of fructose-6-phosphate to fructose-1,6-bisphosphate in the glycolysis pathway. Its activity is inhibited by the binding of Phosphoenolpyruvate (PEP), which regulates the rate of glycolysis. Additionally, Phosphofructokinase is utilized in the measurement of fructose-6-phosphate (fructose-6-phosphate) levels.</p>
    Forma y color:Solid
  • IONIS PTP1BRx

    CAS:
    <p>IONIS PTP1BRx (ISIS 404173) acts as an antisense inhibitor of protein tyrosine phosphatase 1B (PTP-1B). This compound exhibits anti-diabetic properties, making it suitable for research into insulin resistance related to obesity and type 2 diabetes.</p>
    Forma y color:Solid
  • Antibacterial agent 237


    <p>Anti bacterial agent 237 (compound Ru-8) acts as a potent antibacterial agent against Staphylococcus aureus, exhibiting minimum inhibitory concentrations (MICs) ranging from 0.78 to 1.56 μg/mL. It works by disrupting bacterial cell membranes, altering their permeability, and inducing the production of reactive oxygen species, which leads to bacterial cell death without promoting resistance. Additionally, Anti bacterial agent 237 demonstrates low hemolytic toxicity towards rabbit erythrocytes and Raw 264.7 cells. It has shown significant antibacterial activity in models of skin wound infections in mice and larval infections by the greater wax moth, effectively combating Staphylococcus aureus infections.</p>
    Fórmula:C65H69Cl3N10RuS2
    Forma y color:Solid
    Peso molecular:1261.87
  • Imperatoxin A TFA


    <p>Imperatoxin A TFA, a peptide toxin derived from the venom of the African scorpion Pandinus imperator, acts as an activator of Ca2+-release channels/ryanodine receptors (RyRs). It facilitates the influx of Ca2+ from the sarcoplasmic reticulum into the cell.</p>
    Fórmula:C148H254N58O45S6·xC2HF3O2
    Forma y color:Solid
    Peso molecular:3758.35 (free base)
  • NAD Synthetase

    CAS:
    <p>NAD Synthetase is responsible for the final step in the synthesis of Nicotinamide Adenine Dinucleotide (NAD). The enzyme sourced from Escherichia coli exhibits Km values of 200 μM for NAD, 11 μM for ATP, and 0.65 μM for ammonia. Conversely, NAD Synthetase derived from yeast demonstrates Km values of 170 μM for NAD, 190 μM for ATP, and 64 μM for ammonia. This enzyme is applicable in enzymatic assays for ATP, ammonia, urea, or creatinine and can also be used in enzymatic recycling methods. Additionally, NAD Synthetase holds potential for research into metabolic diseases, cancer, aging, and neurodegenerative disorders.</p>
    Forma y color:Solid
  • Oseltamivir carboxylate HCl

    CAS:
    <p>Oseltamivir carboxylate is an active metabolite of oseltamivir phosphate (Tamiflu).</p>
    Fórmula:C14H25ClN2O4
    Forma y color:Solid
    Peso molecular:320.81
  • 10-Formyldihydrofolate

    CAS:
    <p>10-Formyldihydrofolate is a Methotrexate metabolite. It inhibits thymidylate synthetase and glycinamide ribotide transformylase.</p>
    Fórmula:C20H21N7O7
    Forma y color:Solid
    Peso molecular:471.43
  • h15-LOX-2 inhibitor 2


    <p>Compound 10 (h15-LOX-2 inhibitor 2) suppresses h15-LOX activity, exhibiting IC 50 and K i values of 26.9 μM and 16.4 μM, respectively.</p>
    Fórmula:C22H30Cl2N6O3
    Forma y color:Solid
    Peso molecular:497.42
  • N,S-Bis-Fmoc-Glutathione

    CAS:
    <p>N,S-Bis-Fmoc-Glutathione is a potent inhibitor of glyoxalase II, exhibiting a K i of 0.32 mM [1].</p>
    Fórmula:C40H37N3O10S
    Forma y color:Solid
    Peso molecular:751.8
  • Zymostenol

    CAS:
    <p>Zymostenol (5a-Cholest-8-en-3b-ol) is a RORγ agonist with an EC50 of 1 μM.Zymostenol is a late stage precursor of cholesterol biosynthesis.</p>
    Fórmula:C27H46O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:386.65
  • Leuhistin

    CAS:
    Leuhistin is an aminopeptidases N inhibitor isolated from Bacillus laterosporus BMI156-14F1.
    Fórmula:C11H19N3O3
    Pureza:98%
    Forma y color:White To Off-White Solid
    Peso molecular:241.29
  • IONIS PTP1BRx sodium


    <p>IONIS PTP1BRx (ISIS 404173) sodium, an antisense inhibitor of protein tyrene phosphatase 1B (PTP-1B), exhibits antidiabetic properties. This compound is utilzed in researching insulin resistance and type 2 diabetes mellitus associated with obesity.</p>
    Forma y color:Odour Solid
  • Maurocalcine TFA


    <p>Maurocalcine TFA acts as an agonist for ryanodine receptor (RyR) channels 1, 2, and 3, demonstrating cell-penetrating capabilities. It induces binding of [3H]ryanodine to RyR1 with an EC50 of 2558 nM and exhibits an apparent affinity of 14 nM for RyR2. This compound is applicable for in vivo cell tracking or other cellular imaging techniques.</p>
    Fórmula:C156H270N56O46S6·xC2HF3O2
    Forma y color:Solid
    Peso molecular:3858.55 (free base)
  • Epoxide hydrolase

    CAS:
    <p>Epoxide hydrolase, an enzyme responsible for catalyzing the reaction of epoxides with water to convert epoxy groups into diols, plays a crucial role in the metabolism of environmental pollutants and lipids. It is instrumental in detoxification, inflammatory responses, and regulating the health of the cardiovascular system. Additionally, Epoxide hydrolase is used in asymmetric catalytic reactions, such as the asymmetric ring-opening of epoxides, which are important for the synthesis of chiral pharmaceutical molecules.</p>
    Forma y color:Solid
  • PKM2-IN-4


    <p>Compound 5C, referred to as Pkm2-in-4, is a selective PKM2 inhibitor (IC50 = 0.35 µM) that modulates pyruvate-dependent respiration and promotes mitochondrial</p>
    Fórmula:C15H17BrClNO3Se
    Forma y color:Solid
    Peso molecular:453.62
  • 4'-Methoxyisoagarotetrol

    CAS:
    <p>4'-Methoxyisoagarotetrol, a chromone derivative, exhibits moderate phosphodiesterase 3A (PDE3A) inhibitory activity with an IC50 value of 54 μM [1].</p>
    Fórmula:C18H20O7
    Forma y color:Solid
    Peso molecular:348.35
  • ESI1


    <p>ESI1 is a small molecule inhibitor of epigenetic silencing. This compound induces the formation of nuclear aggregates of the key lipid metabolism regulator SREBP1/2, thereby concentrating transcription co-activators to drive lipid/cholesterol biosynthesis. Additionally, ESI1 promotes myelin regeneration in demyelination animal models and facilitates de novo myelination on regenerating CNS axons, reversing age-related cognitive decline.</p>
    Fórmula:C18H18ClN5O
    Forma y color:Solid
    Peso molecular:355.82
  • TSPO/Carbonic Anhydrase Modulator 1


    <p>TSPO/Carbonic Anhydrase Modulator 1 (Compound 3) acts as a dual modulator of mitochondrial translocator protein and carbonic anhydrase, with a TSPOKi of 1.340 μM and a CAVII KA of 10.7 μM. It enhances neurosteroid production, increases BDNF gene expression, and demonstrates neuroprotective activity.</p>
    Fórmula:C35H51N3O3
    Forma y color:Solid
    Peso molecular:561.798
  • 4,5-Dimethylthiazole

    CAS:
    <p>4,5-Dimethylthiazole exhibits inhibitory against mitochondrial respiration in liver cells and can be used in biochemical experiments and drug synthesis.</p>
    Fórmula:C5H7NS
    Forma y color:Solid
    Peso molecular:113.18
  • Galactose 1-dehydrogenase


    <p>Galactose 1-dehydrogenase, pseudomonas fluorescens, a dehydrogenase found in Pseudomonas fluorescens, facilitates the oxidation of L-arabinose and D-galactose, utilizing NADP+/NAD+ as a cofactor. This enzyme is employed in diagnostic assays to quantify total galactose levels and serves as a biocatalyst in the production of galacturonic acid salts.</p>
    Forma y color:Odour Solid
  • N-Desbutyl Dronedarone-d7 HCl


    <p>N-Desbutyl Dronedarone-d7 HCl is the deuterium-labelled isomer of N-Desbutyl Dronedarone HCl, used for isotope tracing. N-Desbutyl Dronedarone is a metabolite of the antiarrhythmic drug Dronedarone.</p>
    Fórmula:C27H30D7ClN2O5S
    Forma y color:Solid
    Peso molecular:544.15
  • Bupirimate

    CAS:
    Bupirimate, a systemic fungicide for powdery mildew in roses and apples, belongs to pyrimidines.
    Fórmula:C13H24N4O3S
    Pureza:99.56%
    Forma y color:Emulsifiable Liquid
    Peso molecular:316.42
  • Cho-Arg (trifluoroacetate salt)

    CAS:
    <p>Cho-Arg is a cholesterol-based cationic lipid that complexes with DNA, aids transfection, and is cytotoxic at 88.5 μg/ml IC50.</p>
    Fórmula:C43H71F6N5O7
    Forma y color:Solid
    Peso molecular:884.059
  • Diacetinase


    <p>Diacetinase, a member of the esterase family, catalyzes the hydrolysis of glyceryl diacetate (Diacetin). It is utilized in the measurement of lipase activity.</p>
    Forma y color:Odour Solid
  • Autophagy inducer 5


    <p>Autophagyinducer 5 (compound 21o) serves as a potent inhibitor of MCF-7 (IC50: 2 μM), making it a potential candidate for breast cancer therapy. It induces autophagy by activating the ROS/JNK signaling pathway, which increases ROS production and JNK phosphorylation, ultimately exerting cytotoxic effects.</p>
    Fórmula:C41H52N4O3
    Forma y color:Solid
    Peso molecular:648.88
  • KKII5

    CAS:
    <p>KKII5 is a potent inhibitor of the lipoxygenase LOX-1 with an IC50 of 19 μM.KKII5 inhibits lipid peroxidation and enhances the ability of the active centers of</p>
    Fórmula:C16H14N2S
    Pureza:99.34%
    Forma y color:Solid
    Peso molecular:266.36
  • Pregnant mare serum gonadotropin

    CAS:
    <p>Pregnant mare serum gonadotropin (PMSG) functions as a gonadotropin that enhances follicular development and ovulation in animals. This compound operates by modulating blood hormones, gonadotropins, and cytoplasmic estradiol receptors in the anterior pituitary and hypothalamus. Commonly employed in livestock to boost reproductive efficiency, PMSG is also valuable for research focused on estrous cycle regulation.</p>
    Forma y color:Solid
  • Kazusamycin A

    CAS:
    <p>Kazusamycin A is a new antitumor antibiotic.</p>
    Fórmula:C33H48O7
    Forma y color:Solid
    Peso molecular:556.74
  • 12α-Hydroxysteroid dehydrogenase

    CAS:
    <p>12α-Hydroxysteroid dehydrogenase, an NAD-dependent enzyme expressed in Bacillus sphaericus, actively processes both free and conjugated bile salts. It is utilized to determine the levels of 12α-hydroxy bile acids in serum.</p>
    Forma y color:Solid
  • Methyl (5α,7α)-7-hydroxy-3-oxocholan-24-oate

    CAS:
    <p>Compound 7a, Methyl (5α,7α)-7-hydroxy-3-oxocholan-24-oate, is a metabolite of bile acid.</p>
    Fórmula:C25H40O4
    Forma y color:Solid
    Peso molecular:404.58
  • Xanthine oxidase-IN-16


    <p>Xanthine oxidase-IN-16 is an effective orally active inhibitor of xanthine oxidase (XO), demonstrating significant therapeutic efficacy in rats with hyperuricemia and an IC50 of 102 nM.</p>
    Forma y color:Odour Solid
  • Sarcinapterin

    CAS:
    <p>Sarcinapterin is a coenzyme isolated from Methanosarcina barkeri.</p>
    Fórmula:C35H48N7O19P
    Forma y color:Solid
    Peso molecular:901.773
  • MPC-IN-1


    <p>MPC-IN-1 (compound 4i), a derivative of UK-5099, is a cyanocinnamate-based inhibitor of the mitochondrial pyruvate transporter (MPC). This compound selectively fosters the development of hair follicle stem cells while not impacting normal cells. It enhances cellular lactate production and has shown significant hair growth promotion in mice, suggesting its potential use in combating hair loss.</p>
    Fórmula:C18H13N3O2
    Forma y color:Solid
    Peso molecular:303.31
  • Creatine kinase (OcCK)

    CAS:
    <p>Creatine kinase (OcCK) converts creatine and ATP into phosphocreatine and ADP, crucial for ATP/ADP balance during high energy demand.</p>
    Forma y color:Solid
  • N-Fmoc-D-glutamine

    CAS:
    <p>N-Fmoc-D-glutamine is Fmoc-protected alpha-glutamine. Alpha-glutamine is an α-amino acid and the most abundant free amino acid in human blood.</p>
    Fórmula:C20H20N2O5
    Pureza:99.14%
    Peso molecular:368.38
  • Mersalyl

    CAS:
    <p>Mersalyl is an organic mercurial diuretic.</p>
    Fórmula:C13H16HgNNaO6
    Forma y color:Solid
    Peso molecular:505.854
  • Lysylcysteine TFA


    <p>Lysylcysteine (L-Lysyl-L-cysteine)TFA is a dipeptide composed of lysine and cysteine.</p>
    Fórmula:C13H21F6N3O7S
    Forma y color:Solid
    Peso molecular:477.10044
  • Alphostatin

    CAS:
    <p>Alphostatin is an alkaline phosphatase inhibitor isolated from Bacillus megaterium.</p>
    Fórmula:C25H45N6O13P
    Forma y color:Solid
    Peso molecular:668.638
  • Tetracosanoyl-sulfatide

    CAS:
    <p>C24 3'-sulfo Galactosylceramide is a key myelin sulfatide, high in leukodystrophy patients, non-immunogenic compared to C24:1 variant.</p>
    Fórmula:C48H93NO11S
    Forma y color:Solid
    Peso molecular:892.32
  • MK-4074

    CAS:
    <p>MK-4074 is a liver-specific acetyl-CoA carboxylase ACC1 and ACC2 inhibitor(IC50 of 3 nM).</p>
    Fórmula:C33H31N3O6
    Forma y color:Solid
    Peso molecular:565.62
  • (Rac)-sn-Glycerol 3-phosphate sodium

    CAS:
    <p>(Rac)-sn-Glycerol 3-phosphate sodium, an a-site substrate analogue, inhibits indole reactions with E(A-A).</p>
    Fórmula:C3H7Na2O6P
    Forma y color:Solid
    Peso molecular:216.04
  • Palitantin

    CAS:
    <p>Palitantin is a useful organic compound for research related to life sciences. The catalog number is T125757 and the CAS number is 15265-28-8.</p>
    Fórmula:C14H22O4
    Forma y color:Solid
    Peso molecular:254.326
  • (1S)-Calcitriol

    CAS:
    <p>(1S)-Calcitriol, a natural 1α,25(OH)2D3 metabolite, regulates VDR actions like keratinocyte growth inhibition.</p>
    Fórmula:C27H44O3
    Forma y color:Solid
    Peso molecular:416.646
  • 15-keto Latanoprost (free acid)

    CAS:
    <p>15-keto Latanoprost, a less potent metabolite and impurity of latanoprost, lowers intraocular pressure in monkeys and constricts pupils in cats.</p>
    Fórmula:C23H32O5
    Forma y color:Solid
    Peso molecular:388.5
  • DSPE-PEG2000-CREKA


    <p>DSPE-PEG3000-CREKA is a PEG compound composed of DSPE and the fibrin-targeting peptide (CREKA). The CREKA peptide targets tumor cells and tumor vasculature, exhibiting antitumor activity. DSPE-PEG3000-CREKA is useful in drug delivery applications.</p>
    Forma y color:Odour Solid
  • N-Benzoyl-L-Leucine

    CAS:
    <p>N-Benzoyl-L-Leucine is a leucine derivative exhibiting antibacterial activity against Staphylococcus aureus.</p>
    Fórmula:C13H17NO3
    Pureza:99.60%
    Forma y color:Soild
    Peso molecular:235.28
  • 5(S)​-​HPETE

    CAS:
    <p>5(S)-HpETE is a PUFA made by 5-LO from arachidonic acid, metabolized into LTA4, a key leukotriene precursor.</p>
    Fórmula:C20H32O4
    Forma y color:Solid
    Peso molecular:336.472
  • Phenylsulfamide

    CAS:
    <p>Phenylsulfamide (Compound 10), acting as an inhibitor of human carbonic anhydrase-II (hCA-II), exhibits a dissociation constant (Kd) of 45.50 μM and an</p>
    Fórmula:C6H8N2O2S
    Forma y color:Solid
    Peso molecular:172.2
  • Phosphate acetyltransferase

    CAS:
    <p>Phosphate acetyltransferase, an enzyme, reversibly transfers acetyl groups to CoA, aiding in acetate assimilation/dissimilation.</p>
    Forma y color:Solid
  • 1,2-Dipalmitoyl-sn-glycero-3-phosphoserine sodium salt

    CAS:
    <p>DPPS is a negatively charged diacyl-phospholipid used to create cationic vesicles and liposomes.</p>
    Fórmula:C38H73NNaO10P
    Pureza:99.54%
    Forma y color:Solid
    Peso molecular:757.95
  • VM4-037

    CAS:
    <p>VM4-037 is a PET imaging agent used for carbonic anhydrase IX.</p>
    Fórmula:C26H29FN6O7S2
    Forma y color:Solid
    Peso molecular:620.67
  • Fumarate hydratase-IN-2 sodium salt

    CAS:
    <p>Fumarate hydratase-IN-2 Na salt: cell-permeable, competitive inhibitor (Ki=4.5μM), nutrient-dependent cytotoxicity.</p>
    Fórmula:C25H25N2NaO4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:440.47
  • Aclimostat

    CAS:
    <p>Aclimostat (ZGN-1061) is a MetAP2 inhibitor with strong preclinical results, improving obesity-related metrics and gene expression.</p>
    Fórmula:C26H42N2O6
    Forma y color:Solid
    Peso molecular:478.63
  • BChE-IN-36


    <p>hBChE-IN-4 (compound 40) serves as an effective activator for hCA and an inhibitor for BChE. It demonstrates affinity for various hCA subtypes with affinity constants (KA) of 266 nM for hCA I, 76.9 nM for hCA II, 918 nM for hCA IV, 893 nM for hCA VB, and 98.0 nM for hCA VII. Inhibition concentrations (IC50) for eeAChE and eqBChE are recorded at 72.1 nM and 4.2 nM, respectively. hBChE-IN-4 is non-cytotoxic and has demonstrated potential cognitive enhancement effects. It holds potential for research in neurodegenerative and other neuropsychiatric disorders.</p>
    Forma y color:Odour Solid
  • Acanthifolicin

    CAS:
    <p>Acanthifolicin, an okadaic acid derivative, has been shown top inhibit protein phosphatase 1 with an IC50= 20 nM (similar to that of okadaic acid at 19 nM).</p>
    Fórmula:C44H68O13S
    Forma y color:Solid
    Peso molecular:837.08
  • ω-Muricholic Acid

    CAS:
    <p>ω-Muricholic acid (ω-MCA) is a murine-specific secondary bile acid.</p>
    Fórmula:C24H40O5
    Forma y color:Solid
    Peso molecular:408.57
  • DSPE-PEG2000-K237


    <p>DSPE-PEG2000-K237 is a PEG compound consisting of DSPE and the KDR-targeting peptide (K237). K237 functionally disrupts the interaction between VEGF and KDR receptors, resulting in significant biological effects such as inhibition of angiogenesis and tumor growth. DSPE-PEG2000-K237 is applicable in drug delivery.</p>
    Forma y color:Odour Solid