Metabolismo
Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.
Subcategorías de "Metabolismo"
- AhR(41 productos)
- Aminopeptidasa(74 productos)
- CETP(20 productos)
- Anhídrido carbónico(185 productos)
- Caseína quinasa(137 productos)
- DHFR(34 productos)
- Descarboxilasa(4 productos)
- Deshidrogenasa(289 productos)
- FAAH(65 productos)
- FXR(59 productos)
- Factor Xa(83 productos)
- Ácido graso sintasa(36 productos)
- Ferroptosis(218 productos)
- GR(3 productos)
- GSNOR(4 productos)
- Glucoquinasa(56 productos)
- HIF / HIF Prolilhidroxilasa(145 productos)
- HMG-CoA reductasa(33 productos)
- Hidroxilasa(34 productos)
- IDO(84 productos)
- LDL(8 productos)
- Lipasa(104 productos)
- Lípido(62 productos)
- Lipoxigenasa(132 productos)
- MAO(87 productos)
- MPO(2 productos)
- NAMPT(38 productos)
- P450(6 productos)
- PAI-1(26 productos)
- PDE(166 productos)
- PED(1 productos)
- PKM(15 productos)
- PPAR(168 productos)
- Fosfolipasa(82 productos)
- ROR(43 productos)
- Receptor de retinoides(28 productos)
- SGK(11 productos)
- Tiorredoxina(12 productos)
- Transferasa(29 productos)
- Transportador(43 productos)
- UGT(4 productos)
- Inhibidores de la xantina oxidasa (XO)(9 productos)
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Se han encontrado 9054 productos de "Metabolismo"
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NPD-1335
CAS:NPD1335: potent TbrPDEB1 inhibitor, submicromolar efficacy, low toxicity, raises cAMP, disrupts cell cycle, kills T. brucei.Fórmula:C28H29N3O3Pureza:98%Forma y color:SolidPeso molecular:455.55Xanthine oxidase-IN-5
CAS:Xanthine oxidase-IN-5: oral XO inhibitor, IC50 = 0.70 μM, LE = 0.33, LLE = 3.41, reduces uric acid in rats.Fórmula:C18H16FN3O3Forma y color:SolidPeso molecular:341.34ICI 153110
CAS:<p>ICI 153110: Oral phosphodiesterase inhibitor for treating congestive heart failure, has inotropic, vasodilator effects.</p>Fórmula:C11H11N3OPureza:98%Forma y color:SolidPeso molecular:201.22PRRSV/CD163-IN-1
CAS:PRRSV/CD163-IN-1 blocks PRRSV GP2a/GP4 and CD163-SRCR5, aiding PRRS research.Fórmula:C25H24FN5O5S2Forma y color:SolidPeso molecular:557.62Xanthine oxidase-IN-4
CAS:<p>Xanthine oxidase-IN-4: an oral XO inhibitor with 0.039 μM IC50, useful for hyperuricemia/gout research.</p>Fórmula:C15H13N5O2Forma y color:SolidPeso molecular:295.3DP00477
CAS:DP00477, a potent inhibitor of indoleamine 2,3-dioxygenase 1 (IDO1), exhibits an inhibitory concentration (IC50) of 7.0 µM.Fórmula:C17H11ClF3N3OSForma y color:SolidPeso molecular:397.8PDE4-IN-11
CAS:<p>PDE4-IN-11: Potent PDE4 inhibitor with strong bronchodilatory and anti-inflammatory effects for airway disease research.</p>Fórmula:C21H19FN2O2Forma y color:SolidPeso molecular:350.39hCAXII-IN-1
CAS:hCAXII-IN-1 selectively inhibits HCA IX/XII, promising for new cancer drug development.Fórmula:C20H17NO5Forma y color:SolidPeso molecular:351.3524(S),25-Epoxycholesterol
CAS:24(S),25-Epoxycholesterol is an oxysterol agonist of the liver X receptor.Fórmula:C27H44O2Forma y color:SolidPeso molecular:400.64FABP-IN-2
CAS:FABP-IN-2, a novel ligand for FABP3, demonstrates inhibition of both FABP3 and FABP4 with IC50 values of 1.16 μM and 4.27 μM, respectively.Fórmula:C25H21ClN2O3Forma y color:SolidPeso molecular:432.9A-908292
CAS:A-908292: potent ACC2 inhibitor with 38 nM IC50, useful for studying fatty acid metabolism.Fórmula:C18H20N2O4SForma y color:SolidPeso molecular:360.43Arasertaconazole
CAS:Arasertaconazole, a sterol-14-alpha demethylation inhibitor, is used potentially for the treatment of vulvovaginal candcanidiasis.Fórmula:C20H15Cl3N2OSForma y color:SolidPeso molecular:437.77Carbonic anhydrase inhibitor 7
CAS:Potent hCA inhibitor; targets hCA IX, II, XII, I with Ki: 6.5, 7.1, 72.1, 255.8 nM respectively.Fórmula:C23H17N3O5SForma y color:SolidPeso molecular:447.46Spirapril
CAS:Spiropril is an ACE inhibitor antihypertensive drug, which belongs to the bicarboxyl group of ACE inhibitors and is used in the treatment of hypertension.Fórmula:C22H30N2O5S2Forma y color:SolidPeso molecular:466.61Antitumor agent-88
CAS:Antitumor agent-88, a potent antimitotic, arrests G2/M phase, disrupts microtubules in breast cancer, and inhibits CYP1A1 (Ki: 1.4 μM).Fórmula:C23H30N2O7SForma y color:SolidPeso molecular:478.56Fmoc-5-aminopentanoic acid
CAS:Fmoc-5-aminopentanoic acid: alkane, Fmoc-protected amine, carboxyl group, PROTAC linker, deprotects to free amine, forms amides with activators.Fórmula:C20H21NO4Forma y color:SolidPeso molecular:339.39hCAIX-IN-14
CAS:hCAIX-IN-14 is a potent inhibitor of human CA IX with a K i value of 134.8 nM .Fórmula:C11H17ClN6O2SForma y color:SolidPeso molecular:332.81ATX inhibitor 8
CAS:ATX inhibitor 8 is an inhibitor of the autocrine motor factor Autotaxin (ATX).Fórmula:C28H26N10OForma y color:SolidPeso molecular:518.57CP 80633
CAS:CP 80633 is a PDE4 inhibitor.Fórmula:C18H24N2O3Pureza:98%Forma y color:SolidPeso molecular:316.39PDE11-IN-1
CAS:PDE11-IN-1 is a PDE11 inhibitor and can be used for adrenal insufficiency research [1].Fórmula:C16H10ClN3O3SForma y color:SolidPeso molecular:359.79Umbralisib tosylate
CAS:Umbralisib tosylate, an oral PI3Kδ/CK1ε inhibitor (EC50: 22.2 nM/6.0 μM), shows promise for CLL research.Fórmula:C38H32F3N5O6SForma y color:SolidPeso molecular:743.75JNJ-61803534
CAS:JNJ-61803534: RORγt inverse agonist, IC50=9.6 nM, oral, anti-inflammatory, reduces IL-17A in T cells.Fórmula:C23H23Cl2F6N3O4SForma y color:SolidPeso molecular:622.41GKA-71
CAS:<p>GKA-71 is an effective glucokinase activator (GKA).</p>Fórmula:C21H23N3O6S2Forma y color:SolidPeso molecular:477.55HIF-1α-IN-3
CAS:<p>HIF-1α-IN-3, also known as Compound (S)-3f, is a hypoxia-selective inhibitor of HIF-1α. It exhibits potent antiestrogenic activity [1].</p>Fórmula:C19H17N5O2Forma y color:SolidPeso molecular:347.37GNX-865
CAS:GNX-865 is an inhibitor of mitochondrial permeability transition pore (mtPTP).Fórmula:C16H14ClNO3Forma y color:SolidPeso molecular:303.74α-Amylase-IN-2
CAS:α-Glucosidase-IN-3, an oxime ester derivative of oleanolic acid (OA), exhibits inhibitory activity against α-glucosidase (IC50 = 1.28 µM) and α-amylase (IC50 =Fórmula:C39H52BrNO4Forma y color:SolidPeso molecular:678.74HIF-PHD-IN-2
CAS:HIF-PHD-IN-2 (compound 25) is a highly effective PHD inhibitor, displaying IC50 values below 100 nM for PHD1, PHD2, and PHD3 [1].Fórmula:C17H15N5O3SForma y color:SolidPeso molecular:369.4Chaetomellic acid A
CAS:Chaetomellic acid A inhibits farnesyltransferase (IC50=55nM), not active in cells, and selective over geranylgeranyltransferases (IC50: 92µM, 34µM).Fórmula:C19H34O4Forma y color:SolidPeso molecular:326.47HX-600
CAS:HX-600 is a synthetic agonist for the RXR-Nurr1 heterodimer complex. HX-600 prevents ischemia-induced neuronal damage.Fórmula:C29H30N2O2Forma y color:SolidPeso molecular:438.56SCD1-IN-1
CAS:SCD1-IN-1, a potent inhibitor of SCD1 (IC50: 5.8 nM), is valuable in dermatologic research [1].Fórmula:C20H20F3NO4Forma y color:SolidPeso molecular:395.37Xanthine oxidoreductase-IN-1
CAS:Xanthine oxidoreductase-IN-1 is a xanthine oxidoreductase (XOR) inhibitor with an IC 50 value of 7.0 nM.Fórmula:C18H20N4O2Forma y color:SolidPeso molecular:324.38JNJ-40413269
CAS:<p>JNJ-40413269 inhibits FAAH, engages central targets, and is effective in rat neuropathic pain.</p>Fórmula:C19H15ClF3N3OForma y color:SolidPeso molecular:393.79hCAIX-IN-7
CAS:<p>hCAIX-IN-7 (6c) selectively inhibits tumor-related isoform hCAIX (KI: 410.6 nM) and weakly affects hCAI/II (KI: >10000 nM).</p>Fórmula:C18H12FNO3Forma y color:SolidPeso molecular:309.29DMPAC-Chol
CAS:DMPAC-Chol, a cationic cholesterol, aids gene transfection, DNA protection, binds DNA, and lowers HepG2 viability at 37.5 μg/ml.Fórmula:C33H58N2O2Forma y color:SolidPeso molecular:514.83Glyoxalase I inhibitor 2
CAS:<p>Glyoxalase I inhibitor 2 (compound 26) blocks GLO1 effectively (IC50: 0.5 μM), promising for depression and anxiety research.</p>Fórmula:C24H23N3O4SForma y color:SolidPeso molecular:449.52Fluindione
CAS:Fluindione is a hematologic drug.Fórmula:C15H9FO2Forma y color:SolidPeso molecular:240.23URB532
CAS:URB532 is an irreversible fatty acid amide hydrolase (FAAH) inhibitor.Fórmula:C18H21NO3Pureza:98%Forma y color:SolidPeso molecular:299.36ALDH3A1-IN-2
CAS:ALDH3A1-IN-2 is a potent inhibitor targeting ALDH3A1 (IC50=1.29µM), potentially useful in cancer research.Fórmula:C11H14N2O3Forma y color:SolidPeso molecular:222.24AChE/hCA I/II-IN-1
CAS:Compound 6: Potent inhibitor for AChE, Hca I & II with IC50s of 22.21, 60.79, 66.64 nM, useful in glaucoma, Alzheimer's, diabetes research.Fórmula:C15H13N3SForma y color:SolidPeso molecular:267.35sEH inhibitor-6
CAS:<p>sEH inhibitor-6 (Compound 3g) is a highly potent soluble epoxide hydrolase (sEH) inhibitor, exhibiting an IC 50 value of 0.5 nM [1].</p>Fórmula:C21H14ClN3O2Forma y color:SolidPeso molecular:375.81OHM1
CAS:OHM1, an analog of HIF1α CTAD, effectively inhibits the interaction between HIF1α CTAD and p300/CBP by targeting the CH1 domain with a binding affinity of 0.53Fórmula:C24H42N6O5Forma y color:SolidPeso molecular:494.63Cholesteryl behenate
CAS:Cholesteryl behenate is a standard in electrospray ionization tandem mass spectrometry for the analysis of cholesteryl esters and cholesterol.Fórmula:C49H88O2Pureza:98%Forma y color:SolidPeso molecular:709.22CYP3A4-IN-3
CAS:CYP3A4-IN-3, a ritonavir analogue, is a potent CYP3A4 inhibitor with an IC50 of 0.075 μM, used as an antiviral and immunosuppressant.Fórmula:C34H39N3O3SForma y color:SolidPeso molecular:569.76CAY10762
CAS:CAY10762, a MAGL inhibitor (IC50=34.1 nM), curbs H2O2-induced LDH in Neuro2a cells and boosts 2-AG in mouse brains at 10 mg/kg.Fórmula:C15H13NOSForma y color:SolidPeso molecular:255.33ASP3662
CAS:ASP3662/SPI-62: Potent, selective CNS-penetrable 11β-HSD1 inhibitor; potential neuropathic pain treatment.Fórmula:C19H16ClF3N4O2Forma y color:SolidPeso molecular:424.8Trandolaprilate hydrate
CAS:Trandolaprilate hydrate, a powerful ACE inhibitor and Trandolapril's main metabolite, is lipophilic with partial c-fos blocking.Fórmula:C22H32N2O6Forma y color:SolidPeso molecular:420.5EDP-305
CAS:<p>EDP-305, an oral FXR agonist, has EC50s of 34 nM/8 nM in CHO/HEK cells, aids in PBC and NASH research with antifibrotic properties.</p>Fórmula:C36H58N2O5SForma y color:SolidPeso molecular:630.92Anserinone B
CAS:Anserinone B: Antifungal, antibacterial; inhibits S.fimicola (50%), A. furfuraceus (37%); cytotoxic to human tumor cells (GI50=4.4 µg/mL).Fórmula:C11H14O4Forma y color:SolidPeso molecular:210.23JBP485
CAS:JBP485 is an inhibitor of renal transporters OAT1 and OAT3. JBP485 is an antihepatitis agent as a substrate for intestinal PEPT1.Fórmula:C8H12N2O4Forma y color:SolidPeso molecular:200.19Kurasoin B
CAS:Kurasoin B is an inhibitor of protein farnesyltransferase.Fórmula:C18H17NO2Forma y color:SolidPeso molecular:279.33CAY10761
CAS:CAY10761 inhibits ENPP1 (IC50: 467 μM human, 429 μM snake), mushroom tyrosinase (Ki: 1.9 μM), and urease from different sources (IC50: 0.093-<0.125 mM).Fórmula:C7H8N4O2S2Forma y color:SolidPeso molecular:244.29FR-221647
CAS:FR-221647: non-nucleoside adenosine deaminase blocker, moderate efficacy, better pharmacokinetics than EHNA/Pentostatin.Fórmula:C14H17N3O2Forma y color:SolidPeso molecular:259.311β-HSD1-IN-10
CAS:11β-HSD1-IN-10, a potent inhibitor of 11β-HSD1 with an IC50 value of 1.8 µM for humans, is suitable for research into obesity, hyperglycemia, and cognitiveFórmula:C16H10F3NO2Forma y color:SolidPeso molecular:305.25IQA
CAS:<p>IQA is a casein kinase 2 (CK2) inhibitor.</p>Fórmula:C17H12N2O3Forma y color:SolidPeso molecular:292.29103D5R
CAS:<p>103D5R selectively inhibits hif-1α, reducing its levels in hypoxia or with cobalt ions, dose- and time-dependently.</p>Fórmula:C20H21N3O2Forma y color:SolidPeso molecular:335.4hCAI/II-IN-2
CAS:hCAI/II-IN-2 (2b) inhibits hCA I/II (Ki: 40.97 nM, 15.15 nM) and IX (61.88 nM), fights AMS with anti-hypoxic effects, but has low cellular activity.Fórmula:C12H12N4O5S2Forma y color:SolidPeso molecular:356.3814-dehydro Zymostenol
CAS:14-dehydro Zymostenol, a cholesterol precursor, boosts MBP+ oligodendrocytes from precursors at 5.8-17 μM.Fórmula:C27H44OForma y color:SolidPeso molecular:384.64TPN729MA
CAS:<p>TPN729MA, a potent PDE5 inhibitor, IC50: 2.28 nM, targets erectile dysfunction research.</p>Fórmula:C29H40N6O8SForma y color:SolidPeso molecular:632.73Loxoprofenol-SRS
CAS:<p>Loxoprofenol-SRS, a potent metabolite of Loxoprofen, is an IV NSAID with enhanced anti-inflammatory and pain relief properties.</p>Fórmula:C15H20O3Forma y color:SolidPeso molecular:248.32MEDS433
CAS:<p>MEDS433 inhibits dihydroorotate dehydrogenase (IC50 1.2 nM) and blocks replication of hCoV-OC43, hCoV-229E, SARS-CoV-2 at nanomolar levels.</p>Fórmula:C20H11F4N3O2Forma y color:SolidPeso molecular:401.31PKM2 activator 3
CAS:PKM2 activator 3, with 90 nM AC50, enhances PKM2. It has good Caco-2 permeability, stable, and aids cancer research.Fórmula:C15H11ClF2N2O3SForma y color:SolidPeso molecular:372.77SHP2 inhibitor LY6
CAS:<p>SHP2 inhibitor LY6 (LY6) is a potent and selective SHP2 inhibitor (IC50: 9.8 μM) that blocks SHP2-mediated cell signaling and proliferation.</p>Fórmula:C30H27Cl2N3O4Forma y color:SolidPeso molecular:564.46LY367385
CAS:LY367385 is a highly effective and selective mGluR1a antagonist.Fórmula:C10H11NO4Pureza:98%Forma y color:SolidPeso molecular:209.2UK-500001
CAS:<p>UK-500001 is a potent PDE4 inhibitor with robust anti-inflammatory activity.</p>Fórmula:C26H24F3N3O4Pureza:98%Forma y color:SolidPeso molecular:499.48IDH-C227
CAS:IDH-C227 is a selective and potent inhibitor of IDH1R132H that exhibits anticancer activity.Fórmula:C30H31FN4O2Forma y color:SolidPeso molecular:498.59hCAI/II-IN-1
CAS:<p>hCAI/II-IN-1 (Compound 3h) is a human carbonic anhydrase I and II (hCA I/II) inhibitor that acts on hCA I (IC50: 0.047 μM) and hCA II (IC50: 0.024 μM).</p>Fórmula:C18H29N5O3S3Forma y color:SolidPeso molecular:459.65TFB-TBOA
CAS:glial glutamate transporter EAAT1 and EAAT2 inhibitorFórmula:C19H17F3N2O6Pureza:98%Forma y color:SolidPeso molecular:426.34Enpp-1-IN-6
CAS:Enpp-1-IN-6, a potent enpp-1 inhibitor, may aid cancer and infectious disease studies (WO2021203772A1, compound 51).Fórmula:C22H28N4O5SForma y color:SolidPeso molecular:460.55Fodipir
CAS:Fodipir, the active metabolite of mangafodipir, plays a crucial role in the mechanism of mangafodipir-mediated cytoprotection, specifically mitigating cellFórmula:C22H32N4O14P2Pureza:98%Forma y color:SolidPeso molecular:638.46CD 2314
CAS:CD2314 is a potent and subtype-selective RARβ receptor agonist with a Kd of 195 nM in S91 melanoma cells [1].Fórmula:C23H24O2SForma y color:SolidPeso molecular:364.5ONO-1603
CAS:<p>ONO-1603, a prolyl endopeptidase inhibitor, is used potentially for the treatment of Alzheimer's disease.</p>Fórmula:C16H19ClN2O3Pureza:98%Forma y color:SolidPeso molecular:322.79hCAIX-IN-11
CAS:<p>hCAIX-IN-11 inhibits carbonic anhydrases IX & XII with Ki of 32.7 nM & 623.5 nM, respectively.</p>Fórmula:C21H15ClN4O3Forma y color:SolidPeso molecular:406.82(Rac)-Etavopivat
CAS:(Rac)-Etavopivat, an oral PKR activator, targets sickle cell disease and haemoglobinopathies.Fórmula:C22H23N3O6SForma y color:SolidPeso molecular:457.5ARL-67156 trisodium salt hydrate
CAS:ARL-67156 trisodium salt hydrate is an ecto-ATPase inhibitor that prevents metabolism of P2 purinoceptor agonists.Fórmula:C15H24Br2N5O12P3Forma y color:SolidPeso molecular:719.11Seviteronel R enantiomer
CAS:Seviteronel R enantiomer (VT-464 R enantiomer) is a Seviteronel isomer produced during the manufacturing process.Fórmula:C18H17F4N3O3Pureza:97.97% - >99.99%Forma y color:SolidPeso molecular:399.34ZSET-845
CAS:<p>ZSET-845 is an enhancer of cognitive which enhances choline acetyltransferase activity in the hippocampus in the rat.</p>Fórmula:C21H18N2OPureza:98%Forma y color:SolidPeso molecular:314.38Mevalonic acid
CAS:Mevalonic acid is essential for cell growth and proliferation,Mevalonic acid is a precursor in the mevalonate pathway.Fórmula:C6H12O4Pureza:98%Forma y color:SolidPeso molecular:148.16HCAIX-IN-2
CAS:HCAIX-IN-2 (compound 9d) is a selective inhibitor of carbonic anhydrase and acts on hCA IX (Ki: 24.6 nM) and hCA XII (Ki: 45.3 nM).Fórmula:C19H16N8O4SForma y color:SolidPeso molecular:452.45Glucosylceramide synthase-IN-2
CAS:T-690: Potent, BBB-permeable, oral GCS inhibitor; human IC50: 15 nM, mouse IC50: 190 nM; non-competitive with C8 ceramide/UDP glucose.Fórmula:C22H20F3N3O4Forma y color:SolidPeso molecular:447.41Fenleuton
CAS:Fenleuton is a 5-lipoxygenase inhibitor.Fórmula:C17H15FN2O3Pureza:98%Forma y color:SolidPeso molecular:314.31L 656224
CAS:L 656224 is a 5-LO inhibitor.Fórmula:C20H21ClO3Pureza:98%Forma y color:SolidPeso molecular:344.83BN-82685
CAS:<p>BN-82685, a quinone-based CDC25 inhibitor, shows in vitro and in vivo efficacy, suggesting potential as an anticancer therapy.</p>Fórmula:C12H15N3O2SPureza:98%Forma y color:SolidPeso molecular:265.33Win-62005
CAS:Win-62005 is an inhibitor of cyclic AMP phosphodiesterase III (PDE III)(Kis: 25 and 26 nM for rat heart and canine aorta).Fórmula:C12H10N4OPureza:98%Forma y color:SolidPeso molecular:226.23Dacisteine
CAS:Dacisteine (N,S-Diacetyl-L-cysteine) is an inhibitor of New Delhi metallo-beta-lactamase-1 (NDM-1, IC50 = 1000 μM).Fórmula:C7H11NO4SPureza:99.57%Forma y color:SolidPeso molecular:205.23PGAM1-IN-1
CAS:PGAM1-IN-1 is an inhibitor of phosphoglycerate mutase 1 ( PGAM1 ) with an IC 50 of 6.4 μM [1].Fórmula:C19H11ClFNO6SPureza:98%Forma y color:SolidPeso molecular:435.81LAZABEMIDE
CAS:Lazabemide (Ro 19-6327) is selective, reversible monoamine oxidase B (MAO-B) inhibitor (IC50 values are 0.03 and > 100 μM for MAO-B and MAO-A respectively).Fórmula:C8H10ClN3OPureza:98%Forma y color:SolidPeso molecular:199.64L-Xylulose
CAS:<p>L-Xylulose: a rare sugar, key in metabolism, α-glucosidase inhibitor, lowers glucose, precursor to antiviral drug components.</p>Fórmula:C5H10O5Forma y color:SolidPeso molecular:150.13IDO1/TDO-IN-2
CAS:<p>IDO1/TDO-IN-2: IDO1/TDO inhibitor; IC50s: IDO1, 0.1μM; TDO, 0.07μM; potential for cancer research.</p>Fórmula:C16H9N3O2Forma y color:SolidPeso molecular:275.26AK-106
CAS:AK-106, or AK106-001616, selectively inhibits cPLA2 and has NSAID-like analgesic effects.Fórmula:C26H25N3O3Forma y color:SolidPeso molecular:427.49Leniquinsin
CAS:Leniquinsin is an antihypertensive compound. It is a phosphodiesterase inhibitor and a potent vasodilator.Fórmula:C20H20N2O4Pureza:98%Forma y color:SolidPeso molecular:352.38KT109
CAS:KT109 is a DAGLβ inhibitor (IC50=42nM), lessens LPS allodynia in mice without tolerance, and has no major side effects.Fórmula:C27H26N4OPureza:98%Forma y color:SolidPeso molecular:422.52Tanogitran
CAS:Tanogitran, a coagulation factor Xa inhibitor, is used potentially for the treatment of septic shock.Fórmula:C25H31N7O3Pureza:98%Forma y color:SolidPeso molecular:477.56TC-E 5008
CAS:TC-E 5008 is a selective inhibitor of mutant isocitrate dehydrogenase 1 (mIDH1).Fórmula:C13H13NO2Forma y color:SolidPeso molecular:215.25α-Glucosidase-IN-3
CAS:α-Glucosidase-IN-3 is an oleanolic acid oxime ester derivative targeting α-glucosidase and α-amylase with an IC50 value of 0.35 μM for α-glucosidase.Fórmula:C39H53NO4Forma y color:SolidPeso molecular:599.84Oosponol
CAS:Oosponol is a dopamine beta-hydroxylase inhibitor exhibiting hypotensive effects.Fórmula:C11H8O5Pureza:98%Forma y color:SolidPeso molecular:220.18M8891
CAS:M8891: Oral, reversible MetAP-2 inhibitor, brain-penetrant (IC50: 54nM; Ki: 4.33nM), hinders endothelial & tumor cell growth, antiangiogenic & antitumor.Fórmula:C20H17F2N3O3Forma y color:SolidPeso molecular:385.36OL-135
CAS:<p>OL-135: CNS-accessible, potent, selective FAAH inhibitor with analgesic effects in animals, no motor impairment.</p>Fórmula:C21H22N2O2Forma y color:SolidPeso molecular:334.41Oleyl Anilide
CAS:"Oleyl analide (OA) inhibits ACAT (IC50 26 μM), linked to toxic oil syndrome (TOS) with eosinophilia, T-cell activation, and high IL-4, IL-2R, IL-5."Fórmula:C24H39NOForma y color:SolidPeso molecular:357.57ARN19874
CAS:ARN19874 is a selective, reversible uncompetitive N-acylphosphatidylethanolamine phospholipase D (NAPE-PLD) activity inhibitor. With an IC50 of ~34 μM[1].Fórmula:C19H14N4O4SPureza:98%Forma y color:SolidPeso molecular:394.4JNJ-42314415
CAS:JNJ-42314415 is a potent, specific, and centrally active inhibitor of PDE10A.Fórmula:C19H23N5O2Pureza:98%Forma y color:SolidPeso molecular:353.42
