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Metabolismo

Metabolismo

Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.

Subcategorías de "Metabolismo"

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Se han encontrado 8628 productos de "Metabolismo"

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  • 2'-Ethyl Simvastatin

    CAS:
    <p>2'-Ethyl Simvastatin is a Mevinolin analog with HMG-CoA reductase inhibition.</p>
    Fórmula:C23H34O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:390.51
  • IDH-C227

    CAS:
    <p>IDH-C227 is a selective and potent inhibitor of IDH1R132H that exhibits anticancer activity.</p>
    Fórmula:C30H31FN4O2
    Forma y color:Solid
    Peso molecular:498.59
  • Indolapril hydrochloride

    CAS:
    <p>Indolapril hydrochloride is a nonsulfhydryl angiotensin converting enzyme (ACE) inhibitor with antihypertensive activity.</p>
    Fórmula:C24H35ClN2O5
    Forma y color:Solid
    Peso molecular:467
  • ML368

    CAS:
    <p>ML368 is a selective inhibitor of CYP3A4.</p>
    Fórmula:C26H18N6O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:430.46
  • Glutamamide

    CAS:
    <p>Glutamamide is an anticancer drug.</p>
    Fórmula:C5H11N3O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:145.16
  • PF-06424439

    CAS:
    <p>PF-06424439 is an oral and selective inhibitor of imidazopyridine diacylglycerol acyltransferase 2 (DGAT2) (IC50 of 14 nM).</p>
    Fórmula:C22H26ClN7O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:439.94
  • UK-500001

    CAS:
    <p>UK-500001 is a potent PDE4 inhibitor with robust anti-inflammatory activity.</p>
    Fórmula:C26H24F3N3O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:499.48
  • 9(R)-HODE

    CAS:
    9(R)-HODE, a linoleic acid product, is made by some human/bovine endothelial cells, but its function and forming enzyme are unknown.
    Fórmula:C18H32O3
    Forma y color:Solid
    Peso molecular:296.44
  • JTV-519

    CAS:
    <p>K201 (JTV-519) is a Ca2+-dependent blocker and prevents abnormal Ca(2+) leak from the sarcoplasmic reticulum in the ischemic heart and skeletal muscle (SkM) by</p>
    Fórmula:C25H33ClN2O2S
    Pureza:99.88%
    Forma y color:Solid
    Peso molecular:461.06
  • Riboflavine phosphate

    CAS:
    <p>Riboflavine phosphate (Flavin mononucleotide) is a derivative of Riboflavin.</p>
    Fórmula:C17H21N4O9P
    Pureza:98%
    Forma y color:Solid
    Peso molecular:456.34
  • LY367385

    CAS:
    <p>LY367385 is a highly effective and selective mGluR1a antagonist.</p>
    Fórmula:C10H11NO4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:209.2
  • PTP1B-IN-4

    CAS:
    <p>PTP1B-IN-4 (NUN-17724) is an allosteric PTP1B inhibitor with an IC50 of 8 μM. PTP1B-IN-4 can be used in studies about obesity and diabetes.</p>
    Fórmula:C26H19Br2N3O7S3
    Pureza:98.19%
    Forma y color:Solid
    Peso molecular:741.45
  • ATX inhibitor 5

    CAS:
    ATX inhibitor 5: potent, oral autotaxin blocker, IC50 15.3 nM, curbs CCl4 liver fibrosis.
    Fórmula:C22H18ClF3N6O
    Pureza:99.73%
    Forma y color:Solid
    Peso molecular:474.87
  • IDO1-IN-2

    CAS:
    <p>IDO1-IN-2 is a potent and selective IDO1 inhibitor with IC50s of 81 nM, 59 nM (mouse), and 28 nM (rat), respectively. It has anti-cancer activity.</p>
    Fórmula:C15H17FN6O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:364.33
  • Otamixaban

    CAS:
    Otamixaban (FXV673) is a selective and highly effective Xa inhibitor that inhibits the generation of thrombin and can be used to study acute coronary syndrome.
    Fórmula:C25H26N4O4
    Pureza:98.08%
    Forma y color:Solid
    Peso molecular:446.5
  • Oosponol

    CAS:
    <p>Oosponol is a dopamine beta-hydroxylase inhibitor exhibiting hypotensive effects.</p>
    Fórmula:C11H8O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:220.18
  • Semotiadil recemate fumarate

    CAS:
    Semotiadil recemate fumarate is the recemate of Semotiadil fumarate. Semotiadil fumarate is a novel antagonist of vasoselective Ca2+ channel.
    Fórmula:C33H36N2O10S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:652.71
  • TP-004

    CAS:
    <p>TP-004 is a potent and reversible methionine aminopeptidase 2 (MetAP2) inhibitor (IC50: 6 nM).</p>
    Fórmula:C17H16F3N5O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:363.34
  • Fadrozole HCl hydrate

    CAS:
    <p>Fadrozole is a selective inhibitor of aromatase. It also effective in the treatment of estrogen-dependent diseases including breast cancer.</p>
    Fórmula:C14H13N3ClHH2O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:268.74
  • Quinapril-d5

    CAS:
    <p>Quinapril-d5: An internal standard for quinapril quantification via GC/LC-MS; a prodrug ACE inhibitor for hypertension and heart failure.</p>
    Fórmula:C25H25D5N2O5
    Forma y color:Solid
    Peso molecular:443.55
  • AK-106

    CAS:
    <p>AK-106, or AK106-001616, selectively inhibits cPLA2 and has NSAID-like analgesic effects.</p>
    Fórmula:C26H25N3O3
    Forma y color:Solid
    Peso molecular:427.49
  • CDK2-IN-12

    CAS:
    <p>CDK2-IN-12 (10b), potent CDK2 inhibitor, IC50: 11.6 μM; inhibits hCA I/II/IX/XII, KI: 3534/638.4/44.3/48.8 nM; anti-cancer properties.</p>
    Fórmula:C20H17N9O2S
    Forma y color:Solid
    Peso molecular:447.47
  • L-(-)-threo-3-Hydroxyaspartic acid

    CAS:
    L-(-)-threo-3-Hydroxyaspartic acid is an EAAT1-4 inhibitor/non-transportable EAAT5 inhibitor.
    Fórmula:C4H7NO5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:149.1
  • ATX inhibitor 14

    CAS:
    <p>ATX inhibitor 14, an indole carbamate, potently blocks self-adhesive proteins (IC50: 0.41 nM), aiding fibrosis research.</p>
    Fórmula:C26H26Cl2N4O3S
    Forma y color:Solid
    Peso molecular:545.48
  • SHP2 inhibitor LY6

    CAS:
    <p>SHP2 inhibitor LY6 (LY6) is a potent and selective SHP2 inhibitor (IC50: 9.8 μM) that blocks SHP2-mediated cell signaling and proliferation.</p>
    Fórmula:C30H27Cl2N3O4
    Forma y color:Solid
    Peso molecular:564.46
  • 2614W94

    CAS:
    2614W94 is a selective inhibitor of MAO-A with IC50 of 5 nM and Ki of 1.6 nM.
    Fórmula:C15H11F3O4S
    Pureza:99.6%
    Forma y color:Solid
    Peso molecular:344.31
  • PF-06471553

    CAS:
    <p>PF-06471553 is an effective and selective inhibitor of monoacylglycerol acyltransferase 3 (IC50: 92 nM).</p>
    Fórmula:C23H25N5O4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:467.54
  • Asterriquinol D dimethyl ether

    CAS:
    <p>Asterriquinol D dimethyl ether inhibits mouse myeloma (IC50: 28 μg/mL) and Tritrichomonas foetus.</p>
    Fórmula:C26H24N2O4
    Forma y color:Solid
    Peso molecular:428.48
  • Methazolamide-d6

    CAS:
    <p>Methazolamide-d6 is a GC/LC-MS standard for measuring methazolamide, a glaucoma drug that lowers eye pressure and fluid, reduces seizures, and combats ROS.</p>
    Fórmula:C5H2D6N4O3S2
    Forma y color:Solid
    Peso molecular:242.31
  • PKM2 activator 3

    CAS:
    <p>PKM2 activator 3, with 90 nM AC50, enhances PKM2. It has good Caco-2 permeability, stable, and aids cancer research.</p>
    Fórmula:C15H11ClF2N2O3S
    Forma y color:Solid
    Peso molecular:372.77
  • CD2665

    CAS:
    <p>CD2665 is an orally active antagonist of retinoic acid receptor (RAR). For RARγ and RARβ, the Kis are 110 nM and 306 nM.</p>
    Fórmula:C31H34O5
    Pureza:99.71%
    Forma y color:Solid
    Peso molecular:486.6
  • Benserazide

    CAS:
    <p>Benserazide blocks dopa decarboxylase; paired with levodopa for Parkinson's to boost CNS dopamine levels and lower dosage.</p>
    Fórmula:C10H15N3O5
    Forma y color:Solid
    Peso molecular:257.24
  • RO6806051

    CAS:
    RO6806051 (compound 12) is a potent dual inhibitor of fatty acid binding proteins 4 and 5 (FABP4 and FABP5), exhibiting excellent selectivity and absorption, distribution, metabolism, and excretion (eADME) properties.
    Fórmula:C21H19ClN6
    Forma y color:Solid
    Peso molecular:390.87
  • CDK2-IN-11

    CAS:
    <p>CDK2-IN-11 inhibits CDK2 (IC50: 6.4 μM) and targets hCA II, IX, XII (Ki: 23.4-56.3 nM); suited for cancer research.</p>
    Fórmula:C18H14ClN7O2S
    Forma y color:Solid
    Peso molecular:427.87
  • FABP4/5-IN-5

    CAS:
    <p>FABP4/5-IN-5 (compound D9) serves as a potent inhibitor of both FABP 4 and FABP 5, demonstrating IC50 values of 4.68 μM and 10.72 μM, respectively. It is notably effective in addressing metabolic disorders such as diabetes mellitus [1].</p>
    Fórmula:C23H14ClF2NO4S
    Forma y color:Solid
    Peso molecular:473.88
  • OMDM-4

    CAS:
    <p>OMDM-4 is a selective and metabolically stable anandamide cellular uptake (ACU)inhibitor(Ki of 17.7 μM).</p>
    Fórmula:C29H43NO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:453.66
  • SQ 27786

    CAS:
    <p>SQ 27786 is an inhibitor of ACE.</p>
    Fórmula:C23H25ClN4O7S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:569.05
  • Fexarine

    CAS:
    <p>Fexarine is a potent, selective agonist of farnesoid X receptor.</p>
    Fórmula:C31H31NO5
    Forma y color:Solid
    Peso molecular:497.58
  • PDE-9 inhibitor

    CAS:
    <p>PDE-9 inhibitor is used for treatment neurodegenerative diseases.</p>
    Fórmula:C22H27N5O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:393.48
  • (3S,5R)-Fluvastatin sodium

    CAS:
    (3S,5R)-Fluvastatin sodium: synthetic HMG-CoA reductase inhibitor, IC50 8 nM, boosts vascular cell antioxidant defense.
    Fórmula:C24H26FNNaO4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:434.463
  • Dehydronitrosonisoldipine

    CAS:
    <p>Dehydronitrosonisoldipine blocks SARM1, slows axon decay &amp; cADPR synthesis; useful in neurodegeneration research.</p>
    Fórmula:C20H22N2O5
    Pureza:99.68%
    Forma y color:Solid
    Peso molecular:370.4
  • ML-148

    CAS:
    <p>ML-148 is a selective inhibitor of 15-hydroxy prostaglandin dehydrogenase (15-PGDH, IC50 = 56 nM).</p>
    Fórmula:C20H21N3O
    Pureza:99.88%
    Forma y color:Solid
    Peso molecular:319.4
  • (R)-Bromoenol lactone

    CAS:
    <p>(R)-Bromoenol lactone (BEL) irreversibly inhibits iPLA2γ with 0.6 μM IC50, not affecting iPLA2β unless at 20-30 μM doses.</p>
    Fórmula:C16H13BrO2
    Forma y color:Solid
    Peso molecular:317.18
  • SGK1-IN-2

    CAS:
    <p>SGK1-IN-2 (14h) is a selective inhibitor of SGK1 (serum and glucocorticoid regulated kinase 1)(with an IC50 of 5 nM at 10 μM ATP concentration).</p>
    Fórmula:C17H12Cl2N6O2S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:435.29
  • AVE-8134

    CAS:
    <p>AVE-8134 is an agonist of PPARα. For human and rodent PPARα receptor, the EC50 values are 100 and 3000 nM, respectively.</p>
    Fórmula:C22H23NO5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:381.42
  • Tebuconazole-d9

    CAS:
    <p>Tebuconazole-d9 is a GC/LC-MS standard for quantifying the triazole fungicide tebuconazole, affecting seed/foliar fungi and androgen receptors.</p>
    Fórmula:C16H13ClD9N3O
    Forma y color:Solid
    Peso molecular:316.87
  • MEDS433

    CAS:
    <p>MEDS433 inhibits dihydroorotate dehydrogenase (IC50 1.2 nM) and blocks replication of hCoV-OC43, hCoV-229E, SARS-CoV-2 at nanomolar levels.</p>
    Fórmula:C20H11F4N3O2
    Forma y color:Solid
    Peso molecular:401.31
  • Arcapillin

    CAS:
    <p>Arcapillin, an anticancer agent, induces apoptosis mediated at least in part by the ERS pathway and inhibits hepatoma tumor growth.</p>
    Fórmula:C18H16O8
    Forma y color:Solid
    Peso molecular:360.31
  • ML218

    CAS:
    ML218 is an inhibitor of T-type Ca2+ channels (Cav3.1, Cav3.2, Cav3.3).ML218 inhibits the synaptic activity of subthalamic nucleus (STN) neurons.
    Fórmula:C19H26Cl2N2O
    Pureza:99.2% - 99.45%
    Forma y color:Solid
    Peso molecular:369.33
  • GW844520

    CAS:
    <p>GW844520 is a potent and selective inhibitor of the cytochrome bc1 complex of mitochondrial electron transport in P. falciparum.</p>
    Fórmula:C20H15ClF3NO3
    Forma y color:Solid
    Peso molecular:409.79
  • Loxoprofenol-SRS

    CAS:
    <p>Loxoprofenol-SRS, a potent metabolite of Loxoprofen, is an IV NSAID with enhanced anti-inflammatory and pain relief properties.</p>
    Fórmula:C15H20O3
    Forma y color:Solid
    Peso molecular:248.32
  • SR1555 HCl

    CAS:
    <p>SR1555: A selective RORγ inverse agonist, hinders TH17 cells, key in autoimmune diseases like RA and MS.</p>
    Fórmula:C22H22F6N2O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:460.41
  • Lipoxygenin

    CAS:
    <p>Lipoxygenin: IC50 of 5 μM inhibits 5-LO, hedgehog, TGF-β, activin A, BMP, Wnt signaling, and boosts cardiac marker TnnT in iPSCs.</p>
    Fórmula:C24H22N2O4
    Forma y color:Solid
    Peso molecular:402.44
  • SHP2-IN-5

    CAS:
    <p>SHP2-IN-5 (compound 1) is a non-receptor protein tyrosine phosphatase inhibitor targeting SHP2 with an IC50 value of 97 nM, associated with regulating cell</p>
    Fórmula:C12H8O6
    Forma y color:Solid
    Peso molecular:248.19
  • Safusidenib

    CAS:
    <p>Safusidenib, oral mutant IDH1 inhibitor, selectively targets IDH1R132H/C mutations with IC50 of 15/130 nM; impairs chondrosarcoma growth.</p>
    Fórmula:C25H18Cl3FN2O4
    Forma y color:Solid
    Peso molecular:535.78
  • IHVR-11029

    CAS:
    <p>IHVR-11029 inhibits ER α-glucosidase, combats hemorrhagic fever viruses, and hinders enveloped virus morphogenesis.</p>
    Fórmula:C18H27F2NO5
    Forma y color:Solid
    Peso molecular:375.41
  • Ro 41-0960

    CAS:
    <p>Ro 41-0960 is used as a reversible and orally-active COMT-inhibitor.</p>
    Fórmula:C13H8FNO5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:277.2
  • Diapocynin

    CAS:
    <p>Diapocynin (Dehydrodiacetovanillone), a dimer of Apocynin, acts as an orally administered inhibitor of NADPH oxidase.</p>
    Fórmula:C18H18O6
    Forma y color:Solid
    Peso molecular:330.33
  • TPN729MA

    CAS:
    <p>TPN729MA, a potent PDE5 inhibitor, IC50: 2.28 nM, targets erectile dysfunction research.</p>
    Fórmula:C29H40N6O8S
    Forma y color:Solid
    Peso molecular:632.73
  • SAHO

    CAS:
    <p>SAHO is a methyl donor cleaved by SAM enzymes into adenosylhomocysteine and thioadenosine derivatives.</p>
    Fórmula:C14H20N6O6S
    Forma y color:Solid
    Peso molecular:400.41
  • BMP-22

    CAS:
    <p>BMP-22 selectively inhibits autotaxin (IC50=170 nM), blocks LPA production and MM1 cell invasion, and reduces lung metastases in mice at 0.5 mg/kg/day.</p>
    Fórmula:C22H39O3P
    Forma y color:Solid
    Peso molecular:382.52
  • GlcN-6-P Synthase-IN-1

    CAS:
    <p>'GlcN-6-P Synthase-IN-1, IC50 3.47 μM, inhibits GlcN-6-P synthase &amp; CYP3A4. Has antimicrobial activity and CNS penetration.'</p>
    Fórmula:C20H21N7S
    Forma y color:Solid
    Peso molecular:391.49
  • PF 4800567 hydrochloride

    CAS:
    <p>casein kinase 1ε inhibitor</p>
    Fórmula:C17H19Cl2N5O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:396.27
  • McN3716

    CAS:
    <p>McN3716 is a carnitine palmitoyltransferase I (CPT-1) inhibitor for the study of metabolic diseases.</p>
    Fórmula:C18H34O3
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:298.46
  • ATX inhibitor 20

    CAS:
    <p>ATX inhibitor 20 is a potent inhibitor of ATX (IC50: 2.3 nM).</p>
    Fórmula:C31H34FN5O3
    Forma y color:Solid
    Peso molecular:543.63
  • Ro-15-2041

    CAS:
    Ro 15-2041 is a selective inhibitor of platelet phosphodiesterase, with antithrombotic properties.
    Fórmula:C12H12BrN3O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:294.15
  • NCX899

    CAS:
    <p>NCX899 shows inhibitory activity against angiotensin-converting enzyme (ACE) activity.</p>
    Fórmula:C23H33N3O8
    Pureza:98%
    Forma y color:Solid
    Peso molecular:479.52
  • 20-HC-Me-Pyrrolidine


    <p>20-HC-Me-Pyrrolidine is a potent Aster protein inhibitor that blocks the ability of Aster proteins to bind and transfer cholesterol.</p>
    Fórmula:C28H47NO2
    Pureza:99.99%
    Forma y color:Solid
    Peso molecular:429.68
  • Sp-Cyclic AMPS (sodium salt)

    CAS:
    <p>Sp-cAMPS Na salt activates PKA I/II and competitively inhibits PDE3A (Ki: 47.6 μM), also binds PDE10 GAF (EC50: 40 μM).</p>
    Fórmula:C10H12N5NaO5PS
    Forma y color:Solid
    Peso molecular:367.25
  • BTX161

    CAS:
    <p>BTX161: potent CKIα degrader, surpasses Lenalidomide in AML, triggers DDR + p53, stabilizes MDM2.</p>
    Fórmula:C15H16N2O3
    Forma y color:Solid
    Peso molecular:272.3
  • ZM223

    CAS:
    <p>ZM223 is an inhibitor of NEDD8 activating enzyme (NAE).</p>
    Fórmula:C23H17F3N4O2S2
    Pureza:99.73%
    Forma y color:Solid
    Peso molecular:502.53
  • N-Methylmoranoline

    CAS:
    N-Methylmoranoline is an inhibitor of α-glucosidase.
    Fórmula:C7H15NO4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:177.2
  • Glyoxalase I inhibitor 7

    CAS:
    <p>Glyoxalase I inhibitor 7 (Compound 6) is a potent inhibitor of glyoxalase I (Glo-I) with an IC50 of 3.65 μM. It exhibits potential as an anticancer agent [1].</p>
    Fórmula:C17H16N4O3S
    Forma y color:Solid
    Peso molecular:356.4
  • hCAXII-IN-5

    CAS:
    <p>hCAXII-IN-5, or compound 6o, is a potent, selective hCAXII inhibitor with Ki values: hCAI &amp; II &gt;10000, hCAIX 286.1, hCAXII 1.0 nM.</p>
    Fórmula:C23H22N2O4
    Forma y color:Solid
    Peso molecular:390.43
  • M77976

    CAS:
    <p>M77976 inhibits PDK4 with an IC50 of 648 μM, targeting obesity and diabetes research.</p>
    Fórmula:C17H16N2O3
    Pureza:99.43%
    Forma y color:Solid
    Peso molecular:296.32
  • Indoleacetyl phenylalanine

    CAS:
    <p>Indoleacetyl phenylalanine is an indole-acetyl-amino acid involved in regulating auxin activity.</p>
    Fórmula:C19H18N2O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:322.36
  • Acetylhydrolase-IN-1

    CAS:
    Acetylhydrolase-IN-1 is an inhibitor of the esterase 1-Alkyl-2-acetylglycerophosphocholine (Alkylacetyl-GPC: acetylhydrolase).
    Fórmula:C23H48NO7P
    Pureza:98%
    Forma y color:Solid
    Peso molecular:481.6
  • L-Canaline

    CAS:
    L-Canaline is a nonprotein amino acid with IC50 of 297 nM against malaria, anticancer properties, and blocks ornithine aminotransferase.
    Fórmula:C4H10N2O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:134.13
  • hDHODH-IN-11

    CAS:
    <p>hDHODH-IN-11: potent hDHODH inhibitor, IC50 7.2 nM, low cytotoxicity, for AML research.</p>
    Fórmula:C24H23N3O3
    Forma y color:Solid
    Peso molecular:401.46
  • VP3.15

    CAS:
    <p>VP3.15 is an orally bioavailable and CNS-penetrant dual inhibitor of phosphodiesterase (PDE)7- GSK3 (IC50s: 1.59 μM and 0.88 μM for PDE7 and GSK-3).</p>
    Fórmula:C20H22N4OS
    Pureza:98%
    Forma y color:Solid
    Peso molecular:366.48
  • Nampt activator-3

    CAS:
    <p>NAMPT activator-3: a NAT derivative, EC50 of 2.6 μM, KD 132 nM, protects cells, prevents FK866 toxicity, and is neuroprotective in CIPN mice.</p>
    Fórmula:C19H20N2O3
    Forma y color:Solid
    Peso molecular:324.37
  • Glyoxalase I inhibitor 4

    CAS:
    <p>Glyoxalase I inhibitor 4 is a potent inhibitor of glyoxalase I (GLO1) (Ki: 10 nM).</p>
    Fórmula:C17H21IN4O8S
    Forma y color:Solid
    Peso molecular:568.34
  • p18SMI-21

    CAS:
    <p>p18SMI-21 is a novel INK4C inhibitor. It also specifically blocking the bioactivity of p18 protein.</p>
    Fórmula:C10H14N2O4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:258.29
  • Anti-hyperglycemic agent-1

    CAS:
    <p>Anti-hyperglycemic agent 1 is a potent inhibitor of alpha-glucosidase (IC50: 0.53 μM). anti-Hyperglycemic agent 1 can be used to study diabetes.</p>
    Fórmula:C20H15BrN2O3
    Forma y color:Solid
    Peso molecular:411.25
  • Trimoxamine hydrochloride

    CAS:
    <p>Trimoxamine hydrochloride is an antihypertensive.</p>
    Fórmula:C15H24ClNO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:301.81
  • PSB069

    CAS:
    NTPDase inhibitor
    Fórmula:C20H13ClN2NaO5S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:451.84
  • SWE101

    CAS:
    <p>SWE101 is a potent human and rat soluble epoxide hydrolase (sEH)-P inhibitor(IC50s of 4 μM and 2.8 μM, respectively).</p>
    Fórmula:C19H15Cl2NO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:376.23
  • MAO-IN-1

    CAS:
    MAO-IN-1 is a potent monoamine oxidase B (MAO B) inhibitor (IC50: 20 nM) for the study of neurologically related diseases.
    Fórmula:C17H19ClO4
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:322.78
  • RORγt agonist 1

    CAS:
    <p>RORγt agonist 1 is a potent, orally bioavailable agonist of RORγt(EC50 of 20.8 nM).</p>
    Fórmula:C24H17F6NO5S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:545.45
  • HZ52

    CAS:
    <p>HZ52: Potent reversible 5-LO inhibitor; IC50 0.7 μM; blocks LTs in human leukocytes.</p>
    Fórmula:C24H26ClN3O2S
    Forma y color:Solid
    Peso molecular:456
  • Enpp-1-IN-10

    CAS:
    <p>Enpp-1-IN-10 inhibits ENPP1 with 3.866 μM Ki, useful in cancer research.</p>
    Fórmula:C13H12N6OS
    Forma y color:Solid
    Peso molecular:300.34
  • VU0155056

    CAS:
    <p>VU0155056 is a dual PLD1/2 inhibitor with IC50 &lt; 1 µM in cellular assays, inhibits breast cancer cell invasion.</p>
    Fórmula:C25H26N4O2
    Pureza:98.6% - 99.15%
    Forma y color:Solid
    Peso molecular:414.5
  • DNS-8254

    CAS:
    <p>DNS-8254: Potent, selective PDE2 inhibitor, enhances memory (IC50=8 nM), effective in rat memory tests.</p>
    Fórmula:C18H15BrF3N5O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:454.24
  • ATX inhibitor 19

    CAS:
    <p>ATX inhibitor 19 is a potent inhibitor of ATX (IC50: 156 nM).</p>
    Fórmula:C28H33ClN6O2S
    Forma y color:Solid
    Peso molecular:553.12
  • Propaquizafop

    CAS:
    <p>Propaquizafop, a phenoxyisopropionic acid derivative, is used as a herbicide.</p>
    Fórmula:C22H22ClN3O5
    Pureza:98%
    Forma y color:Colourless-To-Brown Crystals
    Peso molecular:443.88
  • Disulfamide

    CAS:
    <p>Disulfamide: Oral carbonic anhydrase inhibitor, IC50 0.07 μM, diuretic by blocking Na+/HCO3- reabsorption.</p>
    Fórmula:C7H9ClN2O4S2
    Pureza:98.1%
    Forma y color:Solid
    Peso molecular:284.74
  • Flutolanil

    CAS:
    <p>Flutolanil: a fungicide targeting R. solani in rice, toxic to zebrafish.</p>
    Fórmula:C17H16F3NO2
    Forma y color:Solid
    Peso molecular:323.31
  • Lp-PLA2-IN-4

    CAS:
    <p>Lp-PLA2-IN-4, a potent inhibitor of Lp-PLA2/PAF-AH, may target Alzheimer's, atherosclerosis. (WO2021228159A1, Compound 38)</p>
    Fórmula:C23H18F5N3O4
    Forma y color:Solid
    Peso molecular:495.4
  • FCE 28654

    CAS:
    <p>FCE 28654 is a water-soluble acyl-CoA inhibitor.</p>
    Fórmula:C25H35N2O7P
    Forma y color:Solid
    Peso molecular:506.53
  • Zidovudine glucuronide

    CAS:
    <p>Zidovudine glucuronide: an NRTI antiretroviral for HIV/AIDS treatment; blocks HIV reverse transcriptase, stops viral DNA formation.</p>
    Fórmula:C16H21N5O10
    Forma y color:Solid
    Peso molecular:443.37