
Metabolismo
Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.
Subcategorías de "Metabolismo"
- AhR(41 productos)
- Aminopeptidasa(73 productos)
- CETP(20 productos)
- Anhídrido carbónico(184 productos)
- Caseína quinasa(136 productos)
- DHFR(34 productos)
- Descarboxilasa(4 productos)
- Deshidrogenasa(288 productos)
- FAAH(65 productos)
- FXR(59 productos)
- Factor Xa(83 productos)
- Ácido graso sintasa(36 productos)
- Ferroptosis(218 productos)
- GR(3 productos)
- GSNOR(4 productos)
- Glucoquinasa(56 productos)
- HIF / HIF Prolilhidroxilasa(142 productos)
- HMG-CoA reductasa(34 productos)
- Hidroxilasa(34 productos)
- IDO(84 productos)
- LDL(8 productos)
- Lipasa(104 productos)
- Lípido(61 productos)
- Lipoxigenasa(133 productos)
- MAO(87 productos)
- MPO(2 productos)
- NAMPT(38 productos)
- P450(6 productos)
- PAI-1(26 productos)
- PDE(166 productos)
- PED(1 productos)
- PKM(15 productos)
- PPAR(167 productos)
- Fosfolipasa(82 productos)
- ROR(43 productos)
- Receptor de retinoides(28 productos)
- SGK(12 productos)
- Tiorredoxina(12 productos)
- Transferasa(29 productos)
- Transportador(43 productos)
- UGT(4 productos)
- Inhibidores de la xantina oxidasa (XO)(9 productos)
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Se han encontrado 9007 productos de "Metabolismo"
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Enterostatin(human,mouse,rat) TFA
Enterostatin TFA, a pentapeptide from the intestine, reduces fat intake and body fat.Fórmula:C23H37F3N8O8Peso molecular:610.58Xenin
CAS:Xenin is a 25 amino acid peptide that has been identified in human gastric mucosa in the search for a counterpart to the amphibian octapeptide xenopsin.Fórmula:C139H224N38O32SPureza:98%Forma y color:SolidPeso molecular:2971.5719R(20S)-EpDPA
CAS:19R(20S)-EpDPA: oxylipin, DHA metabolite via CYPs, blocks calcium-induced beats in rat heart cells.Fórmula:C22H32O3Forma y color:SolidPeso molecular:344.495Hypusine HCl
CAS:Hypusine HCl: a unique amino acid in eukaryotes/archaea, absent in bacteria; only in eIF5A protein.Fórmula:C10H25Cl2N3O3Forma y color:SolidPeso molecular:306.23CRT0063465
CRT0063465 is a ligand for both human Phosphoglycerate Kinase 1 (PGK1) and the stress sensor protein DJ-1, exhibiting a dissociation constant (Kd) of 24 μM forForma y color:Odour SolidLEI110
CAS:LEI110 inhibits PLA2G16 and HRASLS enzymes, Ki 20 nM, selectively targets related thiol hydrolases.Fórmula:C25H23F3N2O3Pureza:98.66% - 98.8%Forma y color:SolidPeso molecular:456.46MAGL-IN-21
<p>MAGL-IN-21 (Compound (S)-6) is a selective inhibitor of monoacylglycerol lipase (MAGL) with an IC50 of 1.59 nM.</p>Fórmula:C20H24ClFN2O4Forma y color:SolidPeso molecular:410.8674-Hydroxy Atorvastatin calcium salt
CAS:<p>4-Hydroxy Atorvastatin calcium salt is metabolised by cytochrome P450 CYP3A4 and has antimicrobial and anti-microbial activity.</p>Fórmula:C66H68CaF2N4O12Forma y color:SolidPeso molecular:1187.34hCAII/XII-IN-1
hCAII/XII-IN-1 (compound 4l) is a potent inhibitor of hCAXII and hCAII, with Ki values of 8.4 nM and 9.4 nM, respectively. It plays a significant role in cancer research.Fórmula:C22H20N4O6S2Forma y color:SolidPeso molecular:500.547hCAII/IX-IN-1
<p>hCAII/IX-IN-1 (compound 4o) is a potent inhibitor of hCAII and hCAIX, with Ki values of 7.4 nM and 7.0 nM, respectively. It plays a significant role in cancer research.</p>Fórmula:C23H22N4O7S2Forma y color:SolidPeso molecular:530.573CA IX/VEGFR-2-IN-3
<p>CAIX/VEGFR-2-IN-3 (Compound 6i) is an inhibitor of Carbonic Anhydrase IX and VEGFR-2, with IC50 values of 41 and 48 nM, respectively. It exhibits anticancer activity by inhibiting the growth of MCF-7 breast cancer cells (IC50 of 22.33 μM) and mouse fibroblast cell line 3T3, where cell viability is reduced to below 40% at a concentration of 100 μM. This compound is applicable for research in the field of cancer treatment.</p>Fórmula:C19H16ClN3O5S2Forma y color:SolidPeso molecular:465.93α-Glucosidase-IN-78
<p>α-Glucosidase-IN-78 (Compound 12m) is a reversible competitive inhibitor of α-glucosidase (α-glucosidase) with an IC50 of 6.0 μM. Due to its blood sugar-lowering properties, α-Glucosidase-IN-78 is applicable in diabetes research.</p>Fórmula:C28H22N8O4Forma y color:SolidPeso molecular:534.526LDHA-IN-8
CAS:<p>LDHA-IN-8, an inhibitor, inhibits the proliferation of pancreatic and lung cancer cells, decreasing the intracellular lactate content and increasing ROS levels.</p>Fórmula:C15H14N4O2Pureza:99.73%Forma y color:SolidPeso molecular:282.3Speract
CAS:<p>Speract, a peptide from sea urchin eggs, regulates sperm motility and stimulates sperm mitochondrial metabolism.</p>Fórmula:C38H57N11O14Pureza:98%Forma y color:SolidPeso molecular:891.93Impurity C of Calcitriol
CAS:<p>Impurity C of Calcitriol is an impurity of Calcitriol.Impurity C of Calcitriol is used in the synthesis of vitamin D3.</p>Fórmula:C35H49N3O5Pureza:98%Forma y color:SolidPeso molecular:591.78Ercalcitriol
CAS:<p>Ercalcitriol, active Vitamin D2 metabolite, boosts immunity by regulating CAMP and DEFB4 genes against infections.</p>Fórmula:C28H44O3Pureza:99.02%Forma y color:SolidPeso molecular:428.65Nε,Nε,Nε-Trimethyllysine chloride
CAS:Nε,Nε,Nε-Trimethyllysine chloride (Lys(Me)3-OH Chloride) is a methylated derivative of the amino acid lysine and a component of histone proteins.Fórmula:C9H21ClN2O2Pureza:99.83%Forma y color:SolidPeso molecular:224.7311β-HSD1 inibitor 19
CAS:3-chloro-4-sulfonyl-Benzonitrile inhibits hHSD1/mHSD1, IC50: 16nM/10nM.Fórmula:C19H16ClF4N3O2SPureza:99.58%Forma y color:SoildPeso molecular:461.86

