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Metabolismo

Metabolismo

Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.

Subcategorías de "Metabolismo"

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Se han encontrado 8626 productos de "Metabolismo"

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  • Fondaparinux sodium

    CAS:
    <p>Fondaparinux sodium (SR-90107A) is an antithrombin-dependent factor Xa inhibitor with antithrombotic activity.</p>
    Fórmula:C31H43N3Na10O49S8
    Pureza:98% - >99.99%
    Forma y color:Solid
    Peso molecular:1728.08
  • GNE-617 hydrochloride

    CAS:
    <p>GNE-617 hydrochloride is a specific inhibitor of NAMPT and inhibits NAMPT activity (IC50: 5 nM).</p>
    Fórmula:C21H16ClF2N3O3S
    Forma y color:Solid
    Peso molecular:463.88
  • Edoxaban Tosylate Monohydrate

    CAS:
    <p>Edoxaban(DU-176) is an oral factor Xa (FXa) inhibitor in clinical development for stroke prevention.</p>
    Fórmula:C31H40ClN7O8S2
    Pureza:99.86% - 99.91%
    Forma y color:Solid
    Peso molecular:738.27
  • MP07-66

    CAS:
    MP07-66 is a novel FTY720-analog devoid of immunosuppressive effects leads to the reactivation of PP2A, which in turn triggers apoptosis of CLL cells.
    Fórmula:C19H33NO3
    Pureza:95.678%
    Forma y color:Solid
    Peso molecular:323.47
  • Ivosidenib

    CAS:
    <p>Ivosidenib (AG-120) is an oral IDH1 inhibitor targeting mutated IDH1 to reduce 2-hydroxyglutarate and hinder tumor growth.</p>
    Fórmula:C28H22ClF3N6O3
    Pureza:98.71% - 99.98%
    Forma y color:Solid
    Peso molecular:582.96
  • Tetradecylthioacetic acid

    CAS:
    <p>Synthetic fatty acid TTA has β-sulfur, resists β-oxidation, and activates PPARs, especially PPARα.</p>
    Fórmula:C16H32O2S
    Pureza:99.93%
    Forma y color:Solid
    Peso molecular:288.49
  • Fmoc-Gly-Thr(psi(Me,Me)pro)-OH

    CAS:
    <p>Fmoc-Gly-Thr(psi(Me,Me)pro)-OH is a polypeptide composed of two amino acids.</p>
    Fórmula:C24H26N2O6
    Pureza:97.35%
    Forma y color:Solid
    Peso molecular:438.47
  • LB-60-OF61 hydrochloride

    CAS:
    <p>LB-60-OF61 hydrochloride is a potent NAMPT enzyme inhibitor with cytotoxic effects, targeting MYC-overexpressing cell lines.</p>
    Fórmula:C29H31ClN6O2
    Forma y color:Solid
    Peso molecular:531.06
  • SR1001

    CAS:
    <p>SR 1001 is an inverse agonist for RORα/RORγ (Kis: 172/111 nM).</p>
    Fórmula:C15H13F6N3O4S2
    Pureza:98.93%
    Forma y color:Solid
    Peso molecular:477.4
  • PQ-10

    CAS:
    <p>PQ-10 (A-844337) is a PDE-10 inhibitor. PQ-10 induces brain glucose metabolism patterns, which may be a potential translational biomarker.</p>
    Fórmula:C22H21N5O3
    Pureza:99.86%
    Forma y color:Solid
    Peso molecular:403.43
  • TETRAHYDROPIPERINE

    CAS:
    <p>Tetrahydropiperine (Cosmoperine) is a natural product derived from piperine, can be used to treat convulsion, epilepsy, relieve pain, and control insects.</p>
    Fórmula:C17H23NO3
    Pureza:98.04% - 99.61%
    Forma y color:Off-White Low Melting Solid With Characteristic Odour
    Peso molecular:289.37
  • Varespladib

    CAS:
    <p>Varespladib (LY315920) inhibits hnsPLA2 effectively (IC50=7 nM), studied for sickle cell, VOC, and acute coronary syndrome.</p>
    Fórmula:C21H20N2O5
    Pureza:99.97%
    Forma y color:Solid
    Peso molecular:380.39
  • T863

    CAS:
    T-863(DGAT-1 inhibitor) is an orally active, selective and potent DGAT1 (Acyl-CoA:diacylglycerol acyltransferase 1) inhibitor that interacts with the acyl-CoA
    Fórmula:C22H26N4O3
    Pureza:98.66% - 99.88%
    Forma y color:Solid
    Peso molecular:394.47
  • Genz-123346 free base

    CAS:
    Genz 123346 is an inhibitor of GL1 synthase that blocks the conversion of ceramide to GL1.
    Fórmula:C24H38N2O4
    Pureza:99.41%
    Forma y color:Solid
    Peso molecular:418.57
  • Mirogabalin

    CAS:
    <p>Mirogabalin (DS5565) is a calcium channel blocker with analgesic effects.</p>
    Fórmula:C12H19NO2
    Pureza:98.57%
    Forma y color:Solid
    Peso molecular:209.28
  • Telaglenastat

    CAS:
    <p>Telaglenastat (CB 839) (IC50 of 24 nM), an effective, specific, and oral inhibitor, which is bioavailable glutaminase, for recombinant human GAC.</p>
    Fórmula:C26H24F3N7O3S
    Pureza:97.57% - 99.89%
    Forma y color:Solid
    Peso molecular:571.57
  • JNJ-42041935

    CAS:
    <p>JNJ-42041935 (HIF-PHD Inhibitor II) is a potent (pKi = 7.3-7.9), 2-oxoglutarate competitive, reversible, and selective inhibitor of PHD enzymes.</p>
    Fórmula:C12H6ClF3N4O3
    Pureza:99.58% - ≥95%
    Forma y color:Solid
    Peso molecular:346.65
  • Pargyline

    CAS:
    <p>Pargyline (Pargylamine) is a monoamine oxidase inhibitor with antihypertensive properties.</p>
    Fórmula:C11H13N
    Pureza:95.64% - 97.21%
    Forma y color:Solid
    Peso molecular:159.23
  • PfDHODH-IN-2

    CAS:
    <p>PfDHODH-IN-2: powerful antimalarial, blocks PfDHODH (IC50: 1.11 μM), for malaria research.</p>
    Fórmula:C13H12ClNO3S
    Pureza:98.9%
    Forma y color:Solid
    Peso molecular:297.76
  • Pentamidine isethionate

    CAS:
    <p>Pentamidine isethionate (Pentamidine diisethionate) is a synthetic amidine derivative, Pentamidine Isethionate is an antiprotozoal and antifungal agent.</p>
    Fórmula:C23H36N4O10S2
    Pureza:98% - 99.83%
    Forma y color:Slight Butyric Odor Very Bitter Taste Ph (5% Aqueous Solution) 4 5-6 5 (Ntp 1992)
    Peso molecular:592.68