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Metabolismo

Metabolismo

Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.

Subcategorías de "Metabolismo"

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Se han encontrado 8595 productos de "Metabolismo"

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  • JZL 184

    CAS:
    <p>JZL 184 is a potent and selective inhibitor of MAGL with IC50 of 8 nM and 4 μM for inhibition of MAGL and FAAH in mouse brain membranes respectively.</p>
    Fórmula:C27H24N2O9
    Pureza:97.56% - 99.31%
    Forma y color:Solid
    Peso molecular:520.49
  • LOX-IN-3 dihydrochloride

    CAS:
    <p>LOX-IN-3 dihydrochloride is an inhibitor of lysyl oxidase (LOX).</p>
    Fórmula:C13H15Cl2FN2O2S
    Pureza:99.96%
    Forma y color:Solid
    Peso molecular:353.24
  • Cobicistat

    CAS:
    <p>Cobicistat (GS-9350): A carbamate, thiazole derivative, and CYP3A inhibitor used to boost anti-HIV drugs for treating HIV.</p>
    Fórmula:C40H53N7O5S2
    Pureza:97.36% - 99.62%
    Forma y color:Solid
    Peso molecular:776.02
  • Ethyl potassium malonate

    CAS:
    <p>Ethyl potassium malonate, a competitive inhibitor of the enzyme succinate dehydrogenase, acts as a precursor to produce (trimethylsilyl)ethyl malonate, which is</p>
    Fórmula:C5H7KO4
    Pureza:99.71%
    Forma y color:White Crystals Or Powder
    Peso molecular:170.21
  • Glycerol 3-phosphate biscyclohexylammonium salt

    CAS:
    <p>Glycerol 3-phosphate biscyclohexylammonium salt is an endogenous metabolite produced by cytosolic glycerol 3-phosphate dehydrogenase pathway.</p>
    Fórmula:C15H35N2O6P
    Pureza:99.94%
    Forma y color:Solid
    Peso molecular:370.42
  • SR 16832

    CAS:
    <p>SR 16832: Dual-site PPARγ inhibitor; outperforms GW 9662, T 0070907 in ligand binding, transcription inhibition.</p>
    Fórmula:C17H12ClN3O4
    Pureza:99.6%
    Forma y color:Solid
    Peso molecular:357.75
  • SR3335

    CAS:
    <p>SR3335 (ML 176) is a selective inverse agonist of RORα, competitively inhibiting the binding of 25-hydroxycholesterol to the ligand binding domain (Ki: 220 nM).</p>
    Fórmula:C13H9F6NO3S2
    Pureza:99.77%
    Forma y color:Solid
    Peso molecular:405.34
  • AZ876

    CAS:
    <p>AZ876 is a potent, highly selective LXR agonist with Ki/EC50 of 7/6 nM and 11/73 nM for hLXRα and hLXRβ respectively.</p>
    Fórmula:C24H29N3O3S
    Pureza:99.86%
    Forma y color:Solid
    Peso molecular:439.57
  • ARM1

    CAS:
    <p>ARM1 is a potent inhibitor of aminopeptidase and epoxide hydrolase. The IC50 values are 7.61 µM for aminopeptidase and 12.4 µM for epoxide hydrolase.</p>
    Fórmula:C16H14N2S
    Pureza:99.36%
    Forma y color:Solid
    Peso molecular:266.36
  • Cecropin P1, porcine acetate


    <p>Cecropin P1, porcine acetate is an antibacterial peptide found in Hyalophora cecropia and pig intestine.</p>
    Fórmula:C149H257N45O45
    Pureza:95.4% - 98%
    Forma y color:Solid
    Peso molecular:3398.91
  • Bempedoic acid

    CAS:
    <p>Bempedoic acid (ETC1002) is an orally available, once-daily LDL-C lowering small molecule designed to lower elevated levels of LDL-C.</p>
    Fórmula:C19H36O5
    Pureza:99.85% - 99.94%
    Forma y color:Solid
    Peso molecular:344.49
  • AGI-5198

    CAS:
    <p>AGI-5198 (IDH-C35) is a highly effective and specific inhibitor of IDH1 R132H/R132C mutants (IC50: 0.07/0.16 μM).</p>
    Fórmula:C27H31FN4O2
    Pureza:97.37% - 99.23%
    Forma y color:Solid
    Peso molecular:462.56
  • 1-Ethynylpyrene

    CAS:
    <p>1-Ethynylpyrene is an aryl acetylenic inhibitor of CYTP450 1A1(IC50=0.18 μM), 1A2(IC50 = 0.32 μM), and 2B1(IC50 = 0.04 μM).</p>
    Fórmula:C18H10
    Pureza:98.48%
    Forma y color:Solid
    Peso molecular:226.27
  • Suvecaltamide

    CAS:
    <p>Suvecaltamide (MK-8998) as potent inhibitors of T-type calcium channels.</p>
    Fórmula:C20H23F3N2O2
    Pureza:99.29% - 99.70%
    Forma y color:Solid
    Peso molecular:380.4
  • Diflubenzuron

    CAS:
    <p>Diflubenzuron (Larvakil) is a benzoyl-urea insecticide, found to be a potent inhibitor of melanosome synthesis in mouse melanoma cells.</p>
    Fórmula:C14H9ClF2N2O2
    Pureza:99.58% - 99.96%
    Forma y color:Colorless Crystals Diflubenzuron Is A Colorless To Yellow Crystals Used As A Selective Insecticide
    Peso molecular:310.68
  • Ivosidenib

    CAS:
    <p>Ivosidenib (AG-120) is an oral IDH1 inhibitor targeting mutated IDH1 to reduce 2-hydroxyglutarate and hinder tumor growth.</p>
    Fórmula:C28H22ClF3N6O3
    Pureza:98.71% - 99.98%
    Forma y color:Solid
    Peso molecular:582.96
  • Carbamazepine 10,11-epoxide

    CAS:
    <p>Carbamazepine 10,11-epoxide, an active metabolite with anticonvulsant properties, is created by CYP3A4 and CYP2C8.</p>
    Fórmula:C15H12N2O2
    Pureza:98.64% - 99.75%
    Forma y color:Solid
    Peso molecular:252.27
  • AMG-3969

    CAS:
    <p>AMG-3969 is an effective glucokinase-glucokinase regulatory protein interaction (GK-GKRP) disruptor (IC50: 4 nM).</p>
    Fórmula:C21H20F6N4O3S
    Pureza:99.65%
    Forma y color:Solid
    Peso molecular:522.46
  • DHBP dibromide

    CAS:
    <p>DHBP dibromide (1,1'-DI-N-HEPTYL-4,4'-BIPYRIDINIUM DIBRO) is calcium release and a muscle relaxant inhibitor.</p>
    Fórmula:C24H38Br2N2
    Pureza:99.73%
    Forma y color:Yellow To Yellow-Green Powder Or Flakes
    Peso molecular:514.38
  • Ciprofibrate

    CAS:
    <p>Ciprofibrate (Win35833) is a fibrate derivative with antilipidemic activity.</p>
    Fórmula:C13H14Cl2O3
    Pureza:99.63% - >99.99%
    Forma y color:White Or Almost White Crystalline Powder
    Peso molecular:289.15