
Metabolismo
Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.
Subcategorías de "Metabolismo"
- AhR(41 productos)
- Aminopeptidasa(67 productos)
- CETP(18 productos)
- Anhídrido carbónico(177 productos)
- Caseína quinasa(130 productos)
- DHFR(32 productos)
- Descarboxilasa(4 productos)
- Deshidrogenasa(267 productos)
- FAAH(63 productos)
- FXR(58 productos)
- Factor Xa(80 productos)
- Ácido graso sintasa(32 productos)
- Ferroptosis(215 productos)
- GR(3 productos)
- GSNOR(3 productos)
- Glucoquinasa(53 productos)
- HIF / HIF Prolilhidroxilasa(142 productos)
- HMG-CoA reductasa(32 productos)
- Hidroxilasa(30 productos)
- IDO(82 productos)
- LDL(8 productos)
- Lipasa(96 productos)
- Lípido(59 productos)
- Lipoxigenasa(124 productos)
- MAO(87 productos)
- MPO(2 productos)
- NAMPT(36 productos)
- P450(6 productos)
- PAI-1(25 productos)
- PDE(166 productos)
- PED(1 productos)
- PKM(15 productos)
- PPAR(164 productos)
- Fosfolipasa(82 productos)
- ROR(42 productos)
- Receptor de retinoides(29 productos)
- SGK(11 productos)
- Tiorredoxina(12 productos)
- Transferasa(30 productos)
- Transportador(42 productos)
- UGT(4 productos)
- Inhibidores de la xantina oxidasa (XO)(9 productos)
Mostrar 34 subcategorías más
Se han encontrado 8595 productos de "Metabolismo"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
JZL 184
CAS:<p>JZL 184 is a potent and selective inhibitor of MAGL with IC50 of 8 nM and 4 μM for inhibition of MAGL and FAAH in mouse brain membranes respectively.</p>Fórmula:C27H24N2O9Pureza:97.56% - 99.31%Forma y color:SolidPeso molecular:520.49LOX-IN-3 dihydrochloride
CAS:<p>LOX-IN-3 dihydrochloride is an inhibitor of lysyl oxidase (LOX).</p>Fórmula:C13H15Cl2FN2O2SPureza:99.96%Forma y color:SolidPeso molecular:353.24Cobicistat
CAS:<p>Cobicistat (GS-9350): A carbamate, thiazole derivative, and CYP3A inhibitor used to boost anti-HIV drugs for treating HIV.</p>Fórmula:C40H53N7O5S2Pureza:97.36% - 99.62%Forma y color:SolidPeso molecular:776.02Ethyl potassium malonate
CAS:<p>Ethyl potassium malonate, a competitive inhibitor of the enzyme succinate dehydrogenase, acts as a precursor to produce (trimethylsilyl)ethyl malonate, which is</p>Fórmula:C5H7KO4Pureza:99.71%Forma y color:White Crystals Or PowderPeso molecular:170.21Glycerol 3-phosphate biscyclohexylammonium salt
CAS:<p>Glycerol 3-phosphate biscyclohexylammonium salt is an endogenous metabolite produced by cytosolic glycerol 3-phosphate dehydrogenase pathway.</p>Fórmula:C15H35N2O6PPureza:99.94%Forma y color:SolidPeso molecular:370.42SR 16832
CAS:<p>SR 16832: Dual-site PPARγ inhibitor; outperforms GW 9662, T 0070907 in ligand binding, transcription inhibition.</p>Fórmula:C17H12ClN3O4Pureza:99.6%Forma y color:SolidPeso molecular:357.75SR3335
CAS:<p>SR3335 (ML 176) is a selective inverse agonist of RORα, competitively inhibiting the binding of 25-hydroxycholesterol to the ligand binding domain (Ki: 220 nM).</p>Fórmula:C13H9F6NO3S2Pureza:99.77%Forma y color:SolidPeso molecular:405.34AZ876
CAS:<p>AZ876 is a potent, highly selective LXR agonist with Ki/EC50 of 7/6 nM and 11/73 nM for hLXRα and hLXRβ respectively.</p>Fórmula:C24H29N3O3SPureza:99.86%Forma y color:SolidPeso molecular:439.57ARM1
CAS:<p>ARM1 is a potent inhibitor of aminopeptidase and epoxide hydrolase. The IC50 values are 7.61 µM for aminopeptidase and 12.4 µM for epoxide hydrolase.</p>Fórmula:C16H14N2SPureza:99.36%Forma y color:SolidPeso molecular:266.36Cecropin P1, porcine acetate
<p>Cecropin P1, porcine acetate is an antibacterial peptide found in Hyalophora cecropia and pig intestine.</p>Fórmula:C149H257N45O45Pureza:95.4% - 98%Forma y color:SolidPeso molecular:3398.91Bempedoic acid
CAS:<p>Bempedoic acid (ETC1002) is an orally available, once-daily LDL-C lowering small molecule designed to lower elevated levels of LDL-C.</p>Fórmula:C19H36O5Pureza:99.85% - 99.94%Forma y color:SolidPeso molecular:344.49AGI-5198
CAS:<p>AGI-5198 (IDH-C35) is a highly effective and specific inhibitor of IDH1 R132H/R132C mutants (IC50: 0.07/0.16 μM).</p>Fórmula:C27H31FN4O2Pureza:97.37% - 99.23%Forma y color:SolidPeso molecular:462.561-Ethynylpyrene
CAS:<p>1-Ethynylpyrene is an aryl acetylenic inhibitor of CYTP450 1A1(IC50=0.18 μM), 1A2(IC50 = 0.32 μM), and 2B1(IC50 = 0.04 μM).</p>Fórmula:C18H10Pureza:98.48%Forma y color:SolidPeso molecular:226.27Suvecaltamide
CAS:<p>Suvecaltamide (MK-8998) as potent inhibitors of T-type calcium channels.</p>Fórmula:C20H23F3N2O2Pureza:99.29% - 99.70%Forma y color:SolidPeso molecular:380.4Diflubenzuron
CAS:<p>Diflubenzuron (Larvakil) is a benzoyl-urea insecticide, found to be a potent inhibitor of melanosome synthesis in mouse melanoma cells.</p>Fórmula:C14H9ClF2N2O2Pureza:99.58% - 99.96%Forma y color:Colorless Crystals Diflubenzuron Is A Colorless To Yellow Crystals Used As A Selective InsecticidePeso molecular:310.68Ivosidenib
CAS:<p>Ivosidenib (AG-120) is an oral IDH1 inhibitor targeting mutated IDH1 to reduce 2-hydroxyglutarate and hinder tumor growth.</p>Fórmula:C28H22ClF3N6O3Pureza:98.71% - 99.98%Forma y color:SolidPeso molecular:582.96Carbamazepine 10,11-epoxide
CAS:<p>Carbamazepine 10,11-epoxide, an active metabolite with anticonvulsant properties, is created by CYP3A4 and CYP2C8.</p>Fórmula:C15H12N2O2Pureza:98.64% - 99.75%Forma y color:SolidPeso molecular:252.27AMG-3969
CAS:<p>AMG-3969 is an effective glucokinase-glucokinase regulatory protein interaction (GK-GKRP) disruptor (IC50: 4 nM).</p>Fórmula:C21H20F6N4O3SPureza:99.65%Forma y color:SolidPeso molecular:522.46DHBP dibromide
CAS:<p>DHBP dibromide (1,1'-DI-N-HEPTYL-4,4'-BIPYRIDINIUM DIBRO) is calcium release and a muscle relaxant inhibitor.</p>Fórmula:C24H38Br2N2Pureza:99.73%Forma y color:Yellow To Yellow-Green Powder Or FlakesPeso molecular:514.38Ciprofibrate
CAS:<p>Ciprofibrate (Win35833) is a fibrate derivative with antilipidemic activity.</p>Fórmula:C13H14Cl2O3Pureza:99.63% - >99.99%Forma y color:White Or Almost White Crystalline PowderPeso molecular:289.15
