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Metabolismo

Metabolismo

Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.

Subcategorías de "Metabolismo"

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Se han encontrado 8597 productos de "Metabolismo"

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  • Raphin1 acetate

    CAS:
    <p>Raphin1 acetate is a selective and orally bioavailable regulatory phosphatase PPP1R15B (R15B) inhibitor.</p>
    Fórmula:C10H12Cl2N4O2
    Pureza:99.95%
    Forma y color:Solid
    Peso molecular:291.13
  • Ethyl potassium malonate

    CAS:
    <p>Ethyl potassium malonate, a competitive inhibitor of the enzyme succinate dehydrogenase, acts as a precursor to produce (trimethylsilyl)ethyl malonate, which is</p>
    Fórmula:C5H7KO4
    Pureza:99.71%
    Forma y color:White Crystals Or Powder
    Peso molecular:170.21
  • Dorzolamide hydrochloride

    CAS:
    <p>Dorzolamide hydrochloride (MK507 hydrochloride) is the hydrochloride salt form of dorzolamide, an inhibitor of carbonic anhydrase, a zinc-containing enzyme that</p>
    Fórmula:C10H17ClN2O4S3
    Pureza:99.48% - 99.67%
    Forma y color:White Off-White Crystalline Powder
    Peso molecular:360.9
  • H2S Donor 5a

    CAS:
    <p>H2S Donor 5a is a H2S donor that could mimic the slow and continuous H(2)S generation process.</p>
    Fórmula:C14H11NO2S
    Pureza:99.68%
    Forma y color:Solid
    Peso molecular:257.31
  • AMG-208

    CAS:
    <p>AMG-208 is a highly selective c-Met inhibitor with IC50 of 9 nM. Phase 1.</p>
    Fórmula:C22H17N5O2
    Pureza:98.56%
    Forma y color:Solid
    Peso molecular:383.4
  • Cyclosporine

    CAS:
    <p>Cyclosporine is a calcineurin phosphatase pathway inhibitor, used as an immunosuppressant drug to prevent rejection in organ transplantation.</p>
    Fórmula:C62H111N11O12
    Pureza:99.68%
    Forma y color:White Powder
    Peso molecular:1202.61
  • LJ570

    CAS:
    <p>LJ570 is the first PPARα/γ dual agonist (PPARα,PPARγ with EC50s of 1.05 and 0.12 μM, respectively[)</p>
    Fórmula:C27H22O3
    Pureza:99.64%
    Forma y color:Solid
    Peso molecular:394.46
  • GSK0660

    CAS:
    <p>GSK0660 is an antagonist and inverse agonist of PPARβ/δ.</p>
    Fórmula:C19H18N2O5S2
    Pureza:99.26% - ≥95%
    Forma y color:Solid
    Peso molecular:418.49
  • LDHA-IN-4

    CAS:
    <p>LDHA-IN-4 (AZ33) is an LDHA inhibitor. Binding affinity to 6-His-tagged human LDHA expressed in E.coli BL21 (DE3) by SPR analysis with an active value of 93 nM.</p>
    Fórmula:C25H27N3O6S
    Pureza:98.17% - 99.68%
    Forma y color:Solid
    Peso molecular:497.56
  • N6022

    CAS:
    <p>N6022(IC50 of 8 nM) is an effective, reversible, and selective S-Nitrosoglutathione reductase(GSNOR) inhibitor.</p>
    Fórmula:C24H22N4O3
    Pureza:98.24% - 98.32%
    Forma y color:Solid
    Peso molecular:414.46
  • CDN1163

    CAS:
    <p>CDN1163 is a small molecule activator of sarco/endoplasmic reticulum Ca2+-ATPase (SERCA).</p>
    Fórmula:C20H20N2O2
    Pureza:99.83% - ≥95%
    Forma y color:Solid
    Peso molecular:320.39
  • Anti-Inflammatory Peptide 1 Acetate


    <p>Anti-Inflammatory Peptide 1 Acetate (C45H82N12O14S2) inhibits PLA2 to reduce inflammation and pain.</p>
    Fórmula:C47H86N12O16S2
    Pureza:98.95%
    Forma y color:Solid
    Peso molecular:1139.39
  • Anacetrapib

    CAS:
    <p>Anacetrapib (MK-0859) inhibits rhCETP/CETP(C13S) (IC50: 7.9/11.8 nM), boosts HDL, lowers LDL cholesterol.</p>
    Fórmula:C30H25F10NO3
    Pureza:98.40% - 99.87%
    Forma y color:Solid
    Peso molecular:637.51
  • Fluorometholone Acetate

    CAS:
    <p>Fluorometholone Acetate (Oxylone acetate) is a synthetic corticosteroid, used in the treatment of steroid responsive inflammatory conditions of the eye.</p>
    Fórmula:C24H31FO5
    Pureza:99.76%
    Forma y color:Solid
    Peso molecular:418.50
  • IBMX

    CAS:
    <p>IBMX (Methylisobutylxanthine) is a broad-spectrum phosphodiesterase (PDE) inhibitor with inhibitory activity against PDE3, PDE4, and PDE5 (IC50=6.5/26.3/31.7 μM</p>
    Fórmula:C10H14N4O2
    Pureza:98% - >99.99%
    Forma y color:Off-White
    Peso molecular:222.24
  • FT113

    CAS:
    <p>FT113 is a novel potent inhibitor of fatty acid synthase (fasn, IC50 : 213 nM),and exhibits anti-cancer activity</p>
    Fórmula:C22H20FN3O4
    Pureza:97.05%
    Forma y color:Solid
    Peso molecular:409.41
  • NSC 65809

    CAS:
    <p>NSC-65809 (Raphin1) is a selective inhibitor of R15B.</p>
    Fórmula:C8H8Cl2N4
    Pureza:99.37%
    Forma y color:Solid
    Peso molecular:231.08
  • GW4869

    CAS:
    <p>GW4869 (GW69A) is a selective and non-competitive inhibitor of neutral sphingomyelinase N-SMase (IC50=1 μM).</p>
    Fórmula:C30H30Cl2N6O2
    Pureza:98.12% - 98.47%
    Forma y color:Solid
    Peso molecular:577.5
  • LHW090-A7

    CAS:
    <p>LHW090-A7 is an neutral endopeptidase (NEP) inhibitor, and an enzyme responsible for the metabolic inactivation of enkephalins.</p>
    Fórmula:C20H22ClNO4
    Pureza:98.26%
    Forma y color:Solid
    Peso molecular:375.85
  • JNJ-42165279

    CAS:
    <p>JNJ-42165279 selectively inactivates FAAH without notably affecting other enzymes, ion channels, receptors, or CYPs/hERG at 10 μM.</p>
    Fórmula:C18H17ClF2N4O3
    Pureza:99.67% - 99.88%
    Forma y color:Solid
    Peso molecular:410.8