
Metabolismo
Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.
Subcategorías de "Metabolismo"
- AhR(41 productos)
- Aminopeptidasa(67 productos)
- CETP(18 productos)
- Anhídrido carbónico(178 productos)
- Caseína quinasa(130 productos)
- DHFR(33 productos)
- Descarboxilasa(4 productos)
- Deshidrogenasa(271 productos)
- FAAH(64 productos)
- FXR(58 productos)
- Factor Xa(80 productos)
- Ácido graso sintasa(33 productos)
- Ferroptosis(215 productos)
- GR(3 productos)
- GSNOR(3 productos)
- Glucoquinasa(54 productos)
- HIF / HIF Prolilhidroxilasa(142 productos)
- HMG-CoA reductasa(33 productos)
- Hidroxilasa(30 productos)
- IDO(82 productos)
- LDL(8 productos)
- Lipasa(98 productos)
- Lípido(58 productos)
- Lipoxigenasa(124 productos)
- MAO(87 productos)
- MPO(2 productos)
- NAMPT(36 productos)
- P450(6 productos)
- PAI-1(25 productos)
- PDE(166 productos)
- PED(1 productos)
- PKM(15 productos)
- PPAR(165 productos)
- Fosfolipasa(82 productos)
- ROR(42 productos)
- Receptor de retinoides(29 productos)
- SGK(11 productos)
- Tiorredoxina(12 productos)
- Transferasa(30 productos)
- Transportador(42 productos)
- UGT(4 productos)
- Inhibidores de la xantina oxidasa (XO)(9 productos)
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Se han encontrado 8628 productos de "Metabolismo"
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Benzthiazide
CAS:<p>Benzthiazide treats edema and hypertension by promoting diuresis and inhibiting kidney Na+/Cl- reuptake, but may reduce potassium and raise uric acid.</p>Fórmula:C15H14ClN3O4S3Pureza:99.34% - 99.79%Forma y color:Crystals From Acetone SolidPeso molecular:431.94Pargyline hydrochloride
CAS:Pargyline hydrochloride (Pargylamine hydrochloride) is an irreversible monoamine oxidase(MAO) inhibitor with antihypertensive properties.Fórmula:C11H14ClNPureza:99.41% - 99.91%Forma y color:SolidPeso molecular:195.69Topiramate
CAS:<p>Topiramate (RWJ 17021) is a unique antiseizure medication that is used in the treatment of partial and generalized seizures.</p>Fórmula:C12H21NO8SPureza:99.79% - 99.92%Forma y color:White To Off-White Crystalline PowderPeso molecular:339.36Glucosamine hydrochloride
CAS:<p>Glucosamine hydrochloride (Chitosamine hydrochloride) is commonly used as a treatment for osteoarthritis, although its acceptance as a medical therapy varies.</p>Fórmula:C6H13NO5·HClPureza:99.77%Forma y color:White Solid CrystallinePeso molecular:215.63Sulfameter
CAS:<p>Sulfameter (Sulfametoxydiazine) is a long-acting sulfonamide antibacterial agent used to treat urinary tract infections and leprosy.</p>Fórmula:C11H12N4O3SPureza:99.46% - 99.90%Forma y color:Crystalline SolidPeso molecular:280.3LY195448
CAS:<p>LY 195448 (4-(3-(2-Hydroxy-2-phenyl)ethylamino-3-methylbutyl)benzamide) shows antitumor activity in a mouse tumor model, blocking cells in the mid-stage.</p>Fórmula:C20H26N2O2Pureza:98.11% - 99.04%Forma y color:SolidPeso molecular:326.43Phenylhydantoin
CAS:<p>5-Phenylhydantoin is a Mephenytoin metabolite with anti-epileptic effects, targeting NVSCs.</p>Fórmula:C9H8N2O2Pureza:98.09% - 98.91%Forma y color:White SolidPeso molecular:176.17Opevesostat
CAS:<p>Opevesostat (ODM-208) is an inhibitor of lyase (CYP11A1) (the enzyme cleavage cholesterol side chain).</p>Fórmula:C21H26N2O5SPureza:99.25%Forma y color:SoildPeso molecular:418.51FASN-IN-3
CAS:<p>FASN-IN-3 is an inhibitor of fatty acid synthase (FASN).</p>Fórmula:C24H24N4OPureza:97.41%Forma y color:SolidPeso molecular:384.47Tetracaine hydrochloride
CAS:<p>Tetracaine HCl (Pontocaine), a potent local anesthetic and antipruritic, is used in eye care and for surface/spinal anesthesia.</p>Fórmula:C15H25ClN2O2Pureza:99.72% - 99.94%Forma y color:White Or Off White Crystalline PowderPeso molecular:300.82(-)-Vorozole
CAS:<p>(-)-Vorozole, potent/selective oral non-steroidal aromatase inhibitor, shows antitumor activity, used in breast cancer research.</p>Fórmula:C16H13ClN6Pureza:99.02% - >99.99%Forma y color:SoildPeso molecular:324.77DIPQUO hydrochloride
DIPQUO hydrochloride: ALP activator (EC50=6.27μM, C2C12 cells), induces osteoblast differentiation via p38 MAPK-β.Fórmula:C20H18ClN3OPureza:98.09%Forma y color:SoildPeso molecular:351.83VU533
CAS:<p>VU533 is a NAPE-PLD activator, EC50=0.30 µM, boosts macrophage activity, potential in cardiometabolic diseases.</p>Fórmula:C21H22FN3O3S2Pureza:99.08%Forma y color:SolidPeso molecular:447.55VU534
CAS:<p>VU534 is a NAPE-PLD agonist with an EC50 of 0.30 μM.VU534 is a dual inhibitor of FAAH and sEH, with an IC50 of 1.2 μM for sEH.VU534 is used in diseases related</p>Fórmula:C21H22FN3O3S2Pureza:98.85%Forma y color:SolidPeso molecular:447.552H-Cho-Arg (trifluoroacetate salt)
CAS:<p>2H-Cho-Arg, a cationic lipid, enables gene delivery into cells and shows cytotoxicity at 92.7 μg/ml.</p>Fórmula:C43H73F6N5O7Forma y color:SolidPeso molecular:886.06α-Glycerophosphate Dehydrogenase-Triosephosphate
<p>α-Glycerophosphate Dehydrogenase-Triosephosphate (GDH-TIM) is an enzyme mixture composed of glycerophosphate dehydrogenase (GDH) and triosephosphate isomerase (TIM). This compound is employed to measure transketolase (TK) activity in erythrocyte hemolysates, which helps in assessing vitamin B deficiency.</p>PROTAC NAMPT Degrader-1
<p>PROTACNAMPT Degrader-1 is an effective NAMPT-targeting PROTAC with a DC50 value of 217 nM. It exhibits antiproliferative activity, with an IC50 value of 0.12 μM against A2780 cells.</p>Fórmula:C57H69N13O8S2Peso molecular:1127.48335Galactose 1-dehydrogenase
<p>Galactose 1-dehydrogenase, pseudomonas fluorescens, a dehydrogenase found in Pseudomonas fluorescens, facilitates the oxidation of L-arabinose and D-galactose, utilizing NADP+/NAD+ as a cofactor. This enzyme is employed in diagnostic assays to quantify total galactose levels and serves as a biocatalyst in the production of galacturonic acid salts.</p>Forma y color:Odour SolidCTL-06
<p>CTL-06, a Fatty Acid Synthase (FASN) inhibitor with an IC50 of 3 μM, induces apoptosis, while CTL-12 impedes cell cycle progression in the Sub-G1/S phase and</p>Fórmula:C21H21ClN4O4Forma y color:SolidPeso molecular:428.87FABP4-IN-3
<p>FABP4-IN-3 (Compound C3) is a highly selective inhibitor of FABP4, with an inhibition constant (Ki) of 25 ± 3 nM for FABP4 and a Ki of 15.03 μM for FABP3, showcasing a selectivity factor of 601 times over FABP3. It also demonstrates metabolic stability and potent anti-inflammatory activity in cells, making it a promising candidate for research in metabolic disorders, cardiac dysfunction, and inflammation-related diseases.</p>Fórmula:C20H16ClNO2Peso molecular:337.08696

