
Metabolismo
Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.
Subcategorías de "Metabolismo"
- AhR(41 productos)
- Aminopeptidasa(74 productos)
- CETP(20 productos)
- Anhídrido carbónico(185 productos)
- Caseína quinasa(137 productos)
- DHFR(34 productos)
- Descarboxilasa(4 productos)
- Deshidrogenasa(289 productos)
- FAAH(65 productos)
- FXR(59 productos)
- Factor Xa(83 productos)
- Ácido graso sintasa(36 productos)
- Ferroptosis(218 productos)
- GR(3 productos)
- GSNOR(4 productos)
- Glucoquinasa(56 productos)
- HIF / HIF Prolilhidroxilasa(145 productos)
- HMG-CoA reductasa(33 productos)
- Hidroxilasa(34 productos)
- IDO(84 productos)
- LDL(8 productos)
- Lipasa(104 productos)
- Lípido(62 productos)
- Lipoxigenasa(132 productos)
- MAO(87 productos)
- MPO(2 productos)
- NAMPT(38 productos)
- P450(6 productos)
- PAI-1(26 productos)
- PDE(166 productos)
- PED(1 productos)
- PKM(15 productos)
- PPAR(168 productos)
- Fosfolipasa(82 productos)
- ROR(43 productos)
- Receptor de retinoides(28 productos)
- SGK(11 productos)
- Tiorredoxina(12 productos)
- Transferasa(29 productos)
- Transportador(43 productos)
- UGT(4 productos)
- Inhibidores de la xantina oxidasa (XO)(9 productos)
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Se han encontrado 9054 productos de "Metabolismo"
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UDP-glucosamine disodium
CAS:UDP-GlcNAc disodium is a substrate for O-GlcNAc transferase and removed by O-GlcNAcase, produced in the hexosamine pathway regulated by GFAT.Fórmula:C15H23N3Na2O16P2Forma y color:SolidPeso molecular:609.28Terpendole I
CAS:<p>Terpendole I, from A. yamanashiensis, inhibits ACAT (IC50=145 μM), fights B. cereus/subtilis (MIC=100 μg/ml), and kills HeLa cells (IC50=52.6 μM).</p>Fórmula:C27H35NO5Forma y color:SolidPeso molecular:453.579Calcitroic acid
CAS:<p>Calcitroic acid is a vitamin D receptor (VDR) agonist that activates VDR-mediated transcription. It is the primary metabolite of 1,25-dihydroxyvitamin D3, showing the highest concentrations in the liver and mucosa of mice. The compound exhibits metabolic stability and extremely low toxicity.</p>Fórmula:C23H34O4Forma y color:SolidPeso molecular:374.514tetranor-PGAM
CAS:PGE2 is a biomarker for inflammation and disease; its unstable urinary metabolite, tetranor-PGEM, and its byproduct, tetranor-PGAM, indicate biosynthesis.Fórmula:C16H22O6Forma y color:SolidPeso molecular:310.346FASN-IN-4 tosylate
CAS:FASN-IN-4 tosylate: Fatty acid synthase inhibitor, IC50 10 nM; blocks SARS-CoV-2, EC50 18.6 nM.Fórmula:C33H35N3O7S2Forma y color:SolidPeso molecular:649.78(Rac)-5-Keto Fluvastatin
CAS:<p>(Rac)-5-Keto Fluvastatin (rac 5-Keto Fluvastatin) is an impurity of Fluvastatin which is an inhibitor of HMG-CoA reductase.</p>Fórmula:C24H24FNO4Pureza:95.04%Forma y color:SolidPeso molecular:409.45α-Amylase-IN-4
<p>α-Amylase-IN-4 (Compd 10y) exhibits the highest level of amylase inhibition, demonstrating an IC50 value of 17.83 ± 0.14 μg/mL [1].</p>Forma y color:Odour Solid(±)-threo-3-Methylglutamic acid
CAS:glutamate transport blockerFórmula:C6H11NO4Pureza:98%Forma y color:SolidPeso molecular:161.16Mycophenolate mofetil hydrochloride
CAS:Mycophenolate Mofetil: Non-competitive, selective inhibitor of IMP dehydrogenase I/II, IC50: 39/27 nM.Fórmula:C23H32ClNO7Pureza:98%Forma y color:SolidPeso molecular:469.96Histamine glutarimide
CAS:Histamine glutarimide is a novel QPCT inhibitor that targets inflammatory processes like eosinophil migration, showing anti-asthmatic effects in animal models.Fórmula:C10H13N3O2Pureza:99.79%Forma y color:SolidPeso molecular:207.23DSPE-PEG5000-R8
<p>DSPE-PEG5000-R8 is a PEG compound composed of DSPE and the cell-penetrating peptide (R8). It is utilized for drug delivery applications.</p>Forma y color:Odour SolidHIV-1 inhibitor-58
HIV-1 Inhibitor-58 (Compound 10c) is a non-nucleoside reverse transcriptase inhibitor with broad-spectrum antiviral properties, effective against both wild-typeFórmula:C26H24N6O2Forma y color:SolidPeso molecular:452.51IDO1-IN-7
CAS:IDO1-IN-7 is a potent IDO1 inhibitor with a 6.1 nM IC50 and immunomodulatory effects for cancer research.Fórmula:C22H19ClFN3O3Forma y color:SolidPeso molecular:427.86(±)20-HDHA
CAS:<p>(±)20-HDHA is an autoxidation product and is a racemic mixture of Docosahexaenoic acid (DHA).</p>Fórmula:C22H32O3Pureza:98%Forma y color:SolidPeso molecular:344.49DOTA-XYIMSR-01
CAS:DOTA-XYIMSR-01 is a molecular probe targeting CAIX, capable of being labeled with 177Lu for the treatment and localization of malignant gliomas. The uptake of [177Lu]Lu-XYIMSR-01 in U87MG tumors is 6.19% injected dose per gram (% ID/g), with a tumor-to-muscle uptake ratio of 20.14. In an orthotopic glioma model, co-administration with temozolomide significantly enhances survival rates and inhibits tumor growth in mice. DOTA-XYIMSR-01 shows potential for research in the field of cancer treatment.Fórmula:C61H88N16O22S2Forma y color:SolidPeso molecular:1461.57cis-5-Tetradecenoic acid
CAS:cis-5-Tetradecenoic acid, found in blood, helps study Long Chain 3-Hydroxyacyl-CoA Dehydrogenase Deficiency.Fórmula:C14H26O2Forma y color:SolidPeso molecular:226.36GLX481369
GLX481369 is a redox-active substance that functions as an NOX4 inhibitor, exhibiting antioxidant effects [1].Fórmula:C21H24ClN7OForma y color:SolidPeso molecular:425.91Beauverolide Ka
CAS:<p>Beauverolide Ka, from Beauveria bassiana, enhances glucose uptake and protects HEI-OC1 cells; active in L6 cells/myotubes.</p>Fórmula:C37H50N4O5Forma y color:SolidPeso molecular:630.82Calpinactam
CAS:<p>Calpinactam, from M. alpina, fights M. smegmatis (MIC 0.78 μg/ml), boosts silkworm survival, but ineffective against 13 other species.</p>Fórmula:C38H57N9O8Forma y color:SolidPeso molecular:767.9291,2-Dihexadecyl-sn-glycero-3-PC
CAS:1,2-Dihexadecyl-sn-glycero-3-PC can be used in related research in the field of life sciences. Its product number is T37043 and CAS number is 36314-47-3.Fórmula:C40H84NO6PForma y color:SolidPeso molecular:706.07

