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Metabolismo

Metabolismo

Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.

Subcategorías de "Metabolismo"

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Se han encontrado 8626 productos de "Metabolismo"

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  • KCA-1490

    CAS:
    <p>KCA-1490 is an inhibitor of dual PDE3/4.</p>
    Fórmula:C14H13F3N4O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:326.27
  • BMS-185411

    CAS:
    <p>BMS-185411 is a bio-active chemical.</p>
    Fórmula:C26H23NO3
    Forma y color:Solid
    Peso molecular:397.47
  • SHP394

    CAS:
    <p>SHP394 is an orally efficacious inhibitor of protein tyrosine phosphatase SHP2 (IC50: 23 nM).</p>
    Fórmula:C20H25F3N6O2S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:470.51
  • sEH/AChE-IN-3

    CAS:
    <p>sEH/AChE-IN-3 -15: potent dual sEH &amp; AChE inhibitor; crosses BBB; IC50: hsEH 0.4nM, hAChE 1.94nM, hBChE 615nM, msEH 4.3nM, mAChE 2.61nM.</p>
    Fórmula:C35H39ClF3N5O3
    Forma y color:Solid
    Peso molecular:670.16
  • hCAIX-IN-15

    CAS:
    <p>hCAIX-IN-15 is a potent inhibitor of human carbonic anhydrase IX (hCA IX) with an inhibition constant (Ki) of 38.8 nM, exhibiting broad-spectrum anticancer</p>
    Fórmula:C18H14FN7O2S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:411.41
  • α-Glucosidase-IN-28

    CAS:
    <p>α-Glucosidase-IN-28 (Compound 18) is an α-glucosidase inhibitor with an IC50 of 0.62 μM and Ki value of 3.93 μM.</p>
    Fórmula:C29H22Br2O7
    Pureza:98%
    Forma y color:Solid
    Peso molecular:642.29
  • ICMT-IN-19

    CAS:
    <p>ICMT-IN-19 (compound 53) serves as a potent inhibitor of ICMT, demonstrating an IC50 value of 0.026 μM [1].</p>
    Fórmula:C21H26N2O3
    Forma y color:Solid
    Peso molecular:354.44
  • hCAIX/XII-IN-8

    CAS:
    <p>hCAIX/XII-IN-8 (compound 3g) is a potent inhibitor of the human carbonic anhydrases (CAs) IX and XII, with inhibition constants (K i) of 8.5 nM for CA IX and 6.</p>
    Fórmula:C16H13Cl2N5O3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:426.28
  • UCPH-102

    CAS:
    <p>UCPH-102: Selective EAAT1 inhibitor, IC50 0.43 μM, treats Alzheimer's, ALS, chronic pain, OCD; crosses blood-brain barrier, targets T-ALL cells.</p>
    Fórmula:C21H18N2O2
    Forma y color:Solid
    Peso molecular:330.38
  • Cav 3.2 inhibitor 4

    CAS:
    <p>Cav 3.2 Inhibitor 4 (Compound 21) is a selective and potent inhibitor of the T-type calcium channel (Ca v 3.2), demonstrating peripheral restriction with an</p>
    Fórmula:C21H32Cl2N4O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:459.41
  • Phenylpyropene C

    CAS:
    <p>Phenylpyropene C inhibits JAK/STAT and IFN-γ expression (IC50: 5.4-10.8 μM), also blocks acyl CoA (IC50: 16.0 μM).</p>
    Fórmula:C28H34O5
    Forma y color:Solid
    Peso molecular:450.57
  • ICMT-IN-36

    CAS:
    <p>ICMT-IN-36 (compound 40) serves as an ICMT inhibitor, with an IC50 value of 0.181 μM [1].</p>
    Fórmula:C21H25Cl2NO
    Forma y color:Solid
    Peso molecular:378.34
  • BBT

    CAS:
    <p>BBT has anti-hyperglycemic activity, protecting beta cells from cytokine or streptozotocin-induced cell death, and restoring beta cell function.</p>
    Fórmula:C18H12BrNO2S
    Pureza:99.02%
    Forma y color:Solid
    Peso molecular:386.26
  • ERX-41

    CAS:
    <p>ERX-41 is an orally active, stereospecific small molecule that targets lysosomal acid lipase A (LIPA).</p>
    Fórmula:C38H48N4O9
    Pureza:98%
    Forma y color:Solid
    Peso molecular:704.81
  • BAY-7081


    <p>BAY-7081 is a cyanopyridone-based compound that functions as a potent, selective, and orally active PDE9A inhibitor, demonstrating an inhibition concentration (</p>
    Fórmula:C19H27ClN4O
    Forma y color:Solid
    Peso molecular:362.9
  • H-0106 Dihydrochloride

    CAS:
    <p>H-0106 Dihydrochloride is an inhibitor of ROCK that acts by applying strong intraocular pressure (IOP)-lowering effects into the eyes of monkeys.</p>
    Fórmula:C16H22Cl3N3O2S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:426.79
  • VT-1598 tosylate

    CAS:
    <p>VT-1598 tosylate is a selective, orally active antifungal compound that targets CYP51. It demonstrates efficacy against C. auris.</p>
    Fórmula:C38H28F4N6O5S
    Forma y color:Solid
    Peso molecular:756.72
  • PF-04937319

    CAS:
    <p>PF-04937319 activates glucokinase (EC50=154.4μM) with low hypoglycemia risk, researched for type 2 diabetes treatment.</p>
    Fórmula:C22H20N6O4
    Pureza:99.89%
    Forma y color:Solid
    Peso molecular:432.43
  • Diethyl-pythiDC

    CAS:
    <p>Diethyl-pythiDC is an collagen prolyl 4-hydroxylase inhibitor.</p>
    Fórmula:C14H14N2O4S
    Pureza:99.98%
    Forma y color:Solid
    Peso molecular:306.34
  • GPX4-IN-2

    CAS:
    <p>GPX4-IN-2 is a potent inhibitor of GPX4, exhibiting antiproliferative activity. It holds potential for cancer research applications.</p>
    Fórmula:C30H40N2O
    Forma y color:Solid
    Peso molecular:444.65