
Metabolismo
Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.
Subcategorías de "Metabolismo"
- AhR(41 productos)
- Aminopeptidasa(67 productos)
- CETP(18 productos)
- Anhídrido carbónico(177 productos)
- Caseína quinasa(130 productos)
- DHFR(32 productos)
- Descarboxilasa(4 productos)
- Deshidrogenasa(267 productos)
- FAAH(63 productos)
- FXR(58 productos)
- Factor Xa(80 productos)
- Ácido graso sintasa(32 productos)
- Ferroptosis(215 productos)
- GR(3 productos)
- GSNOR(3 productos)
- Glucoquinasa(53 productos)
- HIF / HIF Prolilhidroxilasa(142 productos)
- HMG-CoA reductasa(32 productos)
- Hidroxilasa(30 productos)
- IDO(82 productos)
- LDL(8 productos)
- Lipasa(96 productos)
- Lípido(59 productos)
- Lipoxigenasa(124 productos)
- MAO(87 productos)
- MPO(2 productos)
- NAMPT(36 productos)
- P450(6 productos)
- PAI-1(25 productos)
- PDE(166 productos)
- PED(1 productos)
- PKM(15 productos)
- PPAR(164 productos)
- Fosfolipasa(82 productos)
- ROR(42 productos)
- Receptor de retinoides(29 productos)
- SGK(11 productos)
- Tiorredoxina(12 productos)
- Transferasa(30 productos)
- Transportador(42 productos)
- UGT(4 productos)
- Inhibidores de la xantina oxidasa (XO)(9 productos)
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Se han encontrado 8595 productos de "Metabolismo"
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Antiproliferative agent-13
CAS:<p>Antiproliferative agent-13 is a compound with antiproliferative activity.</p>Fórmula:C20H18N2O6Pureza:99.723%Forma y color:SolidPeso molecular:382.37Eflucimibe
CAS:<p>Eflucimibe (L0081), an ACAT inhibitor, treats cardiovascular, endocrine, and metabolic diseases, and helps in atherosclerosis and hyperlipidemia research.</p>Fórmula:C29H43NO2SPureza:99.17% - 99.43%Forma y color:SolidPeso molecular:469.72ATX inhibitor 7
CAS:<p>ATX inhibitor 7 is a autotaxin inhibitor and shows good oral exposure.</p>Fórmula:C21H22F3N7O2Forma y color:SolidPeso molecular:461.449Burnettramic Acid A aglycone
CAS:<p>Burnettramic acid A aglycone, from A. burnettii, has anticancer properties; cytotoxic to NS-1 cells (IC50 = 8.4 μg/ml), not to fibroblasts (>100 μg/ml).</p>Fórmula:C35H61NO7Forma y color:SolidPeso molecular:607.873SAICAR
CAS:<p>SAICAR is an intermediate of de novo purine nucleotide biosynthesis, activates pyruvate kinase isoform M2 (PKM2) in an isozyme-selective manner (EC50: 0.3 mM).</p>Fórmula:C13H19N4O12PPureza:98%Forma y color:SolidPeso molecular:454.28α-Glucosidase-IN-60
<p>α-Glucosidase-IN-60 (Compound 5k) acts as a competitive inhibitor of α-Glucosidase, with an IC50 of 10.8 μM.</p>Fórmula:C23H14N2O5Peso molecular:398.09027Ritonavir metabolite
CAS:<p>Ritonavir metabolite is a Ritonavir metabolite, which is a inhibitor of HIV protease.</p>Fórmula:C32H45N5O3SPureza:98%Forma y color:SolidPeso molecular:579.80SGK1-IN-3 hydrochloride
<p>SGK1-IN-3 hydrochloride (compound 3a) is an efficacious, orally bioavailable SGK1 inhibitor. The serine/threonine kinase SGK1 acts as an activator of the β-catenin pathway and strongly stimulates cartilage degradation, being upregulated under genomic control in diseased osteoarthritic cartilage. SGK1-IN-3 hydrochloride holds potential for osteoarthritis research.</p>Fórmula:C23H21Cl3N6O3SPeso molecular:566.04614Garcinone B
CAS:<p>Garcinone B, a xanthone derivative naturally isolated from the pericarp of Mangosteen, serves as a potent inhibitor of ACE2 and Mpro, and is utilized in COVID-</p>Fórmula:C23H22O6Pureza:98%Forma y color:SolidPeso molecular:394.42WVSAV
<p>WVSAV is a ligand for the PDZ2 domain (tyrosine phosphatase) with a dissociation constant (Kd) of 111 μM. It is utilized in studies of protein-ligand interactions.</p>Fórmula:C27H40N6O7Forma y color:SolidPeso molecular:560.64DSPE-PEG1000-pPB
<p>DSPE-PEG1000-pPB is a PEG compound consisting of DSPE and a cyclic oligopeptide (pPB). The pPB component exhibits a strong binding affinity to PDGFRβ, which is overexpressed in activated hepatic stellate cells (HSC). DSPE-PEG1000-pPB is applicable for drug delivery.</p>Forma y color:Odour SolidCasein Kinase Substrates 3
CAS:<p>Casein Kinase Substrates 3 is a substrate of casein kinase.</p>Fórmula:C85H139N27O35SPureza:98%Forma y color:SolidPeso molecular:2131.24Lysylglutamic acid
CAS:<p>Lysylglutamic acid is a dipeptide composed of the amino acids lysine (Lysine, Lys) and glutamic acid (Glutamic acid, Glu), with an inhibitory constant (Ki) of 1.3 mM for the membrane transport protein PEPT1.</p>Fórmula:C11H21N3O5Forma y color:SolidPeso molecular:275.3Ilexoside O
CAS:<p>Ilexoside O, a root-derived triterpene saponin, modestly blocks XOD with an IC50 of 53.05 μM.</p>Fórmula:C53H86O22Forma y color:SolidPeso molecular:1075.249CNBCA
<p>CNBCA, a selective and potent competitive inhibitor of the SHP2 enzyme, exhibits an IC50 value of 0.87 μM.</p>Fórmula:C26H34O5Forma y color:SolidPeso molecular:426.55α-Amylase-IN-4
<p>α-Amylase-IN-4 (Compd 10y) exhibits the highest level of amylase inhibition, demonstrating an IC50 value of 17.83 ± 0.14 μg/mL [1].</p>Forma y color:Odour SolidAdefovir diphosphate 2TEA
<p>Adefovir diphosphate 2TEA,a metabolite of Adefovir, an oral reverse transcriptase inhibitor with antiviral activity against herpes, hepatitis B, and HIV.</p>Fórmula:C20H43N7O7P2Pureza:98.33%Forma y color:SolidPeso molecular:555.55LDHA-IN-8
CAS:<p>LDHA-IN-8, an inhibitor, inhibits the proliferation of pancreatic and lung cancer cells, decreasing the intracellular lactate content and increasing ROS levels.</p>Fórmula:C15H14N4O2Pureza:99.73%Forma y color:SolidPeso molecular:282.31,3-Dipalmitoleoyl-rac-glycerol
CAS:<p>1,3-Dipalmitoleoyl-rac-glycerol: a diacylglycerol inhibiting yeast α-glucosidase over rat's (IC50s: 4.45 vs 9326.5 μM). Used to study membrane potentials.</p>Fórmula:C35H64O5Forma y color:SolidPeso molecular:564.892C18:1 Ceramide (d18:1/18:1(9Z))
CAS:<p>C18:1 Ceramide (d18:1/18:1(9Z)) is a ceramide, and C18:1-Ceramide levels are elevated in overweight and insulin-resistant , advanced ovarian cancer.</p>Fórmula:C36H69NO3Pureza:99.96%Forma y color:SolidPeso molecular:563.94

