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Metabolismo

Metabolismo

Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.

Subcategorías de "Metabolismo"

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Se han encontrado 8626 productos de "Metabolismo"

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  • Calcitriol Derivatives


    <p>Calcitriol Derivatives is an analog of vitamin D3.</p>
    Fórmula:C30H47NO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:469.7
  • α-Amylase/α-Glucosidase-IN-17


    <p>α-Amylase/α-Glucosidase-IN-17 (Compound 3) is an inhibitor of α-amylase and α-glucosidase, with IC50 values of 14.61 μM and 25.38 μM, respectively. It exhibits some inhibitory activity against A549 cancer cells and possesses both antitumor and antidiabetic properties.</p>
    Fórmula:C19H18FNO
    Forma y color:Solid
    Peso molecular:295.35
  • BNTA

    CAS:
    <p>BNTA is a potent extracellular matrix (ECM) modulator.</p>
    Fórmula:C17H11BrClNO3S2
    Pureza:98.87% - 99.79%
    Forma y color:Solid
    Peso molecular:456.76
  • Zifcasiran

    CAS:
    <p>Zifcasiran reduces HIF synthesis, has antitumor properties, useful in renal carcinoma studies.</p>
    Fórmula:C737H972F20N211O349P43S8
    Forma y color:Solid
    Peso molecular:20339.13
  • LH1513


    <p>LH1513 is a dioxalate salt derivative of l-lysine that inhibits CaOx crystallization more effectively than citrate and pyruvate. It shows potential preventive activity in hyperoxaluria models and effectively prevents urinary CaOx crystal formation in Agxt knockout mice. AGXT-1 is a mitochondrial protein involved in metabolic processes.</p>
    Fórmula:C10H11N2Na3O8
    Forma y color:Solid
    Peso molecular:356.17
  • NAMPT activator-7


    <p>NAMPTactivator-7 (Compound 232) is an activator of nicotinamide phosphoribosyltransferase (NAMPT) with an EC50 of less than 0.5 μM. It effectively stimulates NAMPT in U2OS cells, demonstrating a cellular EC50 of less than 0.5 μM.</p>
    Fórmula:C21H17ClN4O3
    Peso molecular:408.09892
  • Carbolactone

    CAS:
    <p>Carbolactone is a biologically active metabolite from fungi [1] .</p>
    Fórmula:C24H36O3
    Forma y color:Solid
    Peso molecular:372.54
  • TMP-778

    CAS:
    <p>TMP-778 is a selective inverse agonist of RORγt.</p>
    Fórmula:C31H30N2O4
    Pureza:99.68%
    Forma y color:Solid
    Peso molecular:494.58
  • NIM811

    CAS:
    <p>NIM811 is an orally bioavailable dual inhibitor of mitochondrial permeability transition and cyclophilin.</p>
    Fórmula:C62H111N11O12
    Pureza:98%
    Forma y color:Solid
    Peso molecular:1202.635
  • (S,S)-GSK321

    CAS:
    <p>(S,S)-GSK321 is a (S,S)-enantiomer of GSK321 [1] .</p>
    Fórmula:C28H28FN5O3
    Forma y color:Solid
    Peso molecular:501.55
  • 5-Lipoxygenase-IN-3

    CAS:
    <p>Compound 14, a &lt;1 μM 5-lipoxygenase inhibitor, researches inflammation, cancer, stroke, Alzheimer's.</p>
    Fórmula:C19H16ClN5O
    Forma y color:Solid
    Peso molecular:365.82
  • Coproporphyrin I

    CAS:
    <p>Coproporphyrin I, an endogenous metabolite found in urine and blood, is utilized in researching liver disease and porphyria [1] [2] [3] [4].</p>
    Fórmula:C36H38N4O8
    Forma y color:Solid
    Peso molecular:654.71
  • NADP+ (sodium salt hydrate)

    CAS:
    <p>NADP+ is the oxidized cofactor form of NADPH, vital for cell survival, redox balance, and signaling; synthesized from NAD+ and ATP.</p>
    Fórmula:C21H30N7NaO18P3
    Forma y color:Solid
    Peso molecular:784.413
  • m-Tyramine

    CAS:
    <p>m-Tyramine has effects on the adrenergic and dopaminergic receptor.m-Tyramine is an endogenous trace amine neuromodulator.</p>
    Fórmula:C8H11NO
    Pureza:98%
    Forma y color:Solid
    Peso molecular:137.18
  • ST6 Sialyltransferase 5


    <p>ST6Sialyltransferase5 (EC:2.4.3.3, ST6GALNAC5, SIAT7E, ST6 N-acetylgalactosaminide alpha-2,6-sialyltransferase 5) transfers sialic acid to N-acetylgalactosamine (GalNAc) residues. It may serve as a biomarker in cervical screening samples.</p>
  • Adaptaquin

    CAS:
    <p>Adaptaquin is an inhibitor of the hypoxia-inducing factor prolyl hydroxylase (HIF-PH) [1] [2].</p>
    Fórmula:C21H16ClN3O2
    Pureza:99.75%
    Forma y color:Solid
    Peso molecular:377.82
  • ACAT-IN-4 hydrochloride

    CAS:
    <p>ACAT-IN-4 hydrochloride is a potent ACAT inhibitor and blocks NF-κB transcription.</p>
    Fórmula:C32H51ClN2O5S
    Forma y color:Solid
    Peso molecular:611.28
  • Cholesteryl arachidonate

    CAS:
    <p>Cholesteryl arachidonate is a human endogenous metabolite.</p>
    Fórmula:C47H76O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:673.11
  • APOL1-IN-2

    CAS:
    <p>APOL1-IN-2 (Compound 467) acts as an inhibitor of apolipoprotein L1 (APOL1). It effectively reduces HEK293 cell death induced by APOL1 G2/G1, with EC50 values of 4.74 nM and 14.3 nM, respectively. Additionally, APOL1-IN-2 decreases the mortality of trypanosomes triggered by APOL1 G2/G1/G0, with EC50 values of 2.24, 6.03, and 3.72 nM, respectively.</p>
    Fórmula:C28H30ClF3N4O5
    Forma y color:Solid
    Peso molecular:595.01
  • Ivabradine impurity 1

    CAS:
    <p>Ivabradine impurity 1, orally bioavailable HCN channel blocker.</p>
    Fórmula:C15H18BrNO3
    Forma y color:Solid
    Peso molecular:340.21