
Metabolismo
Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.
Subcategorías de "Metabolismo"
- AhR(41 productos)
- Aminopeptidasa(67 productos)
- CETP(18 productos)
- Anhídrido carbónico(178 productos)
- Caseína quinasa(130 productos)
- DHFR(33 productos)
- Descarboxilasa(4 productos)
- Deshidrogenasa(270 productos)
- FAAH(64 productos)
- FXR(58 productos)
- Factor Xa(80 productos)
- Ácido graso sintasa(33 productos)
- Ferroptosis(215 productos)
- GR(3 productos)
- GSNOR(3 productos)
- Glucoquinasa(54 productos)
- HIF / HIF Prolilhidroxilasa(142 productos)
- HMG-CoA reductasa(33 productos)
- Hidroxilasa(30 productos)
- IDO(82 productos)
- LDL(8 productos)
- Lipasa(97 productos)
- Lípido(59 productos)
- Lipoxigenasa(125 productos)
- MAO(87 productos)
- MPO(2 productos)
- NAMPT(36 productos)
- P450(6 productos)
- PAI-1(25 productos)
- PDE(166 productos)
- PED(1 productos)
- PKM(15 productos)
- PPAR(164 productos)
- Fosfolipasa(82 productos)
- ROR(42 productos)
- Receptor de retinoides(29 productos)
- SGK(11 productos)
- Tiorredoxina(12 productos)
- Transferasa(30 productos)
- Transportador(42 productos)
- UGT(4 productos)
- Inhibidores de la xantina oxidasa (XO)(9 productos)
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Se han encontrado 8625 productos de "Metabolismo"
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ERAP1 modulator-1
CAS:<p>ERAP1 modulator-1 (Compound 1) is a regulator of endoplasmic reticulum aminopeptidase 1 (ERAP1) with an IC50 of less than 250 nM.</p>Fórmula:C23H23F3N2O5SForma y color:SolidPeso molecular:496.5APOL1-IN-2
CAS:<p>APOL1-IN-2 (Compound 467) acts as an inhibitor of apolipoprotein L1 (APOL1). It effectively reduces HEK293 cell death induced by APOL1 G2/G1, with EC50 values of 4.74 nM and 14.3 nM, respectively. Additionally, APOL1-IN-2 decreases the mortality of trypanosomes triggered by APOL1 G2/G1/G0, with EC50 values of 2.24, 6.03, and 3.72 nM, respectively.</p>Fórmula:C28H30ClF3N4O5Forma y color:SolidPeso molecular:595.01PPARγ agonist 15
<p>PPARγ agonist15 (Compound 7c) functions as an agonist of PPARγ, inhibiting the expression of α-amylase (HPA) and α-glucosidase (HLAG) with IC50 values of 28.35 µM and 26.21 µM, respectively. It enhances glucose uptake in L6 myotubes and improves glucose homeostasis, insulin sensitivity, and lipid metabolism in a rat model of Streptozotocin-induced diabetes.</p>Fórmula:C21H16N4O3S2Forma y color:SolidPeso molecular:436.51APL180
CAS:<p>APL180 (L-4F) is an apolipoprotein A-I mimetic peptide that enhances the anti-inflammatory activity of high-density lipoprotein (HDL). It is applicable for cardiovascular disease research.</p>Fórmula:C114H156N24O28Forma y color:SolidPeso molecular:2310.6Plipastatin A1
CAS:<p>Plipastatin A1, a lipopeptide isolated from B.</p>Fórmula:C72H110N12O20Forma y color:SolidPeso molecular:1463.71hCAI/II-IN-10
<p>hCAI/II-IN-10 (Compound 5d) is an inhibitor of human carbonic anhydrase I and II (hCA I and hCA II), with IC50 values of 4.32 nM and 3.89 nM, respectively.</p>Fórmula:C24H17Cl2N3O3S2Forma y color:SolidPeso molecular:530.446cis-Vitamin K1
CAS:<p>Cis-Vitamin K1 is an endogenous metabolite of Vitamin K [1] .</p>Fórmula:C31H46O2Forma y color:SolidPeso molecular:450.70ZG-2033
CAS:<p>ZG-2033 (Compound 26) is an orally active HIF-2α agonist that exhibits nanomolar activity (EC50 = 490 nM) in a luciferase reporter assay. It demonstrates an anti-anemic effect and shows synergistic effects with AKB-6548 in anemia, making it useful for the study of renal anemia.</p>Fórmula:C15H14N2O2SForma y color:SolidPeso molecular:286.35PPARγ agonist 16
CAS:<p>PPARγ agonist16 (Compound 4G) is a PPARγ agonist that competitively binds to the ligand-binding domain (LBD) of PPARγ with an IC50 of 1790 nM. It reduces ear swelling in mouse models and exhibits antihyperglycemic activity in mice with Streptozotocin-induced diabetes.</p>Fórmula:C19H14BrNO4SForma y color:SolidPeso molecular:432.29Galactose 1-phosphate
CAS:<p>Galactose 1-phosphate, an intermediate substance in both galactose metabolism and nucleotide sugar processes, plays a crucial role in the biochemical pathways</p>Fórmula:C6H13O9PPureza:98%Forma y color:SolidPeso molecular:260.14Hydroxycotinine
CAS:<p>Hydroxycotinine is the main nicotine metabolite detected in smokers' urine.</p>Fórmula:C10H12N2O2Pureza:98%Forma y color:SolidPeso molecular:192.218Calcium Channel antagonist 5
CAS:<p>Calcium Channel antagonist5 (compound 32) is a calcium channel antagonist with a pIC50 of 5.50.</p>Fórmula:C17H18N2O6Forma y color:SolidPeso molecular:346.34Adenosine 3',5'-diphosphate sodium salt
CAS:<p>Adenosine 3',5'-diphosphate sodium inhibits hydroxysteroid sulfotransferases and studies SULT kinetics/structure.</p>Fórmula:C10H15N5NaO10P2Pureza:95%Forma y color:SolidPeso molecular:450.19DSPE-PEG1000-R6H4
<p>DSPE-PEG1000-R6H4 is a PEG compound comprised of DSPE and pH-responsive cell-penetrating peptide (R6H4), designed for pH-sensitive anti-cancer drug delivery. It is utilized in drug delivery applications.</p>Forma y color:Odour SolidAK-4
<p>AK-4 is an antidiabetic agent that functions as a mitochondrial uncoupler.</p>Fórmula:C21H14Cl2N2O4SForma y color:SolidPeso molecular:461.32LYP-IN-3
<p>LYP-IN-3 (compound D34) is a selective Lymphoid-tyrosine phosphatase (LYP) inhibitor (Ki=0.93 μM) that modulates the T-cell receptor (TCR) signaling pathway</p>Fórmula:C35H27NO6SPureza:98%Forma y color:SolidPeso molecular:589.66BDM_92499
<p>BDM_92499 is a nanomolar, selective IRAP inhibitor with an IC50 of 3.4 nM. It also inhibits ERAP1 and ERAP2, with IC50 values of 0.46 μM and 4.2 μM, respectively.</p>Forma y color:Odour SolidL-Isoleucyl-L-arginine
CAS:<p>L-Isoleucyl-L-arginine, a dipeptide composed of L-isoleucine and L-arginine, acts as a potent angiotensin-converting enzyme (ACE) inhibitor and is utilized in</p>Fórmula:C12H25N5O3Pureza:98%Forma y color:SolidPeso molecular:287.36Anticancer agent 232
Anticanceragent 232 (compound 12f) is a sugar hybrid designed from 1-azide glycosides derived from d-glucose, d-galactose, and d-mannose. The IC50 values for this compound are 1.05 μM against MCF-7 cells and 18.03 μM for MDA-MB231 cells.Fórmula:C32H31BrN4O11Peso molecular:726.117271-(2-Quinoxalinyl)-1,2,3,4-butanetetrol
CAS:<p>1-(2-Quinoxalinyl)-1,2,3,4-butanetetrol is a quinoxaline derivative and endogenous metabolite applicable to biochemical experiments and drug synthesis research.</p>Fórmula:C12H14N2O4Pureza:99.49%Forma y color:SolidPeso molecular:250.25

