
Metabolismo
Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.
Subcategorías de "Metabolismo"
- AhR(41 productos)
- Aminopeptidasa(67 productos)
- CETP(18 productos)
- Anhídrido carbónico(178 productos)
- Caseína quinasa(130 productos)
- DHFR(33 productos)
- Descarboxilasa(4 productos)
- Deshidrogenasa(271 productos)
- FAAH(64 productos)
- FXR(58 productos)
- Factor Xa(80 productos)
- Ácido graso sintasa(33 productos)
- Ferroptosis(215 productos)
- GR(3 productos)
- GSNOR(3 productos)
- Glucoquinasa(54 productos)
- HIF / HIF Prolilhidroxilasa(142 productos)
- HMG-CoA reductasa(33 productos)
- Hidroxilasa(30 productos)
- IDO(82 productos)
- LDL(8 productos)
- Lipasa(98 productos)
- Lípido(58 productos)
- Lipoxigenasa(124 productos)
- MAO(87 productos)
- MPO(2 productos)
- NAMPT(36 productos)
- P450(6 productos)
- PAI-1(25 productos)
- PDE(166 productos)
- PED(1 productos)
- PKM(15 productos)
- PPAR(165 productos)
- Fosfolipasa(82 productos)
- ROR(42 productos)
- Receptor de retinoides(29 productos)
- SGK(11 productos)
- Tiorredoxina(12 productos)
- Transferasa(30 productos)
- Transportador(42 productos)
- UGT(4 productos)
- Inhibidores de la xantina oxidasa (XO)(9 productos)
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Se han encontrado 8628 productos de "Metabolismo"
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N-Desmethyl Bendamustine
CAS:<p>N-DesmethylBendamustine is a metabolite of Bendamustine. It exerts cytotoxic effects on various lymphoma cell lines and peripheral blood lymphocytes.</p>Fórmula:C15H19Cl2N3O2Forma y color:SolidPeso molecular:344.24α-Amylase-IN-4
<p>α-Amylase-IN-4 (Compd 10y) exhibits the highest level of amylase inhibition, demonstrating an IC50 value of 17.83 ± 0.14 μg/mL [1].</p>Forma y color:Odour SolidMAGL-IN-8
<p>MAGL-IN-8 (compound 13) serves as a reversible inhibitor of monoacylglycerol lipase (MAGL), exhibiting an inhibitory concentration half-maximal (IC50) value of</p>Pureza:98%Forma y color:Odour SolidDactylocycline A
CAS:<p>Dactylocyclines A: novel antibiotic from Dactylosporangium, effective against tetracycline-resistant microbes.</p>Fórmula:C31H40ClN3O13Pureza:98%Forma y color:SolidPeso molecular:698.11COMT-IN-2
<p>COMT-IN-2 (compound 9) is the most potent inhibitor of COMT, exhibiting selective inhibition for brain (IC50=24 nM) and liver (IC50=81 nM) MB-COMT compared to the liver S-COMT isoform (IC50=620 nM).</p>Forma y color:Odour SolidFABP4-IN-3
<p>FABP4-IN-3 (Compound C3) is a highly selective inhibitor of FABP4, with an inhibition constant (Ki) of 25 ± 3 nM for FABP4 and a Ki of 15.03 μM for FABP3, showcasing a selectivity factor of 601 times over FABP3. It also demonstrates metabolic stability and potent anti-inflammatory activity in cells, making it a promising candidate for research in metabolic disorders, cardiac dysfunction, and inflammation-related diseases.</p>Fórmula:C20H16ClNO2Peso molecular:337.0869618:0,22:6 PS sodium
CAS:<p>Sodium 18:0,22:6 phosphatidylserine (PS) is a lipid found within synaptic vesicles alongside cholesterol, utilized in metabolic research [1].</p>Fórmula:C46H77NNaO10PForma y color:SolidPeso molecular:858.07NADP+ (sodium salt hydrate)
CAS:<p>NADP+ is the oxidized cofactor form of NADPH, vital for cell survival, redox balance, and signaling; synthesized from NAD+ and ATP.</p>Fórmula:C21H30N7NaO18P3Forma y color:SolidPeso molecular:784.413Fumiquinazoline D
CAS:Fumiquinazoline D, from A. fumigatus, inhibits Gram-positive/negative bacteria (MIC 8-16 μg/ml) and F. solani, C. albicans (MIC 32, 64 μg/ml).Fórmula:C24H21N5O4Forma y color:SolidPeso molecular:443.463RORγt inhibitor 1
CAS:<p>RORγt inhibitor 1 is a RORγt allosteric inhibitor with an IC 50 value of 1 nM.</p>Fórmula:C23H21ClFN3O4Forma y color:SolidPeso molecular:457.89PDE10A-IN-5
<p>PDE10A-IN-5 (Compound A30) is an orally active inhibitor of phosphodiesterase 10A (PDE10A) with an IC50 value of 3.5 nM. By inhibiting PDE10A, it activates the cyclic adenosine monophosphate (cAMP)-related signaling pathway, exhibiting activity against pulmonary vascular remodeling. This compound is applicable to research in the field of pulmonary arterial hypertension.</p>Forma y color:Odour Solid1α, 25-Dihydroxy VD2-D6
CAS:<p>1alpha, 25-Dihydroxy VD2-D6 is a deuterated form of vitamin D.</p>Fórmula:C28H44O3Pureza:98%Forma y color:SolidPeso molecular:434.683-Hydroxysebacic acid
CAS:<p>3-Hydroxysebacic acid, an endogenous metabolite found in urine, is utilized in the study of Medium Chain Acyl-CoA Dehydrogenase Deficiency (MCADD) [1] [2].</p>Fórmula:C10H18O5Forma y color:SolidPeso molecular:218.25Thymopentin acetate
CAS:<p>Thymopentin acetate: an immunomodulatory peptide from thymus cells with a 30-sec half-life, boosts T-cell production from hESCs.</p>Fórmula:C32H53N9O11Forma y color:SolidPeso molecular:739.82Irsenontrine maleate
CAS:<p>Irsenontrine (E2027) maleate is a selective and orally active inhibitor of phosphodiesterase 9 (PDE9). It can be utilized in the study of neurological diseases.</p>Fórmula:C26H26N4O7Forma y color:SolidPeso molecular:506.5157-Hydroxyneolamellarin A
CAS:<p>7-Hydroxyneolamellarin A, from Dendrilla nigra, inhibits HIF-1α and VEGF in cancer research.</p>Fórmula:C24H19NO5Forma y color:SolidPeso molecular:401.41LysoFos Glycerol 16
CAS:LysoFos Glycerol 16 is a useful organic compound for research related to life sciences. The catalog number is TF0118 and the CAS number is 326495-22-1.Fórmula:C22H44NaO9PForma y color:SolidPeso molecular:506.54911β-HSD1 inibitor 19
CAS:3-chloro-4-sulfonyl-Benzonitrile inhibits hHSD1/mHSD1, IC50: 16nM/10nM.Fórmula:C19H16ClF4N3O2SPureza:99.58%Forma y color:SoildPeso molecular:461.86PDE1-IN-5
<p>PDE1-IN-5 (Compound 10c) is a selective PDE1C inhibitor with an IC50 of 15 nM, exhibiting anti-inflammatory properties through the inhibition of iNOS, TNF-α, IL</p>Fórmula:C27H29FN4OForma y color:SolidPeso molecular:444.54DSPE-PEG-Maleimide ammonium (MW 2000)
<p>DSPE-PEG-Maleimide (ammonium) (MW 2000) is a compound containing DSPE phospholipids and maleimide, designed for the preparation of nanoscale lipid carriers. It is applicable in the study of drug delivery systems.</p>Forma y color:Odour Solid

