
Metabolismo
Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.
Subcategorías de "Metabolismo"
- AhR(41 productos)
- Aminopeptidasa(67 productos)
- CETP(18 productos)
- Anhídrido carbónico(178 productos)
- Caseína quinasa(130 productos)
- DHFR(33 productos)
- Descarboxilasa(4 productos)
- Deshidrogenasa(270 productos)
- FAAH(64 productos)
- FXR(58 productos)
- Factor Xa(80 productos)
- Ácido graso sintasa(33 productos)
- Ferroptosis(215 productos)
- GR(3 productos)
- GSNOR(3 productos)
- Glucoquinasa(54 productos)
- HIF / HIF Prolilhidroxilasa(142 productos)
- HMG-CoA reductasa(33 productos)
- Hidroxilasa(30 productos)
- IDO(82 productos)
- LDL(8 productos)
- Lipasa(97 productos)
- Lípido(59 productos)
- Lipoxigenasa(125 productos)
- MAO(87 productos)
- MPO(2 productos)
- NAMPT(36 productos)
- P450(6 productos)
- PAI-1(25 productos)
- PDE(166 productos)
- PED(1 productos)
- PKM(15 productos)
- PPAR(164 productos)
- Fosfolipasa(82 productos)
- ROR(42 productos)
- Receptor de retinoides(29 productos)
- SGK(11 productos)
- Tiorredoxina(12 productos)
- Transferasa(30 productos)
- Transportador(42 productos)
- UGT(4 productos)
- Inhibidores de la xantina oxidasa (XO)(9 productos)
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Se han encontrado 8625 productos de "Metabolismo"
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Ingenol disoxate
CAS:<p>Ingenol disoxate (LEO43204) is a compound for treating actinic keratosis, a natural Euphorbia peplus extract.</p>Fórmula:C28H37NO7Forma y color:SolidPeso molecular:499.6XW-032
<p>XW-032 is an apo-IDO1 inhibitor with an IC50 of 21 nM. In the CT26 syngeneic mouse model, XW-032 demonstrates significant in vivo antitumor efficacy with a TGI of 63%, showing potential for cancer research applications.</p>Forma y color:Odour SolidFerroleuton
<p>Ferroleuton is a selective competitive inhibitor of 5-lipoxygenase with an IC50 of 0.21 μM. It demonstrates antioxidant properties, clearing 86% of DPPH at 50 μM and exhibiting activities in ABTS (EC50 = 19.42 μM) and FRAP (EC50 = 3.32 μM) assays.</p>Fórmula:C13H16FeN2O2Forma y color:SolidPeso molecular:288.12m-PEG8-DSPE
<p>m-PEG8-DSPE is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules.</p>Fórmula:C59H116NO17PPureza:98%Forma y color:SolidPeso molecular:1142.52Atocalcitol
CAS:<p>Atocalcitol is a vitamin D analog. It also acts as an agonist of alcitriol receptor.</p>Fórmula:C32H46O4Pureza:98%Forma y color:SolidPeso molecular:494.71GPX4-IN-16
<p>GPX4-IN-16 ((R)-9i) is a potent inhibitor of GPX4 with a KD value of 20.4 nM, exhibiting cytotoxic properties and anticancer activity.</p>Fórmula:C29H24N4O3S2Forma y color:SolidPeso molecular:540.656Naroparcil
CAS:<p>Naroparcil, an oral thioglycoside, has antithrombotic properties and alters thrombin complex formation.</p>Fórmula:C19H17NO4S2Pureza:98.71% - 99.88%Forma y color:SolidPeso molecular:387.47Leuhistin
CAS:Leuhistin is an aminopeptidases N inhibitor isolated from Bacillus laterosporus BMI156-14F1.Fórmula:C11H19N3O3Pureza:98%Forma y color:White To Off-White SolidPeso molecular:241.29Coformycin
CAS:<p>Coformycin is a ribonucleoside antibiotic synergist and adenosine deaminase inhibitor.</p>Fórmula:C11H16N4O5Pureza:98%Forma y color:SolidPeso molecular:284.27Propiverine N-oxide
CAS:<p>Propiverine N-oxide is the primary metabolite of propiverine hydrochloride, and it influences bladder contraction and saliva secretion in miniature pigs.</p>Fórmula:C23H29NO4Forma y color:SolidPeso molecular:383.48ICMT-IN-35
<p>ICMT-IN-35 (compound 10n), an ICMT inhibitor with an IC50 value of 0.8 μM, is a FTPA-triazole derivative.</p>Forma y color:Odour SolidSofosbuvir impurity E
<p>Sofosbuvir impurity E, a less active byproduct, inhibits HCV RNA replication with potent anti-HCV effects.</p>Fórmula:C22H29FN3O9PPureza:98%Forma y color:SolidPeso molecular:529.45α-Glucosidase-IN-83
<p>α-Glucosidase-IN-83 (compound I-1) is a potent inhibitor of α-glucosidase, demonstrating an IC50 of 1.49 μg/mL. This compound effectively reduces blood glucose levels in vivo.</p>Fórmula:C25H20N4O6SForma y color:SolidPeso molecular:504.514PDE5-IN-10
<p>PDE5-IN-10 (compound 4b), a potent phosphodiesterase type 5 (PDE5) inhibitor, exhibits an effective half-maximal inhibitory concentration (IC50) of 20 nM,</p>Fórmula:C21H20N4O2Forma y color:SolidPeso molecular:360.41BE2647
<p>BE2647 is a selective inhibitor of the mitochondrial pyruvate carrier (MPC), with an EC50 of 70 nM. It exhibits good metabolic stability in mouse liver microsomes. BE2647 can be utilized in research related to metabolic diseases, metabolic-associated steatotic liver disease (MASLD), or metabolic-associated steatohepatitis (MASH).</p>Fórmula:C13H7Br2N3O2Forma y color:SolidPeso molecular:397.022α-Glucosidase-IN-82
<p>α-Glucosidase-IN-82 (compound 8l) is a potent inhibitor of α-glucosidase, with an IC50 value of 13.66 μM. Its inhibitory activity is 52 times greater than that of Acarbose.</p>Fórmula:C30H24N4O4Forma y color:SolidPeso molecular:504.536Gluconapin
CAS:<p>Gluconapin serves as a precursor to sulforaphane, an effective anticancer isothiocyanate. It has been found to reduce the increase in plasma triglycerides induced by corn oil consumption in mice.</p>Fórmula:C11H19NO9S2Forma y color:SolidPeso molecular:373.4Ascorbate oxidase
CAS:<p>Ascorbate oxidase, a REDOX enzyme, catalyzes ascorbic acid and oxygen to dehydroascorbic acid, regulating the extracellular matrix.</p>Forma y color:SolidGeranyl pyrophosphate triammonium
CAS:<p>Geranyl pyrophosphate, an intermediary for making cholesterol, terpenes, and others, forms from dimethylallyl and isopentenyl pyrophosphates.</p>Fórmula:C10H29N3O7P2Forma y color:SolidPeso molecular:365.304TDO-IN-2
<p>TDO-IN-2 is an orally active TDO inhibitor with an IC50 of 1.25 μM. It exhibits antitumor activity in a Hepa1-6 liver cancer allograft mouse model. Additionally, TDO-IN-2 works synergistically with PD-1/PD-L1 inhibitor BMS-202, making it useful for studying tumor immune tolerance.</p>Fórmula:C20H15N3O3Forma y color:SolidPeso molecular:345.11134

