
Metabolismo
Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.
Subcategorías de "Metabolismo"
- AhR(41 productos)
- Aminopeptidasa(67 productos)
- CETP(18 productos)
- Anhídrido carbónico(178 productos)
- Caseína quinasa(130 productos)
- DHFR(33 productos)
- Descarboxilasa(4 productos)
- Deshidrogenasa(269 productos)
- FAAH(64 productos)
- FXR(58 productos)
- Factor Xa(80 productos)
- Ácido graso sintasa(32 productos)
- Ferroptosis(215 productos)
- GR(3 productos)
- GSNOR(3 productos)
- Glucoquinasa(54 productos)
- HIF / HIF Prolilhidroxilasa(142 productos)
- HMG-CoA reductasa(33 productos)
- Hidroxilasa(30 productos)
- IDO(82 productos)
- LDL(8 productos)
- Lipasa(97 productos)
- Lípido(59 productos)
- Lipoxigenasa(124 productos)
- MAO(87 productos)
- MPO(2 productos)
- NAMPT(36 productos)
- P450(6 productos)
- PAI-1(25 productos)
- PDE(166 productos)
- PED(1 productos)
- PKM(15 productos)
- PPAR(164 productos)
- Fosfolipasa(82 productos)
- ROR(42 productos)
- Receptor de retinoides(29 productos)
- SGK(11 productos)
- Tiorredoxina(12 productos)
- Transferasa(30 productos)
- Transportador(42 productos)
- UGT(4 productos)
- Inhibidores de la xantina oxidasa (XO)(9 productos)
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Se han encontrado 8626 productos de "Metabolismo"
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ENPP3 Inhibitor 1
CAS:<p>ENPP3 Inhibitor 1 is a selective inhibitor of ENPP3, exhibiting an IC50 value of 0.15 µM, compared to an IC50 of 41.4 µM for ENPP1. It demonstrates antitumor effects against breast and cervical cancers.</p>Fórmula:C20H14F3NO5SForma y color:SolidPeso molecular:437.39PTP1B-IN-27
<p>PTP1B-IN-27 (Compound 7i) is an inhibitor of protein tyrosine phosphatase 1-B (PTP-1B) with an IC50 of 8.2 µM. Additionally, it inhibits α-glucosidase with an IC50 of 120 µM and exhibits competitive inhibition characteristics (Ki=118 µM).</p>Fórmula:C26H24FN7O2SPeso molecular:517.16962α-Glucosidase-IN-89
<p>α-Glucosidase-IN-89 (8g) is an inhibitor of α-glucosidase, with an IC50 of 0.5 μM and a Ki of 0.46 μM.</p>Forma y color:Odour SolidEflucimibe
CAS:<p>Eflucimibe (L0081), an ACAT inhibitor, treats cardiovascular, endocrine, and metabolic diseases, and helps in atherosclerosis and hyperlipidemia research.</p>Fórmula:C29H43NO2SPureza:99.17% - 99.43%Forma y color:SolidPeso molecular:469.72CHEMBL1276927
CAS:<p>CHEMBL1276927 (N-(3-(1H-benzo[d]imidazol-2-yl)phenyl)-3-methylbenzamide) shows antibacterial and antiparasitic activities against Chlamydia pneumoniae and</p>Fórmula:C21H17N3OPureza:99.86%Forma y color:SolidPeso molecular:327.38Desoxycarbadox
CAS:<p>Desoxycarbadox, derived from Carbadox, is a quinoxaline-di-N-oxide antibiotic compound.</p>Fórmula:C11H10N4O2Forma y color:SolidPeso molecular:230.227Ritonavir metabolite
CAS:<p>Ritonavir metabolite is a Ritonavir metabolite, which is a inhibitor of HIV protease.</p>Fórmula:C32H45N5O3SPureza:98%Forma y color:SolidPeso molecular:579.80PLA2-IN-1
<p>PLA2-IN-1 (Compound 7) is a potent and selective inhibitor of phospholipase A (PLA2) with an IC50 value of 1 nM. It effectively inhibits PLA2-induced coagulation disorders in vitro and shows potential for use as an antidote for snake bites caused by cobra venom.</p>Forma y color:Odour Solidα-Amylase/α-Glucosidase-IN-15
<p>α-Amylase/α-Glucosidase-IN-15 (compound 6C) is an orally active inhibitor of α-glucosidase (α-Glucosidase) and α-amylase (α-amylase), with IC50 values of 21 μM and 61 μM, respectively.</p>Fórmula:C26H24N4O3SPeso molecular:472.15691(S)-3-Thienylglycine
CAS:<p>(S)-3-Thienylglycine is a thiophene derivative and can be used to investigate the genotoxicity of the similar structures with thiophene derivatives.</p>Fórmula:C6H7NO2SPureza:99.68%Forma y color:SolidPeso molecular:157.19α-Pyrone
CAS:<p>Alpha-Pyrone exhibits inhibitory activity against tyrosinase, carbonic anhydrase 1, and carbonic anhydrase 9</p>Fórmula:C5H4O2Forma y color:SolidPeso molecular:96.08Fenbendazole sulfone
CAS:<p>Fenbendazole sulfone is a minor metabolite of fenbendazole, exhibiting inhibitory activity against 7-ethoxycoumarin O-deethylase in rat liver.</p>Fórmula:C15H13N3O4SPureza:98.70%Forma y color:SolidPeso molecular:331.35Sarcophine
CAS:<p>Sarcophine is a natural cembranoid from the Red Sea soft coral Sarcophyton glaucum.</p>Fórmula:C20H28O3Forma y color:SolidPeso molecular:316.441D-Sedoheptulose 7-phosphate
CAS:<p>D-Sedoheptulose 7-phosphate, a precursor to group III heptaic acid and group IV hygromycin B, converts to NDP-heptose via similar pathways.</p>Fórmula:C7H15O10PPureza:98%Forma y color:SolidPeso molecular:290.16Mitochondrial respiration-IN-1 hydrobromide
<p>Mitochondrial inhibitor 49 (respiration-IN-1 hydrobromide, IC50=8.8 mg/mL) from US20110301180A1 reduces platelet respiration.</p>Forma y color:SolidPtdIns-(3,4,5)-P3 (1,2-dihexanoyl) (ammonium salt)
CAS:<p>PIP3, a minor yet critical phospholipid for cell signaling, resists PLC cleavage and anchors PH domain proteins, affecting cytoskeletal and membrane dynamics.</p>Fórmula:C21H45NO22P4Forma y color:SolidPeso molecular:787.471Fluticasone dimer impurity
CAS:<p>Fluticasone dimer impurity: a dimer of Fluticasone Propionate, a potent corticosteroid.</p>Fórmula:C43H51F5O8SForma y color:SolidPeso molecular:822.92Cellobiosan
CAS:<p>Cellobiosan is an anhydro sugar formed during biofuel production from the fast pyrolysis of wood.</p>Fórmula:C12H20O10Forma y color:SolidPeso molecular:324.282Terpendole C
CAS:<p>Terpendole C, an indole diterpene from A. yamanashiensis, inhibits ACAT with IC50 of 2.1 μM in rats, 0.46 μM in J774 cells, non-toxic.</p>Fórmula:C32H41NO5Forma y color:SolidPeso molecular:519.682Tetrahydropteroylpentaglutamate
CAS:<p>H4PteGlu5 strongly inhibits itself and tightly binds in vivo, almost irreversibly, as a coenzyme.</p>Fórmula:C39H51N11O18Pureza:98%Forma y color:SolidPeso molecular:961.89

