
Metabolismo
Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.
Subcategorías de "Metabolismo"
- AhR(41 productos)
- Aminopeptidasa(67 productos)
- CETP(18 productos)
- Anhídrido carbónico(178 productos)
- Caseína quinasa(130 productos)
- DHFR(33 productos)
- Descarboxilasa(4 productos)
- Deshidrogenasa(271 productos)
- FAAH(64 productos)
- FXR(58 productos)
- Factor Xa(80 productos)
- Ácido graso sintasa(33 productos)
- Ferroptosis(215 productos)
- GR(3 productos)
- GSNOR(3 productos)
- Glucoquinasa(54 productos)
- HIF / HIF Prolilhidroxilasa(142 productos)
- HMG-CoA reductasa(33 productos)
- Hidroxilasa(30 productos)
- IDO(82 productos)
- LDL(8 productos)
- Lipasa(98 productos)
- Lípido(58 productos)
- Lipoxigenasa(124 productos)
- MAO(87 productos)
- MPO(2 productos)
- NAMPT(36 productos)
- P450(6 productos)
- PAI-1(25 productos)
- PDE(166 productos)
- PED(1 productos)
- PKM(15 productos)
- PPAR(165 productos)
- Fosfolipasa(82 productos)
- ROR(42 productos)
- Receptor de retinoides(29 productos)
- SGK(11 productos)
- Tiorredoxina(12 productos)
- Transferasa(30 productos)
- Transportador(42 productos)
- UGT(4 productos)
- Inhibidores de la xantina oxidasa (XO)(9 productos)
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Se han encontrado 8628 productos de "Metabolismo"
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Daclatasvir Impurity C
CAS:<p>Daclatasvir Impurity C is an impurity found in Daclatasvir, a robust inhibitor of the HCV NS5A protein [1].</p>Fórmula:C29H32N6O3Forma y color:SolidPeso molecular:512.6ALR2-IN-1
CAS:<p>ALR2-IN-1: potent, selective inhibitor of ALR2 (IC50=1.42 μM), antiglycemic, antioxidant; for diabetes research.</p>Fórmula:C16H17N3O2SPureza:98.79%Forma y color:SoildPeso molecular:315.39S-Phenylmercapturic acid
CAS:<p>S-Phenylmercapturic acid is a metabolite of benzene that can be used as a biomarker to assess benzene exposure.</p>Fórmula:C11H13NO3SPureza:99.68%Forma y color:SolidPeso molecular:239.29DSPE-PEG2000-K237
<p>DSPE-PEG2000-K237 is a PEG compound consisting of DSPE and the KDR-targeting peptide (K237). K237 functionally disrupts the interaction between VEGF and KDR receptors, resulting in significant biological effects such as inhibition of angiogenesis and tumor growth. DSPE-PEG2000-K237 is applicable in drug delivery.</p>Forma y color:Odour Solid1,4-DPCA
CAS:<p>1,4-DPCA is an inhibitor of prolyl-hydroxylase with an IC50 of 2.4 µM for collagen hydroxylation in human foreskin fibroblasts and 60 μM for factor inhibiting</p>Fórmula:C13H8N2O3Pureza:97.77%Forma y color:SolidPeso molecular:240.213,3'-Bipyridine
CAS:<p>3,3'-Bipyridine is an inhibitor of CYP2A6, CYP3A4, and CYP2B6, and also inhibits gastric acid secretion in rats.</p>Fórmula:C10H8N2Forma y color:SolidPeso molecular:156.184-Hydroxytryptamine creatinine sulfate
CAS:<p>4-Hydroxytryptamine creatinine sulfate, a derivative of tryptamine, acts as an agonist for neurotransmitters.</p>Fórmula:C14H21N5O6SForma y color:SolidPeso molecular:387.41RORγ inverse agonist 1
CAS:<p>RORγ inverse agonist 1 has anti-inflammatory activity and can be used to treat rheumatism and psoriasis.</p>Fórmula:C22H20F3N3O3SPureza:99.68%Forma y color:SolidPeso molecular:463.47RORγ agonist 1
CAS:<p>RORγ agonist 1 is a highly potent and orally bioavailable compound that activates the RORγ receptor.</p>Fórmula:C29H27ClF4N2O4SForma y color:SolidPeso molecular:611.05PDE2A-IN-1
CAS:<p>PDE2A-IN-1 is a phosphodiesterase 2A (PDE2A) inhibitor with an IC 50 value of 1.3 nM.</p>Fórmula:C23H22F2N6Forma y color:SolidPeso molecular:420.468CB1151
CAS:<p>CB1151 is a 20-epi analogue of 1,25 dihydroxyvitamin D3 with anti-tumor effects. It inhibits MCF-7 cell growth (IC50: 0.82 nM).</p>Fórmula:C28H46O4Pureza:98%Forma y color:SolidPeso molecular:446.661,2-Dilinoleoyl-sn-glycerol
CAS:<p>1,2-Dilinoleoyl-sn-glycerol, a DAG with two linoleic acids, is in rat liver, spinach membranes, and indicates preeclampsia risk in pregnancy.</p>Fórmula:C39H68O5Forma y color:SolidPeso molecular:616.95Tanshinone IIA anhydride
CAS:<p>Tanshinone IIA anhydride: irreversible inhibitor for human CE1 (Ki=1.9 nM) and hiCE (Ki=1.4 nM).</p>Fórmula:C19H18O4Forma y color:SolidPeso molecular:310.34Acetoacetic acid
CAS:<p>Acetoacetic acid(3-oxobutanoic acid) is a oxidative stress inducer, gluconeogenesis, and can be used as an indicator of in ketoacidosis.</p>Fórmula:C4H6O3Pureza:99.59% - 99.85%Forma y color:SolidPeso molecular:102.09MS1262-C3-amide-C10-amine
<p>MS1262-C3-amide-C10-amine is an E3 Ligase Ligand-Linker conjugate. It includes a GLP ligand targeting the E3 ligase SPOP and a PROTAC linker. This compound can be utilized in designing PROTACs such as example [MS479].</p>Forma y color:Odour Solidtetranor-PGAM
CAS:<p>PGE2 is a biomarker for inflammation and disease; its unstable urinary metabolite, tetranor-PGEM, and its byproduct, tetranor-PGAM, indicate biosynthesis.</p>Fórmula:C16H22O6Forma y color:SolidPeso molecular:310.346TKL-IN-1
<p>TKL-IN-1 (compound 7r) serves as an inhibitor of transketolase (Transketolase) and can be utilized as an herbicide. This compound effectively hampers the growth of Digitaria sanguinalis (Ds) and Amaranthus retroflexus (Ar).</p>Fórmula:C20H12ClN5OS2Forma y color:SolidPeso molecular:437.93CALP3 TFA(261969-05-5 free base)
<p>CALP3 TFA is a potent Ca2+ channel blocker that activates EF-hand motifs of Ca2+-binding proteins.</p>Fórmula:C46H69F3N10O11Pureza:98%Forma y color:SolidPeso molecular:995.1ER 50891 quarterhydrate
<p>ER 50891 quarterhydrate is a potent RARα (retinoic acid receptor α) antagonist that markedly diminishes the inhibitory effects of ATRA (all-trans retinoic acid</p>Fórmula:C29H24N2O2H2OForma y color:SolidPeso molecular:437.02ICMT-IN-35
<p>ICMT-IN-35 (compound 10n), an ICMT inhibitor with an IC50 value of 0.8 μM, is a FTPA-triazole derivative.</p>Forma y color:Odour Solid

