Metabolismo
Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.
Subcategorías de "Metabolismo"
- AhR(41 productos)
- Aminopeptidasa(67 productos)
- CETP(18 productos)
- Anhídrido carbónico(177 productos)
- Caseína quinasa(130 productos)
- DHFR(32 productos)
- Descarboxilasa(4 productos)
- Deshidrogenasa(267 productos)
- FAAH(63 productos)
- FXR(58 productos)
- Factor Xa(80 productos)
- Ácido graso sintasa(32 productos)
- Ferroptosis(215 productos)
- GR(3 productos)
- GSNOR(3 productos)
- Glucoquinasa(53 productos)
- HIF / HIF Prolilhidroxilasa(142 productos)
- HMG-CoA reductasa(32 productos)
- Hidroxilasa(30 productos)
- IDO(82 productos)
- LDL(8 productos)
- Lipasa(96 productos)
- Lípido(59 productos)
- Lipoxigenasa(124 productos)
- MAO(87 productos)
- MPO(2 productos)
- NAMPT(36 productos)
- P450(6 productos)
- PAI-1(25 productos)
- PDE(165 productos)
- PED(1 productos)
- PKM(15 productos)
- PPAR(164 productos)
- Fosfolipasa(82 productos)
- ROR(42 productos)
- Receptor de retinoides(29 productos)
- SGK(11 productos)
- Tiorredoxina(12 productos)
- Transferasa(30 productos)
- Transportador(42 productos)
- UGT(4 productos)
- Inhibidores de la xantina oxidasa (XO)(9 productos)
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Se han encontrado 8597 productos de "Metabolismo"
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2,7"-Phloroglucinol-6,6'-bieckol
CAS:<p>2,7"-Phloroglucinol-6,6'-bieckol serves as an effective oral dual α-amylase/α-glucosidase inhibitor, demonstrating IC 50 concentrations of 6.94 μM and 23.35 μM, respectively. This compound is beneficial in mitigating postprandial hyperglycemia among diabetic mice and is applicable in diabetes research [1].</p>Fórmula:C48H30O23Forma y color:SolidPeso molecular:974.742,3-Indolobetulonic Acid
CAS:<p>2,3-Indolobetulonic acid is pentacyclic triterpenoid derivative of betulonic acid and an inhibitor of α-glucosidase (IC50= 1.8 μM).1</p>Fórmula:C36H49NO2Forma y color:SolidPeso molecular:527.793Maltodextrin, dextrose equivalent 16.5-19.5
CAS:<p>Maltodextrin (DE 16.5-19.5) is an inactive pharma excipient that enhances drug stability, solubility, and processing.</p>Fórmula:(C6H10O5)n·xH2OForma y color:SolidN-Acetyl lysyltyrosylcysteine amide acetate
<p>N-Acetyl lysyltyrosylcysteine amide acetate is an effective and selective tripeptide inhibitor of myeloperoxidase (MPO).</p>Fórmula:C22H35N5O7SPureza:98%Forma y color:SolidPeso molecular:513.61β-N-Acetylhexosaminidase
CAS:<p>β-N-Acetylhexosaminidase is an exoglycosidase that catalyzes the hydrolysis of terminal non-reducing β-N-acetylgalactosamine and glucosamine residues in</p>Forma y color:SolidD-Sedoheptulose-7-phosphate (barium salt)
CAS:<p>D-Sedoheptulose-7-phosphate: Key in pentose phosphate path, carbon fixation, and compound biosynthesis.</p>Fórmula:C7H17BaO10PForma y color:SolidPeso molecular:429.504ARL67156 trisodium hydrate
<p>ARL67156 trisodium hydrate inhibits ecto-ATPase, NTPDase1, NTPDase3, NPP1 (Kis 11-18µM), for calcific valve disease, asthma research.</p>Fórmula:C15H23Br2N5Na3O13P3Forma y color:SolidPeso molecular:834.61Avellanin B
CAS:<p>Avellanin B is a fungal metabolite.</p>Fórmula:C30H37N5O5Forma y color:SolidPeso molecular:547.6564-Hydroxy Atorvastatin calcium salt
CAS:<p>4-Hydroxy Atorvastatin calcium salt is metabolised by cytochrome P450 CYP3A4 and has antimicrobial and anti-microbial activity.</p>Fórmula:C66H68CaF2N4O12Forma y color:SolidPeso molecular:1187.34α-Glucosidase-IN-83
<p>α-Glucosidase-IN-83 (compound I-1) is a potent inhibitor of α-glucosidase, demonstrating an IC50 of 1.49 μg/mL. This compound effectively reduces blood glucose levels in vivo.</p>Fórmula:C25H20N4O6SForma y color:SolidPeso molecular:504.514PKM2 activator 6
<p>Compound Z10 (PKM2 activator 6) serves as both a PKM2 activator and a PDK1 inhibitor, exhibiting dissociation constants (K D ) of 121 μM and 19.6 μM,</p>Forma y color:Odour SolidVoclosporin
CAS:<p>Voclosporin (ISAtx-247) is a novel and orally available calcium-modulated phosphatase (CN; PP2B) inhibitor and immunosuppressant for the treatment of lupus</p>Fórmula:C63H111N11O12Pureza:99.85%Forma y color:SolidPeso molecular:1214.622-NP-AMOZ
CAS:<p>2-NP-AMOZ, a 2-nitrophenyl AMOZ, detects protein-bound AMOZ, a Furaltadone metabolite.</p>Fórmula:C15H18N4O5Forma y color:SolidPeso molecular:334.33PTP1B-IN-13
CAS:<p>PTP1B-IN-13 inhibits PTP1B at an allosteric site with 1.59 μM IC50.</p>Fórmula:C24H25N3O3S2Forma y color:SolidPeso molecular:467.6DSPE-PEG1000-LyP-1
<p>DSPE-PEG1000-LyP-1 is a PEG compound composed of DSPE and a nine-residue peptide (LyP-1). LyP-1 specifically targets tumor-associated lymphatic vessels and macrophages.</p>Forma y color:Odour SolidWVSAV
<p>WVSAV is a ligand for the PDZ2 domain (tyrosine phosphatase) with a dissociation constant (Kd) of 111 μM. It is utilized in studies of protein-ligand interactions.</p>Fórmula:C27H40N6O7Forma y color:SolidPeso molecular:560.64DSPE-PEG-Maleimide ammonium (MW 2000)
<p>DSPE-PEG-Maleimide (ammonium) (MW 2000) is a compound containing DSPE phospholipids and maleimide, designed for the preparation of nanoscale lipid carriers. It is applicable in the study of drug delivery systems.</p>Forma y color:Odour SolidBipolamine G
CAS:<p>Bipolamine G is an antibacterial polyketide alkaloid [1] .</p>Fórmula:C21H28N2O4Forma y color:SolidPeso molecular:372.46GSK-3β/CK-1δ-IN-1
<p>GSK-3β/CK-1δ-IN-1 (8d) is a dual inhibitor of GSK-3β and CK-1δ that can cross the blood-brain barrier, with IC50 values of 0.77 μM and 0.57 μM, respectively. GSK-3β/CK-1δ-IN-1 (8d) is applicable in neuroblastoma research.</p>Fórmula:C22H17F3N4OForma y color:SolidPeso molecular:410.39Herbicidal agent 6
<p>Herbicidal agent 6 (D15) functions as a Transketolase (TKL) inhibitor and exhibits herbicidal activity.</p>Forma y color:Odour Solid(-)-OPC-51803
CAS:<p>(-)-OPC-51803 is an antidiuretic hormone V2 receptor agonist used in the treatment of nocturia and urinary incontinence.</p>Fórmula:C26H32ClN3O2Pureza:98.73% - 99.59%Forma y color:SoildPeso molecular:4541-Palmitoyl-2-linoleoyl PE
CAS:<p>Phosphatidylethanolamine PLPE: a cell membrane component, studied for anandamide biosynthesis, sPLA2-IIA activity substrate.</p>Fórmula:C39H74NO8PForma y color:SolidPeso molecular:715.994Adrenocorticotropic Hormone (ACTH) (18-39), human
CAS:<p>ACTH (18-39), or Corticotropin-like Peptide, boosts insulin, amylase, and protein secretion dose-dependently.</p>Fórmula:C112H165N27O36Pureza:98%Forma y color:SolidPeso molecular:2465.67Carbonic anhydrase inhibitor 31
<p>Carbonic anhydrase inhibitor31 is an mtCA2 inhibitor (Ki: 5.2 nM) that can be used in antituberculosis research.</p>Fórmula:C24H20N6O5SForma y color:SolidPeso molecular:504.12159IR-117-17
CAS:<p>IR-117-17 is an ionizable cationic amino lipid that targets the airways. It is degradable via esterase cleavage, making it less likely to accumulate with repeated dosing.</p>Fórmula:C59H110N2O5Forma y color:SolidPeso molecular:927.52Cavosonstat
CAS:<p>Cavosonstat (N91115) is an oral GSNOR inhibitor aiding CFTR in cystic fibrosis.</p>Fórmula:C16H10ClNO3Pureza:98.91%Forma y color:SolidPeso molecular:299.71NMTCA
CAS:<p>NMTCA (NMTPRO) is a sulfur-containing N-nitrosamino acid utilized as an endogenous nitrosation indicator in gas chromatography-thermal energy analysis.</p>Fórmula:C5H8N2O3SForma y color:SolidPeso molecular:176.19Nucleocidin
CAS:<p>Nucleocidin, an antitrypanosomal antibiotic, inhibits the transfer of labeled amino acids from S-RNA to protein.</p>Fórmula:C10H13FN6O6SPureza:98%Forma y color:SolidPeso molecular:364.3111R-CaN-AID
CAS:<p>11R-CaN-AID is a potent, cell-permeant inhibitor of calcineurin [1] [2].</p>Fórmula:C135H248N70O34S2Forma y color:SolidPeso molecular:3459.99Speract
CAS:<p>Speract, a peptide from sea urchin eggs, regulates sperm motility and stimulates sperm mitochondrial metabolism.</p>Fórmula:C38H57N11O14Pureza:98%Forma y color:SolidPeso molecular:891.93Kouitchenside G
CAS:<p>Kouitchenside G, a natural compound extracted from Swertia kouitchensis, demonstrates inhibitory activity against α-Glucosidase, showcasing an IC 50 value of</p>Fórmula:C27H32O15Forma y color:SolidPeso molecular:596.531-Palmitoyl Lysophosphatidic Acid
CAS:<p>1-Palmitoyl Lysophosphatidic Acid boosts antibiotics against P. aeruginosa by binding Ca2+ and Mg2+.</p>Fórmula:C19H39O7PPureza:98%Forma y color:SolidPeso molecular:410.48Lactosylsphingosine (d18:1)
CAS:<p>Lactosylsphingosine (d18:1) is a sphingolipid with a lactose moiety that can inhibit fMetLeuPhe-induced cell aggregation at a concentration of 1 μm.</p>Fórmula:C30H57NO12Forma y color:SolidPeso molecular:623.77ACAT-IN-5
CAS:<p>ACAT-IN-5 inhibits ACAT, suppressing NF-κB-mediated transcription.</p>Fórmula:C32H49N3O5SForma y color:SolidPeso molecular:587.824-Hydroxybenzoic acid-d4
CAS:<p>4-Hydroxybenzoicacid-d4 is a deuterated form of 4-Hydroxybenzoicacid, which is a phenolic derivative of benzoic acid. It is effective in inhibiting most Gram-positive bacteria and some Gram-negative bacteria with an IC50 of 160 μg/mL.</p>Fórmula:C7H6O3Forma y color:SolidPeso molecular:142.15MS-PPOH
CAS:<p>MS-PPOH is a potent and selective inhibitor of cytochrome P450 (CYP) epoxygenase. MS-PPOH inhibits CYP2C8 and CYP2C9 with IC50s of 15 and 11 µM, respectively</p>Fórmula:C16H21NO4SPureza:99.39%Forma y color:SolidPeso molecular:323.41Inulobiose
CAS:<p>Inulobiose, a difructan disaccharide isolated from Pistacia vera L., demonstrates inhibitory effects on α-glycosidase (α-glycosidase) and α-amylase (α-amylase) activities, with IC50 values of 1.87 and 40.72 mg/mL respectively. It is utilized in research related to diabetes and glomerular filtration rate testing.</p>Fórmula:C12H22O11Forma y color:SolidPeso molecular:342.3(rac./meso)-Astaxanthin
CAS:<p>(rac./meso)-Astaxanthin (AstaREAL; AstaXin) is a carotenoid pigment primarily found in marine animals such as shrimp and salmon. It serves as an effective fat-soluble antioxidant.</p>Fórmula:C40H52O4Forma y color:SolidPeso molecular:596.84Lantanose A
CAS:<p>Lantanose A is a bioactive chemical from Lantana cumara roots.</p>Fórmula:C30H52O26Pureza:98%Forma y color:SolidPeso molecular:828.72DSPE-PEG2000-APRPG
<p>DSPE-PEG2000-APRPG is a PEG compound composed of DSPE and the APRPG peptide. It is utilized in drug delivery applications.</p>Forma y color:Odour SolidGirentuximab
CAS:<p>Girentuximab (G250) is an anti-carbonic anhydrase IX (CAIX) monoclonal antibody with anti-cancer activity for the study of uroepithelial carcinoma PET (ZiPUP).</p>Forma y color:LiquidPeso molecular:145.55 kDaCAXII-IN-2
<p>CAXII-IN-2 (compound 3j) is a highly effective inhibitor of CAXII. It demonstrates inhibitory activity against CA IX and CAXII, with Ki values of 27.4 nM and 4.0 nM, respectively.</p>Fórmula:C16H13FNO4PForma y color:SolidPeso molecular:333.05662Pestalotin
CAS:<p>Pestalotin, a fungal derivative, promotes rice seedling growth and sugar release, has antifungal properties, and is cytotoxic to certain cells.</p>Fórmula:C11H18O4Forma y color:SolidPeso molecular:214.26Daclatasvir Impurity B
CAS:<p>Daclatasvir Impurity B, a noted impurity of the antiviral agent Daclatasvir, acts as a potent inhibitor of the HCV NS5A protein [1].</p>Fórmula:C35H41N7O4Forma y color:SolidPeso molecular:623.7418-Hydroxycorticosterone
CAS:<p>18-Hydroxycorticosterone is a corticosteroid and corticosterone derivative, which can lead to serious electrolyte imbalances.</p>Fórmula:C21H30O5Pureza:98%Forma y color:SolidPeso molecular:362.46Trimetazidine-N-oxide
CAS:<p>Trimetazidine-N-oxide, main active metabolite of Trimetazidine, blocks 3-ketoyl CoA thiolase (IC50: 75nM) and has multiple protective properties.</p>Fórmula:C14H22N2O4Pureza:98%Forma y color:SolidPeso molecular:282.34Edoxaban impurity 6
CAS:<p>Edoxaban impurity 6 is a byproduct of the anticoagulant Edoxaban, a potent oral factor Xa inhibitor with Kis of 0.561 nM. Used to prevent stroke.</p>Fórmula:C16H22ClN5O3Forma y color:SolidPeso molecular:367.83hCAI/II-IN-10
<p>hCAI/II-IN-10 (Compound 5d) is an inhibitor of human carbonic anhydrase I and II (hCA I and hCA II), with IC50 values of 4.32 nM and 3.89 nM, respectively.</p>Fórmula:C24H17Cl2N3O3S2Forma y color:SolidPeso molecular:530.446Resveratrol-3-O-sulfate sodium
CAS:<p>Resveratrol-3-O-sulfate reduces IL-1α/β, IL-6, TNF-α in LPS-stimulated U-937 cells, inhibits Caco-2 cell growth, induces apoptosis, and binds mitoNEET.</p>Fórmula:C14H11NaO6SForma y color:SolidPeso molecular:330.29BI 1015550
CAS:<p>Nerandomilast (BI 1015550) is an orally active PDE4B inhibitor with IC50 of 7.2 nM.Cost-effective and quality-assured.</p>Fórmula:C20H25ClN6O2SPureza:98.06% - 99.71%Forma y color:SoildPeso molecular:448.97DSPE-PEG2000-TAASGVRSMH
<p>DSPE-PEG2000-TAASGVRSMH is a PEG compound composed of DSPE and TAASGVRSMH. This compound exhibits strong affinity for the NG2 proteoglycan on PC membranes. DSPE-PEG2000-TAASGVRSMH can be utilized for drug delivery.</p>Forma y color:Odour SolidAcrihellin
CAS:<p>Acrihellin is a cardioactive steroid, a cardiotonic drug.</p>Fórmula:C29H38O7Forma y color:SolidPeso molecular:498.61GQ-16
CAS:<p>GQ-16 is a partial agonist of PPARγ with a Ki of 160 nM. GQ-16 reduces adipogenic actions and promotes insulin Sensitization without weight gain.</p>Fórmula:C19H16BrNO3SPureza:99.84%Forma y color:SolidPeso molecular:418.3SDUY816
<p>SDUY816 is an orally active dual APN/NEP inhibitor, with IC50 values of 0.68 μM for APN and 6.9 μM for NEP. It exhibits analgesic properties and demonstrates good safety and pharmacokinetic profiles, having an oral bioavailability of 27% and a half-life of 4.02 hours in rats (oral, 10 mg/kg). SDUY816 is applicable for research in the field of neuropathic pain disorders.</p>Fórmula:C18H16IN3O3Forma y color:SolidPeso molecular:449.24hCAII/XII-IN-1
<p>hCAII/XII-IN-1 (compound 4l) is a potent inhibitor of hCAXII and hCAII, with Ki values of 8.4 nM and 9.4 nM, respectively. It plays a significant role in cancer research.</p>Fórmula:C22H20N4O6S2Forma y color:SolidPeso molecular:500.547Glucose 1-dehydrogenase
CAS:<p>Glucose 1-dehydrogenase, an enzyme, transforms glucose and NAD(P) into NAD(P)H and gluconic acid.</p>Forma y color:SolidL-739750 2HCl
<p>L-739750 2HCl is a potent inhibitor of peptidomimetic farnesyltransferase, a novel pseudopeptide mimetic with potential anticancer activity.</p>Fórmula:C23H41Cl2N3O6S2Pureza:98.69% - 99.16%Forma y color:SoildPeso molecular:590.62ZG-2305
<p>ZG-2305 is an effective, selective, and orally active inhibitor of FIH (factor inhibiting hypoxia-inducible factor (FIH)), with Ki values of 79.6 nM for FIH and 2786 nM for PHD2. This compound enhances the expression of the EGLN3 gene, reduces cellular triglyceride levels, and decreases lipid accumulation. ZG-2305 holds potential for research into obesity and fatty liver disease.</p>Fórmula:C17H11Cl2N3O5Forma y color:SolidPeso molecular:408.19ERAP1-IN-3
<p>ERAP1-IN-3 (compound 13) is a potent inhibitor of endoplasmic reticulum aminopeptidase 1 (ERAP1), with a pIC50 value of 8.6. ERAP1-IN-3 shows potential for research in cancer immunotherapy and autoimmune disease studies.</p>Fórmula:C22H22N2O4SForma y color:SolidPeso molecular:410.49Dilaurylglycerosulfate
CAS:<p>Dilauryl glycerol sulfate is an auxiliary emulsifier for lipase determination.</p>Fórmula:C27H56O6SPureza:98%Forma y color:SolidPeso molecular:508.811-epi-Chaetomugilin I
CAS:<p>11-epi-Chaetomugilin I, from Chaetomium globosum, has cytotoxic effects against P388, HL-60, L1210 leukemia, and KB carcinoma cells.</p>Fórmula:C22H27ClO5Forma y color:SolidPeso molecular:406.9Liarozole fumarate
CAS:<p>Liarozole fumarate is used as a retinoic acid metabolism blocking agent (RAMBA) and an aromatase inhibitor.</p>Fórmula:C17H13ClN4C4H4O4Pureza:98%Forma y color:SolidPeso molecular:482.88FCPR03
CAS:<p>FCPR03 is a selective inhibitor of phosphodiesterase 4 (PDE4) with IC50s of 31 nM, 47 nM, and 60 nM for PDE4B1, PDE4D7, and PDE4 catalytic domain, respectively.</p>Fórmula:C15H19F2NO3Pureza:99.94%Forma y color:SolidPeso molecular:299.31SHR168442
CAS:<p>SHR168442 is a potent RORγ modulator, exhibiting an IC50 value of 0.035 μM.</p>Fórmula:C23H25Cl2F2N3O3SForma y color:SolidPeso molecular:532.43Ninopterin
CAS:<p>Ninopterin is an experimental antineoplastic and folic acid analog.</p>Fórmula:C20H21N7O6Pureza:98%Forma y color:SolidPeso molecular:455.42(R)-Mephenytoin
CAS:<p>(R)-Mephenytoin ((–)-Mephenytoin) is the the R-enantiomer of Mephenytoin which is an anticonvulsant agent.</p>Fórmula:C12H14N2O2Pureza:99.95%Forma y color:SolidPeso molecular:218.25Coumachlor
CAS:<p>Coumachlor, a first-generation anticoagulant rodenticide, blocks the formation of prothrombin and inhibits blood coagulation causing internal haemorrhage.</p>Fórmula:C19H15ClO4Forma y color:SolidPeso molecular:342.77Nicotinic Acid Adenine Dinucleotide
CAS:<p>Nicotinic Acid Adenine Dinucleotide is a precursor of NAD (Nicotinamide adenine dinucleotide) and a substrate for glutamine-dependent NAD+ synthase</p>Fórmula:C21H26N6O15P2Forma y color:SoildPeso molecular:664.41Octanoyl Coenzyme A (sodium salt)
<p>Octanoyl Coenzyme A (sodium salt) inhibits citrate synthase and glutamate dehydrogenase with an IC50 of 0.4–1.6 mM.</p>Fórmula:C29H49N7NaO17P3SForma y color:SolidPeso molecular:915.71Ono EI-601
CAS:<p>Ono EI-601 is the main metabolite of ONO-5046, the human neutrophil elastase inhibitor .</p>Fórmula:C15H14N2O6SPureza:98%Forma y color:SolidPeso molecular:350.35hCA/VEGFR-2-IN-3
<p>hCA/VEGFR-2-IN-3 (compound 8j) is an indolinonylbenzenesulfonamide with potential as a dual inhibitor of cancer-associated hCA IX/XII and VEGFR-2.</p>Fórmula:C24H28N6O6SPureza:98%Forma y color:SolidPeso molecular:528.58TAK-778
CAS:<p>TAK-778, a derivative of ipriflavone, demonstrates the ability to stimulate bone growth in both in vitro and in vivo models.</p>Fórmula:C24H28NO7PSPureza:98%Forma y color:SolidPeso molecular:505.52BMT-297376
CAS:<p>BMT-297376, the optimized Linrodostat, is a potent IDO1 inhibitor.</p>Fórmula:C23H29F2N3O3Forma y color:SolidPeso molecular:433.5Acanthifolicin
CAS:<p>Acanthifolicin, an okadaic acid derivative, has been shown top inhibit protein phosphatase 1 with an IC50= 20 nM (similar to that of okadaic acid at 19 nM).</p>Fórmula:C44H68O13SForma y color:SolidPeso molecular:837.08N,S-Bis-Fmoc-Glutathione
CAS:<p>N,S-Bis-Fmoc-Glutathione is a potent inhibitor of glyoxalase II, exhibiting a K i of 0.32 mM [1].</p>Fórmula:C40H37N3O10SForma y color:SolidPeso molecular:751.84,8-Dioxa-3H-perfluorononanoic acid
CAS:<p>4,8-Dioxa-3H-perfluorononanoic acid, a type of per- and polyfluoroalkyl substance (PFAS), exhibits affinity for the human pregnane X receptor (hPXR) and demonstrates potential agonistic activity.</p>Fórmula:C7H2F12O4Forma y color:SolidPeso molecular:378.07Palmitoyl tripeptide-38
CAS:<p>Palmitoyl tripeptide-38 is a bioactive peptide renowned for its anti-aging properties [1].</p>Fórmula:C33H65N5O7SPureza:98%Forma y color:SolidPeso molecular:675.96Glycodehydrocholic acid
CAS:<p>Glycodehydrocholic acid is a bile acid compound formed by conjugation of bile acid with glycine.</p>Fórmula:C26H37NO6Forma y color:SolidPeso molecular:459.584-hydroxy Valsartan
CAS:<p>4-hydroxy Valsartan, a key valsartan metabolite, curbs epinephrine and collagen-caused platelet clumping, not ADP's.</p>Fórmula:C24H29N5O4Forma y color:SolidPeso molecular:451.527Phosphate acetyltransferase
CAS:<p>Phosphate acetyltransferase, an enzyme, reversibly transfers acetyl groups to CoA, aiding in acetate assimilation/dissimilation.</p>Forma y color:SolidPAz-PC
CAS:<p>PAz-PC (Azelaoyl PC) is a truncated phospholipid oxidation product that enhances endothelial barrier disruption caused by HKSA.</p>Fórmula:C33H64NO10PForma y color:SolidPeso molecular:665.84Sorbifolin
CAS:<p>Sorbifolin is a flavone glucoside from Pterogyne nitens with myeloperoxidase inhibition (IC50: 19.2 nM) and radical scavenging effects.</p>Fórmula:C16H12O6Forma y color:SolidPeso molecular:300.26Abiraterone N-oxide
CAS:<p>Abiraterone N-oxide is a metabolite of Abiraterone . Abiraterone is a potent and irreversible CYP17A1 inhibitor with antiandrogen activity [1] .</p>Fórmula:C24H31NO2Forma y color:SolidPeso molecular:365.51Fumarate hydratase-IN-2 sodium salt
CAS:<p>Fumarate hydratase-IN-2 Na salt: cell-permeable, competitive inhibitor (Ki=4.5μM), nutrient-dependent cytotoxicity.</p>Fórmula:C25H25N2NaO4Pureza:98%Forma y color:SolidPeso molecular:440.47BTT-266
CAS:<p>BTT-266 is a blocker of voltage-gated calcium channel for pain management.</p>Fórmula:C34H28N4O4Pureza:98.34%Forma y color:SolidPeso molecular:556.61TXA707
CAS:<p>TXA707, the active metabolite of TXA-709, is an FtsZ inhibitor with antibacterial properties. It shows potential for use in research involving S. aureus.</p>Fórmula:C15H8F5N3O2SForma y color:SolidPeso molecular:389.3APL180
CAS:<p>APL180 (L-4F) is an apolipoprotein A-I mimetic peptide that enhances the anti-inflammatory activity of high-density lipoprotein (HDL). It is applicable for cardiovascular disease research.</p>Fórmula:C114H156N24O28Forma y color:SolidPeso molecular:2310.6Betulin ditosylate
CAS:<p>Betulinditosylate is a derivative of Betulin, which functions as an SREBP inhibitor.</p>Fórmula:C44H62O6S2Forma y color:SolidPeso molecular:751.095-Aminoisotonitazene
CAS:<p>5-Aminoisotonitazene is a metabolite of the synthetic opioid analgesic agent, Isotonitazene, found in urine.</p>Fórmula:C23H32N4OForma y color:SolidPeso molecular:380.532-γ-Linolenoyl-1,3-dilinoleoyl-sn-glycerol
CAS:<p>2-γ-Linolenoyl-1,3-dilinoleoyl-sn-glycerol is a triglyceride.</p>Fórmula:C57H96O6Pureza:98%Forma y color:SolidPeso molecular:877.37(3S,5R)-Fluvastatin D6 sodium
CAS:<p>(3S,5R)-Fluvastatin D6 sodium: deuterium-labeled synthetic HMG-CoA reductase inhibitor with 8 nM IC50.</p>Fórmula:C24H25FNNaO4Pureza:98%Forma y color:SolidPeso molecular:439.49Nampt degrader-2
<p>Nampt degrader-2: a fluorescent PROTAC that degrades NAMPT at IC50 41.9 nM, reducing NAD+ and having anti-tumor effects.</p>Fórmula:C59H73N9O7SForma y color:SolidPeso molecular:1052.33BAY-277
<p>BAY-277 is a degrader of METAP2, with IC50 values of 5.8 nM for human METAP2 (hMETAP2) and 5.9 nM for mouse METAP2 (mMETAP2).</p>Fórmula:C44H52N8O5Forma y color:SolidPeso molecular:772.93iso-C15:0 3-OH
CAS:<p>Iso-C15:0 3-OH is a fatty acid that can be isolated from the PLRT strain. PLRT is a rod-shaped, Gram-negative, chemolithoheterotrophic, obligately aerobic bacterium, obtained from the feces of the mollusk Aplysia punctata.</p>Fórmula:C15H30O3Forma y color:SolidPeso molecular:258.397Mono(5-carboxy-2-ethylpentyl) phthalate
CAS:<p>MECPP is a metabolite of DEHP, a major plasticizer used in flexible PVC.</p>Fórmula:C16H20O6Forma y color:SolidPeso molecular:308.33Antidiabetic agent 2
<p>Compound 56 (Antidiabetic agent 2) is a glucose-uptake promoter that inhibits DPP-4, PTP-1B, α-amylase, and α-glucosidase, with IC50 values of 0.036, 0.042, 0.</p>Fórmula:C25H21N5O9S2Pureza:98%Forma y color:SolidPeso molecular:599.59AHK
CAS:<p>AHK, a bioactive peptide known for its antioxidant properties, has been employed as a cosmetic ingredient [1].</p>Fórmula:C15H26N6O4Pureza:98%Forma y color:SolidPeso molecular:354.4ITH12711
<p>ITH12711, a PP2A ligand, can traverse the blood-brain barrier (BBB) and exerts neuroprotection by restoring PP2A-phosphatase activity [1].</p>Fórmula:C12H20O5Pureza:98%Forma y color:SolidPeso molecular:244.28Myr-TAT-CBD3
<p>Myr-TAT-CBD3, a CRMP2-CaV2.2 interaction inhibitor, has been shown to significantly attenuate carrageenan-induced thermal hypersensitivity and reverse thermal</p>Fórmula:C148H269N59O33Pureza:98%Forma y color:SolidPeso molecular:3403.09hCA/Wnt/β-catenin-IN-1
<p>hCA/Wnt/β-catenin-IN-1 (Compd 15) serves as an inhibitor with selective affinity for hCA isoforms II, IX, and XII, exhibiting K i values of 33.6, 24.1, and 6.8</p>Forma y color:Odour Solidα-Amylase/α-Glucosidase-IN-4
<p>α-Amylase/α-Glucosidase-IN-4 (compound 5), a dual inhibitor targeting α-amylase (Amylases) and α-glucosidase (Glucosidase), exhibits potent inhibition with IC50</p>Fórmula:C32H26N6O10Pureza:98%Forma y color:SolidPeso molecular:654.58Prunetin 5-O-β-D-glucopyranoside
CAS:<p>Prunetin 5-O-β-D-glucopyranoside, an isoflavone obtained from Potentilla astracanica extracts, is a potent uncompetitive inhibitor of α-glucosidase (IC 50 = 56.</p>Fórmula:C22H22O10Forma y color:SolidPeso molecular:446.408His-D-β-Nal-Ala-Trp-D-Phe-Lys-NH2 TFA
<p>His-D-beta-Nal-Ala-Trp-D-Phe-Lys-NH2 TFA, a growth hormone releasing peptide and metabolite of GHRP-1 (Ala-His-D-beta-Nal-Ala-Trp-D-Phe-Lys-NH2), stimulates</p>Fórmula:C50H58F3N11O8Pureza:98%Forma y color:SolidPeso molecular:998.06Sucunamostat hydrochloride
<p>Sucunamostat (SCO-792) hydrochloride is an orally active, reversible inhibitor of enteropeptidase, displaying inhibition constants (IC50) of 4.6 nM for rat</p>Fórmula:C22H23ClN4O8Pureza:98%Forma y color:SolidPeso molecular:506.89NADP+ (sodium salt hydrate)
CAS:<p>NADP+ is the oxidized cofactor form of NADPH, vital for cell survival, redox balance, and signaling; synthesized from NAD+ and ATP.</p>Fórmula:C21H30N7NaO18P3Forma y color:SolidPeso molecular:784.413Carbonic anhydrase inhibitor 26
<p>Compound 6T, designated as Carbonic anhydrase inhibitor26, acts as an inhibitor of Carbonic Anhydrase II (Carbonic AnhydraseII), exhibiting an IC50 value of 9.10 ± 0.26 μM.</p>Fórmula:C17H14N6O4Forma y color:SolidPeso molecular:366.33Nepetalactone
CAS:<p>Nepetalactone is found in the plant Nepeta parnassica and has high mosquito repellency properties.</p>Fórmula:C10H14O2Forma y color:SolidPeso molecular:166.22VU533
CAS:<p>VU533 is a NAPE-PLD activator, EC50=0.30 µM, boosts macrophage activity, potential in cardiometabolic diseases.</p>Fórmula:C21H22FN3O3S2Pureza:99.08%Forma y color:SolidPeso molecular:447.55Abieslactone
CAS:<p>Abieslacton possesses anti-tumor promoting activity isolated from several Abies genus.</p>Fórmula:C31H48O3Forma y color:SolidPeso molecular:468.722(R)-ICMT-IN-3
<p>(R)-ICMT-IN-3 (compound ent 2-27) functions as a potent inhibitor of ICMT, exhibiting an IC50 value of 0.01 μM [1].</p>Forma y color:Odour SolidMaurocalcine
CAS:<p>Maurocalcine is a cell-permeable agonist for ryanodine receptor (RyR) subtypes 1, 2, and 3.</p>Fórmula:C156H270N56O46S6Pureza:98%Forma y color:SolidPeso molecular:3858.55D-Ribofuranose1-dihydrogenphosphate dicyclohexanamine
CAS:<p>D-Ribofuranose 1-phosphate is used to synthesize 5-fluorouracil via uridine phosphorylase.</p>Fórmula:C11H24NO8PForma y color:SolidPeso molecular:329.2816α-hydroxy Dehydroepiandrosterone
CAS:<p>16α-hydroxy Dehydroepiandrosterone (16α-OH-DHEA) is a neurosteroid found in the brain and a precursor in the biosynthesis of placental estriol.</p>Fórmula:C19H28O3Forma y color:SolidPeso molecular:304.42tetranor-12(R)-HETE
CAS:<p>Corneal metabolism of 12(R)-HETE yields 8(R)-HHxTrE via β-oxidation, losing four carbons from C-1.</p>Fórmula:C16H26O3Forma y color:SolidPeso molecular:266.381trans-hydroxy Glimepiride
CAS:<p>trans-Hydroxy Glimepiride, an active sulfonylurea glimepiride metabolite, is primarily synthesized in the liver by CYP2C9.</p>Fórmula:C24H34N4O6SForma y color:SolidPeso molecular:506.62α,α-Trehalose 6-phosphate potassium
CAS:<p>α,α-Trehalose 6-phosphate (Tre6P) potassium is an intrinsic 6-phosphate derivative of α,α′-trehalose and acts as an intermediary metabolite.</p>Fórmula:C12H21K2O14PPureza:98%Forma y color:SolidPeso molecular:498.46Myoregulin TFA
<p>Myoregulin (MLN peptide) TFA, belonging to the regulin family, is a regulator of muscle performance through modulation of intracellular calcium dynamics.</p>Fórmula:C239H391N53O67S3·xC2HF3O2Pureza:98%Forma y color:SolidPeso molecular:5175.17 (free base)α-Glycosidase-IN-2
<p>α-Glycosidase-IN-2 (compound 8b) is an inhibitor of α-glycosidase, displaying Ki values of 74.16 nM and 6.09 nM for aldose reductase and α-glycosidase, respectively. This compound is utilized in research related to diabetes.</p>Fórmula:C25H22N6OS2Forma y color:SolidPeso molecular:486.61α-1,4-Galactosyltransferase (LgtC)
CAS:<p>A4GALT (LgtC) adds galactose to lactosylceramide, forming globotriaosylceramide; used in P1 antigen synthesis.</p>Forma y color:SolidCellulose
CAS:<p>Cellulose, an excipient, aids stability, solubility, and processing of drugs and affects their ADME.</p>Fórmula:C12H22O11Forma y color:SolidPeso molecular:342.297D-threo-PPMP
CAS:<p>D-threo-PPMP, a powerful glucosylceramide (GlcCer) synthase inhibitor, effectively impedes karyokinesis and decreases cyst formation.</p>Fórmula:C29H50N2O3Forma y color:SolidPeso molecular:474.73(2-Hydroxyethoxy)acetic acid
CAS:<p>'(2-Hydroxyethoxy)acetic acid is 1,4-Dioxane's primary urine metabolite and a reliable short-term biomarker.'</p>Fórmula:C4H8O4Forma y color:SolidPeso molecular:120.1Endocrocin
CAS:<p>Endocrocin is a useful organic compound for research related to life sciences. The catalog number is T124800 and the CAS number is 481-70-9.</p>Fórmula:C16H10O7Forma y color:SolidPeso molecular:314.249BBOX-IN-1
<p>BBOX-IN-1 (compound 58) is a potent BBOX inhibitor with an IC50 of 0.02 μM, and it is applicable in research related to triple-negative breast cancer (TNBC).</p>Fórmula:C18H17N3O6SForma y color:SolidPeso molecular:403.41sPLA2 inhibitor 3
<p>sPLA2 inhibitor 3 (Compound 6c) functions as a potent α-glucosidase inhibitor (IC50= 0.0953 µM) and has potential applications in diabetes research.</p>Fórmula:C22H16F6N6O4S2Forma y color:SolidPeso molecular:606.52CAY10581
CAS:<p>CAY10581, a derivative of pyranonaphthoquinone, serves as a highly specific and reversible uncompetitive inhibitor of IDO, demonstrating potency with an IC50</p>Fórmula:C22H21NO4Forma y color:SolidPeso molecular:363.41Febuxostat dicarboxylic acid impurity
CAS:<p>Febuxostat dicarboxylic acid impurity is an impurity of Febuxostat. Febuxostat is selective xanthine oxidase inhibitor with a K i of 0.6 nM [1] .</p>Fórmula:C16H17NO5SForma y color:SolidPeso molecular:335.38trans-5-Hydroxyferulic acid
CAS:<p>trans-5-Hydroxyferulic acid is a useful organic compound for research related to life sciences. The catalog number is T126397 and the CAS number is 110642-42-7.</p>Fórmula:C10H10O5Forma y color:SolidPeso molecular:210.185Transketolase-IN-5
<p>Transketolase-IN-5 (compound 6ba) is an inhibitor of transketolase. It exhibits herbicidal activity against Amaranthus retroflexus, Setaria viridis, and Digitaria sanguinalis.</p>Fórmula:C20H24ClN5OPeso molecular:385.16694Xanthine oxidase-IN-9
CAS:<p>Xanthine Oxidase-IN-9 (also known as Icarisids E or Compound 2) effectively inhibits xanthine oxidase (XOD) with an IC50 value of 31.81 μM [1].</p>Fórmula:C38H50O20Forma y color:SolidPeso molecular:826.79L 645164
CAS:<p>L 645164 is an inhibitor of hydroxymethylglutaryl-CoA reductase.</p>Fórmula:C22H23FO3Forma y color:SolidPeso molecular:354.41Vitamin B12a hydrochloride
CAS:<p>Vitamin B12a monohydrochloride (Hydroxocobalamin) is an essential water-soluble vitamin.a cyanide detoxifier and nutritional supplement, injection, inhalation.</p>Fórmula:C62H89CoN13O15P·xHClForma y color:SolidFABP4-IN-3
<p>FABP4-IN-3 (Compound C3) is a highly selective inhibitor of FABP4, with an inhibition constant (Ki) of 25 ± 3 nM for FABP4 and a Ki of 15.03 μM for FABP3, showcasing a selectivity factor of 601 times over FABP3. It also demonstrates metabolic stability and potent anti-inflammatory activity in cells, making it a promising candidate for research in metabolic disorders, cardiac dysfunction, and inflammation-related diseases.</p>Fórmula:C20H16ClNO2Peso molecular:337.08696α-Glucosidase-IN-50
<p>α-Glucosidase-IN-50 (compound 8) acts as an inhibitor of α-Glucosidase.</p>Fórmula:C33H28Cl4N6O6SPeso molecular:776.05451α-Amylase/α-Glucosidase-IN-13
<p>α-Amylase/α-Glucosidase-IN-13 (Compound 5d) is a dual inhibitor of α-amylase and α-glucosidase, and is useful in diabetes research.</p>Fórmula:C22H16N2O5Peso molecular:388.1059210'-Desmethoxystreptonigrin
CAS:<p>'10'-Desmethoxystreptonigrin antibiotic derived from streptonigrin combats various bacteria and cancer cells, and inhibits p21ras farnesylation (IC50 = 21 nM).</p>Fórmula:C24H20N4O7Forma y color:SolidPeso molecular:476.445IDO1-IN-24
<p>IDO1-IN-24 (compound 2c) inhibits the production of IDO1 during cell assays, with an IC50 value of 17 μM.</p>Fórmula:C18H22N2O4Peso molecular:330.15796Casein kinase 1δ-IN-14
CAS:<p>Casein kinase 1δ-IN-14 (WAY-637081) can be used to study atherosclerosis-related cardiovascular disease.</p>Fórmula:C17H11ClN4O2Pureza:99.74%Forma y color:SolidPeso molecular:338.75Erucic acid sodium
CAS:<p>Erucic acid sodium, a monounsaturated fatty acid (MUFA) extracted from the seeds of rapeseed, readily crosses the blood-brain barrier (BBB). It normalizes the accumulation of long-chain fatty acids in the brain, enhances cognitive function, and effectively prevents dementia.</p>Fórmula:C22H42NaO2Forma y color:SolidPeso molecular:361.56α-Cyclopentyl-4-(2-quinolinylmethoxy)benzeneacetic acid
CAS:<p>α-Cyclopentyl-4-(2-quinolinylmethoxy)benzeneacetic acid was identified as possible dual inhibitors for hLTA4H and hLTC4S enzymes by the computer-aided</p>Fórmula:C23H23NO3Pureza:97.19% - 99.36%Forma y color:SoildPeso molecular:361.43PDE4-IN-3
CAS:<p>PDE4-IN-3, a new oral drug, potently blocks PDE4 enzyme with 4.2 nM IC50.</p>Fórmula:C35H33FO8Forma y color:SolidPeso molecular:600.639Perflubutane
CAS:<p>Perfluorobutane is a gas that is colorless.</p>Fórmula:C4F10Pureza:98%Forma y color:Colorless Gas Colorless GasPeso molecular:238.03(-)-Vorozole
CAS:<p>(-)-Vorozole, potent/selective oral non-steroidal aromatase inhibitor, shows antitumor activity, used in breast cancer research.</p>Fórmula:C16H13ClN6Pureza:99.02% - >99.99%Forma y color:SoildPeso molecular:324.77CA IX/VEGFR-2-IN-3
<p>CAIX/VEGFR-2-IN-3 (Compound 6i) is an inhibitor of Carbonic Anhydrase IX and VEGFR-2, with IC50 values of 41 and 48 nM, respectively. It exhibits anticancer activity by inhibiting the growth of MCF-7 breast cancer cells (IC50 of 22.33 μM) and mouse fibroblast cell line 3T3, where cell viability is reduced to below 40% at a concentration of 100 μM. This compound is applicable for research in the field of cancer treatment.</p>Fórmula:C19H16ClN3O5S2Forma y color:SolidPeso molecular:465.93RARα antagonist 1
<p>Compound 21, an orally active and selective RARα antagonist, exhibits a potent inhibition of the retinoic acid receptor α with an IC50 of 4.6 nM [1].</p>Fórmula:C26H23NO4Forma y color:SolidPeso molecular:413.47SGK1-IN-3 hydrochloride
<p>SGK1-IN-3 hydrochloride (compound 3a) is an efficacious, orally bioavailable SGK1 inhibitor. The serine/threonine kinase SGK1 acts as an activator of the β-catenin pathway and strongly stimulates cartilage degradation, being upregulated under genomic control in diseased osteoarthritic cartilage. SGK1-IN-3 hydrochloride holds potential for osteoarthritis research.</p>Fórmula:C23H21Cl3N6O3SPeso molecular:566.04614(24S)-24,25-Dihydroxyvitamin D3
CAS:<p>(24S)-24,25-Dihydroxyvitamin D3 undergoes various levels of hydroxylation to form active vitamin D3 analogs.</p>Fórmula:C27H44O3Pureza:98.98%Forma y color:SolidPeso molecular:416.645A2-SC8 TFA
<p>5A2-SC8 TFA is an ionizable amino lipid used in lipid nanoparticles (LNPs), offering high delivery potential and low in vivo toxicity. It effectively delivers small RNAs, such as siRNA and miRNA, to tumor cells. Moreover, 5A2-SC8 TFA LNPs provide unique delivery paths for RNA within the liver, enhancing therapeutic outcomes in cancer models.</p>Forma y color:Odour SolidLysylglutamic acid
CAS:<p>Lysylglutamic acid is a dipeptide composed of the amino acids lysine (Lysine, Lys) and glutamic acid (Glutamic acid, Glu), with an inhibitory constant (Ki) of 1.3 mM for the membrane transport protein PEPT1.</p>Fórmula:C11H21N3O5Forma y color:SolidPeso molecular:275.3NAADP sodium
<p>NAADP sodium is a Ca2+ motor second messenger that targets Ca(2+) channels and can be used to study cancer and immune dysfunction.</p>Fórmula:C21H27N6O18P3Forma y color:SolidPeso molecular:744.39PR280
<p>PR280 is a potent inhibitor of dihydroceramide desaturase 1 (Des1) with an IC50 of 700 nM. It forms hydrogen bonds with amino acid residues of Des1, while its cyclopropenone group may coordinate with the iron center, stabilizing its binding at Des1's active site. This inhibits the ceramide biosynthesis pathway, preventing dihydroceramide (dhCer) from converting into ceramide. PR280 can be used in research related to sphingolipid metabolism disorders, including cancer and metabolic diseases.</p>Fórmula:C27H49NO4Peso molecular:451.36616OPC18750 HCl
CAS:<p>OPC18750 HCl is a phosphodiesterase inhibitor with positive inotropic effects that can be used to study asthma, cancer, diabetes, and psychiatric disorders.</p>Fórmula:C20H23ClN2O4Pureza:98.92%Forma y color:SoildPeso molecular:390.86(S)-O-Desmethyl Venlafaxine N-Oxide
CAS:<p>(S)-O-Desmethyl Venlafaxine N-Oxide is the N-oxide metabolite of Venlafaxine, an SNRI antidepressant.</p>Fórmula:C16H25NO3Forma y color:SolidPeso molecular:279.37Desmethylene Paroxetine hydrochloride
CAS:<p>Desmethylene Paroxetine hydrochloride is a non-conjugated metabolite of Paroxetine, a catechol intermediate.</p>Fórmula:C18H21ClFNO3Forma y color:SolidPeso molecular:353.82Motapizone
CAS:<p>Motapizone (NAT 05-239), a PDE3 inhibitor, moderates LPS-induced cytokine release and blocks platelet aggregation by boosting cAMP.</p>Fórmula:C12H12N4OSForma y color:SolidPeso molecular:260.3212-Hydroxynevirapine
CAS:<p>12-Hydroxynevirapine, major Nevirapine metabolite; non-toxic but liver/skin SULTs convert it to reactive 12-Sulphoxy-nevirapine.</p>Fórmula:C15H14N4O2Forma y color:SolidPeso molecular:282.3DSPE-PEG1000-M2pep
<p>DSPE-PEG1000-M2pep is a PEG compound comprised of DSPE and the M2 macrophage-targeting peptide (M2pep). M2pep acts as a mono- or multivalent ligand conjugated with pro-apoptotic peptides to focus the peptides' toxic effects on M2 macrophages. DSPE-PEG1000-M2pep can be utilized for drug delivery.</p>Forma y color:Odour SolidVU534
CAS:<p>VU534 is a NAPE-PLD agonist with an EC50 of 0.30 μM.VU534 is a dual inhibitor of FAAH and sEH, with an IC50 of 1.2 μM for sEH.VU534 is used in diseases related</p>Fórmula:C21H22FN3O3S2Pureza:98.85%Forma y color:SolidPeso molecular:447.55Sphingomyelin phosphodiesterase
CAS:<p>Sphingomyelin phosphodiesterase, a hydrolase, converts sphingomyelin into phosphocholine and ceramide, affecting cellular processes and cholesterol metabolism.</p>Forma y color:Solid11β-HSD1 inibitor 19
CAS:<p>3-chloro-4-sulfonyl-Benzonitrile inhibits hHSD1/mHSD1, IC50: 16nM/10nM.</p>Fórmula:C19H16ClF4N3O2SPureza:99.58%Forma y color:SoildPeso molecular:461.86ND-011992
CAS:<p>ND-011992: Quinazoline inhibitor of E. coli respiratory enzymes; IC50s: 0.12-2.47 μM; potential tuberculosis research.</p>Fórmula:C21H14F3N3OPureza:99.7%Forma y color:SoildPeso molecular:381.35MNI caged kainic acid
CAS:<p>Generates large inward currents at resting membrane potential</p>Fórmula:C19H23N3O6Pureza:98%Forma y color:SolidPeso molecular:389.40S-Phenylmercapturic acid
CAS:<p>S-Phenylmercapturic acid is a metabolite of benzene that can be used as a biomarker to assess benzene exposure.</p>Fórmula:C11H13NO3SPureza:99.68%Forma y color:SolidPeso molecular:239.29wt hMLN
<p>Wild-type human myoregulin (wt hMLN) is a microprotein that inhibits the sarcoplasmic reticulum Ca²⁺ pump (SERCA), playing a crucial role in the regulation of</p>Fórmula:C245H404N54O66SPureza:98%Forma y color:SolidPeso molecular:5194.22Ozolinone
CAS:<p>Ozolinone, an etozoline metabolite, is a loop diuretic treating hypertension and edema.</p>Fórmula:C11H16N2O3SForma y color:SolidPeso molecular:256.3213,14-dehydro-15-cyclohexyl Carbaprostacyclin
CAS:<p>13,14-dehydro-15-cyclohexyl Carbaprostacyclin, a stable PGI2 analog, impedes ADP-induced platelet aggregation; ED50 ~40 nM in PRP, 77 nM in washed platelets.</p>Fórmula:C21H30O4Forma y color:SolidPeso molecular:346.46713-cis-Retinyl acetate
CAS:<p>13-cis-Retinyl acetate: active 13-cis isomer of Retinyl acetate, metabolite of vitamin A.</p>Fórmula:C22H32O2Forma y color:SolidPeso molecular:328.49α-Glucosidase-IN-79
<p>α-Glucosidase-IN-79 (Compound 4d9) is a non-competitive α-glucosidase inhibitor with an IC50 of 2.11 μM, demonstrating greater inhibitory potency than the existing α-glucosidase inhibitors Acarbose (IC50 of 327.0 μM) and HXH8r (IC50 of 15.32 μM). It exhibits no cytotoxicity on normal human liver cells (LO2) and shows good metabolic stability in rat plasma. α-Glucosidase-IN-79 holds promise for research in type 2 diabetes.</p>Fórmula:C21H22N2O5SForma y color:SolidPeso molecular:414.475Vardenafil dihydrochloride
CAS:<p>Vardenafil dihydrochloride (Levitra) is a new type PDE inhibitor with IC50 of 0.7 and 180 nM for PDE5 and PDE1, respectively.</p>Fórmula:C23H34Cl2N6O4SPureza:98%Forma y color:SolidPeso molecular:561.52α-Glucosidase-IN-60
<p>α-Glucosidase-IN-60 (Compound 5k) acts as a competitive inhibitor of α-Glucosidase, with an IC50 of 10.8 μM.</p>Fórmula:C23H14N2O5Peso molecular:398.09027hCES2A-IN-2
<p>hCES2A-IN-2 (compound 14n) is an orally active, highly specific, irreversible, covalent inhibitor of hCES2A with an IC50 of 0.04 nM. It targets and covalently binds to the catalytic serine residue (Ser-228) of hCES2A. hCES2A-IN-2 can significantly mitigate irinotecan-induced gastrointestinal toxicity (ITGT) without diminishing the antitumor efficacy of irinotecan in tumor-bearing mice.</p>Forma y color:Odour SolidLEI110
CAS:<p>LEI110 inhibits PLA2G16 and HRASLS enzymes, Ki 20 nM, selectively targets related thiol hydrolases.</p>Fórmula:C25H23F3N2O3Pureza:98.66% - 98.8%Forma y color:SolidPeso molecular:456.46(R)-AS-1
CAS:<p>(R)-AS-1 is a selective positive allosteric modulator of excitatory amino acid transporter 2 (EAAT2), with an EC50 of 11 nM. At doses of 60 and 90 mg/kg, (R)-AS-1 enhances spontaneous locomotor activity in mice. It demonstrates anticonvulsant properties in mouse seizure models induced by maximal electroshock (MES), pentylenetetrazole (PTZ), or electric current stimulation (32 or 44 mA), with ED50 values of 66.3, 36.3, 15.6, and 41.6 mg/kg, respectively. This compound is applicable in neurological disease research.</p>Fórmula:C14H16N2O3Forma y color:SolidPeso molecular:260.2924, 25-Dihydroxy VD2
CAS:<p>24, 25-Dihydroxy VD2 (24,25-Dihydroxy vitamin D2) is a metabolite of vitamin D2 and is an isomer of 25-hydroxyvitamin D.</p>Fórmula:C28H44O3Pureza:99.63%Forma y color:SolidPeso molecular:428.65Abiraterone sulfate
CAS:<p>Abiraterone sulfate is a metabolite of Abiraterone . Abiraterone is a potent and irreversible CYP17A1 inhibitor with antiandrogen activity [1] .</p>Fórmula:C24H31NO4SForma y color:SolidPeso molecular:429.57Phenylsulfamide
CAS:<p>Phenylsulfamide (Compound 10), acting as an inhibitor of human carbonic anhydrase-II (hCA-II), exhibits a dissociation constant (Kd) of 45.50 μM and an</p>Fórmula:C6H8N2O2SForma y color:SolidPeso molecular:172.2(±)8-HDHA
CAS:<p>(±)8-HDHA is an autoxidation product of docosahexaenoic acid (DHA) in vitro.</p>Fórmula:C22H32O3Forma y color:SolidPeso molecular:344.495(S,S)-GSK321
CAS:<p>(S,S)-GSK321 is a (S,S)-enantiomer of GSK321 [1] .</p>Fórmula:C28H28FN5O3Forma y color:SolidPeso molecular:501.55Adenosine deaminase
CAS:<p>Adenosine deaminase is an enzyme that catalyzes the irreversible deamination of 2'-deoxyadenosine and adenosine to 2'-deoxyinosine and inosine, respectively.</p>Pureza:98%Forma y color:Solid6-Azathymine acid
CAS:<p>6-Azathymine is a metabolite of Pymetrozine, an insecticide targeting aphids and whiteflies by disrupting feeding.</p>Fórmula:C4H3N3O4Forma y color:SolidPeso molecular:157.08HIF-1 inhibitor-5
<p>HIF-1 inhibitor-5 (Compound 16e) is a potent inhibitor of HIF-1, exhibiting an IC50 value of 2.38 μM and demonstrating significant anti-angiogenic potential [1</p>Fórmula:C28H35NO5Forma y color:SolidPeso molecular:465.58D-Pro-Phe-Arg-Chloromethylketone
CAS:<p>D-Pro-Phe-Arg-Chloromethylketone, an inhibitor of coagulation factor XII and plasma kallikrein, is significant in the regulation of thrombosis and inflammation</p>Fórmula:C21H31ClN6O3Pureza:98%Forma y color:SolidPeso molecular:450.96LL P880 β
CAS:<p>LL P880 beta is a fungal metabolite.</p>Fórmula:C11H18O5Forma y color:SolidPeso molecular:230.26GP4G
CAS:<p>GP4G, from Artemia salina cysts, regulates epithelial cells & hair growth.</p>Fórmula:C20H28N10O21P4Forma y color:SolidPeso molecular:868.39ROS-IN-3
<p>ROS-IN-3 (compound x38) is an inhibitor of ROS and is utilized in neuro-related research.</p>Fórmula:C25H20F2N2O4Forma y color:SolidPeso molecular:450.43Calcitriol Derivatives
<p>Calcitriol Derivatives is an analog of vitamin D3.</p>Fórmula:C30H47NO3Pureza:98%Forma y color:SolidPeso molecular:469.7Purpactin A
CAS:<p>Purpactin A is a useful organic compound for research related to life sciences. The catalog number is T126026 and the CAS number is 133806-59-4.</p>Fórmula:C23H26O7Forma y color:SolidPeso molecular:414.454Prostaglandin F2β
CAS:<p>Prostaglandin F2β (PGF2β) is the 9β-hydroxy stereoisomer of PGF2α.</p>Fórmula:C20H34O5Forma y color:White SolidPeso molecular:354.48Pepsin A
CAS:<p>Pepsin A is a protease and endopeptidase in the stomach, capable of breaking down proteins in food into small peptide fragments.</p>Forma y color:Solidα-Glucosidase-IN-26
<p>α-Glucosidase-IN-26 (Compound 7i), with an IC50 value of 4.63 µM, functions as an α-glucosidase inhibitor and is utilized in research related to type 2 diabetes</p>Fórmula:C23H22ClN3O5Pureza:98%Forma y color:SolidPeso molecular:455.89Ercalcidiol
CAS:<p>Ercalcidiol is a metabolite of vitamin D2 and can be used in monitoring vitamin D therapy.</p>Fórmula:C28H44O2Pureza:99.62%Forma y color:SolidPeso molecular:412.65L-Lysine, sulfite (2:1)
CAS:<p>L-Lysine, sulfite (2:1) is a drug/ therapeutic agent.</p>Fórmula:C6H14N2O2H2O3SForma y color:SolidPeso molecular:187.2313-epi-12-oxo Phytodienoic Acid
CAS:<p>13-epi-12-oxo PDA is a lipoxygenase derivative of α-linolenic acid in green plant leaves, often isomerizing during extraction and storage.</p>Fórmula:C18H28O3Forma y color:SolidPeso molecular:292.41Epicoccamide
CAS:<p>Epicoccamide is a marine fungal metabolite originally isolated from E. purpurascens.</p>Fórmula:C29H51NO9Forma y color:SolidPeso molecular:557.72FR106969
CAS:<p>FR106969 is a platelet activating factor antagonist isolated from fungus with anti-inflammatory activity.</p>Fórmula:C16H22N2O3S2Pureza:98%Forma y color:SolidPeso molecular:354.491-β-D-Glucosylsphingadienine (d18:2 (4E,8E))
CAS:<p>1-β-D-Glucosylsphingadienine is a glucosylsphingosine, which are deacetylated lysolipid derivatives of glucosylcerebrosides .</p>Fórmula:C24H45NO7Forma y color:SolidPeso molecular:459.624Formate dehydrogenase
CAS:<p>Formate dehydrogenase, found in all life forms, converts formate to CO2 and is categorized by metal content for research.</p>Forma y color:SolidAmidase
CAS:<p>Amidases, belonging to the nitrilase superfamily, catalyze amide hydrolysis to yield carboxylic acid and ammonia.</p>Pureza:98%Forma y color:SolidhCA XII-IN-6
<p>Compound 4d, known as hCA XII-IN-6, is a potent inhibitor of human carbonic anhydrase XII (hCA XII) with a Ki value of 84.2 nM and exhibits anti-proliferative</p>Fórmula:C11H9N5O3S2Pureza:98%Forma y color:SolidPeso molecular:323.35(24R)-MC 976
CAS:<p>(24R)-MC 976 is a derivative of Vitamin D3.</p>Fórmula:C27H42O3Pureza:98%Forma y color:SolidPeso molecular:414.62
