Metabolismo
Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.
Subcategorías de "Metabolismo"
- AhR(42 productos)
- Aminopeptidasa(76 productos)
- CETP(20 productos)
- Anhídrido carbónico(197 productos)
- Caseína quinasa(137 productos)
- DHFR(34 productos)
- Descarboxilasa(4 productos)
- Deshidrogenasa(303 productos)
- FAAH(66 productos)
- FXR(62 productos)
- Factor Xa(87 productos)
- Ácido graso sintasa(37 productos)
- Ferroptosis(226 productos)
- GR(3 productos)
- GSNOR(4 productos)
- Glucoquinasa(57 productos)
- HIF / HIF Prolilhidroxilasa(146 productos)
- HMG-CoA reductasa(33 productos)
- Hidroxilasa(35 productos)
- IDO(84 productos)
- LDL(8 productos)
- Lipasa(107 productos)
- Lípido(61 productos)
- Lipoxigenasa(134 productos)
- MAO(87 productos)
- MPO(2 productos)
- NAMPT(40 productos)
- P450(6 productos)
- PAI-1(26 productos)
- PDE(167 productos)
- PED(1 productos)
- PKM(17 productos)
- PPAR(169 productos)
- Fosfolipasa(83 productos)
- ROR(47 productos)
- Receptor de retinoides(28 productos)
- SGK(11 productos)
- Tiorredoxina(12 productos)
- Transferasa(29 productos)
- Transportador(46 productos)
- UGT(4 productos)
- Inhibidores de la xantina oxidasa (XO)(9 productos)
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Se han encontrado 9271 productos de "Metabolismo"
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PF-04671536
CAS:PF-04671536 inhibits PDE8B/PDE8A, boosts insulin in human pancreatic islets.Fórmula:C14H18N8OSForma y color:SolidPeso molecular:346.41BRD9500
CAS:BRD9500 is an oral PDE3 inhibitor, IC50: 10 nM (PDE3A), 27 nM (PDE3B); effective in SK-MEL-3 cancer model.Fórmula:C15H18FN3O2Forma y color:SolidPeso molecular:291.32JZP-MA-13
JZP-MA-13: selective α/β-hydrolase domain 6 inhibitor, IC 50 392 nM, doesn't inhibit MAGL/ABHD12/FAAH, used in PET imaging.Fórmula:C14H15FN4O3SForma y color:SolidPeso molecular:338.36YM-75440
CAS:YM-75440 is an squalene synthase inhibitor with oral activity.Fórmula:C25H26N2OPureza:98%Forma y color:SolidPeso molecular:370.49Methionine sulfoximine
CAS:Methionine sulfoximine (MSO) is an irreversible glutamine synthetase inhibitor. It is the sulfoximine derivative of methionine with convulsant effects.Fórmula:C5H12N2O3SForma y color:SolidPeso molecular:180.23Cefonicid monosodium
CAS:Cefonicid monosodium, a second-gen cephalosporin, treats UTIs, respiratory, soft tissue, and bone infections by blocking cell wall synthesis.Fórmula:C18H17N6NaO8S3Forma y color:SolidPeso molecular:564.54Flutolanil
CAS:Flutolanil: a fungicide targeting R. solani in rice, toxic to zebrafish.Fórmula:C17H16F3NO2Forma y color:SolidPeso molecular:323.31D,L-erythro-PDMP hydrochloride
CAS:D,L-erythro-PDMP hydrochloride, an isomer of PDMP, inhibits rabbit fibroblast growth and glucosyltransferase.Fórmula:C23H39ClN2O3Forma y color:SolidPeso molecular:427.02Lp-PLA2-IN-4
CAS:Lp-PLA2-IN-4, a potent inhibitor of Lp-PLA2/PAF-AH, may target Alzheimer's, atherosclerosis. (WO2021228159A1, Compound 38)Fórmula:C23H18F5N3O4Forma y color:SolidPeso molecular:495.4hCA I-IN-2
CAS:hCA I-IN-2 (6d) inhibits hCA I (Ki: 18.8 nM) more selectively over II, IX, XII (Ki: 375.1, 1721, 283.9 nM).Fórmula:C26H20BrN5O3SForma y color:SolidPeso molecular:562.44Fenprinast
CAS:Fenprinast is a tryptophan-like bronchodilator utilized in the study of allergic and exercise-induced asthma. It exhibits oral activity.Fórmula:C16H16ClN5OPeso molecular:329.78MitoPBN
CAS:MitoPBN: mitochondria-targeted antioxidant, inhibits UCP1-3 at 250 nM, traps hydroxyl & carbon radicals, prevents lipid peroxidation.Fórmula:C33H37BrNO2PForma y color:SolidPeso molecular:590.542Phosphodiesterase 4 Inhibitor
CAS:Phosphodiesterase 4 (PDE4) inhibitor is an inhibitor of PDE4 with an IC50 value of 0.10 μM for the human recombinant enzyme.Fórmula:C14H15N3O4Forma y color:SolidPeso molecular:289.29Lisinopril, ε-biotinamidocaproyl-
CAS:Lisinopril, epsilon-biotinamidocaproyl- is an angiotensin converting enzyme (ACE) inhibitor.Fórmula:C37H56N6O8SForma y color:SolidPeso molecular:744.94S-(-)-Etomoxir
CAS:S-(-)-Etomoxir is an inhibitor of carnitine palmitoyltransferase A (CPT1) -- a molecule required for the oxidation of long-chain acyl CoA esters.Fórmula:C17H23ClO4Forma y color:SolidPeso molecular:326.82l-trans-Phenothrin
CAS:l-trans-Phenothrin, as a synthetic pyrethroid, can kill adult fleas and ticks.Fórmula:C23H26O3Forma y color:SolidPeso molecular:350.45Lombricine
CAS:Lombricine, as a phosphodiester of 2-guanidinoethanol and D-serine in structure, is a phosphagen that is unique to earthworms.Fórmula:C6H15N4O6PForma y color:SolidPeso molecular:270.18Vorozole
CAS:<p>Vorozole (R83842) is an orally active, potent, and selective nonsteroidal aromatase inhibitor.Vorozole exhibits antitumor activity in vivo and may be used in</p>Fórmula:C16H13ClN6Pureza:99.65% - 99.94%Forma y color:SolidPeso molecular:324.77SAHO2
CAS:SAHO2, a sulfone methyl donor, is cleaved by NosL/NosN into 5'-deoxyadenosine and sulfinic acid.Fórmula:C14H20N6O7SForma y color:SolidPeso molecular:416.41hCAXII-IN-4
CAS:hCAXII-IN-4 is a selective and potent CA XII inhibitor with a Ki value of 6.4 nM for human CA XII.Fórmula:C22H27N5O6SForma y color:SolidPeso molecular:489.54UCCF-029
CAS:UCCF-029 is an activator of cystic fibrosis transmembrane conductance regulator (CFTR).Fórmula:C18H11NO2Forma y color:SolidPeso molecular:273.29CP-220629
CAS:CP 220629 is a potent inhibitor of phosphodiesterase IV (PDE4).Fórmula:C20H25N3OForma y color:SolidPeso molecular:323.43Glucocerebrosidase-IN-1
CAS:Glucocerebrosidase-IN-1 inhibits GCase with IC50 of 29.3 μM, Ki 18.5 μM, useful for Gaucher's and Parkinson's research.Fórmula:C13H27NO3Forma y color:SolidPeso molecular:245.36BMS-351
CAS:BMS-351: potent, selective CYP17A1 inhibitor, promising for prostate cancer, minimal side effects.Fórmula:C15H12F3N3Forma y color:SolidPeso molecular:291.27Choline theophyllinate
CAS:Choline theophyllinate (Oxtriphylline) is the choline salt of theophylline, a small molecule PDE inhibitor that can be used to treat immune system disorders andFórmula:C12H21N5O3Pureza:98%Forma y color:SolidPeso molecular:283.3311β-HSD1-IN-9
CAS:<p>11β-HSD1-IN-9 is a potent inhibitor of 11β-HSD1, displaying IC50 values of 0.48 µM for human and 1.3 µM for murine variants, respectively.</p>Fórmula:C13H9F3N2OForma y color:SolidPeso molecular:266.22CL 242817
CAS:CL 242817 is an inhibitor of angiotensin converting enzyme (ACE).Fórmula:C18H21NO5SForma y color:SolidPeso molecular:363.43Inamrinone lactate
CAS:Inamrinone lactate: a cardiotonic vasodilator, inhibits phosphodiesterase, and boosts cardiac calcium influx.Fórmula:C13H15N3O4Forma y color:SolidPeso molecular:277.28Lutropin
CAS:Lutropin is a heterodimeric glycoprotein, a hormone produced by anterior pituitary gonadotrophs, which stimulates follicle development.Forma y color:Solid(±)-γ-Tocopherol
CAS:(±)-γ-Tocopherol is a form of vitamin E with antioxidant and anti-inflammatory properties.Fórmula:C28H48O2Forma y color:SolidPeso molecular:416.68Sitamaquine tosylate
CAS:Sitamaquine: antileishmanial, targets L. donovani species, EC50 = 9.5-19.8 μM, inhibits mitochondrial complex II, induces apoptosis in promastigotes.Fórmula:C28H41N3O4SForma y color:SolidPeso molecular:515.71MK-0952 Sodium
CAS:MK-0952 Sodium is a salt form of MK-0952, which is a selective PDE4 inhibitor.Fórmula:C28H22FN3NaO4Forma y color:SolidPeso molecular:506.4893-Allylphenol
CAS:3-Allylphenol is an inhibitor of dopamine β-hydroxylase (DBH; Ki = 12 mM).Fórmula:C9H10OForma y color:SolidPeso molecular:134.18N-Phenylthiourea
CAS:N-Phenylthiourea (Phenylthiocarbamide) is EC 1.14.18.1 (tyrosinase) inhibitor, a diphenolase inhibitor, and a non-competitive inhibitor of the PvdP tyrosinase.Fórmula:C7H8N2SPureza:99.71%Forma y color:SolidPeso molecular:152.22Endothall
CAS:Endothall is an effective protein phosphatase 2A (PP2A) inhibitor, exerting inhibitory effects on both PP2A and PP1, with IC50 values of 90 nM and 5 µM,Fórmula:C8H10O5Pureza:98.89% - ≥98%Forma y color:Cyrstalline White Solid The Monohydrate Is In The Form Of Colorless Crystals Non Corrosive Used As A Selective HerbicidePeso molecular:186.16ERAP2-IN-1
CAS:ERAP2-IN-1 is a specific non-competitive ERAP2 inhibitor with IC50s of 27 μM for Arg-AMC and 44 μM for peptides.Fórmula:C20H21F3N2O5SForma y color:SolidPeso molecular:458.4511β-HSD1-IN-6
CAS:11β-HSD1-IN-6 is a potent inhibitor of 11β hydroxysteroid dehydrogenase enzymes (11β-HSDs).Fórmula:C21H19ClN4OForma y color:SolidPeso molecular:378.86hCAIX/XII-IN-4
CAS:hCAIX/XII-IN-4 inhibits CAIX/XII with Ki: 4.5 nM (CAXII), 23.6 nM (CAIX), and >10000 nM (CAI/CAII).Fórmula:C20H16N2O5Forma y color:SolidPeso molecular:364.35Carbonic anhydrase inhibitor 11
CAS:Potent carbonic anhydrase inhibitor VI targets CA II, IX, XII with Ki: 40, 39, 900 nM respectively.Fórmula:C19H15F3N4O3S2Forma y color:SolidPeso molecular:468.47PTP1B-IN-15
CAS:PTP1B-IN-15 is a potent and selective protein tyrosine phosphatase 1B (PTP1B) inhibitor that has shown research potential in type II diabetes and obesity.Fórmula:C19H17Br2NO5SForma y color:SolidPeso molecular:531.22(S)-Bromoenol lactone
CAS:(S)-BEL, a chiral inhibitor of iPLA2β, blocks vasopressin-induced arachidonate release in A10 cells; IC50 = 2μM.Fórmula:C16H13BrO2Forma y color:SolidPeso molecular:317.18Oxythiamine diphosphate
CAS:Oxythiamine diphosphate is a competitivethiamine pyrophosphate inhibitor(Ki of 30 nM).Fórmula:C12H17N3O8P2SPureza:98%Forma y color:SolidPeso molecular:425.29CM39
CAS:CM39 inhibits ALDH, linked to cancer stem-like cells & chemoresistance.Fórmula:C19H15FN4OSForma y color:SolidPeso molecular:366.41ABD-1970
CAS:ABD-1970 is a highly potent and selective MGLL inhibitor.Fórmula:C21H24ClF6N3O3Forma y color:SolidPeso molecular:515.88Deoxyhypusine
CAS:Deoxyhypusine is a enzyme.Fórmula:C10H23N3O2Forma y color:SolidPeso molecular:217.31ATX inhibitor 16
CAS:ATX inhibitor 16 is a potent inhibitor of ATX (IC50: 0.0021 μM). ATX inhibitor 16 exhibits a significant anti-proliferative effect on breast cancer cells.Fórmula:C28H27F3N6OS2Forma y color:SolidPeso molecular:584.68ICI 211965
CAS:ICI 211965 is a selective and orally potent of 5-Lipoxygenase (5-LPO).Fórmula:C24H23NO2SPureza:98%Forma y color:SolidPeso molecular:389.51SCH-42354
CAS:SCH-42354: potent oral NEP inhibitor, activates ANP & leu-enkephalin, has anti-hypertensive properties, IC50s of 8.3 & 10.0 nM.Fórmula:C16H23NO3S2Forma y color:SolidPeso molecular:341.49F-1394
CAS:F-1394 is an ACAT inhibitor that reduces atherosclerosis and neointimal thickening without changing serum cholesterol.Fórmula:C33H61N3O6Forma y color:SolidPeso molecular:595.85S6821
CAS:S6821 is a non-mutagenic TAS2R8 antagonist; no clastogenic or micronuclei induction found.Fórmula:C19H19N5O4Forma y color:SolidPeso molecular:381.39
