Metabolismo
Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.
Subcategorías de "Metabolismo"
- AhR(41 productos)
- Aminopeptidasa(75 productos)
- CETP(20 productos)
- Anhídrido carbónico(188 productos)
- Caseína quinasa(137 productos)
- DHFR(34 productos)
- Descarboxilasa(4 productos)
- Deshidrogenasa(296 productos)
- FAAH(65 productos)
- FXR(59 productos)
- Factor Xa(85 productos)
- Ácido graso sintasa(37 productos)
- Ferroptosis(221 productos)
- GR(3 productos)
- GSNOR(4 productos)
- Glucoquinasa(56 productos)
- HIF / HIF Prolilhidroxilasa(146 productos)
- HMG-CoA reductasa(33 productos)
- Hidroxilasa(35 productos)
- IDO(84 productos)
- LDL(8 productos)
- Lipasa(105 productos)
- Lípido(62 productos)
- Lipoxigenasa(133 productos)
- MAO(87 productos)
- MPO(2 productos)
- NAMPT(40 productos)
- P450(6 productos)
- PAI-1(26 productos)
- PDE(166 productos)
- PED(1 productos)
- PKM(15 productos)
- PPAR(169 productos)
- Fosfolipasa(82 productos)
- ROR(45 productos)
- Receptor de retinoides(28 productos)
- SGK(11 productos)
- Tiorredoxina(12 productos)
- Transferasa(29 productos)
- Transportador(46 productos)
- UGT(4 productos)
- Inhibidores de la xantina oxidasa (XO)(9 productos)
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Se han encontrado 9132 productos de "Metabolismo"
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YCT529 free acid
CAS:YCT529 free acid is a potent, selective and orally active RAR-α inhibitor .Fórmula:C29H25NO3Forma y color:SolidPeso molecular:435.51hCAIX/XII-IN-6
hCAIX/XII-IN-6: Oral carbonic anhydrase inhibitor, targets hCA I/II/IV/IX/XII, aids rheumatoid arthritis research. Ki: 6697/2950/4093/4.1/7.7 nM.Fórmula:C26H23N3O6S4Forma y color:SolidPeso molecular:601.74hCAI/II-IN-3
CAS:"hCAI/II-IN-3 (compound 5b) is a potent dual hCA I/II inhibitor with Ki: 51.25nM (I), 13.15nM (II), helps treat AMS."Fórmula:C16H18N4O4S2Forma y color:SolidPeso molecular:394.47Sp-cAMPS
CAS:Rp-cAMPS TEA salt is a cAMP-dependent protein kinase (PKA) activator.Fórmula:C10H12N5O5PSForma y color:SolidPeso molecular:345.27CAY10761
CAS:CAY10761 inhibits ENPP1 (IC50: 467 μM human, 429 μM snake), mushroom tyrosinase (Ki: 1.9 μM), and urease from different sources (IC50: 0.093-<0.125 mM).Fórmula:C7H8N4O2S2Forma y color:SolidPeso molecular:244.29FR-221647
CAS:FR-221647: non-nucleoside adenosine deaminase blocker, moderate efficacy, better pharmacokinetics than EHNA/Pentostatin.Fórmula:C14H17N3O2Forma y color:SolidPeso molecular:259.311β-HSD1-IN-10
CAS:11β-HSD1-IN-10, a potent inhibitor of 11β-HSD1 with an IC50 value of 1.8 µM for humans, is suitable for research into obesity, hyperglycemia, and cognitiveFórmula:C16H10F3NO2Forma y color:SolidPeso molecular:305.25hCAI/II-IN-2
CAS:hCAI/II-IN-2 (2b) inhibits hCA I/II (Ki: 40.97 nM, 15.15 nM) and IX (61.88 nM), fights AMS with anti-hypoxic effects, but has low cellular activity.Fórmula:C12H12N4O5S2Forma y color:SolidPeso molecular:356.38PF 04671536 hydrochloride
CAS:Potent PDE8B/8A inhibitor; IC50: PDE8B-1.3nM, PDE8A-1.9nM; selective over other PDEs; enhances insulin secretion; orally bioavailable.Fórmula:C14H19ClN8OSForma y color:SolidPeso molecular:382.87TAK 21d
CAS:Potent FAAH inhibitorFórmula:C19H17F2N7OPureza:98%Forma y color:SolidPeso molecular:397.3814-dehydro Zymostenol
CAS:14-dehydro Zymostenol, a cholesterol precursor, boosts MBP+ oligodendrocytes from precursors at 5.8-17 μM.Fórmula:C27H44OForma y color:SolidPeso molecular:384.64TPN729MA
CAS:<p>TPN729MA, a potent PDE5 inhibitor, IC50: 2.28 nM, targets erectile dysfunction research.</p>Fórmula:C29H40N6O8SForma y color:SolidPeso molecular:632.73Quetiapine sulfoxide
CAS:Quetiapine sulfoxide: Main metabolite of Quetiapine, a 5-HT agonist & dopamine antagonist antipsychotic.Fórmula:C21H25N3O3SPureza:98%Forma y color:Pale Yellow SolidPeso molecular:399.51DNJNAc
CAS:DNJNAc (2-Acetamido-1,2-dideoxynojirimycin) is a potent β-hexosaminidase inhibitor, reducing cartilage matrix degradation, relevant in glycoconjugate studies.Fórmula:C8H16N2O4Pureza:98.65% - 99.37%Forma y color:SolidPeso molecular:204.22Loxoprofenol-SRS
CAS:Loxoprofenol-SRS, a potent metabolite of Loxoprofen, is an IV NSAID with enhanced anti-inflammatory and pain relief properties.Fórmula:C15H20O3Forma y color:SolidPeso molecular:248.32N-Oleoyl Leucine
CAS:N-Oleoyl Leucine (Oleoyl-L-leucine) is an N-fatty acyl amino acid present in plasma.Fórmula:C24H45NO3Pureza:98.25%Forma y color:SolidPeso molecular:395.62LB42908
CAS:LB42908 is a highly potent Ras farnesyltransferase inhibitor(IC(50)=0.9 nM against H-Ras and 2.4 nM against K-Ras) with potential anticancer activity.Fórmula:C32H31N5O3Forma y color:SolidPeso molecular:533.62TPN729
CAS:TPN729, a PDE5 inhibitor, has an IC50 of 2.28 nM, used to research erectile dysfunction.Fórmula:C25H36N6O4SForma y color:SolidPeso molecular:516.66(R)-MLN-4760
CAS:(R)-MLN-4760, the R-enantiomer of MLN-4760, functions as an ACE2 inhibitor and exhibits a half maximal inhibitory concentration (IC50) of 8.4 μM, identifying itFórmula:C19H23Cl2N3O4Forma y color:SolidPeso molecular:428.31LY367385
CAS:LY367385 is a highly effective and selective mGluR1a antagonist.Fórmula:C10H11NO4Pureza:98%Forma y color:SolidPeso molecular:209.2hCAI/II-IN-1
CAS:<p>hCAI/II-IN-1 (Compound 3h) is a human carbonic anhydrase I and II (hCA I/II) inhibitor that acts on hCA I (IC50: 0.047 μM) and hCA II (IC50: 0.024 μM).</p>Fórmula:C18H29N5O3S3Forma y color:SolidPeso molecular:459.65LY 56110
CAS:LY 56110 is a novel nonsteroidal aromatase inhibitor.Fórmula:C17H12Cl2N2Pureza:98%Forma y color:SolidPeso molecular:315.2TFB-TBOA
CAS:glial glutamate transporter EAAT1 and EAAT2 inhibitorFórmula:C19H17F3N2O6Pureza:98%Forma y color:SolidPeso molecular:426.34Enpp-1-IN-6
CAS:Enpp-1-IN-6, a potent enpp-1 inhibitor, may aid cancer and infectious disease studies (WO2021203772A1, compound 51).Fórmula:C22H28N4O5SForma y color:SolidPeso molecular:460.55PDE1-IN-3
CAS:PDE1-IN-3 is a selective inhibitor of human phosphodiesterase 1 (PDE1).Fórmula:C18H24N4OPureza:98%Forma y color:SolidPeso molecular:312.41Carbazomycin B
CAS:Carbazomycin B, a Streptomyces metabolite, combats fungi, bacteria, P. falciparum, C. albicans, and some cancer cells; inhibits 5-LO (IC50=1.5µM).Fórmula:C15H15NO2Forma y color:SolidPeso molecular:241.29Fodipir
CAS:Fodipir, the active metabolite of mangafodipir, plays a crucial role in the mechanism of mangafodipir-mediated cytoprotection, specifically mitigating cellFórmula:C22H32N4O14P2Pureza:98%Forma y color:SolidPeso molecular:638.46GS 389
CAS:GS 389, a tetrahydroisoquinoline, relaxes blood vessels by inhibiting brain PDE and raising aorta cGMP.Fórmula:C19H23NO3Pureza:98%Forma y color:SolidPeso molecular:313.39Darexaban glucuronide
CAS:Darexaban glucuronide is the major component in plasma after oral administration of darexaban to humans. Darexaban (YM150) is a direct inhibitor of factor Xa.Fórmula:C33H38N4O10Forma y color:SolidPeso molecular:650.68(Rac)-Etavopivat
CAS:(Rac)-Etavopivat, an oral PKR activator, targets sickle cell disease and haemoglobinopathies.Fórmula:C22H23N3O6SForma y color:SolidPeso molecular:457.5ARL-67156 trisodium salt hydrate
CAS:ARL-67156 trisodium salt hydrate is an ecto-ATPase inhibitor that prevents metabolism of P2 purinoceptor agonists.Fórmula:C15H24Br2N5O12P3Forma y color:SolidPeso molecular:719.11Seviteronel R enantiomer
CAS:Seviteronel R enantiomer (VT-464 R enantiomer) is a Seviteronel isomer produced during the manufacturing process.Fórmula:C18H17F4N3O3Pureza:97.97% - >99.99%Forma y color:SolidPeso molecular:399.34ZSET-845
CAS:<p>ZSET-845 is an enhancer of cognitive which enhances choline acetyltransferase activity in the hippocampus in the rat.</p>Fórmula:C21H18N2OPureza:98%Forma y color:SolidPeso molecular:314.38γ-Methylleucine
CAS:Gamma-Methylleucine (2-Amino-3-tert-butylpropionic acid) is an auxiliary for copper-catalyzed asymmetric Michael reactions.Fórmula:C7H15NO2Pureza:≥98%Forma y color:SolidPeso molecular:145.2Mevalonic acid
CAS:Mevalonic acid is essential for cell growth and proliferation,Mevalonic acid is a precursor in the mevalonate pathway.Fórmula:C6H12O4Pureza:98%Forma y color:SolidPeso molecular:148.16LP117
CAS:LP117 is a novel and effective inhibitor of 5-Lipoxygenase (5-LO) product synthesis (IC50: 1.1 μM).Fórmula:C21H23ClN4O2SPureza:98%Forma y color:SolidPeso molecular:430.95IDO-IN-5
CAS:IDO-IN-5 is an indoleamine 2,3-dioxygenase (IDO) inhibitor (IC50: 1-10 μM).Fórmula:C18H21FN2O2Pureza:98%Forma y color:SolidPeso molecular:316.37GKA-22
CAS:GKA-22 is a human glucokinase allosteric activator in the absence of glucose.Fórmula:C22H22N2O5SPureza:98%Forma y color:SolidPeso molecular:426.49Dimethyl-bisphenol A
CAS:<p>DMBPA inhibits HIF-1α, promotes its degradation by detaching Hsp90, and reduces Vegfa mRNA expression.</p>Fórmula:C17H20O2Forma y color:SolidPeso molecular:256.34BN-82685
CAS:<p>BN-82685, a quinone-based CDC25 inhibitor, shows in vitro and in vivo efficacy, suggesting potential as an anticancer therapy.</p>Fórmula:C12H15N3O2SPureza:98%Forma y color:SolidPeso molecular:265.33Win-62005
CAS:Win-62005 is an inhibitor of cyclic AMP phosphodiesterase III (PDE III)(Kis: 25 and 26 nM for rat heart and canine aorta).Fórmula:C12H10N4OPureza:98%Forma y color:SolidPeso molecular:226.23Dacisteine
CAS:Dacisteine (N,S-Diacetyl-L-cysteine) is an inhibitor of New Delhi metallo-beta-lactamase-1 (NDM-1, IC50 = 1000 μM).Fórmula:C7H11NO4SPureza:99.57%Forma y color:SolidPeso molecular:205.23PGAM1-IN-1
CAS:PGAM1-IN-1 is an inhibitor of phosphoglycerate mutase 1 ( PGAM1 ) with an IC 50 of 6.4 μM [1].Fórmula:C19H11ClFNO6SPureza:98%Forma y color:SolidPeso molecular:435.81Abiraterone decanoate
CAS:Abiraterone decanoate is a prodrug of Abiraterone that provides controlled release and prolonged inhibition of the enzyme CYP17 through intramuscular.Fórmula:C34H49NO2Pureza:99.69%Forma y color:SolidPeso molecular:503.76NPD-001
CAS:<p>NPD-001 is an effective inhibitor of TbrPDEB1. NPD-001 is 10-fold more potent on hPDE4 (hPDE4B1 IC50 = 0.6 nM) than on TbrPDEB1 (IC50 = 4 nM).</p>Fórmula:C33H40N6O4Pureza:98%Forma y color:SolidPeso molecular:584.71Leniquinsin
CAS:Leniquinsin is an antihypertensive compound. It is a phosphodiesterase inhibitor and a potent vasodilator.Fórmula:C20H20N2O4Pureza:98%Forma y color:SolidPeso molecular:352.381E7-03
CAS:<p>1E7-03 is an inhibitor of HIV-1 transcription, by targeting host Protein Phosphatase-1 (PP1).</p>Fórmula:C28H29N3O6Forma y color:SolidPeso molecular:503.55KT109
CAS:KT109 is a DAGLβ inhibitor (IC50=42nM), lessens LPS allodynia in mice without tolerance, and has no major side effects.Fórmula:C27H26N4OPureza:98%Forma y color:SolidPeso molecular:422.52Tanogitran
CAS:Tanogitran, a coagulation factor Xa inhibitor, is used potentially for the treatment of septic shock.Fórmula:C25H31N7O3Pureza:98%Forma y color:SolidPeso molecular:477.56TC-E 5008
CAS:TC-E 5008 is a selective inhibitor of mutant isocitrate dehydrogenase 1 (mIDH1).Fórmula:C13H13NO2Forma y color:SolidPeso molecular:215.25
