Metabolismo
Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.
Subcategorías de "Metabolismo"
- AhR(41 productos)
- Aminopeptidasa(67 productos)
- CETP(18 productos)
- Anhídrido carbónico(178 productos)
- Caseína quinasa(130 productos)
- DHFR(33 productos)
- Descarboxilasa(4 productos)
- Deshidrogenasa(270 productos)
- FAAH(64 productos)
- FXR(58 productos)
- Factor Xa(80 productos)
- Ácido graso sintasa(33 productos)
- Ferroptosis(215 productos)
- GR(3 productos)
- GSNOR(3 productos)
- Glucoquinasa(54 productos)
- HIF / HIF Prolilhidroxilasa(142 productos)
- HMG-CoA reductasa(33 productos)
- Hidroxilasa(30 productos)
- IDO(82 productos)
- LDL(8 productos)
- Lipasa(97 productos)
- Lípido(59 productos)
- Lipoxigenasa(125 productos)
- MAO(87 productos)
- MPO(2 productos)
- NAMPT(36 productos)
- P450(6 productos)
- PAI-1(25 productos)
- PDE(166 productos)
- PED(1 productos)
- PKM(15 productos)
- PPAR(164 productos)
- Fosfolipasa(82 productos)
- ROR(42 productos)
- Receptor de retinoides(29 productos)
- SGK(11 productos)
- Tiorredoxina(12 productos)
- Transferasa(30 productos)
- Transportador(42 productos)
- UGT(4 productos)
- Inhibidores de la xantina oxidasa (XO)(9 productos)
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Se han encontrado 8626 productos de "Metabolismo"
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ω-Conotoxin MVIID
<p>ω-Conotoxin MVIID (SNX-238) is a peptide from the Conus genus that inhibits the ω-Conotoxin-GVIA-sensitive, high-threshold calcium (Ca 2+) current in fish</p>Fórmula:C99H164N42O33S7Pureza:98%Forma y color:SolidPeso molecular:2695.08ITH12711
<p>ITH12711, a PP2A ligand, can traverse the blood-brain barrier (BBB) and exerts neuroprotection by restoring PP2A-phosphatase activity [1].</p>Fórmula:C12H20O5Pureza:98%Forma y color:SolidPeso molecular:244.28Calcium 2-oxoglutarate
CAS:<p>Calcium 2-oxoglutarate is an intermediate in the production of GTP or ATP in the Krebs cycle. It is a reversible inhibitor of tyrosinase (IC50: 15 mM).</p>Fórmula:C5H8CaO5Pureza:98%Forma y color:SolidPeso molecular:188.192Hydroxocobalamin
CAS:<p>Hydroxocobalamin (Vitamin B12a) is a naturally occurring, injectable form of vitamin B12 used as a dietary supplement to treat B12 deficiency, including</p>Fórmula:C62H89CoN13O15PPureza:98%Forma y color:SolidPeso molecular:1346.36α-Hydroxytamoxifen
CAS:<p>α-Hydroxytamoxifen is a metabolite of tamoxifen. It reacts with DNA and causes the formation of DNA adducts.</p>Fórmula:C26H29NO2Pureza:98%Forma y color:SolidPeso molecular:387.51CAIX Inhibitor S4
CAS:<p>CAIX Inhibitor S4 (S4) is an effective inhibitor of carbonic anhydrase IX/XII with a Ki of 7 nM and 2 nM, respectively.</p>Fórmula:C15H17N3O4SPureza:99.07%Forma y color:SolidPeso molecular:335.38Glycolithocholic acid, sodium salt
CAS:<p>Sodium glycolithocholate is a bile acid salt used to diagnose UC, NASH, and PSC.</p>Fórmula:C26H42NNaO4Pureza:99.95%Forma y color:SolidPeso molecular:455.61Bz-Ala-Arg
CAS:<p>Bz-Ala-Arg, a dipeptide, serves as a spectrophotometric substrate (0.4 M pyridine formate, pH 4.25) for human pancreatic carboxypeptidase B and plasma</p>Fórmula:C16H23N5O4Pureza:98%Forma y color:SolidPeso molecular:349.38ω-Conotoxin CVIE
<p>ω-Conotoxin CVIE selectively inhibits voltage-gated Ca^2+ channels (Ca_v 2.2) [1].</p>Fórmula:C98H164N40O34S6Pureza:98%Forma y color:SolidPeso molecular:2638.99(±)13(14)-EpDPA
CAS:<p>Cytochrome P450 metabolism of polyunsaturated fatty acids produces numerous bioactive epoxide regioisomers.</p>Fórmula:C22H32O3Forma y color:SolidPeso molecular:344.495ω-Conotoxin Bu8
<p>ω-Conotoxin Bu8 is a 25-amino-acid-residue ω-conotoxin that features three disulfide bridges.</p>Fórmula:C103H174N42O35S6Pureza:98%Forma y color:SolidPeso molecular:2753.13UDP-3-O-acyl-GlcNAc diammonium
<p>UDP-3-O-acyl-GlcNAc diammonium serves as a metabolite in E. coli, playing a critical role in the biosynthesis pathway of 3-deoxy-D-manno-octulosonate (KDO) [1].</p>Fórmula:C31H59N5O19P2Pureza:98%Forma y color:SolidPeso molecular:867.77ω-Conotoxin CnVIIA
CAS:<p>ω-Conotoxin CnVIIA, a 27-amino-acid neuropeptide toxin, serves as an N-type calcium current blocker [1].</p>Fórmula:C110H179N39O36S7Pureza:98%Forma y color:SolidPeso molecular:2848.29Histone acetyltransferase p300 Inhibitor 4c
CAS:<p>2-Amino-4-(4-chlorophenyl)thiazole blocks hCA I/II, AChE, BChE with Ki: ~0.008, 0.124, 0.129, 0.083 µM.</p>Fórmula:C9H7ClN2SPureza:99.76%Forma y color:SolidPeso molecular:210.68Isocrenatoside
CAS:<p>Isocrenatoside (compound 6), a cyclic octapeptide derived from the ethanolic extract of Microtoena prainiana stems, functions as an angiotensin-converting</p>Fórmula:C29H34O15Pureza:98%Forma y color:SolidPeso molecular:622.57Coumachlor
CAS:<p>Coumachlor, a first-generation anticoagulant rodenticide, blocks the formation of prothrombin and inhibits blood coagulation causing internal haemorrhage.</p>Fórmula:C19H15ClO4Forma y color:SolidPeso molecular:342.77Casuarictin
CAS:<p>Casuarictin, a potent competitive inhibitor of α-glucosidase, exhibits an IC50 of 0.21 μg/mL and functions as a presenilin stabilization factor-like (PSFL)</p>Fórmula:C41H28O26Pureza:98%Forma y color:SolidPeso molecular:936.653'-sulfo Galactosylsphingosine (ammonium salt)
CAS:<p>Sulfatide derivative inhibits cell migration, adhesion, PKC, cytochrome c; accumulates in metachromatic leukodystrophy; used for LC-MS quantification.</p>Fórmula:C24H50N2O10SForma y color:SolidPeso molecular:558.73Endo-1,3-β-glucanase
CAS:<p>Endo-1,3-β-glucanase (Lyticase) is a glucanase from fungi and Chlamydomonas reinhardtii that displays lytic activity on fungal cells.</p>Forma y color:SolidMersalyl
CAS:<p>Mersalyl is an organic mercurial diuretic.</p>Fórmula:C13H16HgNNaO6Forma y color:SolidPeso molecular:505.854MeIQx
CAS:<p>MeIQx, a carcinogenic compound in cooked fish/meat, triggers DNA-reactive metabolites and rat tumors.</p>Fórmula:C11H11N5Forma y color:SolidPeso molecular:213.244Clostripain
CAS:<p>Clostripain is a protease from Clostridium with esterase, amidase activities, targeting arginine.</p>Forma y color:Solidω-Tbo-IT1
<p>ω-Tbo-IT1, a peptide toxin extracted from the venom of Tibellus oblongus, functions as an inhibitor of insect calcium channels [1].</p>Fórmula:C171H285N61O53S9Pureza:98%Forma y color:SolidPeso molecular:4332.05Decanoyl coenzyme A
CAS:<p>Decanoyl coenzyme A (Decanoyl CoA) serves as a primer for the fatty acid elongation system in Mycobacterium smegmatis [1].</p>Fórmula:C31H54N7O17P3SForma y color:SolidPeso molecular:921.78Systemin
CAS:<p>Systemin is an 18-amino acid polypeptide with the sequence AVQSKPPSKRDPPKMQTD that is found in Solanaceae plants (such as tomato and potato).</p>Fórmula:C85H144N26O28SPureza:98%Forma y color:SolidPeso molecular:2010.28α-Glucosidase-IN-80
<p>α-Glucosidase-IN-80 (Compound 10n) is a potent competitive inhibitor of α-glucosidase, with an IC50 of 48.4 μM. It exhibits favorable pharmacokinetic properties and toxicity profiles, making it suitable for research in diabetes-related conditions.</p>Fórmula:C24H24N8OS2Forma y color:SolidPeso molecular:504.63PP5-IN-2
<p>PP5-IN-2, a selective and orally active inhibitor of protein phosphatase 5 (PP5), exhibits an IC 50 of 0.9 μM. This compound activates p53 and leads to the downregulation of cyclin D1 and MGMT, thereby inducing cell cycle arrest and reversing Temozolomide (TMZ) resistance in the U87 MG cell line. Additionally, PP5-IN-2 has demonstrated effective inhibition of tumor growth in the xenograft mouse model.</p>Fórmula:C16H15NO4Forma y color:SolidPeso molecular:285.29Imatinib Impurity E
CAS:<p>Imatinib Impurity E, a derivative of orally taken Imatinib, inhibits tyrosine kinases BCR/ABL, PDGFR, c-kit, and SARS/MERS-CoV.</p>Fórmula:C52H48N12O2Forma y color:SolidPeso molecular:873.02Prostaglandin F2β
CAS:<p>Prostaglandin F2β (PGF2β) is the 9β-hydroxy stereoisomer of PGF2α.</p>Fórmula:C20H34O5Forma y color:White SolidPeso molecular:354.48Nε,Nε,Nε-Trimethyllysine chloride
CAS:<p>Nε,Nε,Nε-Trimethyllysine chloride (Lys(Me)3-OH Chloride) is a methylated derivative of the amino acid lysine and a component of histone proteins.</p>Fórmula:C9H21ClN2O2Pureza:99.83%Forma y color:SolidPeso molecular:224.73GSK-3β/CK-1δ-IN-1
<p>GSK-3β/CK-1δ-IN-1 (8d) is a dual inhibitor of GSK-3β and CK-1δ that can cross the blood-brain barrier, with IC50 values of 0.77 μM and 0.57 μM, respectively. GSK-3β/CK-1δ-IN-1 (8d) is applicable in neuroblastoma research.</p>Fórmula:C22H17F3N4OForma y color:SolidPeso molecular:410.39Pestalotin
CAS:<p>Pestalotin, a fungal derivative, promotes rice seedling growth and sugar release, has antifungal properties, and is cytotoxic to certain cells.</p>Fórmula:C11H18O4Forma y color:SolidPeso molecular:214.26Lantanose A
CAS:<p>Lantanose A is a bioactive chemical from Lantana cumara roots.</p>Fórmula:C30H52O26Pureza:98%Forma y color:SolidPeso molecular:828.72D-galactosyl-β1-3-N-acetyl-D-hexosamine phosphorylase (BiGalHexNAcP)
<p>D-galactosyl-β1-3-N-acetyl-D-hexosamine phosphorylase (BiGalHexNAcP), belonging to the CAZy glycoside hydrolase family GH112, plays a pivotal role in</p>Forma y color:SolidCAXII-IN-2
<p>CAXII-IN-2 (compound 3j) is a highly effective inhibitor of CAXII. It demonstrates inhibitory activity against CA IX and CAXII, with Ki values of 27.4 nM and 4.0 nM, respectively.</p>Fórmula:C16H13FNO4PForma y color:SolidPeso molecular:333.05662(+)-Geodin
CAS:<p>(+)-Geodin, a fungal metabolite, boosts fibrinolysis in BAECs (50-150 μM) and glucose uptake in rat adipocytes (1-100 μg/ml).</p>Fórmula:C17H12Cl2O7Forma y color:SolidPeso molecular:399.18DSPE-PEG5000-ANG
<p>DSPE-PEG5000-ANG is a PEGylated compound formed by DSPE and the dual-targeting ligand (Angiopep-2, ANG). ANG exhibits high binding efficacy to LRP1 and has been utilized for targeting glioma delivery. DSPE-PEG5000-ANG is applicable in drug delivery.</p>Forma y color:Odour SolidMethyl gerfelin
CAS:<p>Methyl gerfelin, a flavonoid, hinders osteoclast formation by targeting GLO1, SCP2, and SGTA proteins.</p>Fórmula:C16H16O6Forma y color:SolidPeso molecular:304.29Octanoyl Coenzyme A (sodium salt)
<p>Octanoyl Coenzyme A (sodium salt) inhibits citrate synthase and glutamate dehydrogenase with an IC50 of 0.4–1.6 mM.</p>Fórmula:C29H49N7NaO17P3SForma y color:SolidPeso molecular:915.71Plipastatin A1
CAS:<p>Plipastatin A1, a lipopeptide isolated from B.</p>Fórmula:C72H110N12O20Forma y color:SolidPeso molecular:1463.7113,14-dehydro-15-cyclohexyl Carbaprostacyclin
CAS:<p>13,14-dehydro-15-cyclohexyl Carbaprostacyclin, a stable PGI2 analog, impedes ADP-induced platelet aggregation; ED50 ~40 nM in PRP, 77 nM in washed platelets.</p>Fórmula:C21H30O4Forma y color:SolidPeso molecular:346.467α-Amylase/α-Glucosidase-IN-11
<p>α-Amylase/α-Glucosidase-IN-11 (Compound 5d) is an isoxazoline-indigo hybrid with notable antidiabetic properties. It acts as a competitive inhibitor of the key digestive enzymes α-amylase (IC50 = 30.39 μM) and α-glucosidase (IC50 = 65.1 μM). Additionally, it does not penetrate the blood-brain barrier.</p>Fórmula:C33H40ClN5O5Peso molecular:621.2718DSPE-PEG5000-NYZL1
<p>DSPE-PEG5000-NYZL1 is a PEG compound composed of DSPE and NYZL1, where NYZL1 specifically binds to bladder cancer tissues and cells. DSPE-PEG5000-NYZL1 is applicable for drug delivery.</p>Forma y color:Odour SolidCMP-Sialic acid
CAS:<p>CMP-Sialic acid inhibits UDP-GlcNAc 2-epimerase and is a key substrate for sialic acid biosynthesis.</p>Fórmula:C20H31N4O16PForma y color:SolidPeso molecular:614.45hCAI/II-IN-10
<p>hCAI/II-IN-10 (Compound 5d) is an inhibitor of human carbonic anhydrase I and II (hCA I and hCA II), with IC50 values of 4.32 nM and 3.89 nM, respectively.</p>Fórmula:C24H17Cl2N3O3S2Forma y color:SolidPeso molecular:530.446Glycidamide
CAS:<p>Glycidamide is a carcinogen and metabolite of acrylamide that induces DNA adduct formation and mutations.</p>Fórmula:C3H5NO2Forma y color:SolidPeso molecular:87.08(Rac)-5-Keto Fluvastatin
CAS:<p>(Rac)-5-Keto Fluvastatin (rac 5-Keto Fluvastatin) is an impurity of Fluvastatin which is an inhibitor of HMG-CoA reductase.</p>Fórmula:C24H24FNO4Pureza:95.04%Forma y color:SolidPeso molecular:409.45SGK1-IN-4
CAS:<p>SGK1-IN-4 is a selective inhibitor of SGK1 and can be used in studies about osteoarthritis.</p>Fórmula:C23H21ClFN5O4SPureza:97.03%Forma y color:SolidPeso molecular:517.969AzNue5Ac
CAS:<p>9AzNue5Ac is a Neu5Ac analog that is metabolized in vivo in living cells and in mice.9AzNue5Ac binds to sialoglycans.</p>Fórmula:C11H18N4O8Pureza:≥98%Forma y color:SolidPeso molecular:334.2815-LOX-1 inhibitor 1
CAS:<p>9c(i472) blocks 15-LO-1 (IC50=0.19μM), lowers NF-κB in RAW-Blue cells, & cuts Nos2/lipid peroxidation in RAW 264.7 at 0.2-5μM.</p>Fórmula:C22H21ClN2O4Forma y color:SolidPeso molecular:412.87
