
Metabolismo
Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.
Subcategorías de "Metabolismo"
- AhR(42 productos)
- Aminopeptidasa(76 productos)
- CETP(20 productos)
- Anhídrido carbónico(197 productos)
- Caseína quinasa(139 productos)
- DHFR(30 productos)
- Descarboxilasa(4 productos)
- Deshidrogenasa(303 productos)
- FAAH(64 productos)
- FXR(63 productos)
- Factor Xa(87 productos)
- Ácido graso sintasa(37 productos)
- Ferroptosis(233 productos)
- GR(3 productos)
- GSNOR(3 productos)
- Glucoquinasa(56 productos)
- HIF / HIF Prolilhidroxilasa(146 productos)
- HMG-CoA reductasa(36 productos)
- Hidroxilasa(36 productos)
- IDO(84 productos)
- LDL(7 productos)
- Lipasa(107 productos)
- Lípido(62 productos)
- Lipoxigenasa(134 productos)
- MAO(84 productos)
- MPO(2 productos)
- NAMPT(40 productos)
- P450(6 productos)
- PAI-1(26 productos)
- PDE(169 productos)
- PED(1 productos)
- PKM(17 productos)
- PPAR(170 productos)
- Fosfolipasa(84 productos)
- ROR(47 productos)
- Receptor de retinoides(16 productos)
- SGK(10 productos)
- Tiorredoxina(12 productos)
- Transferasa(30 productos)
- Transportador(43 productos)
- UGT(4 productos)
- Inhibidores de la xantina oxidasa (XO)(9 productos)
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Se han encontrado 9205 productos de "Metabolismo"
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DG172 dihydrochloride
CAS:DG172 dihydrochloride (DG-172 dihydrochloride) is an antagonist of PPARβ/δ(IC50 : 27 nM).
Fórmula:C20H22BrCl2N3Pureza:99.87%Forma y color:SolidPeso molecular:455.2PT-2385
CAS:PT-2385 is a selective HIF-2α inhibitor (Kd<50 nM).Fórmula:C17H12F3NO4SPureza:98.91% - 99.55%Forma y color:SolidPeso molecular:383.34Ref: TM-T7848
1mg63,00€2mg93,00€1mL*10mM (DMSO)119,00€5mg144,00€10mg222,00€25mg379,00€50mg532,00€100mg740,00€200mg982,00€Firsocostat
CAS:Firsocostat (GS-0976) is an inhibitor of acetyl-CoA carboxylase (ACC) dimerization that inhibits human ACC1 and ACC2 activity (IC50s of 2.1 and 6.1 nM).Fórmula:C28H31N3O8SPureza:98% - 99.39%Forma y color:SolidPeso molecular:569.63Ref: TM-T7184
1mg92,00€2mg120,00€5mg200,00€1mL*10mM (DMSO)251,00€10mg334,00€25mg484,00€50mg622,00€100mg859,00€500mg1.701,00€Lofemizole
CAS:Lofemizole is an antagonist of CYP1A2.Fórmula:C10H9ClN2Pureza:97.11%Forma y color:SolidPeso molecular:192.64Ref: TM-T50053
1mg34,00€1mL*10mM (DMSO)60,00€5mg71,00€10mg95,00€25mg161,00€50mg234,00€100mg331,00€200mg455,00€PDE10-IN-1
CAS:PDE10-IN-1 (SEP-0372814) is used for treating CNS and metabolic disorders.Fórmula:C21H19N7Pureza:99.65%Forma y color:SolidPeso molecular:369.42IOX4
CAS:IOX4 is a potent PHD2 inhibitor (IC50 = 1.6 nM)Fórmula:C15H16N6O3Pureza:99.97%Forma y color:SolidPeso molecular:328.33Amifostine trihydrate
CAS:Amifostine trihydrate (WR2721) is the first approved radioprotective drug, used to decrease the risk of kidney problems caused by treatment with cisplatin.Fórmula:C5H15N2O3PS·3H2OPureza:99.71% - 99.80%Forma y color:SolidPeso molecular:268.27DMU-2139
CAS:DMU2139 is a specific CYP1B1 inhibitor (CYP1B1 and CYP1A1 with IC50 of 9 nM and 795 nM, respectively).Fórmula:C19H15NO2Pureza:98.88%Forma y color:SolidPeso molecular:289.33Ref: TM-T8728
1mg35,00€5mg75,00€1mL*10mM (DMSO)75,00€10mg110,00€25mg215,00€50mg316,00€100mg470,00€200mg682,00€PSB-1434
CAS:PSB-1434 is a selective and competitive monoamine oxidase B inhibitor with IC50 of 1.59 nM, selectivity versus MAO-A>6000-fold.Fórmula:C14H9F2N3OPureza:99.57%Forma y color:SolidPeso molecular:273.24Ref: TM-T24679
1mg86,00€1mL*10mM (DMSO)167,00€5mg177,00€10mg268,00€25mg439,00€50mg628,00€100mg870,00€200mg1.153,00€SR0987
CAS:SR0987 is a RORγt agonist,Fórmula:C16H10ClF6NO2Pureza:99.43%Forma y color:SolidPeso molecular:397.7MJN110
CAS:MJN110 (Cravatt Reagent) is a potent and selective MAGL inhibitor. MJN110 Produces Opioid-Sparing Effects in a Mouse Neuropathic Pain Model.Fórmula:C22H21Cl2N3O4Pureza:99.406%Forma y color:SolidPeso molecular:462.33DCBA
CAS:DCBA, an endogenous metabolite of the insect repellent N-N-diethyl-meta-toluamide (DEET), is utilized to evaluate DEET exposure through its concentration levelsFórmula:C12H15NO3Pureza:98.95%Forma y color:SolidPeso molecular:221.25Eliglustat
CAS:Eliglustat (Genz 99067) is an oral inhibitor of glucosylceramide synthase which is used in the therapy of type 1 Gaucher disease.Fórmula:C23H36N2O4Pureza:99% - 99.70%Forma y color:SolidPeso molecular:404.54Ref: TM-T3663
1mg54,00€2mg71,00€1mL*10mM (DMSO)88,00€5mg89,00€10mg117,00€25mg173,00€50mg226,00€100mg421,00€500mg945,00€RMC-4550
CAS:RMC-4550 is an effective and allosteric inhibitor of SHP2 (IC50: 0.583 nM).Fórmula:C21H26Cl2N4O2Pureza:98.95% - 99.65%Forma y color:SolidPeso molecular:437.36Ref: TM-T16762
1mg58,00€5mg113,00€1mL*10mM (DMSO)124,00€10mg178,00€25mg409,00€50mg605,00€100mg860,00€ATP disodium salt hydrate
CAS:ATP disodium salt hydrate (Adenosine disodium triphosphate) is a nucleoside triphosphate used in cells as a coenzyme.Fórmula:C10H16N5Na2O14P3Pureza:98.79% - >99.99%Forma y color:SolidPeso molecular:569.163-Methylglutaric acid
CAS:Methylglutaric acid, a leucine byproduct, is linked to two metabolic disorders, detected in patient urine.Fórmula:C6H10O4Pureza:98.64%Forma y color:SolidPeso molecular:146.14CAY10650
CAS:CAY10650 is an effective inhibitor of cytosolic phospholipase A2α (cPLA2α, IC50: 12 nM).Fórmula:C28H25NO6Pureza:97.33%Forma y color:SolidPeso molecular:471.5Ref: TM-TQ0105
1mg49,00€5mg114,00€1mL*10mM (DMSO)118,00€10mg172,00€25mg334,00€50mg467,00€100mg620,00€Enterostatin, human, mouse, rat acetate
Enterostatin, human, mouse, rat acetate is a pentapeptide mainly formed in the intestine by the cleavage of secreted pancreatic procolipase.Fórmula:C23H40N8O8Pureza:99.91%Forma y color:SolidPeso molecular:556.61LW6
CAS:LW6 (HIF-1α inhibitor) is a novel HIF-1 inhibitor.Fórmula:C26H29NO5Pureza:98.1% - 98.22%Forma y color:SolidPeso molecular:435.51Ref: TM-T3494
2mg44,00€5mg65,00€1mL*10mM (DMSO)65,00€10mg94,00€25mg173,00€50mg281,00€100mg424,00€500mg888,00€Glutamyl-glutamic acid
CAS:Glutamyl-glutamic acid (Glu-glu) is an Interpeptide Bridge in the Murein of Some Micrococci and Arthrobacter sp..Fórmula:C10H16N2O7Pureza:≥98%Forma y color:SolidPeso molecular:276.24
