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Metabolismo

Metabolismo

Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.

Subcategorías de "Metabolismo"

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Se han encontrado 8626 productos de "Metabolismo"

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  • PD0176078

    CAS:
    PD0176078 () is a newly blocker of N-type Calcium channel.
    Fórmula:C23H30F2N2O
    Pureza:99.72%
    Forma y color:Solid
    Peso molecular:388.49
  • RYL-552

    CAS:
    <p>RYL-552 is a potent inhibitor of PfNDH2.</p>
    Fórmula:C24H17F4NO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:427.39
  • YZ9

    CAS:
    <p>Y29 is a potent PFKFB3 inhibitor with an IC50 of 0.183 µM, and acts as a competitive inhibitor against Fru-6-P with a Ki of 0.094 µM[1].</p>
    Fórmula:C12H10O5
    Pureza:99.59%
    Forma y color:Solid
    Peso molecular:234.2
  • KB 5666

    CAS:
    <p>KB 5666, a quinazoline derivative, is a lipid peroxidation inhibitor. It protects the brain from both cellular and functional consequences of ischemia.</p>
    Fórmula:C24H32N4O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:456.54
  • PF04471141 HCl

    CAS:
    <p>PF-04471141 is an effective and selective inhibitor of the calcium-activated phosphodiesterase PDE1 (IC50 = 35 nM).</p>
    Fórmula:C16H24ClN3O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:341.83
  • Afegostat HCl

    CAS:
    <p>Afegostat: GCase inhibitor, Ki ~30 nM for wild-type/mutant, experimental Gaucher's disease drug.</p>
    Fórmula:C6H14ClNO3
    Forma y color:Solid
    Peso molecular:183.63
  • BRD6897

    CAS:
    BRD6897 is a mitochondrial content inducer that increases the cellular content of mitochondria.
    Fórmula:C25H21N3O2S2
    Pureza:97.74%
    Forma y color:Solid
    Peso molecular:459.58
  • Liarozole HCl

    CAS:
    <p>Liarozole HCl: antineoplastic, boosts ATRA levels, impedes cell growth, promotes differentiation, aromatase inhibitor.</p>
    Fórmula:C17H14Cl2N4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:345.23
  • Risarestat

    CAS:
    <p>Risarestat (CT-112) is a potent aldose reductase inhibitor and thyroid hormone receptor (TR) antagonist for the treatment of hypoglycemia.</p>
    Fórmula:C16H21NO4S
    Pureza:98.39%
    Forma y color:Solid
    Peso molecular:323.41
  • Rentiapril racemate

    CAS:
    <p>Rentiapril racemate (SA-446 racemate) is the racemate of Rentiapril.Rentiapril racemate has anti-inflammatory activity and may be used in glaucoma research.</p>
    Fórmula:C13H15NO4S2
    Pureza:98.96% - >99.99%
    Forma y color:Solid
    Peso molecular:313.39
  • Umbralisib sulfate

    CAS:
    <p>Umbralisib sulfate, an oral dual PI3Kδ/CK1ε inhibitor (EC50: 22.2 nM/6.0 μM), targets CLL T cells for blood cancer research.</p>
    Fórmula:C31H26F3N5O7S
    Forma y color:Solid
    Peso molecular:669.63
  • CP-319340(free base)

    CAS:
    <p>CP-319340 free base is a inhibitor of microsomal triglyceride transfer protein (MTP) .</p>
    Fórmula:C27H23F3N4O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:476.49
  • SYN20028567

    CAS:
    <p>SYN20028567, an aromatase (CYP19) inhibitor, exhibits an IC50 value of 9.4 nM. It has potential applications in breast cancer research [1].</p>
    Fórmula:C20H29N3O3S
    Forma y color:Solid
    Peso molecular:391.53
  • PKM2 activator 5

    CAS:
    <p>PKM2 activator 5 is a novel and potent PKM2 activator (AC50: 0.316 µM) with potential anticancer activity for the study of cancer metabolism-related diseases.</p>
    Fórmula:C18H19FN2O6S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:442.48
  • UCK2 Inhibitor-2

    CAS:
    <p>UCK2 Inhibitor-2 is a non-competitive inhibitor of uridine-cytidine kinase 2 (UCK2) with IC50=3.8 µM that inhibits UCK2-mediated nucleoside recycling in cells.</p>
    Fórmula:C28H23N3O4S
    Pureza:98.76% - 99.25%
    Forma y color:Solid
    Peso molecular:497.57
  • 4&prime;-Deoxyphlorizin

    CAS:
    <p>4'-Deoxyphlorizin inhibits glucose transport; Km 0.59 nM, Ki 0.33 nM for phlorizin hydrolase.</p>
    Fórmula:C21H24O9
    Forma y color:Solid
    Peso molecular:420.41
  • mEH-IN-1

    CAS:
    <p>mEH-IN-1 (Compound 62) is a potent mEH enzyme inhibitor with an IC50 of 2.2 nM, relevant in preeclampsia, hypercholanemia, and cancer research.</p>
    Fórmula:C16H17F6NOS
    Forma y color:Solid
    Peso molecular:385.37
  • MDK-0738

    CAS:
    <p>MDK-0738 is a potent and selective aldo-keto reductase 1C3 inhibitor.</p>
    Fórmula:C15H16O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:244.29
  • Glutathione sulfonate

    CAS:
    Glutathione sulfonate, a PAO-derived hydrophilic compound, inhibits angiogenesis and tumor growth.
    Fórmula:C10H17N3O9S2
    Forma y color:Solid
    Peso molecular:387.39
  • Antitumor agent-88

    CAS:
    <p>Antitumor agent-88, a potent antimitotic, arrests G2/M phase, disrupts microtubules in breast cancer, and inhibits CYP1A1 (Ki: 1.4 μM).</p>
    Fórmula:C23H30N2O7S
    Forma y color:Solid
    Peso molecular:478.56