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Metabolismo

Metabolismo

Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.

Subcategorías de "Metabolismo"

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Se han encontrado 8595 productos de "Metabolismo"

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  • C16 1-Deoxyceramide (m18:1/16:0)

    CAS:
    <p>C16 1-Deoxyceramide (m18:1/16:0) is a lipid molecule that can be used in life science related research. The CAS number of C16 1-Deoxyceramide (m18:1/16:0) is 1246298-56-5.</p>
    Fórmula:C34H67NO2
    Forma y color:Solid
    Peso molecular:521.9
  • GSK356278

    CAS:
    <p>GSK356278: selective PDE4A/B/D inhibitor, pIC50~8.7, anti-inflammatory, anxiolytic, cognition-enhancing.</p>
    Fórmula:C21H25N7O2S
    Pureza:99.90% - 99.97%
    Forma y color:Solid
    Peso molecular:439.53
  • 4′-DTMP

    CAS:
    <p>4′-DTMP (4-Demethyltrimethoprim) is a DHFR inhibitor with antimicrobial activity against Escherichia coli.</p>
    Fórmula:C13H16N4O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:276.29
  • ICMT-IN-36

    CAS:
    <p>ICMT-IN-36 (compound 40) serves as an ICMT inhibitor, with an IC50 value of 0.181 μM [1].</p>
    Fórmula:C21H25Cl2NO
    Forma y color:Solid
    Peso molecular:378.34
  • Cis-22a

    CAS:
    <p>Cis-22a: selective TRPV6 inhibitor (IC50=0.32μM), halts T47D breast cancer cell growth.</p>
    Fórmula:C24H30F3N3O2
    Pureza:99.07%
    Forma y color:Solid
    Peso molecular:449.51
  • Ecopladib

    CAS:
    <p>Ecopladib inhibits cPLA2α with IC50 of 0.15 μM (micelles) &amp; 0.11 μM (rat blood).</p>
    Fórmula:C39H33Cl3N2O5S
    Pureza:95.15%
    Forma y color:Solid
    Peso molecular:748.11
  • Fluspirilene

    CAS:
    <p>Fluspirilene is a long-acting antipsychotic for schizophrenia, inhibiting L-type calcium channels (IC50: 0.03 μM).</p>
    Fórmula:C29H31F2N3O
    Pureza:99.59%
    Forma y color:Solid
    Peso molecular:475.57
  • Varespladib methyl

    CAS:
    <p>Varespladib methyl (LY333013), a bioavailable prodrug of Varespladib, is a selective group II secretory phospholipase A2 inhibitor.</p>
    Fórmula:C22H22N2O5
    Pureza:99.42% - 99.97%
    Forma y color:Solid
    Peso molecular:394.42
  • PXS-6302 hydrochloride

    CAS:
    <p>PXS-6302 hydrochloride is a potent irreversible lysine oxidase (LOX) inhibitor, inhibiting Bovine LOX, rh LOXL1, rh LOXL2, rh LOXL3, and rh LOXL4 with IC50 of 3</p>
    Fórmula:C10H11ClF3NO2S
    Pureza:99.89%
    Forma y color:Soild
    Peso molecular:301.71
  • PDE9-IN-(S)-C33

    CAS:
    <p>PDE9-IN-(S)-C33: potent PDE9 inhibitor with 11 nM IC50, for CNS diseases and diabetes study.</p>
    Fórmula:C18H20ClN5O
    Pureza:98.75%
    Forma y color:Solid
    Peso molecular:357.84
  • Inolitazone

    CAS:
    <p>Inolitazone (RS5444) a high-affinity PPARγ agonist. Inolitazone exhibits IC50 for growth inhibition is ~0.8 nM in vitro.</p>
    Fórmula:C27H26N4O4S
    Pureza:99.41% - 99.53%
    Forma y color:Solid
    Peso molecular:502.58
  • Enpp-1-IN-16

    CAS:
    <p>Enpp-1-IN-16 is an ENPP1 inhibitor, yo anti-cancer activity.Enpp-1-IN-16 can be used to study insulin resistance and chondrocalcinosis.</p>
    Fórmula:C23H32N4O4
    Pureza:99.87%
    Forma y color:Solid
    Peso molecular:428.52
  • OGT 2115

    CAS:
    <p>OGT 2115 blocks heparanase (IC50=0.4µM), cleaving heparan sulfate; antiangiogenic (IC50=1µM).</p>
    Fórmula:C24H16BrFN2O4
    Pureza:97.17%
    Forma y color:Solid
    Peso molecular:495.3
  • TP-10

    CAS:
    <p>TP-10 is a selective inhibitor of PDE10A against other PDEs with IC50 of 0.8 nM.</p>
    Fórmula:C26H19F3N4O
    Pureza:99.21%
    Forma y color:Solid
    Peso molecular:460.45
  • Rilapladib

    CAS:
    <p>Rilapladib (SB 659032) is a selective inhibitor of Lipoprotein-Associated Phospholipase A2(Lp-PLA2, IC50 = 230 pM) and an antagonist of the platelet activating</p>
    Fórmula:C40H38F5N3O3S
    Pureza:99.92%
    Forma y color:Solid
    Peso molecular:735.8
  • NEP-IN-1

    CAS:
    <p>NEP-IN-1 is an inhibitor of neutral endopeptidase (NEP, IC50 = 2 nM) and can be used in studies about female sexual arousal disorders.</p>
    Fórmula:C21H30ClNO4
    Pureza:99.69%
    Forma y color:Solid
    Peso molecular:395.92
  • BI-3231

    CAS:
    <p>BI-3231 is a hydroxysteroid 17ß-dehydrogenase 13 HSD17B13 inhibitor that inhibits hHSD17B13 .BI-3231 can be used to study cirrhosis.</p>
    Fórmula:C16H14F2N4O3S
    Pureza:98.2%
    Forma y color:Solid
    Peso molecular:380.37
  • WAY-620147

    CAS:
    <p>WAY-620147 inhibits Monoamine Oxidase and can be used for the study of neurological disorders.</p>
    Fórmula:C12H16BrN3O2
    Pureza:99.55%
    Forma y color:Solid
    Peso molecular:314.18
  • Calcium channel-modulator-1

    CAS:
    <p>Calcium channel-modulator-1 is a calcium channel-modulator (IC50:0.8 μM) with specialisation to block aortic constriction.</p>
    Fórmula:C26H24Cl2N2O7S
    Pureza:99.95%
    Forma y color:Solid
    Peso molecular:579.45
  • AMG 579

    CAS:
    <p>AMG 579 is an efficacious and selective inhibitor of PDE10A (IC50 = 0.1 nM).</p>
    Fórmula:C25H23N5O3
    Pureza:99.87%
    Forma y color:Solid
    Peso molecular:441.48