
Metabolismo
Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.
Subcategorías de "Metabolismo"
- AhR(42 productos)
- Aminopeptidasa(76 productos)
- CETP(20 productos)
- Anhídrido carbónico(196 productos)
- Caseína quinasa(138 productos)
- DHFR(32 productos)
- Descarboxilasa(4 productos)
- Deshidrogenasa(302 productos)
- FAAH(64 productos)
- FXR(62 productos)
- Factor Xa(85 productos)
- Ácido graso sintasa(37 productos)
- Ferroptosis(226 productos)
- GR(3 productos)
- GSNOR(3 productos)
- Glucoquinasa(57 productos)
- HIF / HIF Prolilhidroxilasa(146 productos)
- HMG-CoA reductasa(34 productos)
- Hidroxilasa(36 productos)
- IDO(84 productos)
- LDL(7 productos)
- Lipasa(107 productos)
- Lípido(61 productos)
- Lipoxigenasa(134 productos)
- MAO(87 productos)
- MPO(2 productos)
- NAMPT(40 productos)
- P450(6 productos)
- PAI-1(26 productos)
- PDE(169 productos)
- PED(1 productos)
- PKM(17 productos)
- PPAR(170 productos)
- Fosfolipasa(86 productos)
- ROR(47 productos)
- Receptor de retinoides(22 productos)
- SGK(10 productos)
- Tiorredoxina(12 productos)
- Transferasa(29 productos)
- Transportador(45 productos)
- UGT(4 productos)
- Inhibidores de la xantina oxidasa (XO)(9 productos)
Mostrar 34 subcategorías más
Se han encontrado 9185 productos de "Metabolismo"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
1,2-Dioctanoyl-sn-glycerol
CAS:ZKN14489, also known as 08:0 DG and 1,2-dioctanoyl-sn-glycerol, is a short-chain, cell-permeable diacylglycerol that serves as a lipid cofactor for activating protein kinase C.Fórmula:C19H36O5Forma y color:SolidPeso molecular:344.492ICMT-IN-27
CAS:ICMT-IN-27, also known as compound 64, is an inhibitor of the enzyme ICMT, demonstrating potent activity with an IC50 value of 0.1 µM [1].Fórmula:C22H28FNO2Forma y color:SolidPeso molecular:357.46Cintirorgon sodium
CAS:Cintirorgon (LYC-55716) is an oral RORgamma agonist with immunomodulatory and anticancer effects.Fórmula:C27H23F6NNaO6SPureza:98%Forma y color:SolidPeso molecular:626.52BMS-795311
CAS:Potent CETP inhibitor, boosts HDL-C levels, orally active; IC50=4nM.Fórmula:C33H23F10NO3Forma y color:SolidPeso molecular:671.52Cav 3.2 inhibitor 4
CAS:Cav 3.2 Inhibitor 4 (Compound 21) is a selective and potent inhibitor of the T-type calcium channel (Ca v 3.2), demonstrating peripheral restriction with an
Fórmula:C21H32Cl2N4O3Pureza:98%Forma y color:SolidPeso molecular:459.4119(R)-hydroxy Prostaglandin F2α
CAS:19(R)-hydroxy PGF2α, an ω-1 hydroxylase metabolite of PGF2α present in human semen, exhibits a concentration of approximately 20 µg/ml for both 19(R)-hydroxy PG compounds (F2α and F1α) in fresh samples. This compound demonstrates no activity at the FP receptor of the cat iris sphincter muscle at concentrations up to 1 µM.Fórmula:C20H34O6Forma y color:SolidPeso molecular:370.51-Palmitoyl-2-Arachidoyl-3-Oleoyl-rac-glycerol
CAS:1-Palmitoyl-2-arachidoyl-3-oleoyl-rac-glycerol, a triacylglycerol, incorporates palmitic acid, arachidic acid, and oleic acid at the sn-1, sn-2, and sn-3 positions, respectively, and is identified in cod liver oil.Fórmula:C57H108O6Forma y color:SolidPeso molecular:889.46hCAIX/XII-IN-8
CAS:hCAIX/XII-IN-8 (compound 3g) is a potent inhibitor of the human carbonic anhydrases (CAs) IX and XII, with inhibition constants (K i) of 8.5 nM for CA IX and 6.Fórmula:C16H13Cl2N5O3SPureza:98%Forma y color:SolidPeso molecular:426.28Ionizable lipid-2
CAS:Ionizable Lipid-2 (Compound 1) serves as an ionizable lipid, essential for nucleic acid delivery and the construction of lipid nanoparticles (LNPs) [1].Fórmula:C50H99NO7Forma y color:SolidPeso molecular:826.32Autotaxin-IN-4
CAS:Autotaxin-IN-4 is an Autotaxin inhibitor. It has the potential to treat idiopathic pulmonary fibrosis.Fórmula:C22H21N9O2Pureza:98%Forma y color:SolidPeso molecular:443.46Pentadecanoyl ethanolamide
CAS:Pentadecanoyl ethanolamide, a derivative of the endogenous lipid amides (N-acylethanolamines), demonstrates anticonvulsant efficacy in electroshock-induced seizures in mice, exhibiting minimal toxicity [1].Fórmula:C17H35NO2Forma y color:SolidPeso molecular:285.472α-Glucosidase-IN-28
CAS:α-Glucosidase-IN-28 (Compound 18) is an α-glucosidase inhibitor with an IC50 of 0.62 μM and Ki value of 3.93 μM.Fórmula:C29H22Br2O7Pureza:98%Forma y color:SolidPeso molecular:642.29AZD1092
CAS:AZD1092 is the glucokinase enzyme activator.Fórmula:C24H26N4O5Pureza:98%Forma y color:SolidPeso molecular:450.49hCAIX-IN-15
CAS:hCAIX-IN-15 is a potent inhibitor of human carbonic anhydrase IX (hCA IX) with an inhibition constant (Ki) of 38.8 nM, exhibiting broad-spectrum anticancerFórmula:C18H14FN7O2SPureza:98%Forma y color:SolidPeso molecular:411.411,2-Dimyristoyl-sn-glycero-3-PA sodium
CAS:DMPA, a derivative of phosphatidic acid (PA), constitutes a significant component of cellular membranes.Fórmula:C31H59Na2O8PForma y color:SolidPeso molecular:636.7585(S)-HETrE
CAS:5(S)-HETrE, made by 5-LO from mead acid, has unknown biological activity and metabolic fate.Fórmula:C20H34O3Forma y color:SolidPeso molecular:322.48TAS2R14 agonist-1
CAS:TAS2R14 agonist is a potent partial agonist of TAS2R14, displaying an EC50 value of 116.6 ± 23.6 nM [1].Fórmula:C15H9F6N5Forma y color:SolidPeso molecular:373.26TMP778
CAS:TMP778 is an effective and selective RORγt inverse agonist (IC50: 7 nM in FRET assay).Fórmula:C31H30N2O4Pureza:98%Forma y color:SolidPeso molecular:494.589(E),11(E)-9-nitro Conjugated Linoleic Acid
CAS:9(E),11(E)-9-nitro Conjugated Linoleic Acid (9E,11E-9-nitro CLA) is a nitrated fatty acid produced from 9Z,11E-CLA through exposure to acidified nitrite, peroxynitrite, gaseous nitrogen dioxide, or the combined action of myeloperoxidase, hydrogen peroxide, and nitrite. Additionally, it forms in LPS-stimulated RAW 264.7 macrophages, a process that can be inhibited by the nitric oxide synthase (NOS) inhibitor L-NAME. This compound has also been detected in human plasma.Fórmula:C18H31NO4Forma y color:SolidPeso molecular:325.443'-hydroxy Lidocaine
CAS:3'-Hydroxy Lidocaine, an active metabolite of Lidocaine, is produced through the metabolism by the cytochrome P450 (CYP) isoforms CYP1A2 and CYP3A4.Fórmula:C14H22N2O2Forma y color:SolidPeso molecular:250.342

