
Metabolismo
Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.
Subcategorías de "Metabolismo"
- AhR(42 productos)
- Aminopeptidasa(76 productos)
- CETP(20 productos)
- Anhídrido carbónico(197 productos)
- Caseína quinasa(137 productos)
- DHFR(34 productos)
- Descarboxilasa(4 productos)
- Deshidrogenasa(303 productos)
- FAAH(66 productos)
- FXR(62 productos)
- Factor Xa(87 productos)
- Ácido graso sintasa(37 productos)
- Ferroptosis(226 productos)
- GR(3 productos)
- GSNOR(4 productos)
- Glucoquinasa(57 productos)
- HIF / HIF Prolilhidroxilasa(146 productos)
- HMG-CoA reductasa(33 productos)
- Hidroxilasa(35 productos)
- IDO(84 productos)
- LDL(8 productos)
- Lipasa(107 productos)
- Lípido(61 productos)
- Lipoxigenasa(134 productos)
- MAO(87 productos)
- MPO(2 productos)
- NAMPT(40 productos)
- P450(6 productos)
- PAI-1(26 productos)
- PDE(167 productos)
- PED(1 productos)
- PKM(17 productos)
- PPAR(169 productos)
- Fosfolipasa(83 productos)
- ROR(47 productos)
- Receptor de retinoides(28 productos)
- SGK(11 productos)
- Tiorredoxina(12 productos)
- Transferasa(29 productos)
- Transportador(46 productos)
- UGT(4 productos)
- Inhibidores de la xantina oxidasa (XO)(9 productos)
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Se han encontrado 9282 productos de "Metabolismo"
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h15-LOX-2 inhibitor 3
CAS:Compound 13, identified as h15-LOX-2 inhibitor 3, exhibits inhibitory activity against h15-LOX, with IC50 and Ki values of 25 μM and 15.1 μM, respectively.Fórmula:C22H13N5O3Forma y color:SolidPeso molecular:395.37CHI3L1-IN-2
CAS:CHI3L1-IN-2 (Compound 36), a potent inhibitor of CHI3L1 (YKL-40), effectively blocks the interaction between CHI3L1 and heparan sulfate (CHI3L1:HSIII), demonstrating an IC 50 of 26 nM [1].Fórmula:C26H37ClN4Peso molecular:441.05ent-8-iso-15(S)-Prostaglandin F2α
CAS:Isoprostanes are produced by the non-enzymatic, free radical peroxidation of phospholipid-esterified arachidonic acid.Fórmula:C20H34O5Forma y color:SolidPeso molecular:354.48Carbonic anhydrase inhibitor 2
CAS:Compound 7c inhibits carbonic anhydrase II, lowering intraocular pressure in glaucomatous rabbits.Fórmula:C12H16N4O6SForma y color:SolidPeso molecular:344.34NPD10084
CAS:NPD10084 is an inhibitor of pyruvate kinase PKM2 that blocks non-glycolytic signaling in cancer cells by disrupting PKM2's interaction with β-catenin or STAT3, thus inhibiting downstream pathways. It demonstrates antiproliferative effects against colorectal cancer cells both in vitro and in vivo [1].Fórmula:C21H19N3O2Peso molecular:345.39trans-Doxercalciferol
CAS:trans-Doxercalciferol is an isomer of Doxercalciferol. Doxercalciferol is an activator of the Vitamin D receptor and prevents renal disease.Fórmula:C28H44O2Pureza:98%Forma y color:SolidPeso molecular:412.65AV-5080
CAS:AV-5080 is an orally active neuraminidase (neuraminidase) inhibitor that is utilized in the research of both Type A and Type B influenza viruses.Fórmula:C15H25FN4O4Forma y color:SolidPeso molecular:344.38Glycerophosphoglycerol
CAS:Glycerophosphoglycerol is a precursor in phospholipid synthesis. By enhancing phospholipid formation, it aids in the reconstruction and proliferation of membrane structures in tumor cells. Glycerophosphoglycerol holds promise for research in breast cancer cells.Fórmula:C6H15O8PForma y color:SolidPeso molecular:246.15AD015
CAS:AD015 is a dual inhibitor of angiotensin-converting enzyme (ACE) and neprilysin (NEP), effectively inhibiting NEP, nACE, and cACE with IC50 values of 0.009, 0.019, and 0.0008 μM, respectively.Fórmula:C23H26N2O4SForma y color:SolidPeso molecular:426.534-(4-Bromophenyl)-4-hydroxypiperidine
CAS:<p>4-(4-Bromophenyl)-4-hydroxypiperidine (BPHP) is a metabolite of Bromperidol (BRO), produced through the N-dealkylation of BRO.</p>Fórmula:C11H14BrNOForma y color:SolidPeso molecular:256.139DSM705 hydrochloride
DSM705 hydrochloride: potent antimalarial, pyrrole-based DHODH inhibitor effective against Plasmodium, non-toxic to mammalian DHODH.Fórmula:C19H20ClF3N6OForma y color:SolidPeso molecular:440.85BLT-4
CAS:BLT-4 is a specific and reversible inhibitor of scavenger receptor class B type I (SR-BI). It effectively blocks the SR-BI-mediated transfer of lipids between high-density lipoprotein (HDL) and cells.Fórmula:C18H16N2O2Forma y color:SolidPeso molecular:292.332Casein kinase 1δ-IN-26
CAS:<p>Casein kinase1δ-IN-26 (compound 505) is a potent inhibitor of casein kinase 1δ. This compound is applicable in research related to neurodegenerative disorders such as Alzheimer’s disease.</p>Fórmula:C16H13N3O4SForma y color:SolidPeso molecular:343.357CYP2C1/CYP2C19-IN-2
CYP2C1/CYP2C19-IN-2 is a potent inhibitor of CYP2C9/CYP2C19 without liver toxicity or genotoxicity and can be used to study Zika virus (ZIKV) infection.Fórmula:C27H28N2O6SForma y color:SolidPeso molecular:508.59JTZ-951 HCl
CAS:JTZ-951 is a potent and orally active inhibitor of hypoxia inducible factor prolyl hydroxylase (PHD).Fórmula:C17H17ClN4O4Pureza:98%Forma y color:SolidPeso molecular:376.79Glucokinase activator 7
CAS:Glucokinase activator7 is an activator of glucose kinase (Glucokinase) and can be utilized in research on diabetes and hyperglycemia [refer to compound on page 176].Fórmula:C14H13N3O2SForma y color:SolidPeso molecular:287.337AChE/PDE4-IN-1
AChE/PDE4-IN-1, compound 12c, dual inhibitor; IC50: 0.28μM for AChE, 1.88μM for PDE4D, may reduce Alzheimer's neuroinflammation.Fórmula:C23H28N2O3Forma y color:SolidPeso molecular:380.48FAAH/MAGL-IN-3
FAAH/MAGL-IN-3 irreversibly inhibits FAAH (IC50: 179 nM) & MAGL (IC50: 759 nM) with low PAMPA permeability.Fórmula:C21H25N3O6SForma y color:SolidPeso molecular:447.5BRD2879
CAS:BRD2879 is a potent and cell-active inhibitor of IDH1-R132H (IC50 = 50 nM).Fórmula:C30H38FN3O5SPureza:98%Forma y color:SolidPeso molecular:571.70HIF-2α-IN-5
CAS:HIF-2α-IN-5 is a potent HIF-2α inhibitor with an IC 50 of < 50 nM [1].Fórmula:C15H12F4O3S2Forma y color:SolidPeso molecular:380.38

