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Neurociencia

Neurociencia

Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.

Subcategorías de "Neurociencia"

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Se han encontrado 5398 productos de "Neurociencia"

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  • SEP-363856

    CAS:
    <p>SEP-363856, a non-D2/5-HT2A, orally active CNS psychotropic may treat schizophrenia.</p>
    Fórmula:C9H13NOS
    Pureza:98%
    Forma y color:Solid
    Peso molecular:183.27
  • Echothiophate Iodide

    CAS:
    <p>Echothiophate iodide is an effective long-acting cholinesterase inhibitor for the treatment of glaucoma.</p>
    Fórmula:C9H23INO3PS
    Forma y color:Solid
    Peso molecular:383.23
  • hMAO-B-IN-3

    CAS:
    <p>hMAO-B-IN-3: potent hMAO-B inhibitor, IC50 of 47.4 nM, good drug properties, safe, ideal for lead optimization.</p>
    Fórmula:C20H15NO4
    Forma y color:Solid
    Peso molecular:333.34
  • DR4485 hydrochloride

    CAS:
    <p>5-HT7 antagonist</p>
    Fórmula:C26H29Cl3N2O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:491.88
  • 3-Methyl-GABA

    CAS:
    <p>3-Methyl-GABA activates GABA aminotransferase, fits GABAaR, stimulates GAD, and acts as an anticonvulsant.</p>
    Fórmula:C20H30N2O10S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:522.59
  • CP-601932

    CAS:
    <p>CP-601932 (free base) is a selective base α( 4) β( 2) Nicotinic acetylcholine receptor agonist.</p>
    Fórmula:C12H12F3N
    Forma y color:Solid
    Peso molecular:227.23
  • YIAD-0205

    CAS:
    <p>YIAD-0205, an orally administered inhibitor of Aβ(1-42) aggregation, has exhibited in vivo efficacy in a 5XFAD transgenic mouse model that harbors five familial</p>
    Fórmula:C26H16Br2ClN3
    Forma y color:Solid
    Peso molecular:565.69
  • LY320135

    CAS:
    <p>CB1 receptor antagonist/inverse agonist</p>
    Fórmula:C24H17NO4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:383.4
  • NFPS

    CAS:
    <p>NFPS exerts neuroprotection via glyR alpha1 subunit in the rat model of transient focal cerebral ischaemia and reperfusion.</p>
    Fórmula:C24H24FNO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:393.45
  • Alaproclate hydrochloride, (S)-

    CAS:
    <p>Alaproclate hydrochloride, (S)- is a selective inhibitor of serotonin reuptake.</p>
    Fórmula:C13H19Cl2NO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:292.2
  • JNJ-46356479

    CAS:
    <p>JNJ-46356479: Selective, oral mGlu2 receptor PAM, EC50=78 nM, Emax=256%.</p>
    Fórmula:C22H22F5N5
    Forma y color:Solid
    Peso molecular:451.44
  • AZD 9272

    CAS:
    <p>AZD 9272 is a brain-permeable mGluR5 antagonist for the study of gastroesophageal reflux.</p>
    Fórmula:C14H6F2N4O
    Pureza:98.29%
    Forma y color:Solid
    Peso molecular:284.22
  • Alpidem

    CAS:
    <p>Alpidem (Ananxyl), a non-sedative imidazopyridine anxiolytic, treats anxiety with high benzodiazepine receptor affinity.</p>
    Fórmula:C21H23Cl2N3O
    Pureza:99.56% - 99.97%
    Forma y color:White To Off-White Solid
    Peso molecular:404.33
  • TAK-137

    CAS:
    <p>TAK-137 is an AMPA receptor enhancer with antidepressant effects. TAK-137 has the ability to improve cognition and could be used to study schizophrenia.</p>
    Fórmula:C19H16N2O3S
    Pureza:99.18%
    Forma y color:Solid
    Peso molecular:352.41
  • Faxeladol

    CAS:
    <p>Faxeladol: adrenergic, serotonin inhibitor &amp; opioid agonist for neurological studies.</p>
    Fórmula:C15H23NO
    Pureza:98.09% - 98.77%
    Forma y color:Solid
    Peso molecular:233.35
  • Litoxetine

    CAS:
    <p>Litoxetine: a selective 5-HT inhibitor &amp; 5-HT3 antagonist, used as an antidepressant with antiemetic effects, Ki=85 nM.</p>
    Fórmula:C16H19NO
    Pureza:99.47%
    Forma y color:Solid
    Peso molecular:241.33
  • Selurampanel

    CAS:
    <p>Selurampanel (BGG492), an oral AMPA antagonist for epilepsy, migraine, and tinnitus studies.</p>
    Fórmula:C16H19N5O4S
    Pureza:99.60% - 99.78%
    Forma y color:Solid
    Peso molecular:377.42
  • Teniloxazine

    CAS:
    <p>Teniloxazine is an orally available antidepressant compound with anti-hypoxic properties.</p>
    Fórmula:C16H19NO2S
    Pureza:99.23%
    Forma y color:Solid
    Peso molecular:289.39
  • Fananserin

    CAS:
    <p>Fananserin: Oral 5-HT2A antagonist (Ki=0.37 nM, rat), blocks human D4 receptor (Ki=2.93 nM).</p>
    Fórmula:C23H24FN3O2S
    Pureza:99.88%
    Forma y color:Solid
    Peso molecular:425.52
  • CT-179

    CAS:
    <p>CT-179 is a potent and selective inhibitor of OLIG2, reduces tumor cell proliferation and induces apoptosis, fpr medulloblastoma and glioblastoma.</p>
    Fórmula:C17H22Cl2N6O
    Pureza:98.67%
    Forma y color:Solid
    Peso molecular:397.3
  • RS 67333 hydrochloride

    CAS:
    <p>RS 67333 hydrochloride is a selective 5-HT4R partial agonist (pKi=8.7) with neuroprotective properties for Alzheimer's research.</p>
    Fórmula:C19H30Cl2N2O2
    Pureza:98.78%
    Forma y color:Solid
    Peso molecular:389.36
  • Masupirdine free base

    CAS:
    <p>Masupirdine free base (SUVN-502 free base) is a 5-HT6 receptor antagonist that can be used to study neurological disorders like Alzheimer's disease.</p>
    Fórmula:C21H24BrN3O3S
    Pureza:98.36% - 99.65%
    Forma y color:Solid
    Peso molecular:478.4
  • SB-215505

    CAS:
    <p>SB215505: potent 5-HT2B/2C blocker, enhances rat wakefulness/motor activity. (pKi: 5-HT2B - 8.3, 5-HT2C - 7.66, 5-HT2A - 6.77).</p>
    Fórmula:C19H16ClN3O
    Pureza:98.33%
    Forma y color:Solid
    Peso molecular:337.8
  • Muscimol HBr

    CAS:
    <p>Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.</p>
    Fórmula:C4H7BrN2O2
    Pureza:98.13%
    Forma y color:Off-White Powder
    Peso molecular:195.01
  • (E/Z)-SIB-1893

    CAS:
    <p>(E/Z)-SIB-1893 (SIB 1893) is the racemate of (E)-SIB-1893 and (Z)-SIB-1893.</p>
    Fórmula:C14H13N
    Pureza:99.92%
    Forma y color:Solid
    Peso molecular:195.26
  • SPD-473 citrate

    CAS:
    <p>SPD-473 citrate is an inhibitior of serotonin/dopamine/norepinephrine reuptake.</p>
    Fórmula:C23H31Cl2NO8S
    Pureza:99.37%
    Forma y color:Solid
    Peso molecular:552.47
  • SCH-900271

    CAS:
    <p>SCH-900271 treats dyslipidemia by targeting nicotinic acid receptors, addressing hyperlipidaemia.</p>
    Fórmula:C14H16N2O4
    Pureza:98.82% - 99.93%
    Forma y color:Solid
    Peso molecular:276.29
  • ASM-024

    CAS:
    <p>ASM-024, a synthetic piperazine, activates nicotinic and β2-adrenergic receptors for potential asthma and bronchitis treatment with anti-inflammatory effects.</p>
    Fórmula:C15H25N2
    Pureza:99.74%
    Forma y color:Solid
    Peso molecular:233.37
  • Valiglurax

    CAS:
    <p>Valiglurax (VU2957), potent mGlu4 PAM, crosses blood-brain barrier, orally available; promising for Parkinson's treatment.</p>
    Fórmula:C16H10F3N5
    Pureza:98.29%
    Forma y color:Solid
    Peso molecular:329.28
  • Xanomeline oxalate

    CAS:
    <p>Xanomeline oxalate (LY246708), a potent SMRA, boosts phosphoinositide hydrolysis; key for Alzheimer's research.</p>
    Fórmula:C16H25N3O5S
    Pureza:99.1%
    Forma y color:Solid
    Peso molecular:371.45
  • Perphenazine dihydrochloride

    CAS:
    <p>Perphenazine dihydrochloride: Oral dopamine, histamine-1 antagonist; targets D2, D3, 5-HT2A, Alpha-1A; may treat psychiatric disorders, cancer.</p>
    Fórmula:C21H28Cl3N3OS
    Pureza:99.67%
    Forma y color:Solid
    Peso molecular:476.89
  • Panadiplon

    CAS:
    <p>Panadiplon (FG 10571) is a selective gamma-aminobutyric acid receptor agonist and partial agonist of 5GABAA, a benzodiazepine receptor, used in the treatment of</p>
    Fórmula:C18H17N5O2
    Pureza:98.30% - 98.94%
    Forma y color:Solid
    Peso molecular:335.36
  • Apyramide

    CAS:
    <p>Apyramide, an NSAID and prodrug of indomethacin, inhibits COX1/COX2 and permeates the blood-brain barrier.</p>
    Fórmula:C27H23ClN2O5
    Pureza:99.93%
    Forma y color:Solid
    Peso molecular:490.93
  • Piromelatine

    CAS:
    <p>Piromelatine is an agonist of melatonin MT1/MT2 receptors, 5-HT1A and 5-HT1D, and an antagonist of 5-HT2B.Piromelatine has antinociceptive activity with</p>
    Fórmula:C17H16N2O4
    Pureza:99.89%
    Forma y color:Solid
    Peso molecular:312.32
  • AMPA receptor antagonist-2

    CAS:
    <p>AMPA receptor antagonist-2 is an AMPA receptor antagonist.</p>
    Fórmula:C18H17N3O4
    Pureza:98.76%
    Forma y color:Solid
    Peso molecular:339.35
  • PF-03635659

    CAS:
    <p>PF-03635659: potent M3 antagonist, Ki=0.2 nM, long half-life, potential COPD treatment.</p>
    Fórmula:C28H32N2O3
    Pureza:98.39% - 99.83%
    Forma y color:Solid
    Peso molecular:444.57
  • MM 77 dihydrochloride

    CAS:
    <p>MM 77 dihydrochloride is an effecitve 5-HT1A receptor postsynaptic antagonist with anxiolytic-like activity.</p>
    Fórmula:C19H29Cl2N3O3
    Pureza:99.91%
    Forma y color:Solid
    Peso molecular:418.36
  • SB228357

    CAS:
    <p>SB228357 is a potent and selective antagonist of the 5-HT receptor with pKis of 6.9, 8.0, and 9.0 for 5-HT2A, 5-HT2B, and 5-HT2C, respectively.</p>
    Fórmula:C22H17F4N3O2
    Pureza:99.82%
    Forma y color:Solid
    Peso molecular:431.38
  • NNC 05-711

    CAS:
    <p>NNC 05-711 (NO-711 hydrochloride) is a potent and selective inhibitor of GAT-1 (GABA transporter 1), exerting anticonvulsant and analgesic effects.</p>
    Fórmula:C21H23ClN2O3
    Pureza:99.92%
    Forma y color:Solid
    Peso molecular:386.87
  • RS 42358-197

    CAS:
    <p>RS 42358-197 (RS 25259-007) is a competitive 5-HT3 receptor antagonist.</p>
    Fórmula:C19H23ClN2O
    Pureza:99.70%
    Forma y color:Solid
    Peso molecular:330.85
  • RWJ-51204

    CAS:
    <p>RWJ-51204: potent adenosine A2A blocker, GABA(A) partial agonist (IC50: 0.2-2 nM), neuroprotective, may treat Parkinson's.</p>
    Fórmula:C21H19F2N3O3
    Pureza:99.57% - 99.95%
    Forma y color:Solid
    Peso molecular:399.39
  • 5-HT6/7 antagonist 1

    CAS:
    <p>5-HT6/7 antagonist 1 is a dual 5-HT6/7/2A and D2 receptor antagonist for the study of dementia and Alzheimer's disease.</p>
    Fórmula:C22H20FN3O3
    Pureza:98.78% - 99.26%
    Forma y color:Solid
    Peso molecular:393.41
  • ALX-1393

    CAS:
    <p>ALX-1393 is a selective GlyT2 inhibitor that effectively reduces neuronal action potential activity in a concentration-dependent manner and inhibits the</p>
    Fórmula:C23H22FNO4
    Pureza:99.83%
    Forma y color:Solid
    Peso molecular:395.42
  • Gavestinel sodium

    CAS:
    <p>Gavestinel (GV 150526): potent, selective oral NMDA antagonist; binds glycine site, pKi 8.5; studied for acute ischemic stroke.</p>
    Fórmula:C18H11Cl2N2NaO3
    Pureza:99.04%
    Forma y color:Solid
    Peso molecular:397.19
  • 5-HT1A modulator 1

    CAS:
    <p>5-HT1A modulator 1 displays very high affinities for the 5-HT1A, α1-adrenergic receptor, and D2 receptor (IC50s = 2 nM, 10 nM, and 40 nM).</p>
    Fórmula:C21H25N3O2S
    Pureza:99.68%
    Forma y color:Solid
    Peso molecular:383.51
  • Lesopitron

    CAS:
    <p>Lesopitron: anxiolytic, 5-HT1A agonist, treats rodent anxiety, counters benzodiazepine withdrawal, low toxicity, no alcohol/barbiturate interaction.</p>
    Fórmula:C15H21ClN6
    Pureza:99.15% - 99.38%
    Forma y color:Solid
    Peso molecular:320.82
  • Cianopramine

    CAS:
    <p>Cianopramine (Ro 112465) is a selective 5-hydroxytryptamine uptake inhibitor and a tricyclic antidepressant used in the study of neurological disorders.</p>
    Fórmula:C20H23N3
    Pureza:99.92% - 99.92%
    Forma y color:Solid
    Peso molecular:305.42
  • Riluzole hydrochloride

    CAS:
    <p>Riluzole hydrochloride, an anticonvulsant Na+ channel blocker, inhibits GABA uptake (IC50: 43 µM).</p>
    Fórmula:C8H6ClF3N2OS
    Pureza:99.76%
    Forma y color:Solid
    Peso molecular:270.66
  • Lirequinil

    CAS:
    <p>Lirequinil (Ro 41-3696) is a small molecule GABAA receptor agonist used to study neurological disorders.</p>
    Fórmula:C26H25ClN2O3
    Pureza:98.54%
    Forma y color:Solid
    Peso molecular:448.94
  • Adoprazine

    CAS:
    <p>Adoprazine (SLV313) is a potential atypical antipsychotic bearing potent D2 receptor antagonist and 5-HT1A receptor agonist properties.</p>
    Fórmula:C24H24FN3O2
    Pureza:99.83%
    Forma y color:Solid
    Peso molecular:405.46
  • Ezeprogind disulfate

    CAS:
    <p>Ezeprogind disulfate: neurotrophic inducer targeting neurodegeneration causes like Abeta, tau; for neurological disorder research.</p>
    Fórmula:C25H48N6O8S2
    Pureza:99.72%
    Forma y color:Solid
    Peso molecular:624.81
  • Pimethixene maleate

    CAS:
    <p>Pimethixene maleate (Pimetixene maleate) is a 5-HT2B receptor antagonist with sedative activity that can be used to study dry cough in children.</p>
    Fórmula:C23H23NO4S
    Pureza:99.55%
    Forma y color:Solid
    Peso molecular:409.5
  • CP 96021

    CAS:
    <p>"CP 96021 is an antagonist of 5-HT1/2 receptors, with anti-inflammatory and anti-ulcer effects for treating GI tract and asthma."</p>
    Fórmula:C29H21FN4OS
    Pureza:97.81% - 99.62%
    Forma y color:Soild
    Peso molecular:492.57
  • L-838417

    CAS:
    <p>L-838417 is a GABAA receptor subtype-selective benzodiazepine site-selective ligand and GABAA receptor-positive modulator used in the study of anxiety disorders</p>
    Fórmula:C19H19F2N7O
    Pureza:98.12% - 99.70%
    Forma y color:Solid
    Peso molecular:399.4
  • 2-BFI hydrochloride

    CAS:
    <p>2-BFI hydrochloride: High-affinity I2 agonist; used in researching stroke and immune disease protection.</p>
    Fórmula:C11H11ClN2O
    Pureza:99.94%
    Forma y color:Solid
    Peso molecular:222.67
  • Repinotan

    CAS:
    <p>Repinotan (BAY x 3702 free base) is a 5-HT1A receptor agonist used in acute ischemic stroke studies.</p>
    Fórmula:C21H24N2O4S
    Pureza:99%
    Forma y color:Solid
    Peso molecular:400.49
  • NKY80

    CAS:
    <p>NKY80 regulates the adenylyl cyclase catalytic activity in heart and lung tissues.</p>
    Fórmula:C12H11N3O2
    Pureza:99.88%
    Forma y color:Solid
    Peso molecular:229.23
  • amyloid P-IN-1

    CAS:
    <p>amyloid P-IN-1 can be used in studies about diseases with depletion of serum amyloid P components such as Alzheimer's disease, amyloidosis, osteoarthritis, and</p>
    Fórmula:C30H44N2O14
    Pureza:99.76%
    Forma y color:Solid
    Peso molecular:656.68
  • BL-1020 Mesylate

    CAS:
    <p>BL-1020 Mesylate (CYP-1020 Mesylate) is a GABA A receptor agonist and D2 antagonist used in studies of neurodegeneration.</p>
    Fórmula:C28H45ClN4O11S4
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:777.39
  • Desformylflustrabromine hydrochloride

    CAS:
    <p>Desformylflustrabromine hydrochloride (dFBr hydrochloride) is a selective agonist of nicotinic acetylcholine receptor (nAChR) in α4β2 neurons, with pEC50 of 6.</p>
    Fórmula:C17H12INO5
    Pureza:98.12%
    Forma y color:Solid
    Peso molecular:437.19
  • E6801

    CAS:
    <p>E6801: selective 5-HT6 agonist for research in dementia, Parkinson's, depression, obesity, epilepsy, anxiety, etc.</p>
    Fórmula:C17H18ClN5O2S2
    Pureza:96.32% - 99.53%
    Forma y color:Solid
    Peso molecular:423.94
  • CPCCOEt

    CAS:
    <p>CPCCOEt is a low affinity, selective, non-competitive and reversible antagonist of mGluR1b</p>
    Fórmula:C13H13NO4
    Pureza:99.91%
    Forma y color:Solid
    Peso molecular:247.25
  • Suriclone

    CAS:
    <p>Suriclone (RP 31264), a cyclic pyrrolidone for anxiety, modulates GABA-A receptors without major sedation.</p>
    Fórmula:C20H20ClN5O3S2
    Pureza:99.21% - 99.73%
    Forma y color:Solid
    Peso molecular:477.99
  • Cilansetron

    CAS:
    <p>Cilansetron is an effective and selective 5-HT3 receptor antagonist that can be used for related diseases caused by colitis.</p>
    Fórmula:C20H21N3O
    Pureza:99.82% - 99.98%
    Forma y color:Solid
    Peso molecular:319.4
  • DSS30

    CAS:
    <p>DSS30 is a P25/CDK5 inhibitor that reduces β-amyloid secretion to help prevent Alzheimer's.</p>
    Fórmula:C16H14ClNO3S2
    Pureza:99.19% - 99.4%
    Forma y color:Solid
    Peso molecular:367.87
  • Lecozotan HCl

    CAS:
    <p>Lecozotan HCl is a selective 5-HT antagonist boosting glutamate and acetylcholine release without causing 5-HT(1A) tolerance.</p>
    Fórmula:C28H30ClN5O3
    Pureza:99.04%
    Forma y color:Solid
    Peso molecular:520.02
  • Ensaculin

    CAS:
    <p>Ensaculin, a benzopyrone-piperazine compound, enhances memory, protects neurons, and may treat dementia.</p>
    Fórmula:C26H32N2O5
    Pureza:99.17% - 99.67%
    Forma y color:Solid
    Peso molecular:452.54
  • Aβ-IN-1

    CAS:
    <p>Aβ-IN-1 is a novel, potent and orally active γ-secretase modulator (GSM).</p>
    Fórmula:C35H49N
    Pureza:99.1%
    Forma y color:Soild
    Peso molecular:483.77
  • Roxindole

    CAS:
    <p>Roxindole: dopamine agonist, serotonin reuptake inhibitor, 5-HT1A agonist, developed for schizophrenia.</p>
    Fórmula:C23H26N2O
    Pureza:98.03% - 98.93%
    Forma y color:Solid
    Peso molecular:346.47
  • Ru-32514

    CAS:
    <p>Ru-32514 is a benzodiazepine receptor agonist.</p>
    Fórmula:C18H17N3O2
    Pureza:99.21%
    Forma y color:Solid
    Peso molecular:307.35
  • ELB-139

    CAS:
    <p>ELB-139 is a GABA A receptor agonist. ELB139 increases 5-HT in the striatum and prefrontal cortex of rats.</p>
    Fórmula:C14H16ClN3O
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:277.75
  • Quinupramine

    CAS:
    <p>Quinupramine: an oral antidepressant targeting the serotonin system; penetrates CNS; doesn’t affect β-adrenergic system.</p>
    Fórmula:C21H24N2
    Pureza:99.77%
    Forma y color:Solid
    Peso molecular:304.43
  • Agomelatine hydrochloride

    CAS:
    <p>Agomelatine HCl is a MT1/MT2 receptor agonist (Ki: 0.1-0.27 nM) and a 5-HT2C antagonist (pKi: 6.2-6.4).</p>
    Fórmula:C15H18ClNO2
    Pureza:99.57%
    Forma y color:Solid
    Peso molecular:279.76
  • Femoxetine hydrochloride

    CAS:
    <p>Femoxetine hydrochloride is a selective 5-hydroxytryptamine reuptake inhibitor used in the study of migraine, depression and eating disorders.</p>
    Fórmula:C20H26ClNO2
    Pureza:99.63%
    Forma y color:Solid
    Peso molecular:347.88
  • GSK-1482160

    CAS:
    <p>GSK-1482160 is a CNS-penetrant negative allosteric modulator of P2X7 receptor with oral activity.</p>
    Fórmula:C14H14ClF3N2O2
    Pureza:99.57%
    Forma y color:Solid
    Peso molecular:334.72
  • Sudoxicam

    CAS:
    <p>Sudoxicam (4-Hydroxy-2-methyl-N-2-thiazolyl-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxide) is a reversible antagonist of COX with anti-inflammatory, anti-edema</p>
    Fórmula:C13H11N3O4S2
    Pureza:99.93%
    Forma y color:Solid
    Peso molecular:337.37
  • Fengabine

    CAS:
    <p>Fengabine (SL-79229) is a GABA receptor agonist with antidepressant activity and is used to treat depression.</p>
    Fórmula:C17H17Cl2NO
    Pureza:99%
    Forma y color:Solid
    Peso molecular:322.23
  • Lenumlostat

    CAS:
    <p>Lenumlostat is a lysyl oxidase-like protein 2 (LOXL2) inhibitor with inhibitory effects on hLOXL2, hLOXL3 and LOXL2 for the study of fibrotic diseases.</p>
    Fórmula:C18H17F4N3O3
    Pureza:99.11%
    Forma y color:Solid
    Peso molecular:399.34
  • Ecopipam

    CAS:
    <p>Ecopipam: orally active, selective dopamine D1/D5 antagonist (Ki: 1.2 nM/2.0 nM). 40x more selective over D2/D4/5-HT/α2a. For schizophrenia, obesity research.</p>
    Fórmula:C19H20ClNO
    Pureza:99.68%
    Forma y color:Solid
    Peso molecular:313.82
  • Sarizotan HCl

    CAS:
    <p>Sarizotan HCl (EMD 128130 HCl) is a 5-HT1A receptor and dopamine receptor agonist and an hERG channel inhibitor used in Parkinson;s disease research.</p>
    Fórmula:C22H22ClFN2O
    Pureza:96%
    Forma y color:Solid
    Peso molecular:384.87
  • CP-810123

    CAS:
    <p>CP-810123 is an α7 nAChR agonist used to treat cognitive deficits associated with psychiatric or neurological disorders such as schizophrenia.</p>
    Fórmula:C14H18N4O
    Pureza:98.63% - 99.60%
    Forma y color:Solid
    Peso molecular:258.32
  • AZD6538

    CAS:
    <p>AZD6538 is an mGluR5 negative allosteric modulator used in the study of CNS-related diseases such as Alzheimer's disease.</p>
    Fórmula:C15H6FN5O
    Pureza:98.68%
    Forma y color:Solid
    Peso molecular:291.24
  • LY 272015 hydrochloride

    CAS:
    <p>LY 272015 hydrochloride is a 5-HT2B receptor antagonist.</p>
    Fórmula:C21H25ClN2O2
    Pureza:99.47%
    Forma y color:Solid
    Peso molecular:372.89
  • Golexanolone

    CAS:
    <p>Golexanolone can be used to study neurological diseases.</p>
    Fórmula:C21H31NO2
    Pureza:99.90% - 99.99%
    Forma y color:Solid
    Peso molecular:329.48
  • Ticalopride

    CAS:
    <p>Ticalopride: 5-HT3 agonist for digestive, orofacial, ENT disorders, and bulimia, GERD, IBS research.</p>
    Fórmula:C14H20ClN3O3
    Pureza:99.51%
    Forma y color:Solid
    Peso molecular:313.78
  • Eltenac

    CAS:
    <p>Eltenac, a cyclooxygenase (COX) inhibitor, is used potentially for the treatment of pain.</p>
    Fórmula:C12H9Cl2NO2S
    Pureza:98.53%
    Forma y color:Solid
    Peso molecular:302.18
  • ADR-851 free base

    CAS:
    <p>ADR-851 free base is an antagonist of the HT3 receptor.</p>
    Fórmula:C14H18ClN3O2
    Pureza:97.88% - 98.39%
    Forma y color:Solid
    Peso molecular:295.77
  • Aplindore Fumarate

    CAS:
    <p>Aplindore Fumarate (DAB-452), a selective dopamine D2/D3 partial agonist, is used in Parkinson's and schizophrenia research.</p>
    Fórmula:C22H22N2O7
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:426.42
  • ATC 0175 hydrochloride

    CAS:
    <p>ATC 0175 hydrochloride is an orally active melanocyte concentrating hormone 1 receptor antagonist that is potent and selective.</p>
    Fórmula:C23H26ClF2N5O
    Pureza:99.98%
    Forma y color:Solid
    Peso molecular:461.93
  • NB001

    CAS:
    <p>NB001 (HTS 09836) is an inhibitor of adenyl cyclase 1 exhibiting effects on neural and non-neural pain.</p>
    Fórmula:C12H20N6O
    Pureza:99.69%
    Forma y color:Off-White To Pale Pink Solid
    Peso molecular:264.33
  • Liafensine

    CAS:
    <p>Liafensine(BMS-820836): Selective inhibitor for serotonin, norepinephrine, dopamine reuptake; targets major depression, CNS disorders.</p>
    Fórmula:C24H22N4
    Pureza:99.91%
    Forma y color:Solid
    Peso molecular:366.46
  • BMY-14802 hydrochloride

    CAS:
    <p>BMY-14802 hydrochloride (BMS 181100 hydrochloride) is a selective antagonist of σ receptor (IC50 = 112 nM) with antipsychotic effects.</p>
    Fórmula:C18H23ClF2N4O
    Pureza:99.97%
    Forma y color:Solid
    Peso molecular:384.85
  • 5-HT2 antagonist 1

    CAS:
    <p>5-HT2 antagonist 1 is a potent 5-HT2 receptor antagonist, has weak α1 adrenoceptor blocking activity.</p>
    Fórmula:C22H29FN4O2
    Pureza:99.76%
    Forma y color:Solid
    Peso molecular:400.49
  • GR 46611

    CAS:
    <p>GR 46611 is a selective 5-HT1B and 5-HT1D receptor agonist and can be used in studies about the treatment of epilepsy.</p>
    Fórmula:C23H27N3O2
    Pureza:99.75%
    Forma y color:Solid
    Peso molecular:377.48
  • CGP 37849

    CAS:
    <p>CGP 37849: oral NMDA antagonist (Ki=35 nM), anticonvulsant, with antidepressant/anxiolytic effects.</p>
    Fórmula:C6H12NO5P
    Pureza:99.87%
    Forma y color:White Solid
    Peso molecular:209.14
  • DSP-0565

    CAS:
    <p>DSP-0565 is a broad-spectrum anti-epileptic with a high safety margin and effectiveness in several convulsant models.</p>
    Fórmula:C14H12FNO
    Pureza:99.51% - 99.56%
    Forma y color:Solid
    Peso molecular:229.25
  • CBiPES hydrochloride

    CAS:
    <p>CBiPES hydrochloride (CBiPES HCl) is an orthosteric modulator of the mGlu2 receptor and is used to study neurological disorders like epilepsy.</p>
    Fórmula:C21H20ClN3O2S
    Pureza:99.66%
    Forma y color:Solid
    Peso molecular:413.92
  • VU 0285683

    CAS:
    <p>VU 0285683 is a specific negative allosteric modulator of mGluR5 with a high affinity for the MPEP binding site. VU 0285683 shows anxiolytic-like activity.</p>
    Fórmula:C14H7FN4O
    Pureza:99.98%
    Forma y color:Solid
    Peso molecular:266.23
  • Landipirdine

    CAS:
    <p>Landipirdine (RO-5025181) is a selective 5-HT6R antagonist for the study of central nervous system disorders such as dementia.</p>
    Fórmula:C18H19FN2O3S
    Pureza:97.61% - 99.37%
    Forma y color:Solid
    Peso molecular:362.42
  • LY266097 hydrochloride

    CAS:
    <p>LY266097 hydrochloride is a 5-HT2 antagonist with pKi of 7.7/9.8/7.6 for 5-HT2A/B/C, used in depression research.</p>
    Fórmula:C21H24Cl2N2O2
    Pureza:98.58%
    Forma y color:Solid
    Peso molecular:407.33