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Neurociencia

Neurociencia

Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.

Subcategorías de "Neurociencia"

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Se han encontrado 5398 productos de "Neurociencia"

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  • RWJ-51204

    CAS:
    <p>RWJ-51204: potent adenosine A2A blocker, GABA(A) partial agonist (IC50: 0.2-2 nM), neuroprotective, may treat Parkinson's.</p>
    Fórmula:C21H19F2N3O3
    Pureza:99.57% - 99.95%
    Forma y color:Solid
    Peso molecular:399.39
  • SPD-473 citrate

    CAS:
    <p>SPD-473 citrate is an inhibitior of serotonin/dopamine/norepinephrine reuptake.</p>
    Fórmula:C23H31Cl2NO8S
    Pureza:99.37%
    Forma y color:Solid
    Peso molecular:552.47
  • Roxindole

    CAS:
    <p>Roxindole: dopamine agonist, serotonin reuptake inhibitor, 5-HT1A agonist, developed for schizophrenia.</p>
    Fórmula:C23H26N2O
    Pureza:98.03% - 98.93%
    Forma y color:Solid
    Peso molecular:346.47
  • Aplindore Fumarate

    CAS:
    <p>Aplindore Fumarate (DAB-452), a selective dopamine D2/D3 partial agonist, is used in Parkinson's and schizophrenia research.</p>
    Fórmula:C22H22N2O7
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:426.42
  • Femoxetine hydrochloride

    CAS:
    <p>Femoxetine hydrochloride is a selective 5-hydroxytryptamine reuptake inhibitor used in the study of migraine, depression and eating disorders.</p>
    Fórmula:C20H26ClNO2
    Pureza:99.63%
    Forma y color:Solid
    Peso molecular:347.88
  • GSK-1482160

    CAS:
    <p>GSK-1482160 is a CNS-penetrant negative allosteric modulator of P2X7 receptor with oral activity.</p>
    Fórmula:C14H14ClF3N2O2
    Pureza:99.57%
    Forma y color:Solid
    Peso molecular:334.72
  • AQW051

    CAS:
    <p>AQW051 (VQW-765) is an oral α7-nAChR activator for cognitive impairments, used in anxiety disorder studies.</p>
    Fórmula:C19H22N2O
    Pureza:99.94%
    Forma y color:Solid
    Peso molecular:294.39
  • Masupirdine free base

    CAS:
    <p>Masupirdine free base (SUVN-502 free base) is a 5-HT6 receptor antagonist that can be used to study neurological disorders like Alzheimer's disease.</p>
    Fórmula:C21H24BrN3O3S
    Pureza:98.36% - 99.65%
    Forma y color:Solid
    Peso molecular:478.4
  • Divaplon

    CAS:
    <p>Divaplon is a GABA receptor agonist (IC50: 0.056 µM) that displays non-sedating anxiolytic behavioral characteristics in a rat model of anxiety.</p>
    Fórmula:C17H17N3O2
    Pureza:97.44% - 98.25%
    Forma y color:Solid
    Peso molecular:295.34
  • Cilansetron

    CAS:
    <p>Cilansetron is an effective and selective 5-HT3 receptor antagonist that can be used for related diseases caused by colitis.</p>
    Fórmula:C20H21N3O
    Pureza:99.82% - 99.98%
    Forma y color:Solid
    Peso molecular:319.4
  • MAO-B-IN-9

    CAS:
    <p>MAO-B-IN-9 is a monoamine oxidase B MAO-B inhibitor (IC50: 0.18 μM) that crosses the blood-brain barrier with potency, selectivity and time-dependence.</p>
    Fórmula:C18H24N2O2
    Pureza:99.93%
    Forma y color:Solid
    Peso molecular:300.4
  • 8-OH-Dpat

    CAS:
    <p>8-OH-Dpat (8-Hydroxy-DPAT) is a serotonin 1A-receptor agonist that is used experimentally to test the effects of serotonin.</p>
    Fórmula:C16H25NO
    Pureza:98%
    Forma y color:Solid
    Peso molecular:247.38
  • CGP 37849

    CAS:
    <p>CGP 37849: oral NMDA antagonist (Ki=35 nM), anticonvulsant, with antidepressant/anxiolytic effects.</p>
    Fórmula:C6H12NO5P
    Pureza:99.87%
    Forma y color:White Solid
    Peso molecular:209.14
  • (Z)-Thiothixene

    CAS:
    <p>(Z)-Thiothixene (Thiothixene) is an antagonist of serotonergic receptor.</p>
    Fórmula:C23H29N3O2S2
    Pureza:99.21%
    Forma y color:Yellow To Yellow With A Tan Cast Powder
    Peso molecular:443.63
  • SCH-900271

    CAS:
    <p>SCH-900271 treats dyslipidemia by targeting nicotinic acid receptors, addressing hyperlipidaemia.</p>
    Fórmula:C14H16N2O4
    Pureza:98.82% - 99.93%
    Forma y color:Solid
    Peso molecular:276.29
  • (E/Z)-SIB-1893

    CAS:
    <p>(E/Z)-SIB-1893 (SIB 1893) is the racemate of (E)-SIB-1893 and (Z)-SIB-1893.</p>
    Fórmula:C14H13N
    Pureza:99.92%
    Forma y color:Solid
    Peso molecular:195.26
  • Selurampanel

    CAS:
    <p>Selurampanel (BGG492), an oral AMPA antagonist for epilepsy, migraine, and tinnitus studies.</p>
    Fórmula:C16H19N5O4S
    Pureza:99.60% - 99.78%
    Forma y color:Solid
    Peso molecular:377.42
  • UK-240455

    CAS:
    <p>UK-240455: Potent NMDA glycine antagonist with neuroprotection and motor function benefits in Parkinson's.</p>
    Fórmula:C11H11Cl2N3O5S
    Pureza:98.34% - 99.84%
    Forma y color:Solid
    Peso molecular:368.19
  • Muscimol HBr

    CAS:
    <p>Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.</p>
    Fórmula:C4H7BrN2O2
    Pureza:98.13%
    Forma y color:Off-White Powder
    Peso molecular:195.01
  • DSP-0565

    CAS:
    <p>DSP-0565 is a broad-spectrum anti-epileptic with a high safety margin and effectiveness in several convulsant models.</p>
    Fórmula:C14H12FNO
    Pureza:99.51% - 99.56%
    Forma y color:Solid
    Peso molecular:229.25
  • Buntanetap

    CAS:
    <p>Buntanetap ((+)-Phenserine) is an inhibitor of TINAPs used in the study of neurological disorders, endocrine and metabolic disorders, and cardiovascular disease</p>
    Fórmula:C20H23N3O2
    Pureza:98.2%
    Forma y color:Solid
    Peso molecular:337.42
  • NNC 05-711

    CAS:
    <p>NNC 05-711 (NO-711 hydrochloride) is a potent and selective inhibitor of GAT-1 (GABA transporter 1), exerting anticonvulsant and analgesic effects.</p>
    Fórmula:C21H23ClN2O3
    Pureza:99.92%
    Forma y color:Solid
    Peso molecular:386.87
  • Panadiplon

    CAS:
    <p>Panadiplon (FG 10571) is a selective gamma-aminobutyric acid receptor agonist and partial agonist of 5GABAA, a benzodiazepine receptor, used in the treatment of</p>
    Fórmula:C18H17N5O2
    Pureza:98.30% - 98.94%
    Forma y color:Solid
    Peso molecular:335.36
  • DSS30

    CAS:
    <p>DSS30 is a P25/CDK5 inhibitor that reduces β-amyloid secretion to help prevent Alzheimer's.</p>
    Fórmula:C16H14ClNO3S2
    Pureza:99.19% - 99.4%
    Forma y color:Solid
    Peso molecular:367.87
  • Mibampator

    CAS:
    <p>Mibampator (LY451395) is an effective and selective AMPA receptor potentiator.</p>
    Fórmula:C21H30N2O4S2
    Pureza:99.34%
    Forma y color:Solid
    Peso molecular:438.6
  • ALX-1393

    CAS:
    <p>ALX-1393 is a selective GlyT2 inhibitor that effectively reduces neuronal action potential activity in a concentration-dependent manner and inhibits the</p>
    Fórmula:C23H22FNO4
    Pureza:99.83%
    Forma y color:Solid
    Peso molecular:395.42
  • LM-1685

    CAS:
    <p>LM-1685是一种有效且具有选择性的人单核细胞和全血中COX-2抑制剂,IC50分别为0.65 µM 和IC50 = 4.3 μM,是治疗炎症的潜在化合物。</p>
    Fórmula:C18H16ClNO4S
    Pureza:98.16%
    Forma y color:Solid
    Peso molecular:377.84
  • ABP688

    CAS:
    <p>ABP688 is a non-competitive and selective mGluR5 antagonist(Ki = 1.7 nM). ABP688 can be used as a PET tracer for clinical imaging.</p>
    Fórmula:C15H16N2O
    Pureza:98.63%
    Forma y color:Solid
    Peso molecular:240.3
  • Cirsimaritin

    CAS:
    <p>Cirsimaritin has anti-bacterial, anti-inflammatory, anti-tumor, antioxidant effects, and protects kidneys; it weakly targets GABAA receptors.</p>
    Fórmula:C17H14O6
    Pureza:99.9%
    Forma y color:Solid
    Peso molecular:314.29
  • SB 699551 dihydrochloride

    CAS:
    <p>SB 699551 dihydrochloride is a 5-ht5a receptor antagonist.</p>
    Fórmula:C34H47Cl2N3O
    Pureza:99.83%
    Forma y color:Solid
    Peso molecular:584.66
  • 2-BFI hydrochloride

    CAS:
    <p>2-BFI hydrochloride: High-affinity I2 agonist; used in researching stroke and immune disease protection.</p>
    Fórmula:C11H11ClN2O
    Pureza:99.94%
    Forma y color:Solid
    Peso molecular:222.67
  • Piromelatine

    CAS:
    <p>Piromelatine is an agonist of melatonin MT1/MT2 receptors, 5-HT1A and 5-HT1D, and an antagonist of 5-HT2B.Piromelatine has antinociceptive activity with</p>
    Fórmula:C17H16N2O4
    Pureza:99.89%
    Forma y color:Solid
    Peso molecular:312.32
  • CPCCOEt

    CAS:
    <p>CPCCOEt is a low affinity, selective, non-competitive and reversible antagonist of mGluR1b</p>
    Fórmula:C13H13NO4
    Pureza:99.91%
    Forma y color:Solid
    Peso molecular:247.25
  • Aceclidine

    CAS:
    <p>Aceclidine (1-azabicyclo[2.2.2]octan-3-yl acetate) is a modulator of M3 mAChR and can be used in studies about treating glaucoma by reducing intraocular</p>
    Fórmula:C9H15NO2
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:169.22
  • ML 10302 hydrochloride

    CAS:
    <p>ML 10302 hydrochloride is a specific agonist 5-HT4 and binds 5-HT receptors with Kis of 1.07 nM and 782 nM for 5-HT4 and 5-HT3.</p>
    Fórmula:C15H22Cl2N2O3
    Pureza:99.99%
    Forma y color:Solid
    Peso molecular:349.25
  • DMCM hydrochloride

    CAS:
    <p>DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine.</p>
    Fórmula:C17H19ClN2O4
    Pureza:99.56%
    Forma y color:Solid
    Peso molecular:350.8
  • Valiglurax

    CAS:
    <p>Valiglurax (VU2957), potent mGlu4 PAM, crosses blood-brain barrier, orally available; promising for Parkinson's treatment.</p>
    Fórmula:C16H10F3N5
    Pureza:98.29%
    Forma y color:Solid
    Peso molecular:329.28
  • NKY80

    CAS:
    <p>NKY80 regulates the adenylyl cyclase catalytic activity in heart and lung tissues.</p>
    Fórmula:C12H11N3O2
    Pureza:99.88%
    Forma y color:Solid
    Peso molecular:229.23
  • LY-2624803

    CAS:
    <p>LY-2624803 is a 5-HT2A receptor antagonist and histamine receptor inverse agonist that can be used to improve slow wave sleep.</p>
    Fórmula:C22H25N3O3
    Pureza:99.78% - 99.97%
    Forma y color:Solid
    Peso molecular:379.45
  • Lesopitron

    CAS:
    <p>Lesopitron: anxiolytic, 5-HT1A agonist, treats rodent anxiety, counters benzodiazepine withdrawal, low toxicity, no alcohol/barbiturate interaction.</p>
    Fórmula:C15H21ClN6
    Pureza:99.15% - 99.38%
    Forma y color:Solid
    Peso molecular:320.82
  • PF-03635659

    CAS:
    <p>PF-03635659: potent M3 antagonist, Ki=0.2 nM, long half-life, potential COPD treatment.</p>
    Fórmula:C28H32N2O3
    Pureza:98.39% - 99.83%
    Forma y color:Solid
    Peso molecular:444.57
  • 5-HT2 antagonist 1

    CAS:
    <p>5-HT2 antagonist 1 is a potent 5-HT2 receptor antagonist, has weak α1 adrenoceptor blocking activity.</p>
    Fórmula:C22H29FN4O2
    Pureza:99.76%
    Forma y color:Solid
    Peso molecular:400.49
  • Suriclone

    CAS:
    <p>Suriclone (RP 31264), a cyclic pyrrolidone for anxiety, modulates GABA-A receptors without major sedation.</p>
    Fórmula:C20H20ClN5O3S2
    Pureza:99.21% - 99.73%
    Forma y color:Solid
    Peso molecular:477.99
  • PPI-1019

    CAS:
    <p>PPI-1019 is an APP (β-amyloid A4) inhibitor for the treatment of neurological disorders and the study of Alzheimer's disease (AD).</p>
    Fórmula:C36H54N6O5
    Pureza:95.16% - 98.16%
    Forma y color:Solid
    Peso molecular:650.85
  • CP-810123

    CAS:
    <p>CP-810123 is an α7 nAChR agonist used to treat cognitive deficits associated with psychiatric or neurological disorders such as schizophrenia.</p>
    Fórmula:C14H18N4O
    Pureza:98.63% - 99.60%
    Forma y color:Solid
    Peso molecular:258.32
  • Perphenazine dihydrochloride

    CAS:
    <p>Perphenazine dihydrochloride: Oral dopamine, histamine-1 antagonist; targets D2, D3, 5-HT2A, Alpha-1A; may treat psychiatric disorders, cancer.</p>
    Fórmula:C21H28Cl3N3OS
    Pureza:99.67%
    Forma y color:Solid
    Peso molecular:476.89
  • RS 67333 hydrochloride

    CAS:
    <p>RS 67333 hydrochloride is a selective 5-HT4R partial agonist (pKi=8.7) with neuroprotective properties for Alzheimer's research.</p>
    Fórmula:C19H30Cl2N2O2
    Pureza:98.78%
    Forma y color:Solid
    Peso molecular:389.36
  • Agomelatine hydrochloride

    CAS:
    <p>Agomelatine HCl is a MT1/MT2 receptor agonist (Ki: 0.1-0.27 nM) and a 5-HT2C antagonist (pKi: 6.2-6.4).</p>
    Fórmula:C15H18ClNO2
    Pureza:99.57%
    Forma y color:Solid
    Peso molecular:279.76
  • Itasetron

    CAS:
    <p>Itasetron, a 5-HT3 antagonist, prevents memory loss in rats and has antiemetic effects in cancer treatments.</p>
    Fórmula:C16H20N4O2
    Pureza:98.58% - 99.33%
    Forma y color:Solid
    Peso molecular:300.36
  • Ricasetron

    CAS:
    <p>Ricasetron (Brl 46470) is a 5-HT3 receptor antagonist with pro-axonal lysing properties and is used in the study of anxiety disorders and anxiety disorders.</p>
    Fórmula:C19H27N3O
    Pureza:99.52%
    Forma y color:Solid
    Peso molecular:313.44
  • RS 42358-197

    CAS:
    <p>RS 42358-197 (RS 25259-007) is a competitive 5-HT3 receptor antagonist.</p>
    Fórmula:C19H23ClN2O
    Pureza:99.70%
    Forma y color:Solid
    Peso molecular:330.85
  • SB228357

    CAS:
    <p>SB228357 is a potent and selective antagonist of the 5-HT receptor with pKis of 6.9, 8.0, and 9.0 for 5-HT2A, 5-HT2B, and 5-HT2C, respectively.</p>
    Fórmula:C22H17F4N3O2
    Pureza:99.82%
    Forma y color:Solid
    Peso molecular:431.38
  • BL-1020 Mesylate

    CAS:
    <p>BL-1020 Mesylate (CYP-1020 Mesylate) is a GABA A receptor agonist and D2 antagonist used in studies of neurodegeneration.</p>
    Fórmula:C28H45ClN4O11S4
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:777.39
  • GR 46611

    CAS:
    <p>GR 46611 is a selective 5-HT1B and 5-HT1D receptor agonist and can be used in studies about the treatment of epilepsy.</p>
    Fórmula:C23H27N3O2
    Pureza:99.75%
    Forma y color:Solid
    Peso molecular:377.48
  • Lecozotan HCl

    CAS:
    <p>Lecozotan HCl is a selective 5-HT antagonist boosting glutamate and acetylcholine release without causing 5-HT(1A) tolerance.</p>
    Fórmula:C28H30ClN5O3
    Pureza:99.04%
    Forma y color:Solid
    Peso molecular:520.02
  • Lensiprazine

    CAS:
    <p>Lensiprazine (SLV314) is a potent dopamine D(2) receptor antagonist that acts as a serotonin reuptake inhibitor , and can be used to study bipolar disorder and</p>
    Fórmula:C24H27FN4O2
    Pureza:98.04%
    Forma y color:Solid
    Peso molecular:422.5
  • BMY-14802 hydrochloride

    CAS:
    <p>BMY-14802 hydrochloride (BMS 181100 hydrochloride) is a selective antagonist of σ receptor (IC50 = 112 nM) with antipsychotic effects.</p>
    Fórmula:C18H23ClF2N4O
    Pureza:99.97%
    Forma y color:Solid
    Peso molecular:384.85
  • H-9 dihydrochloride

    CAS:
    <p>H-9 dihydrochloride: Strong PKA inhibitor, curbs 5-HT response and EGF signaling, affects pharyngeal function.</p>
    Fórmula:C11H15Cl2N3O2S
    Pureza:97.3%
    Forma y color:Solid
    Peso molecular:324.23
  • JNJ-54175446

    CAS:
    <p>JNJ-54175446 (JNJ-5446) is a P2X7 receptor antagonist that attenuates the release of IL-1β/IL-18 from microglia and is used in the study of depression.</p>
    Fórmula:C18H13ClF4N6O
    Pureza:97.98% - 99.79%
    Forma y color:Solid
    Peso molecular:440.78
  • Riluzole hydrochloride

    CAS:
    <p>Riluzole hydrochloride, an anticonvulsant Na+ channel blocker, inhibits GABA uptake (IC50: 43 µM).</p>
    Fórmula:C8H6ClF3N2OS
    Pureza:99.76%
    Forma y color:Solid
    Peso molecular:270.66
  • (±)-Fabesetron hydrochloride

    CAS:
    <p>FK1052 hydrochloride is a potent 5-HT3 and 5-HT4 receptor dual antagonist.</p>
    Fórmula:C18H20ClN3O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:329.82
  • Aβ/tau aggregation-IN-3

    CAS:
    <p>Aβ/tau aggregation-IN-3 is a potent inhibitor of amyloid protein aggregation, exhibiting an IC50 value of 0.85 µM in an Aβ-Thioflavin T (Aβ-ThT) functional</p>
    Fórmula:C23H22N4O3
    Forma y color:Solid
    Peso molecular:402.45
  • SB 258719

    CAS:
    <p>SB 258719 is a selective antagonist of 5-HT7 receptor with pKi of 7.5.</p>
    Fórmula:C18H30N2O2S
    Pureza:99.73%
    Forma y color:Solid
    Peso molecular:338.51
  • VU0029251

    CAS:
    <p>VU0029251 serves as a partial antagonist of mGluR5, exhibiting a binding affinity with a K i of 1.07 μM.</p>
    Fórmula:C10H11N3S2
    Forma y color:Solid
    Peso molecular:237.34
  • AAK1-IN-3

    CAS:
    <p>AAK1-IN-3: Brain-penetrant AAK1 inhibitor for neuropathic pain research; IC50=11 nM.</p>
    Fórmula:C20H20N4
    Forma y color:Solid
    Peso molecular:316.4
  • AChE-IN-31

    CAS:
    <p>AChE-IN-31 (compound 1), a non-competitive acetylcholinesterase (AChE) inhibitor, exhibits potential for Alzheimer's disease research [1].</p>
    Fórmula:C27H44Na2O9S2
    Forma y color:Solid
    Peso molecular:622.74
  • Tiotropium Bromide hydrate

    CAS:
    <p>Tiotropium Bromide hydrate is a potent, long-lasting anticholinergic bronchodilator for COPD, with high affinity for muscarinic receptors M1, M2, and M3.</p>
    Fórmula:C19H24BrNO5S2
    Pureza:98.44% - 99.41%
    Forma y color:Solid
    Peso molecular:490.43
  • AAK1-IN-5

    CAS:
    <p>AAK1-IN-5: Potent, selective AAK1 inhibitor; CNS-penetrant; oral; IC50: 1.2 nM; Ki: 0.05 nM; cell IC50: 0.5 nM. Useful in neuropathic pain research.</p>
    Fórmula:C19H23F4N3O
    Forma y color:Solid
    Peso molecular:385.4
  • Quinolactacin A1

    CAS:
    <p>Quinolactacin A1, a strong AChE inhibitor from Penicillium citrinum, aids Alzheimer's research.</p>
    Fórmula:C16H18N2O2
    Forma y color:Solid
    Peso molecular:270.33
  • VU0360172

    CAS:
    <p>VU0360172 is a positive allosteric modulator of mGlu5 receptors (EC50 = 16 nM; Ki = 195 nM).</p>
    Fórmula:C18H15FN2O
    Pureza:99.56%
    Forma y color:Solid
    Peso molecular:294.32
  • AChE-IN-30

    CAS:
    <p>AChE-IN-30 is an acetylcholinesterase (AChE) inhibitor exhibiting neuroprotective effects with an inhibitory concentration (IC 50) of 4.4 μM.</p>
    Fórmula:C22H24N4O2
    Forma y color:Solid
    Peso molecular:376.45
  • AAK1-IN-2

    CAS:
    <p>AAK1-IN-2, a potent (IC50=5.8 nM) AAK1 inhibitor, selective &amp; brain-penetrant, is used for neuropathic pain studies.</p>
    Fórmula:C20H20N4
    Forma y color:Solid
    Peso molecular:316.4
  • Thioflosulide

    CAS:
    <p>Thioflosulide (L-745337) is a selective and potent COX2 inhibitor (IC50: 2.3 nM) with anti-inflammatory activity for the study of gastric ulcers.</p>
    Fórmula:C16H13F2NO3S2
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:369.41
  • 3β-Hydroxy-lup-20(29)-en-16-one

    CAS:
    <p>3β-Hydroxy-lup-20(29)-en-16-one (compound 9) serves as a dual inhibitor of both AChE and BChE, displaying a preference for BChE with an IC50 of 28.9 μM [1].</p>
    Fórmula:C30H48O2
    Forma y color:Solid
    Peso molecular:440.7
  • CAY10649

    CAS:
    <p>1CAY10649, a thiazolinone compound, directly inhibits 5-lipoxygenase (5-LO) product formation in intact polymorphonuclear leukocytes (PMNL) with an IC50 value of 0.28 μM and in a soluble fraction of an S100 PMNL cell lysate with an IC50 value of 0.09 μM, following stimulation by calcium and arachidonic acid. This activity highlights its potential in mitigating inflammatory responses by targeting the biosynthesis of leukotrienes, substances implicated in various inflammatory processes such as neutrophil chemotaxis, increased vascular permeability, and smooth muscle contraction.</p>
    Fórmula:C17H12ClNO2S
    Forma y color:Solid
    Peso molecular:329.8
  • Velusetrag

    CAS:
    <p>Velusetrag(TD-5108), a potent 5-HT4 agonist, is in development for gastroparesis, constipation, and IBS.</p>
    Fórmula:C25H36N4O5S
    Forma y color:Solid
    Peso molecular:504.64
  • P11149

    CAS:
    <p>P11149: oral AChE inhibitor, crosses BBB, IC50 1.3 μM, based on Galanthamine, aims Alzheimer's research.</p>
    Fórmula:C27H34ClNO4
    Forma y color:Solid
    Peso molecular:472.02
  • Indeloxazine hydrochloride

    CAS:
    <p>Indeloxazine HCl: Serotonin releaser, NE reuptake inhibitor, NMDA antagonist; antidepressant that boosts acetylcholine in rats.</p>
    Fórmula:C14H18ClNO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:267.75
  • Frovatriptan

    CAS:
    <p>Frovatriptan, potent 5-HT 1B/D agonist, shows high cerebroselectivity and efficacy for migraine with aura.</p>
    Fórmula:C14H17N3O
    Forma y color:Solid
    Peso molecular:243.3
  • 5-HT2A antagonist 1

    CAS:
    <p>5-HT2A antagonist 1, from US5728835A &amp; JP 1007727, may treat gastrointestinal and circulatory issues.</p>
    Fórmula:C26H28N4O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:428.53
  • RAGE/SERT-IN-1

    CAS:
    <p>RAGE/SERT-IN-1 is a potent, orally active inhibitor of advanced glycation end products (RAGE) and serotonin transporter (SERT), with IC50 values of 8.26 μM and</p>
    Fórmula:C38H41ClN4OS
    Forma y color:Solid
    Peso molecular:637.28
  • cis-PDA

    CAS:
    <p>cis-PDA (cis PDA) is a general ionotropic receptor antagonist. cis-PDA acts by blocking NMDA, AMPA, and kainate-mediated responses.</p>
    Fórmula:C7H11NO4
    Pureza:98.71%
    Forma y color:White Solid
    Peso molecular:173.17
  • GR 127935 hydrochloride

    CAS:
    <p>5-HT1B/1D receptor antagonist</p>
    Fórmula:C29H32ClN5O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:534.05
  • NAD 299 hydrochloride

    CAS:
    <p>Selective, high affinity 5-HT1A receptor antagonist</p>
    Fórmula:C18H24ClFN2O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:354.85
  • LY-426965

    CAS:
    <p>LY-426965 is a selective, potent, orally bioavailable 5-HT1A antagonist.</p>
    Fórmula:C28H38N2O2
    Forma y color:Solid
    Peso molecular:434.61
  • NO-711ME

    CAS:
    <p>NO-711ME (N-O711 Methyl ester) is a prodrug of NO-711. It also is a potent and selective GABA uptake inhibitor.</p>
    Fórmula:C22H24N2O3
    Pureza:99.54%
    Forma y color:Solid
    Peso molecular:364.44
  • 2-Methyl-5-HT

    CAS:
    <p>2-Methyl-5-HT (2-Methyl-5-hydroxytryptamine) is a potent and selective 5-HT3 receptor agonist with anti-depressive-like effects.</p>
    Fórmula:C11H14N2O
    Pureza:97.18%
    Forma y color:Solid
    Peso molecular:190.24
  • ABT-418 hydrochloride

    CAS:
    <p>ABT-418 HCl enhances cognition and reduces anxiety as a selective nAChRs agonist, researched for Alzheimer's.</p>
    Fórmula:C9H15ClN2O
    Forma y color:Solid
    Peso molecular:202.68
  • Dothiepin

    CAS:
    <p>Dothiepin (Dosulepin; Dothep), an antidepressant with sedative/anxiolytic properties, preferentially inhibits noradrenaline over serotonin uptake, enhancing</p>
    Fórmula:C19H21NS
    Pureza:98%
    Forma y color:Solid
    Peso molecular:295.44
  • LY108742

    CAS:
    <p>LY108742 is an antagonist of 5-HT2.</p>
    Fórmula:C21H28N2O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:356.46
  • Befiradol

    CAS:
    <p>Befiradol (NLX-112) is an agonist of 5-HT1A receptor.</p>
    Fórmula:C20H22ClF2N3O
    Forma y color:Solid
    Peso molecular:393.86
  • BACE1-IN-1

    CAS:
    <p>BACE1-IN-1 is a high brain penetrant BACE1 inhibitor (IC50s: 32 and 47 nM for human BACE1 and BACE2).</p>
    Fórmula:C18H14F3N5O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:389.33
  • Muscarine tosylate

    CAS:
    <p>Muscarine ((+)-Muscarine) tosylate, a prototype mAChR agonist, serves as a parasympathetic nervous system stimulant and is recognized for its toxic properties [1] [2].</p>
    Fórmula:C16H27NO5S
    Forma y color:Solid
    Peso molecular:345.45
  • L 663581

    CAS:
    <p>L 663581 is the benzodiazepine receptor partial agonist.</p>
    Fórmula:C17H16ClN5O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:357.79
  • BMS-983970

    CAS:
    <p>BMS-983970 is an oral inhibitor of pan-Notch, and for the treatment of multiplecancers.</p>
    Fórmula:C26H26F4N4O3
    Forma y color:Solid
    Peso molecular:518.5
  • JNJ-46281222

    CAS:
    <p>JNJ-46281222: mGlu2-selective, potent PAM, Kd = 1.7 nM, pEC50 = 7.71.</p>
    Fórmula:C23H25F3N4
    Forma y color:Solid
    Peso molecular:414.47
  • mAChR antagonist 1

    CAS:
    <p>Compound 4a, a mAChR antagonist, exhibits K i values of 255 nM for M1 and M5 subtypes, and lower values of 121 nM and 158 nM for M3 and M4 subtypes,</p>
    Fórmula:C19H22N2O2
    Forma y color:Solid
    Peso molecular:310.39
  • Lanabecestat

    CAS:
    <p>Lanabecestat (AZD3293) is a BACE1 inhibitor (Ki: 0.4 nM), Lanabecestat is used in the study of neurological diseases like Alzheimer's disease.</p>
    Fórmula:C26H28N4O
    Pureza:98.55%
    Forma y color:Solid
    Peso molecular:412.53
  • (2R,4R)-APDC

    CAS:
    <p>(2R,4R)-APDC is a selective group II metabotropic glutamate receptors (mGluRs) agonist. It has anticonvulsant and neuroprotective effects.</p>
    Fórmula:C6H10N2O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:174.15
  • UNC9994 hydrochloride

    CAS:
    <p>UNC9994 hydrochloride is a selective β-arrestin-biased D2R agonist, Ki of 79 nM, that stimulates β-arrestin and modulates cAMP.</p>
    Fórmula:C21H23Cl3N2OS
    Forma y color:Solid
    Peso molecular:457.84