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Neurociencia

Neurociencia

Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.

Subcategorías de "Neurociencia"

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Se han encontrado 5400 productos de "Neurociencia"

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  • Risperidone hydrochloride

    CAS:
    <p>Risperidone hydrochloride blocks 5-HT2, inhibits P-glycoprotein, and antagonizes D2 receptors (Ki: 5-HT2A - 4.8 nM, D2 - 5.9 nM).</p>
    Fórmula:C23H28ClFN4O2
    Forma y color:Solid
    Peso molecular:446.95
  • Rivanicline hemioxalate


    <p>Rivanicline hemioxalate is a selective α4β2 nicotinic receptor agonist (K i =26 nM), over 1,000x preference to α7 (K i =3.6 μM), with limited side effects.</p>
    Fórmula:C12H16N2O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:207.23
  • Acotiamide

    CAS:
    <p>Acotiamide, an oral AChE inhibitor (IC50: 1.79μM), improves gastric motility, targeting functional dyspepsia.</p>
    Fórmula:C21H30N4O5S
    Forma y color:Solid
    Peso molecular:450.55
  • Piperazine

    CAS:
    <p>Piperazine (1,4-Diazacyclohexane), a gamma-aminobutyric acid (GABA) agonist, serves as a crucial building block and core component in a wide range of marketed drugs known for their varied pharmacological activities.</p>
    Fórmula:C4H10N2
    Forma y color:Solid
    Peso molecular:86.14
  • Ginkgolide A

    CAS:
    <p>Ginkgolide A (BN-52020), from Ginkgo biloba leaves, is an active PAF antagonist with potential in treating inflammation and immune disorders.</p>
    Fórmula:C20H24O9
    Pureza:98.76% - 99.81%
    Forma y color:White Powder
    Peso molecular:408.4
  • Syk Inhibitor II dihydrochloride dihydrate

    CAS:
    <p>Potent, selective ATP-competitive Syk Inhibitor II (IC50: 41 nM), with anti-allergic properties, in dihydrochloride dihydrate form.</p>
    Fórmula:C14H21Cl2F3N6O3
    Forma y color:Solid
    Peso molecular:449.26
  • Prifinium bromide

    CAS:
    <p>Prifinium bromide is a quaternary ammon antimuscarinic. It inhibits hyperkinesia of the digestive organs and urinary tract and has a spasmolytic action.</p>
    Fórmula:C22H28BrN
    Pureza:97.99%
    Forma y color:Solid
    Peso molecular:386.37
  • Ziprasidone mesylate

    CAS:
    <p>Ziprasidone mesylate (CP-88059), an oral 5-HT &amp; dopamine blocker, binds D2, 5-HT2A, 5-HT1A with Ki values: 4.8, 0.42, 3.4 nM.</p>
    Fórmula:C22H25ClN4O4S2
    Forma y color:Solid
    Peso molecular:509.04
  • JHU37152

    CAS:
    <p>JHU37152 is a DREADD agonist; Ki: 1.8 nM at hM3Dq, 8.7 nM at hM4Di; EC50: 5 nM (hM3Dq), 0.5 nM (hM4Di) in HEK-293 cell assays.</p>
    Fórmula:C19H20ClFN4
    Pureza:99.72%
    Forma y color:Solid
    Peso molecular:358.84
  • A-582941 dihydrochloride

    CAS:
    <p>A-582941 dihydrochloride (A 582941) is a Selective agonist of α7 nAChR partial</p>
    Fórmula:C17H22Cl2N4
    Pureza:99.55%
    Forma y color:Solid
    Peso molecular:353.29
  • Aripiprazole monohydrate

    CAS:
    <p>Aripiprazole (OPC-14597) is a potent D2 partial agonist and inverse agonist of 5-HT2 receptors, used for schizophrenia and COVID-19 studies.</p>
    Fórmula:C23H29Cl2N3O3
    Forma y color:Solid
    Peso molecular:466.4
  • Dolasetron Mesylate hydrate

    CAS:
    <p>Dolasetron Mesylate hydrate blocks 5HT3 to prevent chemo and radiotherapy nausea.</p>
    Fórmula:C20H26N2O7S
    Pureza:99.86% - 99.9%
    Forma y color:Solid
    Peso molecular:438.49
  • m-Chlorophenylbiguanide hydrochloride

    CAS:
    <p>m-Chlorophenylbiguanide hydrochloride is a 5-HT3 receptor agonist.</p>
    Fórmula:C8H11Cl2N5
    Pureza:99.43% - 99.87%
    Forma y color:Solid
    Peso molecular:248.11
  • Donepezil

    CAS:
    <p>Donepezil (Aricept) is a piperidine-based, potent, specific, and reversible inhibitor of acetylcholinesterase (AChE).</p>
    Fórmula:C24H29NO3
    Pureza:99.69%
    Forma y color:White Or Almost White Crystal Powder
    Peso molecular:379.49
  • CNQX disodium

    CAS:
    <p>CNQX disodium is a competitive non-NMDA receptor antagonist and competitive AMPA/kainate receptor antagonist in neuronal cultures.</p>
    Fórmula:C9H2N4Na2O4
    Pureza:97.77%
    Forma y color:Solid
    Peso molecular:276.12
  • Ritanserin

    CAS:
    <p>Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.</p>
    Fórmula:C27H25F2N3OS
    Pureza:99.77% - 99.89%
    Forma y color:Solid
    Peso molecular:477.57
  • Aminooxyacetic acid hemihydrochloride

    CAS:
    <p>Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABA</p>
    Fórmula:C2H5NO3·5HCl
    Pureza:98.03%
    Forma y color:Light Beige Crystalline Powder
    Peso molecular:109.3
  • Frentizole

    CAS:
    <p>Frentizole, an immunosuppressive agent, is an inhibitor of the Aβ-ABAD interaction</p>
    Fórmula:C15H13N3O2S
    Pureza:99.82%
    Forma y color:Solid
    Peso molecular:299.35
  • α-Conotoxin MII acetate


    <p>α-Conotoxin MII acetate is a 16-amino acid peptide from the venom of the marine snail Conus magus.</p>
    Fórmula:C69H107N23O24S4
    Pureza:94.82% - 97.79%
    Forma y color:Solid
    Peso molecular:1770.99
  • PHA 543613 hydrochloride

    CAS:
    <p>PHA-543613 hydrochloride, a potent α7 nicotinic receptor agonist, may treat schizophrenia-related cognitive deficits.</p>
    Fórmula:C15H18ClN3O2
    Forma y color:Solid
    Peso molecular:307.78