
Neurociencia
Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.
Subcategorías de "Neurociencia"
- Receptor 5-HT(1.025 productos)
- ACK(1 productos)
- AChR(647 productos)
- ATP Citrato Liasa(17 productos)
- Receptor adrenérgico(3.023 productos)
- BACE(37 productos)
- Beta amiloide(228 productos)
- CAMK(73 productos)
- Inhibidores de ciclooxigenasa (COX)(600 productos)
- Receptor de dopamina(445 productos)
- Receptor GABA(373 productos)
- Gamma-secretasa(61 productos)
- GluR(265 productos)
- GlyT(26 productos)
- Receptor de histamina(385 productos)
- LRRK2(43 productos)
- Receptor de melatonina(26 productos)
- NMDAR(10 productos)
- Receptor de OX(41 productos)
- Receptor de opioides(327 productos)
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Se han encontrado 5612 productos de "Neurociencia"
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2,3-Dehydrosilybin A
CAS:2,3-Dehydrosilybin A is a useful organic compound for research related to life sciences and the catalog number is T125202.Fórmula:C25H20O10Forma y color:SolidPeso molecular:480.43L-AP3
CAS:L-AP3 blocks mGluR, inhibits D/L-phosphoserine (IC50: 368/2087 μM).Fórmula:C3H8NO5PForma y color:White Hygroscopic SolidPeso molecular:169.073AChE-IN-60
AChE-IN-60 (compound 6k) is a potent inhibitor of acetylcholinesterase (AChE) and butyrylcholinesterase (BChE), with IC50 values of 27 nM and 43 nM, respectively. It also inhibits monoamine oxidase MAO-A and MAO-B, with IC50 values of 353 nM and 716 nM, respectively.Fórmula:C24H29N3O4S3Peso molecular:519.13202(Iso)-Landipirdine
CAS:(Iso)-Landipirdine((Iso)-RO5025181) is a selective and potent 5-HT6R antagonist.Fórmula:C18H19FN2O3SPureza:98.94%Forma y color:SoildPeso molecular:362.42Pozanicline hydrochloride
Pozanicline hydrochloride is an oral α4β2 nAChR agonist with a 16.7 nM Ki, insignificantly binding to α7 nAChR.Fórmula:C11H17ClN2OPureza:97.13% - 99.81%Forma y color:SolidPeso molecular:228.72Ref: TM-T16563L
1mg73,00€1mL*10mM (DMSO)127,00€5mg146,00€10mg208,00€25mg319,00€50mg447,00€100mg600,00€200mg808,00€(+)-Cinchonaminone
CAS:(+)-Cinchonaminone shows monoamine oxidase (MAO) inhibitory activity.Fórmula:C19H24N2O2Forma y color:SolidPeso molecular:312.413Heliosupine N-oxide
Heliosupine N-oxide is a useful organic compound for research related to life sciences and the catalog number is T125058.Fórmula:C20H31NO8Forma y color:SolidPeso molecular:413.467SB-408124
CAS:SB408124: Non-peptide, OX1 receptor antagonist, Ki 57 nM (whole cell) and 27 nM (membrane), 50x more selective than OX2.Fórmula:C19H18F2N4OPureza:99.81%Forma y color:SolidPeso molecular:356.37BChE-IN-19
BChE-IN-19 (Compound 7b), a para-substituted indone derivative, exhibits potent inhibitory activity against butyryl cholinesterase (BChE) with an IC50 value ofFórmula:C25H31NO5Forma y color:SolidPeso molecular:425.52SIB 1553A
CAS:SIB 1553A is an agonist of nAChRs, a cognitive enhancer that can be used to study diseases associated with neurodegeneration.Fórmula:C13H19NOSPureza:99.79%Forma y color:SoildPeso molecular:237.36CPN-351
CAS:CPN-351 (compound 9a) is a pentapeptide that acts as a selective antagonist for human NMUR1, with a pA2 value of 7.35. It exhibits ten times greater antagonistic activity toward human NMUR1 compared to NMUR2. CPN-351 is applicable in inflammation research.Fórmula:C45H61N13O6SPeso molecular:912.11Millmerranone A
Millmerranone A shows the acetylcholinesterase inhibitory property.Fórmula:C27H28O9Forma y color:SolidPeso molecular:496.51Mosapride citrate dihydrate
CAS:Mosapride Citrate, a 5-HT4 agonist, boosts gut movement by enhancing acetylcholine release.Fórmula:C27H35ClFN3O11Pureza:98%Forma y color:SolidPeso molecular:632.04Paecilomide
CAS:Paecilomide is a pyridone alkaloid and acetylcholinesterase inhibitor [1] .Fórmula:C12H15NO4Forma y color:SolidPeso molecular:237.25Aβ-IN-7
Aβ-IN-7 (compound 5a) acts as a potent inhibitor of Aβ aggregation, stabilizing Aβ monomers at 50 μM concentration to prevent them from forming larger oligomersFórmula:C14H10N2SForma y color:SolidPeso molecular:238.31LY 344864 racemate
CAS:LY 344864 racemate is a 5-HT1F receptor agonist.Fórmula:C21H22FN3OPureza:99.75%Forma y color:SoildPeso molecular:351.42SB236057
CAS:SB236057: potent selective inverse agonist at 5-HT autoreceptors; increases brain 5-HT; teratogen causing musculoskeletal defects in rodents.Fórmula:C33H34N4O3Pureza:98%Forma y color:SolidPeso molecular:534.65Aβ-IN-8
Aβ-IN-8, also known as compound 7e, is a potent inhibitor of Aβ aggregation [1].Fórmula:C22H16F3N3O3SForma y color:SolidPeso molecular:459.44rac-Desethyl Oxybutynin (hydrochloride)
CAS:rac-Desethyl oxybutynin, active oxybutynin metabolite, binds to mAChRs; K_i values 3.12-16 nM; lowers rat micturition pressure.Fórmula:C20H28ClNO3Forma y color:SolidPeso molecular:365.89α-Bungarotoxin
CAS:Neurotoxin that blocks neuromuscular transmission via irreversible inhibition of nicotinic ACh receptors (nAChRs).Fórmula:C338H529N97O105S11Pureza:98%Forma y color:SolidPeso molecular:7984.14

