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Neurociencia

Neurociencia

Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.

Subcategorías de "Neurociencia"

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Se han encontrado 5516 productos de "Neurociencia"

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  • Methiothepin mesylate

    CAS:
    Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an antipsychotic.
    Fórmula:C21H28N2O3S3
    Pureza:98% - 99.92%
    Forma y color:Solid
    Peso molecular:452.65
  • Urapidil

    CAS:
    <p>Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.</p>
    Fórmula:C20H29N5O3
    Pureza:99.85% - >99.99%
    Forma y color:Solid
    Peso molecular:387.48
  • Clomipramine

    CAS:
    <p>Clomipramine treats OCD, depression, chronic pain, and may lower suicide risk in seniors; works by hindering serotonin reuptake.</p>
    Fórmula:C19H23ClN2
    Pureza:99.31% - 99.71%
    Forma y color:Solid
    Peso molecular:314.85
  • (-)-Dizocilpine maleate

    CAS:
    <p>(-)-Dizocilpine maleate ((-)-MK 801 (Maleate)) is a potent, selective and non-competitive NMDA receptor antagonist with Kd of 37.2 nM in rat brain membranes.</p>
    Fórmula:C20H19NO4
    Pureza:>99.99%
    Forma y color:White Solid
    Peso molecular:337.37
  • MTEP

    CAS:
    MTEP: potent, selective mGluR5 antagonist; IC50=5 nM, Ki=16 nM; may have antidepressant/anxiolytic effects; useful in Parkinson's research.
    Fórmula:C11H8N2S
    Forma y color:Solid
    Peso molecular:200.26
  • Intepirdine

    CAS:
    <p>Intepirdine (GSK-742457) is a highly selective 5-HT6 receptor antagonist, used in trials studying the treatment of Alzheimer's Disease.</p>
    Fórmula:C19H19N3O2S
    Pureza:98% - 98.63%
    Forma y color:Solid
    Peso molecular:353.44
  • Zacopride

    CAS:
    Zacopride is a selective agonist of inward rectifier potassium current (I K1) channel, inhibiting ventricular arrhythmias without affecting atrial arrhythmias.
    Fórmula:C15H20ClN3O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:309.79
  • Semagacestat

    CAS:
    Semagacestat (LY450139) (LY450139) is a γ-secretase blocker for Aβ42/Aβ40/Aβ38 (IC50: 10.9/12.1/12.0 nM) and also inhibits Notch signaling (IC50: 14.1 nM).
    Fórmula:C19H27N3O4
    Pureza:97.1% - 99.9%
    Forma y color:Solid
    Peso molecular:361.44
  • PiB

    CAS:
    <p>PiB (Pittsburgh Compound-B) is a standard for analysis of 11C-PiB. 11C-PiB is a β-amyloid PET imaging tracer for Alzheimer's disease diagnosis.</p>
    Fórmula:C14H12N2OS
    Pureza:97.02%
    Forma y color:Solid
    Peso molecular:256.32
  • SC-560

    CAS:
    <p>SC-560 is a member of the diaryl heterocycle class of cyclooxygenase (COX) inhibitors.</p>
    Fórmula:C17H12ClF3N2O
    Pureza:99.97%
    Forma y color:Solid
    Peso molecular:352.74
  • β-Amyloid (31-35)

    CAS:
    <p>β-Amyloid (31-35) (β-Amyloid 31-35) is the shortest sequence of native Amyloid-β peptide.</p>
    Fórmula:C25H47N5O6S
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:545.74
  • Benzetimide hydrochloride

    CAS:
    <p>Benzetimide hydrochloride (R4929) is an antagonist of muscarinic acetylcholine receptor.treatment neuroleptic-induced parkinsonism.</p>
    Fórmula:C23H27ClN2O2
    Pureza:99.32%
    Forma y color:Off-White Powder
    Peso molecular:398.93
  • Verubecestat tosylate

    CAS:
    Verubecestat (MK-8931/SCH 900931) is a potent BACE1 inhibitor, promising for Alzheimer’s, reducing Aβ in CSF by up to 92%.
    Fórmula:C25H26N4O4S2
    Forma y color:Solid
    Peso molecular:510.627
  • Rotundine

    CAS:
    <p>Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.</p>
    Fórmula:C21H25NO4
    Pureza:99.8% - 99.91%
    Forma y color:Off-White Solid
    Peso molecular:355.43
  • MK-0752 Sodium

    CAS:
    Sodium MK-0752 is a novel and potent gamma-secretase inhibitor that has been evaluated in clinical trials for the treatment of various types of cancer.
    Fórmula:C21H21ClF2NaO4S
    Forma y color:Solid
    Peso molecular:465.89
  • Metadoxine

    CAS:
    Metadoxine (Metadoxil) is a neurotransmitter stimulant.
    Fórmula:C8H11NO3·C5H7NO3
    Pureza:99.19%
    Forma y color:Off-White Powder
    Peso molecular:298.29
  • PRX-08066

    CAS:
    PRX-08066 is a selective 5-hydroxytryptamine receptor 2B (5-HT2BR, IC50= 3.4 nM) antagonist that induces selective vasodilation of pulmonary arteries.
    Fórmula:C19H17ClFN5S
    Pureza:97.79% - 98.07%
    Forma y color:Solid
    Peso molecular:401.89
  • Citalopram oxalate

    CAS:
    Citalopram oxalate: a serotonin uptake inhibitor, treats depression, lessens alcohol intake, favored for tardive dyskinesia over tricyclics.
    Fórmula:C22H23FN2O5
    Forma y color:Solid
    Peso molecular:414.43
  • CALP1 acetate


    <p>CALP1 acetate is a calmodulin (CaM) agonist (Kd of 88 µM) that binds to the CaM EF-hand/Ca2+-binding site.</p>
    Fórmula:C42H79N9O12
    Pureza:99.63%
    Forma y color:Solid
    Peso molecular:902.13
  • Isopropamide Iodide

    CAS:
    <p>Isopropamide iodide: long-acting anticholinergic, treats peptic ulcers, GI disorders, Alzheimer's.</p>
    Fórmula:C23H33IN2O
    Pureza:99.67%
    Forma y color:Solid
    Peso molecular:480.43