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Neurociencia

Neurociencia

Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.

Subcategorías de "Neurociencia"

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Se han encontrado 5516 productos de "Neurociencia"

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  • MPEP

    CAS:
    MPEP is a selective mGlu5 receptor antagonist with IC50 of 36 nM, exhibits no appreciable activity at mGlu1b/2/3/4a/7b/8a/6 receptors.
    Fórmula:C14H11N
    Pureza:99.54%
    Forma y color:Solid
    Peso molecular:193.24
  • Cyclodrine hydrochloride

    CAS:
    Cyclodrine hydrochloride is a dual cholinergic muscarinic receptor (mAChR) and nicotinic receptor (nAChR) antagonist that can be used in the study of
    Fórmula:C19H30ClNO3
    Pureza:98.59%
    Forma y color:Solid
    Peso molecular:355.9
  • RO-3

    CAS:
    <p>RO3 is a selective antagonist of homomeric P2X3 and heteromeric P2X2/3 receptor</p>
    Fórmula:C16H22N4O2
    Pureza:99.63%
    Forma y color:Solid
    Peso molecular:302.37
  • Syntide 2 acetate(108334-68-5 free base)


    <p>Syntide-2 acetate is a synthetic peptide recognized as a substrate by Ca2+/calmodulin-dependent protein kinase II (CaMKII; Km = 12 μM).</p>
    Fórmula:C70H126N20O20
    Pureza:99.74%
    Forma y color:Solid
    Peso molecular:1567.85
  • Amitriptyline

    CAS:
    <p>Amitriptyline: a tricyclic antidepressant used for depression and neuropathic pain.</p>
    Fórmula:C20H23N
    Pureza:98.24% - 99.64%
    Forma y color:Crystals Solid
    Peso molecular:277.4
  • Piboserod

    CAS:
    Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.
    Fórmula:C22H31N3O2
    Pureza:97.21% - 99.49%
    Forma y color:Solid
    Peso molecular:369.5
  • Phenibut (hydrochloride)

    CAS:
    Phenibut hydrochloride (3-Amino-4-phenylbutyric acid hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors.
    Fórmula:C10H14ClNO2
    Pureza:99.93%
    Forma y color:White Crystalline Powder
    Peso molecular:215.68
  • Nemifitide acetate(173240-15-8 free base)


    <p>Nemifitide acetate, synthetic 5-amino acid antidepressant, has quick effect, mimics MIF.</p>
    Fórmula:C35H47FN10O8
    Pureza:97.97%
    Forma y color:Solid
    Peso molecular:754.85
  • Lurasidone

    CAS:
    Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6
    Fórmula:C28H36N4O2S
    Pureza:99.78% - 99.91%
    Forma y color:Solid
    Peso molecular:492.68
  • Opiranserin hydrochloride

    CAS:
    Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μM
    Fórmula:C21H35ClN2O5
    Pureza:99.33%
    Forma y color:Solid
    Peso molecular:430.97
  • AF-353

    CAS:
    AF-353 (Ro-4), an effective and orally bioavailable antagonist of the P2X3/P2X2/3 receptor, inhibits human and rat P2X3 (pIC50= 8.0).
    Fórmula:C14H17IN4O2
    Pureza:92.98% - 99.356%
    Forma y color:Solid
    Peso molecular:400.21
  • LY2886721

    CAS:
    <p>LY2886721, a BACE inhibitor, is used for the therapy of Alzheimer's Disease.</p>
    Fórmula:C18H16F2N4O2S
    Pureza:99% - 99.75%
    Forma y color:Solid
    Peso molecular:390.41
  • Flibanserin

    CAS:
    <p>Flibanserin (Girosa) is a serotonergic antidepressant used to treat hypoactive sexual desire disorder.</p>
    Fórmula:C20H21F3N4O
    Pureza:99.37% - 99.93%
    Forma y color:White Powder
    Peso molecular:390.4
  • Ramosetron

    CAS:
    Ramosetron 是一种血清素 5-HT3 受体拮抗剂,用于治疗恶心和呕吐。它被认为比其他一代 5-HT3 拮抗剂如昂丹司琼具有更高的效力和更长的止吐作用。它还适用于治疗“男性以腹泻为主的肠易激综合征”。它仅获准在日本和选定的东南亚国家使用。
    Fórmula:C17H17N3O
    Pureza:98.84%
    Forma y color:Solid
    Peso molecular:279.34
  • PNU-282987 S enantiomer free base

    CAS:
    PNU-282987 S enantiomer free base is an agonist of α7 nicotinic acetylcholine receptor (α7 nAChR).
    Fórmula:C14H17ClN2O
    Pureza:99.74%
    Forma y color:Solid
    Peso molecular:264.75
  • SKF89976A hydrochloride

    CAS:
    <p>SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = 0.28 μM), GAT-2 (IC50s = 137.34 μM) and</p>
    Fórmula:C22H26ClNO2
    Pureza:98.02%
    Forma y color:Solid
    Peso molecular:371.9
  • Revefenacin

    CAS:
    Revefenacin (TD-4208) is a mAChR antagonist has a high affinity on M3 receptor( Ki : 0.18 nM),and potentially useful for the treatment of respiratory disease.
    Fórmula:C35H43N5O4
    Pureza:98.12%
    Forma y color:Solid
    Peso molecular:597.75
  • Sofpironium bromide

    CAS:
    <p>Sofpironium bromide (BBI4000) belongs to a class of drugs called anticholinergics, which exert their effect by blocking the action of acetylcholine.</p>
    Fórmula:C22H32BrNO5
    Pureza:98.85%
    Forma y color:Solid
    Peso molecular:470.4
  • Dinotefuran

    CAS:
    <p>Dinotefuran (MTI-446), a neonicotinoid insecticide, targets pests by blocking their nervous system.</p>
    Fórmula:C7H14N4O3
    Pureza:99.89%
    Forma y color:White Crystalline Powder
    Peso molecular:202.21
  • IC87201

    CAS:
    <p>IC87201 is a nNOS-PDZ/PSD-95-PDZ inhibitor. IC87201 showed great promise in cellular experiments and animal models of ischemic stroke and pain.</p>
    Fórmula:C13H10Cl2N4O
    Pureza:97.44%
    Forma y color:Solid
    Peso molecular:309.15