
Neurociencia
Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.
Subcategorías de "Neurociencia"
- Receptor 5-HT(993 productos)
- ACK(1 productos)
- AChR(612 productos)
- ATP Citrato Liasa(17 productos)
- Receptor adrenérgico(3.004 productos)
- BACE(36 productos)
- Beta amiloide(216 productos)
- CAMK(71 productos)
- Inhibidores de ciclooxigenasa (COX)(592 productos)
- Receptor de dopamina(433 productos)
- Receptor GABA(355 productos)
- Gamma-secretasa(63 productos)
- GluR(261 productos)
- GlyT(24 productos)
- Receptor de histamina(381 productos)
- LRRK2(41 productos)
- Receptor de melatonina(26 productos)
- NMDAR(15 productos)
- Receptor de OX(41 productos)
- Receptor de opioides(310 productos)
Mostrar 12 subcategorías más
Se han encontrado 5516 productos de "Neurociencia"
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MPEP
CAS:MPEP is a selective mGlu5 receptor antagonist with IC50 of 36 nM, exhibits no appreciable activity at mGlu1b/2/3/4a/7b/8a/6 receptors.Fórmula:C14H11NPureza:99.54%Forma y color:SolidPeso molecular:193.24Cyclodrine hydrochloride
CAS:Cyclodrine hydrochloride is a dual cholinergic muscarinic receptor (mAChR) and nicotinic receptor (nAChR) antagonist that can be used in the study ofFórmula:C19H30ClNO3Pureza:98.59%Forma y color:SolidPeso molecular:355.9RO-3
CAS:<p>RO3 is a selective antagonist of homomeric P2X3 and heteromeric P2X2/3 receptor</p>Fórmula:C16H22N4O2Pureza:99.63%Forma y color:SolidPeso molecular:302.37Syntide 2 acetate(108334-68-5 free base)
<p>Syntide-2 acetate is a synthetic peptide recognized as a substrate by Ca2+/calmodulin-dependent protein kinase II (CaMKII; Km = 12 μM).</p>Fórmula:C70H126N20O20Pureza:99.74%Forma y color:SolidPeso molecular:1567.85Amitriptyline
CAS:<p>Amitriptyline: a tricyclic antidepressant used for depression and neuropathic pain.</p>Fórmula:C20H23NPureza:98.24% - 99.64%Forma y color:Crystals SolidPeso molecular:277.4Piboserod
CAS:Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.Fórmula:C22H31N3O2Pureza:97.21% - 99.49%Forma y color:SolidPeso molecular:369.5Phenibut (hydrochloride)
CAS:Phenibut hydrochloride (3-Amino-4-phenylbutyric acid hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors.Fórmula:C10H14ClNO2Pureza:99.93%Forma y color:White Crystalline PowderPeso molecular:215.68Nemifitide acetate(173240-15-8 free base)
<p>Nemifitide acetate, synthetic 5-amino acid antidepressant, has quick effect, mimics MIF.</p>Fórmula:C35H47FN10O8Pureza:97.97%Forma y color:SolidPeso molecular:754.85Lurasidone
CAS:Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6Fórmula:C28H36N4O2SPureza:99.78% - 99.91%Forma y color:SolidPeso molecular:492.68Opiranserin hydrochloride
CAS:Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μMFórmula:C21H35ClN2O5Pureza:99.33%Forma y color:SolidPeso molecular:430.97AF-353
CAS:AF-353 (Ro-4), an effective and orally bioavailable antagonist of the P2X3/P2X2/3 receptor, inhibits human and rat P2X3 (pIC50= 8.0).Fórmula:C14H17IN4O2Pureza:92.98% - 99.356%Forma y color:SolidPeso molecular:400.21LY2886721
CAS:<p>LY2886721, a BACE inhibitor, is used for the therapy of Alzheimer's Disease.</p>Fórmula:C18H16F2N4O2SPureza:99% - 99.75%Forma y color:SolidPeso molecular:390.41Flibanserin
CAS:<p>Flibanserin (Girosa) is a serotonergic antidepressant used to treat hypoactive sexual desire disorder.</p>Fórmula:C20H21F3N4OPureza:99.37% - 99.93%Forma y color:White PowderPeso molecular:390.4Ramosetron
CAS:Ramosetron 是一种血清素 5-HT3 受体拮抗剂,用于治疗恶心和呕吐。它被认为比其他一代 5-HT3 拮抗剂如昂丹司琼具有更高的效力和更长的止吐作用。它还适用于治疗“男性以腹泻为主的肠易激综合征”。它仅获准在日本和选定的东南亚国家使用。Fórmula:C17H17N3OPureza:98.84%Forma y color:SolidPeso molecular:279.34PNU-282987 S enantiomer free base
CAS:PNU-282987 S enantiomer free base is an agonist of α7 nicotinic acetylcholine receptor (α7 nAChR).Fórmula:C14H17ClN2OPureza:99.74%Forma y color:SolidPeso molecular:264.75SKF89976A hydrochloride
CAS:<p>SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = 0.28 μM), GAT-2 (IC50s = 137.34 μM) and</p>Fórmula:C22H26ClNO2Pureza:98.02%Forma y color:SolidPeso molecular:371.9Revefenacin
CAS:Revefenacin (TD-4208) is a mAChR antagonist has a high affinity on M3 receptor( Ki : 0.18 nM),and potentially useful for the treatment of respiratory disease.Fórmula:C35H43N5O4Pureza:98.12%Forma y color:SolidPeso molecular:597.75Sofpironium bromide
CAS:<p>Sofpironium bromide (BBI4000) belongs to a class of drugs called anticholinergics, which exert their effect by blocking the action of acetylcholine.</p>Fórmula:C22H32BrNO5Pureza:98.85%Forma y color:SolidPeso molecular:470.4Dinotefuran
CAS:<p>Dinotefuran (MTI-446), a neonicotinoid insecticide, targets pests by blocking their nervous system.</p>Fórmula:C7H14N4O3Pureza:99.89%Forma y color:White Crystalline PowderPeso molecular:202.21IC87201
CAS:<p>IC87201 is a nNOS-PDZ/PSD-95-PDZ inhibitor. IC87201 showed great promise in cellular experiments and animal models of ischemic stroke and pain.</p>Fórmula:C13H10Cl2N4OPureza:97.44%Forma y color:SolidPeso molecular:309.15
